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Adrenergic Receptor

The adrenergic receptors or adrenoceptors are a class of G protein-coupled receptors that are targets of many catecholamines like norepinephrine (noradrenaline) and epinephrine (adrenaline) produced by the body, but also many medications like beta blockers, β2 agonists and α2 agonists, which are used to treat high blood pressure and asthma, for example.
Signaling Pathways | Target | TargetMol
Cat. No. Product name CAS No. Purity Chemical Structure
TN3507 Beta-Yohimbine 549-84-8 98%
beta-Yohimbine
Beta-Yohimbine has approximately twice as toxic as yohimbine and corynanthine about one fifth as toxic. Beta-yohimbine has alpha-1 and alpha-2 adrenoceptor block...
T21411 Isoproterenol 7683-59-2 98%
Isoproterenol
Isoproterenol (Norisodrine) is a non-selective and orally active β-adrenoceptor agonist.Isoproterenol is a potent peripheral vasodilator and bronchodilator.Isopr...
T68129 Picumeterol 130641-36-0 98%
Picumeterol
Picumeterol(GR 114297A) is a potent and selective β2 adrenergic receptor agonist. In vitro and in vivo trials, Picumeterol produced long-lasting airway smooth mu...
T14287 Ancarolol 75748-50-4 98%
Ancarolol
Ancarolol is a blocking agent of beta-adrenergic.
TN5061 Stephanine 517-63-5 98%
Stephanine
l-Stephanine is a potent and highly selective alpha 1 adrenoceptor blocker, inhibits anococcygeus muscle contraction induced by phenylephrine with pA2 values of ...
T11010 Detomidine carboxylic acid 115664-39-6 98%
Detomidine carboxylic acid
Detomidine carboxylic acid is the main urine metabolite of detomidine. Detomidine is a synthetic α2-adrenergic agonist and an animal analgesic. Detomidine also h...
T68023 Tolnapersine 70312-00-4 98%
Tolnapersine
Tolnapersine is a mixed dopamine agonist and alpha-adrenoceptor antagonist.
T0101 Doxazosin mesylate 77883-43-3 99.98%
Doxazosin mesylate
Doxazosin mesylate (UK 33274 mesylate)(UK 33274) is a quinazoline-derivative. It is a selectively antagonizes postsynaptic α1-adrenergic receptors.
T1619 Trazodone hydrochloride 25332-39-2 99.98%
Trazodone hydrochloride
Trazodone hydrochloride (Trazodone HCl) is a serotonin uptake inhibitor that is used as an antidepressive agent. It has been shown to be effective in patients wi...
T2142 Yohimbine hydrochloride 65-19-0 99.98%
Yohimbine hydrochloride
Yohimbine hydrochloride (Antagonil) is a plant alkaloid with alpha-2-adrenergic blocking activity. Yohimbine has been used as a mydriatic and in the treatment of...
T1282 Carteolol hydrochloride 51781-21-6 99.97%
Carteolol hydrochloride
Carteolol hydrochloride (Abbott-43326) is a synthetic quinolinone derivative, antihypertensive Carteolol Hydrochloride is a nonselective beta-adrenoceptor blocki...
T6701 Terazosin hydrochloride dihydrate 70024-40-7 99.97%
Terazosin hydrochloride dihydrate
Terazosin hydrochloride dihydrate (Heitrin dihydrate) is a selective α1-adrenoceptor antagonist, used for treatment of symptoms of an enlarged prostate (BPH).
T21066 Norepinephrine bitartrate salt 3414-63-9 99.97%
Norepinephrine bitartrate salt
Norepinephrine bitartrate salt is an adrenergic neurotransmitter.
T0871 Noradrenaline bitartrate 69815-49-2 99.97%
Noradrenaline bitartrate
Norepinephrine bitartrate acts directly on the α- and β-adrenergic receptors. Norepinephrine Bitartrate is a bitartrate salt of norepinephrine, a synthetic pheny...
T6703 Tetrahydrozoline hydrochloride 522-48-5 99.97%
Tetrahydrozoline hydrochloride
Tetrahydrozoline hydrochloride (Murine Plus) is an imidazoline derivative with alpha receptor agonist activity.
T2524 Dexmedetomidine 113775-47-6 99.96%
Dexmedetomidine
Dexmedetomidine is a Central alpha-2 Adrenergic Agonist. The mechanism of action of dexmedetomidine is as an Adrenergic alpha2-Agonist. The physiologic effect of...
T1539 Iloperidone 133454-47-4 99.96%
Iloperidone
Iloperidone (HP 873) is an atypical antipsychotic agent that is used for treatment of schizophrenia.
