T80161 |
ω-Conotoxin SO3
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441284-32-8
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98%
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ω-Conotoxin SO3 is an analgesic peptide that functions as an antagonist to N-type voltage-sensitive calcium channels, and can be isolated from the venom of Conus...
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T80185 |
Huwentoxin I
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769973-37-7
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98%
|
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Huwentoxin I (HWTX-I) is a peptide toxin that targets and inhibits both voltage-gated sodium channels and N-type calcium channels. It effectively inhibits sodium...
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T80247 |
Caloxin 3A1
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98%
|
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Caloxin 3A1, a biologically active peptide, is a member of the caloxins, which are inhibitors of the extracellular plasma membrane (PM) Ca2+ pumps. Specifically,...
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T80441 |
FS-2
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98%
|
|
FS-2 is a potent, specific inhibitor of L-type CaV channels, effectively impeding high K+ or glucose-induced L-type Ca2+ influx in RIN beta cells [1].
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T80443 |
ω-Conotoxin MVIID
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98%
|
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ω-Conotoxin MVIID (SNX-238) is a peptide from the Conus genus that inhibits the ω-Conotoxin-GVIA-sensitive, high-threshold calcium (Ca 2+) current in fish retina...
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T80446 |
ω-Conotoxin FVIA
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|
98%
|
|
ω-Conotoxin FVIA is an inhibitor of N-type Ca²⁺ channels (Caᵥ2.2), shown to alleviate mechanical and thermal pain abnormalities in a rat model of caudal nerve in...
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T80448 |
ω-Conotoxin CVIF
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|
98%
|
|
ω-Conotoxin CVIF is a selective inhibitor of Ca v 2.2 channels, demonstrating an IC50 value of 34.3 nM in isolated rat DRG neurons. Its blockade of Cav2.2 channe...
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T80449 |
ω-Conotoxin CVIE
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98%
|
|
ω-Conotoxin CVIE selectively inhibits voltage-gated Ca^2+ channels (Ca_v 2.2) [1].
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T80457 |
ω-Conotoxin Bu8
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98%
|
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ω-Conotoxin Bu8 is a 25-amino-acid-residue ω-conotoxin that features three disulfide bridges. It selectively and potently inhibits rat CaV2.2-mediated depolariza...
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T80458 |
ω-Conotoxin CVIA
|
325164-06-5
|
98%
|
|
ω-Conotoxin CVIA, a 27-amino acid neuropeptide, functions as a blocker of voltage-sensitive calcium channels (VSCCs) [1].
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T80459 |
ω-Conotoxin CnVIIA
|
760212-36-0
|
98%
|
|
ω-Conotoxin CnVIIA, a 27-amino-acid neuropeptide toxin, serves as an N-type calcium current blocker [1].
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T80496 |
Kurtoxin
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98%
|
|
Kurtoxin is a selective Cav3 (T-type) voltage-gated Ca2+ channel gating inhibitor, exhibiting a dissociation constant (Kd) of 15 nM for the Cav3.1 (α1G T-type) C...
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T80501 |
Myr-TAT-CBD3
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98%
|
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Myr-TAT-CBD3, a CRMP2-CaV2.2 interaction inhibitor, has been shown to significantly attenuate carrageenan-induced thermal hypersensitivity and reverse thermal hy...
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T80520 |
ω-conotoxin MoVIA
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|
98%
|
|
ω-Conotoxin MVIIA is a potent, selective inhibitor of Ca_v2.2, exhibiting an IC_50 of 0.33 μM in the SH-SY5Y fluorimetric hCa_v2.2 assay [1].
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T80554 |
Myoregulin
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98%
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Myoregulin (MLN peptide), a regulin family member, modulates muscle performance through intracellular calcium handling. It directly interacts with the sarcoplasm...
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T80555 |
Myoregulin TFA
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98%
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Myoregulin (MLN peptide) TFA, belonging to the regulin family, is a regulator of muscle performance through modulation of intracellular calcium dynamics. It spec...
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T80556 |
Wt hMLN
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98%
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Wild-type human myoregulin (wt hMLN) is a microprotein that inhibits the sarcoplasmic reticulum Ca²⁺ pump (SERCA), playing a crucial role in the regulation of ca...
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T80681 |
γ-Glutamylserine TFA
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98%
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γ-Glutamylserine TFA (γ-Glu-Ser TFA) serves as a calcium receptor activator and is utilized in research focused on Parkinson's disease, diabetes, and obesity [1]...
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T80975 |
TMDJ-035
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2681302-83-8
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98%
|
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TMDJ-035 is a selective inhibitor of the RyR2 (ryanodine receptor 2). It effectively suppresses abnormal calcium (Ca^2+) waves and transients in isolated cardiom...
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T12358 |
Palonidipine
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96515-73-0
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98%
|
|
Palonidipine is an antagonist of calcium, is potential for the therapy of angina-pectoris and hypertension.
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