Adrenergic Receptor

The adrenergic receptors or adrenoceptors are a class of G protein-coupled receptors that are targets of many catecholamines like norepinephrine (noradrenaline) and epinephrine (adrenaline) produced by the body, but also many medications like beta blockers, β2 agonists and α2 agonists, which are used to treat high blood pressure and asthma, for example.

Cat. No.	Product name	CAS No.	Purity
T5159	Olodaterol hydrochloride	869477-96-3	99.58%
T5159	Olodaterol hydrochloride (BI-1744 HCl) is a novel, long-acting β2-adrenergic agonist (EC50s: 97.7 nM for the human β2-adrenoceptor) that exerts its pharmacologic...
T7056	Dronedarone	141626-36-0	99.58%
T7056	Dronedarone (SR 33589) is an amiodarone analogue which has an effective and promising treatment for Atrial fibrillation.
T6565	Levobetaxolol hydrochloride	116209-55-3	99.57%
T6565	Levobetaxolol hydrochloride ((S)-Betaxolol hydrochloride) is a beta-adrenergic receptor inhibitor (beta blocker), used to lower the pressure in the eye in treati...
T13106	TD-5471 hydrochloride	530084-35-6	99.57%
T13106	TD-5471 hydrochloride is a selective and potent long-acting human β2-adrenergic receptor agonist for the treatment of chronic obstructive pulmonary disease (COPD...
T0226	Betaxolol hydrochloride	63659-19-8	99.56%
T0226	Betaxolol hydrochloride (SL 75212 HCl) is a cardioselective beta-blocker used in the treatment of hypertension.Betaxolol hydrochloride has not been linked to ins...
T0279	Metaraminol tartrate	33402-03-8	99.53%
T0279	Metaraminol tartrate (Metaradrine tartrate) is a sympathomimetic agent that acts predominantly at alpha-1 adrenergic receptors. It has been used primarily as a v...
T0031L2	Ziprasidone	146939-27-7	99.53%
T0031L2	Ziprasidone (Geodon) is a united 5-HT (serotonin) and dopamine receptor antagonist which shows potent effects of antipsychotic activity.
T1496	Amiodarone hydrochloride	19774-82-4	99.49%
T1496	Amiodarone hydrochloride (Amiodarone HCl) is an antianginal and class III antiarrhythmic drug. It increases the duration of ventricular and atrial muscle action ...
TN1922	Meranzin hydrate	5875-49-0	99.49%
TN1922	Meranzin hydrate exhibits antidepressive and prokinetic-like effects through the regulation of the common mediator, the alpha 2-adrenoceptor , and α±-amino-3-hyd...
T2889	Isoferulic acid	537-73-5	99.49%
T2889	Isoferulic acid (Hesperetate) exhibits hypoglycemic properties.
T22882	JP1302	80259-18-3	99.48%
T22882	JP1302 is a selective α2C adrenoceptor antagonist with a Kb value of 16 nM and a Ki of 28 nM for human α2C receptors.JP1302 has antidepressant activity, disrupts...
T68161L	Tienoxolol FA		99.47%
T68161L	Tienoxolol FA is a small molecule beta-adrenergic receptor antagonist used in the treatment of cardiovascular disease and in the study of hypertension and cardia...
T13016	SR59230A	174689-39-5	99.46%
T13016	SR59230A is a potent, selective antagonist of β3-adrenergic receptor(β3, β1, and β2 receptors with IC50s of 40, 408, and 648 nM , respectively).
T30586L	Brefonalol HCl		99.45%
T30586L	Brefonalol HCl is an ADRA antagonist used in the treatment of neurological disorders and cardiovascular diseases and can be used in the study of angina pectoris,...
T10998	Deriglidole	122830-14-2	99.45%
T10998	Deriglidole (SL 86-0715) is a peripheral adrenergic receptor antagonist that is a selective inhibitor of alpha2 receptors. Deriglidole inhibits colistin and Idaz...
T77565	Fluparoxan hydrochloride	105227-44-9	99.44%
T77565	Fluparoxan hydrochloride is a highly selective and potent α2-adrenoceptor antagonist for the prevention, amelioration or treatment of neurodevelopmental disorder...
T6408	Betaxolol	63659-18-7	99.43%
T6408	Betaxolol (Kerlone) is a selective beta1 adrenergic receptor blocker used in the treatment of hypertension and glaucoma.
T13376	YS-49	132836-42-1	99.42%
T13376	YS-49 is an activator of PI3K/Akt (a downstream target of RhoA).
T5S2059	Glaucine	475-81-0	99.42%
T5S2059	Glaucine has antitussive, antioxidative potential and antiviral activities, it may be an anti-arthritic agent, it can enhance LPS and zymosan-induced IL-10 produ...
T0696	Naftopidil	57149-07-2	99.4%
T0696	Naftopidil (KT-611) (INN, marketed under the brand name Flivas), an antihypertensive medicine, is used as a selective α1-adrenergic receptor antagonist or α-bloc...