T5457 |
SN 6
|
415697-08-4
|
98%
|
|
SN 6 (SN6) is a selective Na+/Ca2+ exchanger (NCX) inhibitor (IC50s of NCX1: 2.9 μM , NCX2: 16 μM ,NCX3: 8.6 μM)
|
T7540 |
2,5-Di-tert-butylhydroquinone
|
88-58-4
|
98%
|
|
2,5-Di-tert-butylhydroquinone (BHQ) is an effective and selective endoplasmic reticulum Ca2+-ATPase inhibitor.
|
T10884 |
CRAC intermediate 1
|
1249343-86-9
|
97.92%
|
|
CRAC intermediate 1 (5-(S)-Fluorowillardiine) is a key intermediate in the chemical synthesis of a series of CRAC channel inhibitors.
|
TN2078 |
Pinocembrin chalcone
|
4197-97-1
|
97.82%
|
|
Pinocembrin chalcone is an inhibitor of tyrosinase with antimutagenic effects. Pinocembrin chalcone can be used in studies about the prevention of gastric ulcers...
|
T22788 |
FPL64176
|
120934-96-5
|
97.78%
|
|
FPL64176 is a L-type calcium channels activator.
|
T12385 |
PD0176078
|
248922-46-5
|
97.76%
|
|
PD0176078 () is a newly blocker of N-type Calcium channel.
|
T6856 |
Halofuginone
|
55837-20-2
|
97.67%
|
|
Halofuginone (RU-19110), the competitive inhibitor of prolyl-tRNA synthetase(Ki=18.3 nM), could also down-regulate Smad3 and blocked TGF-β signaling at 10 ng/ml ...
|
T34782 |
Tamolarizine
|
93035-32-6
|
97.46%
|
|
Tamolarizine (Tamolarizine free base) free base is a novel calcium antagonist.
|
T8867 |
RO2959 Hydrochloride
|
1219927-22-6
|
97.42%
|
|
RO2959 Hydrochloride (RO2959 HCl) is a potent and selective inhibitor of CRAC channel(IC50: 402 nM). It is also a potent inhibitor of human IL-2.
|
T25263 |
Clopimozide
|
53179-12-7
|
97.18%
|
|
Clopimozide (R-29764) acts as a calcium channel antagonist and inhibits [3H] nilandipine binding.Clopimozide is a novel and orally available long-acting antischi...
|
T37705 |
1,2,4-Trihydroxybenzene
|
533-73-3
|
97.16%
|
|
1,2,4-Trihydroxybenzene (Benzene-1,2,4-triol) is a by-product of coffee bean roasting and is found in mouse, arabica coffee.1,2,4-Trihydroxybenzene is a benzotri...
|
T15553 |
Iganidipine
|
119687-33-1
|
96.85%
|
|
Iganidipine(NKY 722) is a new water-soluble Ca2+ antagonist with antihypertensive activity for research and neurological related diseases.
|
TP1911L |
CALP3 acetate(261969-05-5 free base)
|
TP1911L
|
96.49%
|
|
CALP3 acetate is a potent Ca2+ channel blocker that activates EF hand motifs of Ca2+-binding proteins. CALP3 acetate can functionally mimic increased [Ca2+]i by ...
|
T6848 |
GSK1016790A
|
942206-85-1
|
96.25%
|
|
GSK1016790A (GSK101) (GSK101) is a novel, potent activator of TRPV4 (transient receptor potential vanilloid 4) with EC50 of 34 nM in choroid plexus epithelial ce...
|
T24984 |
5J-4
|
827001-82-1
|
96.12%
|
|
5J-4 is a potent a blocker of calcium release-activated calcium (CRAC) channel and store-operated calcium entry (SOCE). 5J-4 reduces the production of IL-17 and ...
|
T10814 |
Cinacalcet metabolite M4
|
104774-87-0
|
95.28%
|
|
Cinacalcet metabolite M4 (Rarechem AL BW 1078) is a metabolite of Cinacalcet. Cinacalcet is an allosteric agonist of Ca receptor.
|
TN5073 |
Strophanthidin
|
66-28-4
|
93%
|
|
Strophanthidin (Strophanthidine) can induce calcium overload in vivo.
|
T1215 |
Nicardipine hydrochloride
|
54527-84-3
|
100%
|
|
Nicardipine hydrochloride (YC-93 Hydrochloride) is the hydrochloride salt form of nicardipine, a synthetic derivative of nitrophenyl-pyridine and potent calcium ...
|
T1641 |
Strontium ranelate
|
135459-87-9
|
100%
|
|
Strontium ranelate (S12911), a strontium (II) salt of the ranelic acid, is a medication for osteoporosis. Studies indicate it can also slow the course of osteoar...
|
T0207 |
Ranolazine dihydrochloride
|
95635-56-6
|
100%
|
|
Ranolazine dihydrochloride (Ranolazine 2HCl) , an antianginal agent, can treat arrhythmia via a novel mechanism of action (inhibition of the late phase of the in...
|