Adrenergic Receptor

The adrenergic receptors or adrenoceptors are a class of G protein-coupled receptors that are targets of many catecholamines like norepinephrine (noradrenaline) and epinephrine (adrenaline) produced by the body, but also many medications like beta blockers, β2 agonists and α2 agonists, which are used to treat high blood pressure and asthma, for example.

Cat. No.	Product name	CAS No.	Purity
T23283	2-Methoxyidazoxan monohydrochloride	109544-45-8	99.13%
T23283	L-Albizziin (2-Methoxyidazoxan monohydrochloride) is a highly potent selective antagonist of the alpha 2r adrenergic receptor, with little or no antagonistic eff...
T31750	Faxeladol	433265-65-7	99.13%
T31750	Faxeladol, a potent adrenergic absorption inhibitor and serotonin reuptake inhibitor, is a small-molecule Opioid receptor agonist that can be used to study neuro...
T10631L	Bucindolol Formate		99.11%
T10631L	Bucindolol Formatel is a blocker of β1-adrenergic receptor. Bucindolol exhibits intrinsic sympathomimetic activity. Bucindolol can be used in the research of hea...
T0445	Promethazine	60-87-7	99.11%
T0445	Promethazine (Proazamine) is an analogue of anti-glaucoma prostaglandin (PG) .
T28922	Taprizosin	210538-44-6	99.11%
T28922	Taprizosin（UK-338003） is a selective and orally active α1-adrenoceptor antagonist for vasodilatation in the treatment of benign prostatic hyperplasia.
T2226	Pergolide mesylate	66104-23-2	99.09%
T2226	Pergolide mesylate salt(LY127809) is a long-acting dopamine agonist which has been used to treat PARKINSON DISEASE and HYPERPROLACTINEMIA but withdrawn from some...
T3284	Carazolol	57775-29-8	99.08%
T3284	Carazolol (Suacron) is a high-affinity antagonist/partial inverse agonist (also referred to as a beta blocker) of the β-adrenergic receptor.
T7160	Lofexidine	31036-80-3	99.08%
T7160	Lofexidine is a selective α2-receptor agonist, Lofexidine reduces narcotic withdrawal symptoms.
T62893	SM-2470	99899-45-3	99.05%
T62893	SM-2470 is an α1-adrenoceptor antagonist with antihypertensive activity that decreases anterior ganglionic adrenal nerve activity and aortic descending nerve act...
T6872	L755507	159182-43-1	99.04%
T6872	L755507 is an effective, selective agonist of β3-AR（IC50=35 nM）.
T8389	Trifluoperazine	117-89-5	99.03%
T8389	Trifluoperazine (trifluoroperazine) is a Dopamine D2 receptor inhibitor(IC50 : 1.2 nM), and Treatment of schizophrenia.
T23302	(S)-(-)-Propranolol hydrochloride	4199-10-4	99.02%
T23302	(S)-(-)-Propranolol hydrochloride is an adrenergic receptor antagonist with potential anticancer activity that may improve the prognosis of burn patients.
T20898	(R)-Propranolol hydrochloride	13071-11-9	99.01%
T20898	(R)-Propranolol hydrochloride (Dexpropranolol hydrochloride) is the less active enantiomer of the anti-adrenoceptor (β-adrenoceptor) antagonist propranolol. Prop...
T0270	Hydrocortisone 17-butyrate	13609-67-1	99.01%
T0270	Hydrocortisone 17-butyrate (Cortisol 17-butyrate) is a synthetic glucocorticoid receptor agonist with antiinflammatory, antipruritic and vasoconstrictive effects...
T1139	Salbutamol	18559-94-9	99%
T1139	Salbutamol (Albuterol) stimulates beta2-adrenergic receptors in the lungs, thereby activating the enzyme adenylate cyclase that catalyzes the conversion of ATP t...
T12970	Solabegron	252920-94-8	98.99%
T12970	Solabegron (GW 427353) is a selective agonist of β3-adrenergic receptor, stimulating cAMP accumulation in Chinese hamster ovary cells expressing the human β3-AR(...
T12643	(R)-Terazosin	109351-34-0	98.96%
T12643	(R)-Terazosin is an active R-enantiomer of Terazosin. (R)-Terazosin is a potent antagonist of α1-adrenoceptor (α1a, α1b and α1d-adrenoceptor with Ki values of 6....
T30027	Amosulalol	85320-68-9	98.91%
T30027	Amosulalol is a combined alpha and beta adrenoceptor antagonist.
T26822	Bisaramil hydrochloride	96480-44-3	98.90%
T26822	Bisaramil hydrochloride (Bisaramil) is a novel diazabicyclononane antiarrhythmic compound that inhibits the generation of free radicals.Bisaramil hydrochloride b...
T1738	Taxifolin	480-18-2	98.9%
T1738	Taxifolin (Dihydroquercetin) is a flavonoid in many plants such as Taxus chinensis, Siberian larch, Cedrus deodara and so on.