T8389 |
Trifluoperazine
|
117-89-5
|
99.03%
|
|
Trifluoperazine (trifluoroperazine) is a Dopamine D2 receptor inhibitor(IC50 : 1.2 nM), and Treatment of schizophrenia.
|
T3546 |
STO-609
|
52029-86-4
|
98.95%
|
|
STO-609 is a specific and cell-permeable inhibitor of the Ca2+/calmodulin-dependent protein kinase kinase (CaM-KK) for recombinant CaM-KKα/KKβ (Ki: 80/15 ng/mL)....
|
T23525 |
W-9 hydrochloride
|
69762-85-2
|
98.9%
|
|
W-9 hydrochloride is a calmodulin antagonist.
|
T2694 |
KN-62
|
127191-97-3
|
98.77%
|
|
KN-62 is a potent and specific Ca2+/calmodulin-dependent protein kinase II (CaMKII) inhibitor with Ki of 0.9 μM.
|
T1659 |
Melatonin
|
73-31-4
|
98.71%
|
|
Melatonin (Melatonine) is a biogenic amine that is found in animals and plants. In mammals, melatonin is produced by the PINEAL GLAND. Its secretion increases in...
|
T23522 |
W-13 hydrochloride
|
88519-57-7
|
98.51%
|
|
W-13 hydrochloride (W-13 HCl) is a calmodulin antagonist.
|
T68064 |
Elziverine
|
95520-81-3
|
98.43%
|
|
Elziverine is an orally available small molecule calmodulin antagonist.Elziverine in vitro treatment inhibited Ca-loading-induced acanthocyte formation in SHRSP,...
|
T14860 |
CaMKII-IN-1
|
1208123-85-6
|
98.35%
|
|
CaMKII-IN-1 is a potent and highly selective CaMKII inhibitor (IC50: 63 nM). It has significantly high selectivity against CaMKIV, p38a, MLCK, Akt1, and PKC.
|
TN1008 |
Psoralenoside
|
905954-17-8
|
98.17%
|
|
Psoralenoside is a natural product isolated from the fruits of Psoralea corylifolia, shows estrogen-like activity, osteoblastic proliferation accelerating activi...
|
T10667 |
Calmidazolium chloride
|
57265-65-3
|
98.06%
|
|
Calmidazolium chloride (R 24571) is a calmodulin (CaMK) antagonist (Kd = 3 nM), antagonizing CaM-dependent phosphodiesterase(IC50 = 0.15 μM) and calmodulin-induc...
|
T1158 |
Phenoxybenzamine hydrochloride
|
63-92-3
|
98.04%
|
|
Phenoxybenzamine hydrochloride (NCI-c01661) is the hydrochloride salt form of phenoxybenzamine, a synthetic, dibenzamine alpha-adrenergic antagonist with antihyp...
|
TP1217L |
Autocamtide 2 TFA(129198-88-5 free base)
|
TP1217L
|
98%
|
|
Autocamtide 2 TFA is a highly selective peptide substrate of calcium/calmodulin-dependent protein kinase II (CaMKII). Autocamtide 2 TFA can be used in the CaMKII...
|
T4185 |
Lavendustin C
|
125697-93-0
|
97.77%
|
|
lavendustin C (NSC 666251) is a potent inhibitor of epidermal growth factor (EGF) receptor-associated tyrosine kinase.
|
TQ0137 |
A-484954
|
142557-61-7
|
97.47%
|
|
A-484954 (A 484954) is a highly specific eukaryotic elongation factor-2 (eEF2, IC50: 280 nM) inhibitor.
|
TP1921L1 |
Autocamtide-2-related inhibitory peptide, myristoylated acetate(201422-04-0 free base)
|
TP1921L1
|
97.03%
|
|
Autocamtide-2-related inhibitory peptide, myristoylated acetate is a CaM kinase II inhibitor; enhanced cell permeable derivative of Autocamtide-2-related inhibit...
|
TP1271L |
Calmodulin-Dependent Protein Kinase II 290-309 acetate
|
|
96.7%
|
|
Calmodulin-Dependent Protein Kinase II 290-309 acetate is an effective antagonist of Ca2+/calmodulin-dependent protein kinase II (IC50 = 52 nM).
|
T2159 |
CaMKP Inhibitor
|
52789-62-5
|
96.55%
|
|
CaMKP Inhibitor can inhibit CaMKP.
|
TP1216 |
CaM kinase II inhibitor TFA salt
|
TP1216
|
100%
|
|
CaM kinase II inhibitor TFA salt (Autocamtide-2-related inhibitory peptide (TFA)) is a highly specific and potent inhibitor of CaMKII with an IC50 of 40 nM.
|
T1222 |
Trifluoperazine dihydrochloride
|
440-17-5
|
100%
|
|
Trifluoperazine dihydrochloride (SKF5019) is a potent dopamine D2 receptor inhibitor used as an antipsychotic and an antiemetic.
|
T16791 |
Rottlerin
|
82-08-6
|
|
|
Rottlerin (NSC-56346) is a natural product purified from Mallotus Philippinensis and is a specific PKC inhibitor (IC50: PKCδ of 3-6 μM, PKCα,β,γ of 30-42 μM, PKC...
|