T2410 |
Nedaplatin
|
95734-82-0
|
98.69%
|
|
Nedaplatin is a derivative of cisplatin and DNA damage agent for tumor colony forming units (IC50: 94 μM). Containing a novel ring structure in which glycolate i...
|
T4010 |
Juglone
|
481-39-0
|
98.73%
|
|
Juglone is a natural naphthoquinone found in the black walnut (J. nigra) and other plants in the Juglandaceae family. Juglone also irreversibly inhibits peptidyl...
|
T4593 |
ISOPIMPINELLIN
|
482-27-9
|
98.74%
|
|
Antiviral, anti HIV.
|
T13791 |
2-(Methylamino)-1H-purin-6(7H)-one
|
10030-78-1
|
98.74%
|
|
2-(Methylamino)-1H-purin-6(7H)-one is an endogenous methylated nucleoside found in human fluids, is a modified nucleoside.
|
TN2202 |
Sempervirine
|
6882-99-1
|
98.81%
|
|
Sempervirine can unwind circular DNA, it shows selective inhibition of in vitro synthesis of cancer DNA .
|
T9150 |
SCR130
|
2377858-38-1
|
98.9%
|
|
1,7,9-Triazaspiro[4.5]dec-1-ene-6,10-dione, 2,4-bis(4-chlorophenyl)-8-thioxo- is enzyme inhibition, antiproliferative effects and antifungal activity.
|
TQ0184 |
Chebulinic acid
|
18942-26-2
|
98.91%
|
|
Chebulinic acid is a potent inhibitor of M. tuberculosis DNA gyrase. It also can inhibit SMAD-3 phosphorylation and H+ K+-ATPase activity.
|
T3157 |
COH29
|
1190932-38-7
|
98.92%
|
|
COH29 is an orally available, aromatically substituted thiazole and inhibitor of the human ribonucleotide reductase (RNR), with potential antineoplastic activity...
|
T2504 |
Pritelivir
|
348086-71-5
|
98.92%
|
|
Pritelivir (BAY 57-1293) is a potent helicase-primase inhibitor with active against HSV-1 and HSV-2 (IC50: 20 nM).
|
TN1990 |
Norathyriol
|
3542-72-1
|
98.93%
|
|
Norathyriol is a potent PTP1B inhibitor with good cell permeability and oral availability.
|
T9103 |
BVDV-IN-1
|
345651-04-9
|
98.93%
|
|
BVDV-IN-1 is a non-nucleoside inhibitor (NNI) of bovine viral diarrhea virus (BVDV), with an EC50 of 1.8 μM. It directly binds to a hydrophobic pocket of the BVD...
|
TN1134 |
Euscaphic acid
|
53155-25-2
|
98.93%
|
|
Euscaphic acid has anti-diabetic, and anti-inflammatory activities, it inhibits LPS-induced inflammatory responses by interference with the clustering of TRAF6 w...
|
T1120 |
Dacarbazine
|
4342-03-4
|
99%
|
|
Dacarbazine is an antineoplastic agent. It has significant activity against melanomas.
|
T2069 |
TH287
|
1609960-30-6
|
99%
|
|
TH287 is a potent inhibitor of MTH1 (NUDT1), less potent for MTH2, NUDT5, NUDT12, NUDT14, and NUDT16.
|
T0802 |
Procaine hydrochloride
|
51-05-8
|
99%
|
|
Procaine Hydrochloride is the hydrochloride salt form of procaine, a benzoic acid derivative with local anesthetic and antiarrhythmic properties. Procaine binds ...
|
T10936 |
D-I03
|
688342-78-1
|
99.04%
|
|
D-I03 is a selective RAD52 inhibitor with a Kd of 25.8 µM. D-I03 specifically inhibits RAD52-dependent single-chain annealing (SSA) and D-loop formation, with IC...
|
T12006 |
Metarrestin
|
1443414-10-5
|
99.04%
|
|
Metarrestin is a first-in-class perinucleolar compartment inhibitor with a favorable PK profile, which effectively suppresses metastasis. Metarrestin disrupts th...
|
T6632 |
Raltitrexed
|
112887-68-0
|
99.06%
|
|
Raltitrexed(IC50 of 9 nM), a thymidylate synthase inhibitor, is used for the inhibition of L1210 cell growth.
|
T13174 |
TMPyP4 tosylate
|
36951-72-1
|
99.11%
|
|
TMPyP4 tosylate is a quadruplex-specific ligand and is a telomerase inhibitor with antitumor effects in osteosarcoma cell lines.
|
T13231L |
Trovafloxacin mesylate
|
147059-75-4
|
99.12%
|
|
Trovafloxacin mesylate is an effective and selective inhibitor of pannexin 1 channel (PANX1, IC50 = 4 μM). Trovafloxacin mesylate exhibits potent activity agains...
|