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Adrenergic Receptor

The adrenergic receptors or adrenoceptors are a class of G protein-coupled receptors that are targets of many catecholamines like norepinephrine (noradrenaline) and epinephrine (adrenaline) produced by the body, but also many medications like beta blockers, β2 agonists and α2 agonists, which are used to treat high blood pressure and asthma, for example.
Signaling Pathways | Target | TargetMol
Cat. No. Product name CAS No. Purity Chemical Structure
T80477 Muscarinic toxin 3 873336-87-9 98%
Muscarinic toxin 3
Muscarinic toxin 3 (MT3), a potent non-competitive antagonist of mAChR and adrenoceptors, exhibits pIC50 values of 6.71 for M1, 8.79 for M4, 8.86 for α1A, 7.57 f...
TN1797 Isorhoifolin 552-57-8 98%
Isorhoifolin
Isorhoifolin and vicenin II are main compounds of ethyl acetate fraction (EAcF) obtained from Erythrina velutina leaves, EAcF increases the cardiac contractile f...
T81798 Mibenratide TFA 98%
Mibenratide TFA
Mibenratide TFA, a small cyclic peptide, functions as an adrenergic β1 receptor antagonist and has potential applications in heart failure research [1].
T15042 D2343 72734-63-5 98%
D2343
D2343 is an agonist of β2-adrenoceptor. It also is an inhibitor of α1- adrenoceptor.
T6663 Scopine hydrochloride 85700-55-6 98%
Scopine hydrochloride
Scopine hydrochloride (6,7-Epoxytropine hydrochloride), a metabolite of anisodine, acts as an α1-adrenergic receptor agonist and is utilized in managing acute ci...
T16769 Ro 363 74513-77-2 98%
Ro 363
RO 363 is an effective inotropic stimulant and is a cardiovascular modulator that decreases diastolic blood pressure and pronounces increases in myocardial contr...
TN2267 Tetrahydroalstonine 6474-90-4 98%
Tetrahydroalstonine
Tetrahydroalstonine is an indole alkaloid extracted from the fruit of Rhazya stricta and is a selective α2-adrenoceptor antagonist. tetrahydroalstonine has shown...
TN3368 Akuammigine 642-17-1 98%
Akuammigine
Akuammigine has in vitro antimalarial activity. Akuammigine competitively antagonizes the effect of noradrenaline on postsynaptic alpha-adrenoceptors, yielding p...
T11786 KUL-7211 racemate 911196-40-2 98%
KUL-7211 racemate
KUL 7211, a selective β-adrenoceptor agonist, exists as a racemate, referred to as KUL 7211 racemate, which is the mixture of its enantiomers.
T12815 (S)-Terazosin 109351-33-9 98%
(S)-Terazosin
(S)-Terazosin is an active S-enantiomer of Terazosin. (S)-Terazosin is a potent and high-affinity antagonist of α-adrenoceptor(α1a, α1b and α1d-adrenoceptor with...
T13285 Vatinoxan hydrochloride 130466-38-5 98%
Vatinoxan hydrochloride
Vatinoxan hydrochloride is an antagonist of the peripheral α2 adrenergic receptors.
TN3507 Beta-Yohimbine 549-84-8 98%
beta-Yohimbine
Beta-Yohimbine has approximately twice as toxic as yohimbine and corynanthine about one fifth as toxic. Beta-yohimbine has alpha-1 and alpha-2 adrenoceptor block...
T21411 Isoproterenol 7683-59-2 98%
Isoproterenol
Isoproterenol (Norisodrine) is a non-selective and orally active β-adrenoceptor agonist.Isoproterenol is a potent peripheral vasodilator and bronchodilator.Isopr...
T68129 Picumeterol 130641-36-0 98%
Picumeterol
Picumeterol(GR 114297A) is a potent and selective β2 adrenergic receptor agonist. In vitro and in vivo trials, Picumeterol produced long-lasting airway smooth mu...
T14287 Ancarolol 75748-50-4 98%
Ancarolol
Ancarolol is a blocking agent of beta-adrenergic.
TN5061 Stephanine 517-63-5 98%
Stephanine
l-Stephanine is a potent and highly selective alpha 1 adrenoceptor blocker, inhibits anococcygeus muscle contraction induced by phenylephrine with pA2 values of ...
T11010 Detomidine carboxylic acid 115664-39-6 98%
Detomidine carboxylic acid
Detomidine carboxylic acid is the main urine metabolite of detomidine. Detomidine is a synthetic α2-adrenergic agonist and an animal analgesic. Detomidine also h...
