T24239 |
K201
|
1038410-88-6
|
99.8%
|
|
K201 (JTV-519) is a Ca2+-dependent blocker and prevents abnormal Ca(2+) leak from the sarcoplasmic reticulum in the ischemic heart and skeletal muscle (SkM) by s...
|
TNU0864 |
HUP30
|
312747-21-0
|
99.8%
|
|
HUP30 is a potent vasodilating agent. HUP30 can stimulate soluble guanylyl cyclase, activate K+ channels, and block extracellular Ca2+ influx.
|
T2604 |
1-EBIO
|
10045-45-1
|
99.79%
|
|
1-EBIO (1-EBIO) is a calium channel agonist.
|
T1010 |
Verapamil hydrochloride
|
152-11-4
|
99.79%
|
|
Verapamil hydrochloride (Verapamil HCl) is a calcium channel blocker that is a class IV anti-arrhythmia agent.
|
T4727 |
Taurolithocholic acid sodium salt
|
6042-32-6
|
99.79%
|
|
Taurolithocholic acid sodium salt (Sodium taurolithocholate) is the major human metabolite, a bile acid which inhibits radioligand binding to muscarinic M1, but ...
|
T1234 |
5,5-Dimethyloxazolidine-2,4-dione
|
695-53-4
|
99.78%
|
|
5,5-Dimethyloxazolidine-2,4-dione (Dimethadione) is an anticonvulsant that is the active metabolite of TRIMETHADIONE.
|
T15423 |
GSK-7975A
|
1253186-56-9
|
99.78%
|
|
GSK-7975A is a potent and orally available inhibitor of CRAC channel.
|
T73587 |
KT-362 free base
|
93392-97-3
|
99.78%
|
|
KT-362 is a calcium channel blocker with antihypertensive properties that can be used in the study of cardiovascular disease.
|
TN1121 |
Evocarpine
|
15266-38-3
|
99.77%
|
|
Evocarpine shows antimycobacterial, and vasorelaxant effects, it can inhibit Ca2+ influx through voltage-dependent calcium channels.
|
T5120 |
Rhamnose
|
3615-41-6
|
99.77%
|
|
Addition of the Rhamnose (6-Deoxy-L-mannose)-rich polysaccharide, RROP-1, to normal human dermal fibroblasts (NHDFs) and human endothelial cells produced a dose-...
|
T27357 |
FPL-62129
|
95445-79-7
|
99.76%
|
|
FPL-62129 is a calcium channel antagonist and a novel angiotensin-converting enzyme inhibitor with vasodilator activity for the study of cardiovascular disease.
|
T1197 |
Trimebutine maleate
|
34140-59-5
|
99.76%
|
|
Trimebutine maleate (Polibutin) is a weak mu-opioid agonist and has antimuscarinic effects. Trimebutine is an agonist of peripheral mu, delta, and kappa opiate r...
|
T5114 |
Pyridaben
|
96489-71-3
|
99.75%
|
|
Pyridaben is a METI acaricide that inhibits mitochondrial electron transport at complex I (METI; Ki = 0.36 nmol/mg protein in rat brain mitochondria).
|
T28164 |
Nexopamil
|
136033-49-3
|
99.74%
|
|
Nexopamil (LU-49938) is a calcium channel antagonist and a 5-hydroxytryptamine 2A receptor antagonist. Nexopamil inhibits 5-HT-induced contraction and proliferat...
|
T8143 |
Bevantolol hydrochloride
|
42864-78-8
|
99.74%
|
|
Bevantolol hydrochloride (NC-1400 hydrochloride) is a β1-adrenoceptor antagonist that treatment angina pectoris and hypertension.
|
T4S1419 |
(±)-Praeruptorin A
|
73069-25-7
|
99.73%
|
|
1. (±)-Praeruptorin A could exhibit its anti-osteoclastogenic activity by inhibiting p38/Akt-c-Fos-NFATc1 signaling and PLCγ-independent Ca(2+) oscillation 2. Pr...
|
T76373L |
Ser-Ala-alloresact acetate
|
|
99.73%
|
|
Ser-Ala-alloresact acetate is a sperm-activating peptide (SAP) that is released by marine invertebrate eggs and plays an important role in fertilization.
|
T25372 |
EMD57033
|
147527-31-9
|
99.72%
|
|
EMD57033 is a cardiac troponin C (cTnC) activator, a dominant Ca2+ sensitizer, which functions by binding to cardiac/slow skeletal troponin C heterodimers to pro...
|
TQ0139 |
VU 0240551
|
893990-34-6
|
99.72%
|
|
VU 0240551 is a selective antagonist of neuronal K-Cl cotransporter KCC2 inhibitor with an IC50 of 560 nM. VU 0240551 inhibits L-type calcium channels and hERG.
|
T0728 |
Ethosuximide
|
77-67-8
|
99.72%
|
|
Ethosuximide (Zarontin) is an anticonvulsant, blocks the low voltage-activated T-type calcium channel used in the treatment of absence seizures unaccompanied by ...
|