T1071L DL-Adrenaline Hydrochloride 329-63-5 99.95%
DL-Adrenaline Hydrochloride
DL-Adrenaline Hydrochloride is the hydrochloride salt of the naturally occurring sympathomimetic amine with vasoconstricting, intraocular pressure-reducing activ...
T0210 Tamsulosin hydrochloride 106463-17-6 99.95%
Tamsulosin hydrochloride
Tamsulosin hydrochloride (Flomax hydrochloride) is the hydrochloride salt of tamsulosin, a sulfonamide derivative with α1 adrenergic antagonist activity.
T9220 Naftopidil hydrochloride 1164469-60-6 99.95%
Naftopidil hydrochloride
Naftopidil hydrochloride (BM-15275 hydrochloride) is a selective alpha1-adrenoceptor antagonist with Ki of 3.7 nM, 20 nM and 1.2 nM for the cloned human α1a-adre...
beta-Yohimbine
TN3507
Beta-Yohimbine has approximately twice as toxic as yohimbine and corynanthine about one fifth as toxic. Beta-yohimbine has alpha-1 and alpha-2 adrenoceptor block...
Isoproterenol
T21411
Isoproterenol (Norisodrine) is a non-selective and orally active β-adrenoceptor agonist.Isoproterenol is a potent peripheral vasodilator and bronchodilator.Isopr...
Picumeterol
T68129
Picumeterol(GR 114297A) is a potent and selective β2 adrenergic receptor agonist. In vitro and in vivo trials, Picumeterol produced long-lasting airway smooth mu...
Ancarolol
T14287
Ancarolol is a blocking agent of beta-adrenergic.
Stephanine
TN5061
l-Stephanine is a potent and highly selective alpha 1 adrenoceptor blocker, inhibits anococcygeus muscle contraction induced by phenylephrine with pA2 values of ...
Detomidine carboxylic acid
T11010
Detomidine carboxylic acid is the main urine metabolite of detomidine. Detomidine is a synthetic α2-adrenergic agonist and an animal analgesic. Detomidine also h...
Tolnapersine
T68023
Tolnapersine is a mixed dopamine agonist and alpha-adrenoceptor antagonist.
Doxazosin mesylate
T0101
Doxazosin mesylate (UK 33274 mesylate)(UK 33274) is a quinazoline-derivative. It is a selectively antagonizes postsynaptic α1-adrenergic receptors.
Trazodone hydrochloride
T1619
Trazodone hydrochloride (Trazodone HCl) is a serotonin uptake inhibitor that is used as an antidepressive agent. It has been shown to be effective in patients wi...
Yohimbine hydrochloride
T2142
Yohimbine hydrochloride (Antagonil) is a plant alkaloid with alpha-2-adrenergic blocking activity. Yohimbine has been used as a mydriatic and in the treatment of...
Carteolol hydrochloride
T1282
Carteolol hydrochloride (Abbott-43326) is a synthetic quinolinone derivative, antihypertensive Carteolol Hydrochloride is a nonselective beta-adrenoceptor blocki...
Terazosin hydrochloride dihydrate
T6701
Terazosin hydrochloride dihydrate (Heitrin dihydrate) is a selective α1-adrenoceptor antagonist, used for treatment of symptoms of an enlarged prostate (BPH).
Norepinephrine bitartrate salt
T21066
Norepinephrine bitartrate salt is an adrenergic neurotransmitter.
Noradrenaline bitartrate
T0871
Norepinephrine bitartrate acts directly on the α- and β-adrenergic receptors. Norepinephrine Bitartrate is a bitartrate salt of norepinephrine, a synthetic pheny...
Tetrahydrozoline hydrochloride
T6703
Tetrahydrozoline hydrochloride (Murine Plus) is an imidazoline derivative with alpha receptor agonist activity.
Dexmedetomidine
T2524
Dexmedetomidine is a Central alpha-2 Adrenergic Agonist. The mechanism of action of dexmedetomidine is as an Adrenergic alpha2-Agonist. The physiologic effect of...
Iloperidone
T1539
Iloperidone (HP 873) is an atypical antipsychotic agent that is used for treatment of schizophrenia.
DL-Adrenaline Hydrochloride
T1071L
DL-Adrenaline Hydrochloride is the hydrochloride salt of the naturally occurring sympathomimetic amine with vasoconstricting, intraocular pressure-reducing activ...
Tamsulosin hydrochloride
T0210
Tamsulosin hydrochloride (Flomax hydrochloride) is the hydrochloride salt of tamsulosin, a sulfonamide derivative with α1 adrenergic antagonist activity.
Naftopidil hydrochloride
T9220
Naftopidil hydrochloride (BM-15275 hydrochloride) is a selective alpha1-adrenoceptor antagonist with Ki of 3.7 nM, 20 nM and 1.2 nM for the cloned human α1a-adre...
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TargetMol