T61807 |
5-HT6/7 antagonist 1
|
131999-28-5
|
98.78%
|
|
5-HT6/7 antagonist 1 is a dual 5-HT6/7/2A and D2 receptor antagonist for the study of dementia and Alzheimer's disease.
|
TN1217 |
2'-O-Methylisoliquiritigenin
|
51828-10-5
|
98.75%
|
|
2'-O-Methylisoliquiritigenin, a compound synthesized by enzymes specifically induced in NR.2'-O-Methylisoliquiritigenin, isolated from the Arachis species, up-re...
|
T3431 |
Pardoprunox hydrochloride
|
269718-83-4
|
98.73%
|
|
Pardoprunox hydrochloride (SLV-308 hydrochloride) is a novel partial dopamine D2 and D3 receptor agonist and serotonin 5-HT1A receptor agonist, D2 (pKi = 8.1) an...
|
T1322 |
Bendazol
|
621-72-7
|
98.7%
|
|
Bendazol (Dibazol) is always used as the drug for hypertension and cerebral Angiospasm.
|
T14490 |
Talipexole dihydrochloride
|
36085-73-1
|
98.64%
|
|
Talipexole dihydrochloride (Domnin) is a dopamine D2 receptor agonist, α2-adrenoceptor agonist, and 5-HT3 receptor antagonist in both rat cortical and intestinal...
|
T10213 |
A-437203
|
220519-06-2
|
98.62%
|
|
A-437203 (Lu201640) is A kind of based on 1 h - pyrimidin - 2 - one sca ff old, selective, new powerful d3 receptor antagonist, on D2, d3, and D4 receptor, Ki val...
|
T12861 |
SB-277011
|
215803-78-4
|
98.61%
|
|
SB-277011 (SB-277011A) is a specific antagonist of the dopamine D3 receptor with pKi values of 8.0, 6.0, 5.0, and <5.2 for D3 receptor, D2 receptor, 5-HT1D, and ...
|
T7635 |
Raclopride
|
84225-95-6
|
98.6%
|
|
Raclopride is a selective antagonist of dopamine D2/D3 receptor.
|
TQ0084 |
Lumateperone Tosylate
|
1187020-80-9
|
98.57%
|
|
lumateperone Tosylate (ITI-007) is a 5-HT2A receptor antagonist (Ki: 0.54 nM), a SERT blocker (Ki: 61 nM), a partial agonist of presynaptic D2 receptors and an a...
|
T1476 |
Pramipexole
|
104632-26-0
|
98.54%
|
|
Pramipexole (SND 919) is a selective dopamine receptor agonist used in the therapy of Parkinson disease. Pramipexole therapy is associated with a low rate of tra...
|
T11079 |
NMI 8739
|
129024-87-9
|
98.51%
|
|
NMI 8739 (n-docosahexaenoyl dopamine) is an agonist of D2 autoreceptor. NMI 8739 reduces NO production and elicits concentration-dependent suppression of CCL-20,...
|
T31602 |
Ecopipam
|
112108-01-7
|
98.5%
|
|
Ecopipam (UNII-0X748O646K) is a potent, selective and orally active antagonist of dopamine D1/D5 receptor, with Kis of 1.2 nM and 2.0 nM, respectively. Ecopipam ...
|
T7070 |
Nomifensine maleate
|
32795-47-4
|
98.46%
|
|
Nomifensine maleate (Nomifensine (maleate)) is a selective inhibitor of dopamine uptake. Nomifensine maleate is used in adult attention deficit disorder.
|
T60835 |
SKF83959
|
80751-85-5
|
98.45%
|
|
SKF83959, a benzazepine analog, is a selective and potent partial agonist of the dopamine D1 receptor with Ki values of 1.18, 7.56, 920, and 399 nM for rat D1, D...
|
T5158 |
N-Desmethylclozapine
|
6104-71-8
|
98.45%
|
|
N-Desmethylclozapine (Desmethylclozapine) is an antagonist of serotonin (5-HT) receptor subtype 5-HT2C (IC50: 7.1 nM). It also is an antagonist at dopamine D4 re...
|
T60107 |
N-0500 HCl
|
100935-99-7
|
98.42%
|
|
N-0500 HCl ((-)-Propyl-9-hydroxynaphthoxazine Hydrochloride) is a very potent centrally acting DA receptor agonist. N-0500 HCl is a potent displacer of the speci...
|
T0990 |
Droperidol
|
548-73-2
|
98.38%
|
|
Droperidol (Dehydrobenzperidol) is a Dopamine-2 Receptor Antagonist. The mechanism of action of droperidol is as a Dopamine D2 Antagonist.
|
T24444 |
Medifoxamine
|
32359-34-5
|
98.35%
|
|
Medifoxamine (LG 152) is a selective non-monoamine oxidase inhibitor that exhibits antidepressant activity through inhibition of 5 HT reuptake.Medifoxamine prefe...
|
T71707L |
Romergoline 2HCl
|
|
98.33%
|
|
Romergoline 2HCl is a D1 agonist and D2 antagonist used in the study of Parkinson's disease.
|
T24613 |
PF-00217830
|
846032-02-8
|
98.30%
|
|
PF-00217830 is a serotonin 1A receptor agonist, dopamine D2 receptor agonist, and serotonin 2A receptor antagonist.PF-00217830 may be used in the study of schizo...
|