TN3260 |
8(14),15-Isopimaradien-3-ol
|
4728-30-7
|
98%
|
|
ent-8(14),15-pimaradien-3beta-ol (8(14),15-Isopimaradien-3-ol) can induce vascular relaxation. It displays high antibacterial activities (MIC values lower than 1...
|
TN1913 |
Marmin
|
14957-38-1
|
98%
|
|
Marmin have anti-ulcer effects, which are ascribed primarily to the maintenance of the mucosal barrier integrity and inhibition of gastric motor activity and sec...
|
T10713 |
CCR4 antagonist 2
|
2206788-99-8
|
98%
|
|
CCR4 antagonist 2 (Compound 31) is a novel potent, orally bioavailable small molecule antagonists of CC chemokine receptor 4 (CCR4) that inhibits Treg traffickin...
|
TN1367 |
Alismol
|
87827-55-2
|
98%
|
|
Alismol has antihypertensive action, it decreases cardiac output, heart rate and left ventricular pressure, but it increases coronary flow, it has been used for ...
|
TQ0153 |
Mibefradil
|
116644-53-2
|
98%
|
|
Mibefradil is a calcium channel blocker with moderate selectivity for T-type Ca2+ channels (IC50s: 2.7 μM and 18.6 μM for T-type and L-type currents).
|
T35935 |
D-myo-Inositol-1,4,5-triphosphate trisodium
|
141611-10-1
|
98%
|
|
D-myo-Inositol-1,4,5-triphosphate trisodium (Inositol 1,4,5-trisphosphate trisodium) is a second messenger produced in cells by phospholipase C-mediated hydrolys...
|
T11080 |
Dopropidil
|
79700-61-1
|
98%
|
|
Dopropidil is a new anti-angina pectoris calcium regulator, which has intracellular calcium antagonist activity and anti-ischemic effects in various predicted an...
|
T12625 |
(R)-Lercanidipine-d3 hydrochloride
|
1217724-52-1
|
98%
|
|
(R)-lercanidipine D3 hydrochloride is a deuterium labeled (R)-Lercanidipine hydrochloride. (R)-Lercanidipine D3 (hydrochloride) is a calcium channel blocker.
|
TN5109 |
Taxezopidine L
|
219749-76-5
|
98%
|
|
Taxezopidines K and taxezopidine L can markedly inhibit Ca2+-induced depolymerization of microtubules.
|
TN2641 |
15-Methoxypinusolidic acid
|
769928-72-5
|
98%
|
|
15-Methoxypinusolidic acid has anti-inflammatory effects, it inhibits LPS-induced iNOS expression and NO production, independent on MAPK and NF-kappaB. 15-Methox...
|
T12205L |
Trans-Ned 19
|
1354235-96-3
|
98%
|
|
trans-Ned 19 is a NAADP antagonist and TPC blocker and inhibits the calcium signal in human umbilical vein endothelial cells and the rat aorta relaxation in resp...
|
T19882 |
Bryonolic acid
|
24480-45-3
|
98%
|
|
Bryonolic acid (20-epi-Bryonolic acid), a triterpenoid extracted from Sandoricum indicum, possesses immunomodulatory, anti-inflammatory, antioxidant and anticanc...
|
T15366 |
Gabapentin enacarbil
|
478296-72-9
|
98%
|
|
Gabapentin enacarbil (XP-13512) is a prodrug for the anticonvulsant and analgesic drug gabapentin. Gabapentin enacarbil provides sustained dose-proportional expo...
|
T13879 |
(S)-Verapamil hydrochloride
|
36622-28-3
|
98%
|
|
(S)-Verapamil hydrochloride is an inhibitor of leukotriene C4 (LTC4) and calcein transport by MRP1,and leads to the death of potentially resistant tumor cells.
|
TN4051 |
Fargesone B
|
116424-70-5
|
98%
|
|
Fargesone B inhibits the vascular smooth muscle contraction by suppressing the voltage- and receptor-activated calcium influxes in a nonselective manner.
|
TN3568 |
Calceolarioside A
|
84744-28-5
|
98%
|
|
Calceolarioside A shows potent activity against visceral leishmaniasis. It can induce a dose-related aggregant effect on rabbit platelets, which may be partly re...
|
T12244 |
Norverapamil
|
67018-85-3
|
98%
|
|
Norverapamil is a blocker of L-type calcium channel and an inhibitor of P-glycoprotein (P-gp) function .
|
T2782L |
Catharanthine Tartrate(2468-21-5(free base))
|
T2782L
|
99.98%
|
|
Catharanthine Tartrate is a natural product isolated from Madagascar periwinkle, Catharanthine Tartrate inhibits voltage-operated L-type Ca2+ channel, with anti-...
|
T6777 |
Bay K 8644
|
71145-03-4
|
99.97%
|
|
Bay K 8644 (SQ 28,873) is a potent, selective activator of L-type Ca2+ channel with IC50 of 17.3 nM.
|
T14844 |
BX430
|
688309-70-8
|
99.95%
|
|
BX430 is used for chronic pain and cardiovascular disease and it is a potent and selective noncompetitive allosteric human P2X4 receptor channels antagonist with...
|