T68023 Tolnapersine 70312-00-4 98%
Tolnapersine
Tolnapersine is a mixed dopamine agonist and alpha-adrenoceptor antagonist.
T0101 Doxazosin mesylate 77883-43-3 99.98%
Doxazosin mesylate
Doxazosin mesylate (UK 33274 mesylate)(UK 33274) is a quinazoline-derivative. It is a selectively antagonizes postsynaptic α1-adrenergic receptors.
T1619 Trazodone hydrochloride 25332-39-2 99.98%
Trazodone hydrochloride
Trazodone hydrochloride (Trazodone HCl) is a serotonin uptake inhibitor that is used as an antidepressive agent. It has been shown to be effective in patients wi...
Muscarinic toxin 3
T80477
Muscarinic toxin 3 (MT3), a potent non-competitive antagonist of mAChR and adrenoceptors, exhibits pIC50 values of 6.71 for M1, 8.79 for M4, 8.86 for α1A, 7.57 f...
Isorhoifolin
TN1797
Isorhoifolin and vicenin II are main compounds of ethyl acetate fraction (EAcF) obtained from Erythrina velutina leaves, EAcF increases the cardiac contractile f...
Mibenratide TFA
T81798
Mibenratide TFA, a small cyclic peptide, functions as an adrenergic β1 receptor antagonist and has potential applications in heart failure research [1].
D2343
T15042
D2343 is an agonist of β2-adrenoceptor. It also is an inhibitor of α1- adrenoceptor.
Scopine hydrochloride
T6663
Scopine hydrochloride (6,7-Epoxytropine hydrochloride), a metabolite of anisodine, acts as an α1-adrenergic receptor agonist and is utilized in managing acute ci...
Ro 363
T16769
RO 363 is an effective inotropic stimulant and is a cardiovascular modulator that decreases diastolic blood pressure and pronounces increases in myocardial contr...
Tetrahydroalstonine
TN2267
Tetrahydroalstonine is an indole alkaloid extracted from the fruit of Rhazya stricta and is a selective α2-adrenoceptor antagonist. tetrahydroalstonine has shown...
Akuammigine
TN3368
Akuammigine has in vitro antimalarial activity. Akuammigine competitively antagonizes the effect of noradrenaline on postsynaptic alpha-adrenoceptors, yielding p...
KUL-7211 racemate
T11786
KUL 7211, a selective β-adrenoceptor agonist, exists as a racemate, referred to as KUL 7211 racemate, which is the mixture of its enantiomers.
(S)-Terazosin
T12815
(S)-Terazosin is an active S-enantiomer of Terazosin. (S)-Terazosin is a potent and high-affinity antagonist of α-adrenoceptor(α1a, α1b and α1d-adrenoceptor with...
Vatinoxan hydrochloride
T13285
Vatinoxan hydrochloride is an antagonist of the peripheral α2 adrenergic receptors.
beta-Yohimbine
TN3507
Beta-Yohimbine has approximately twice as toxic as yohimbine and corynanthine about one fifth as toxic. Beta-yohimbine has alpha-1 and alpha-2 adrenoceptor block...
Isoproterenol
T21411
Isoproterenol (Norisodrine) is a non-selective and orally active β-adrenoceptor agonist.Isoproterenol is a potent peripheral vasodilator and bronchodilator.Isopr...
Picumeterol
T68129
Picumeterol(GR 114297A) is a potent and selective β2 adrenergic receptor agonist. In vitro and in vivo trials, Picumeterol produced long-lasting airway smooth mu...
Ancarolol
T14287
Ancarolol is a blocking agent of beta-adrenergic.
Stephanine
TN5061
l-Stephanine is a potent and highly selective alpha 1 adrenoceptor blocker, inhibits anococcygeus muscle contraction induced by phenylephrine with pA2 values of ...
Detomidine carboxylic acid
T11010
Detomidine carboxylic acid is the main urine metabolite of detomidine. Detomidine is a synthetic α2-adrenergic agonist and an animal analgesic. Detomidine also h...
Tolnapersine
T68023
Tolnapersine is a mixed dopamine agonist and alpha-adrenoceptor antagonist.
Doxazosin mesylate
T0101
Doxazosin mesylate (UK 33274 mesylate)(UK 33274) is a quinazoline-derivative. It is a selectively antagonizes postsynaptic α1-adrenergic receptors.
Trazodone hydrochloride
T1619
Trazodone hydrochloride (Trazodone HCl) is a serotonin uptake inhibitor that is used as an antidepressive agent. It has been shown to be effective in patients wi...
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TargetMol