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Adenosine Receptor

The adenosine receptors are a class of purinergic G protein-coupled receptors with adenosine as the endogenous ligand. There are four known types of adenosine receptors in humans: A1, A2A, A2B and A3; each is encoded by a different gene.
Signaling Pathways | Target | TargetMol
Cat. No. Product name CAS No. Purity Chemical Structure
T0853L Adenosine 5'-monophosphate monohydrate 18422-05-4 97.68%
Adenosine 5'-monophosphate monohydrate
Adenosine 5'-monophosphate monohydrate (5'-AMP) , also known as 5'-adenylic acid, is a nucleotide that is used as a monomer in RNA. It is an ester of phosphoric ...
T23518 VUF 5574 280570-45-8 97.63%
VUF 5574
VUF 5574 is a selective antagonist of adenosine A3 receptor with a Ki of 4.03 nM for the recombinant human receptor.
T5081 Adenine monohydrochloride hemihydrate 6055-72-7 97.61%
Adenine monohydrochloride hemihydrate
Adenine monohydrochloride hemihydrate is a high affinity adenine receptor agonist (Ki = 18 nM at rat adenine receptor). It inhibits forskolin-stimulated cAMP for...
T16140 MRS 1754 264622-58-4 97.48%
MRS 1754
MRS 1754 is a selective antagonist radioligand for the A2B adenosine receptor. It has a very low affinity for A1 and A3 receptors of both humans and rats.
T27629 ISAM-140 932191-62-3 97.41%
ISAM-140
ISAM-140 is a potent and highly selective antagonist of A2B adenosine receptor.
T23203 PSB-603 1092351-10-4 97.13%
PSB-603
PSB-603 is a selective antagonist of Adenosine A2B receptor(Ki = 0.553 nM) with anti-inflammatory effects.
T67972L Amp579 TFA 96.67%
Amp579 TFA
Amp579 TFA is a novel adenosine A1/A2a receptor agonist that induces acute and delayed preconditioning against myocardial shock in vivo.
T23016 MRS1220 183721-15-5 96.59%
MRS1220
MRS1220, a highly potent and selective human A3 adenosine receptor (hA3AR) antagonist with a Ki of 0.59 nM, has therapeutic potential for the research of disease...
T68132L Quercetin-3'-o-phosphate TEA 95.50%
Quercetin-3'-o-phosphate TEA
Quercetin-3'-o-phosphate TEA (Quercetin 3'-phosphate TEA) is an adenosine A receptor antagonist that can be used to prevent and treat metabolic disorders.
T7021 ZM241385 139180-30-6 95.28%
ZM241385
ZM-241385 is a high-affinity antagonist ligand selective for the adenosine A2A receptor.
T14127 Adenosine A1 receptor activator T62 40312-34-3 95.00%
Adenosine A1 receptor activator T62
Adenosine A1 receptor activator T62 is an allosteric enhancer of adenosine A1 receptor, and it produces antinociception in animal models of acute pain and also r...
T0665 Xanthine 69-89-6 89.06%
Xanthine
Xanthine (Isoxanthine) is a product on the pathway of purine degradation. Xanthine is subsequently converted to uric acid by the action of the Xanthine oxidase e...
T2671 Regadenoson 313348-27-5 100%
Regadenoson
Regadenoson (CVT-3146) is an adenosine derivative and selective A2A adenosine receptor agonist with coronary vasodilating activity. Upon administration, regadeno...
T9180 LUF6096 1116652-18-6 100%
LUF6096
LUF6096 (CF-602) is a potent allosteric enhancer of the adenosine A3 receptor. LUF6096 is able to allosterically enhance agonist binding. LUF6096 shows low ortho...
T10248 Adenosine antagonist-1 431040-19-6 100%
Adenosine antagonist-1
Adenosine antagonist-1 acts as an adenosine A3 receptor (AA3R) antagonist.
T72067 DPTN dihydrochloride 325767-87-1 100%
DPTN dihydrochloride
DPTN dihydrochloride is a potent and selective A3AR antagonist with Ki values of 1.65, 9.61 and 8.53 nM in human, mouse and rat, respectively.
T8613 1-Ethyl-6-aminouracil 41862-09-3
1-Ethyl-6-aminouracil
1-Ethyl-6-aminouracil (6-AMINO-1-ETHYL-1H-PYRIMIDINE-2,4-DIONE) is an intermediate in the synthesis of a series of new substituted Xanthines which have high affi...
T16263 N6-Cyclopentyladenosine 41552-82-3 98%
N6-Cyclopentyladenosine
N6-Cyclopentyladenosine (CPA) is a selective agonist of the adenosine A1 receptor and can be used to mimic the action of the adenosine A1 receptor, with Ki's of ...
T29112 VPC171 1018830-99-3 98%
VPC171
VPC171 is a novel adenosine A1 receptor positive allosteric modulator (PAM).
T15715 LAS101057 925676-48-8 98%
LAS101057
LAS101057 is a novel orally available and potent and selective A2B receptor antagonist for the study of asthma.
Adenosine 5'-monophosphate monohydrate
T0853L
Adenosine 5'-monophosphate monohydrate (5'-AMP) , also known as 5'-adenylic acid, is a nucleotide that is used as a monomer in RNA. It is an ester of phosphoric ...
VUF 5574
T23518
VUF 5574 is a selective antagonist of adenosine A3 receptor with a Ki of 4.03 nM for the recombinant human receptor.
Adenine monohydrochloride hemihydrate
T5081
Adenine monohydrochloride hemihydrate is a high affinity adenine receptor agonist (Ki = 18 nM at rat adenine receptor). It inhibits forskolin-stimulated cAMP for...
MRS 1754
T16140
MRS 1754 is a selective antagonist radioligand for the A2B adenosine receptor. It has a very low affinity for A1 and A3 receptors of both humans and rats.
ISAM-140
T27629
ISAM-140 is a potent and highly selective antagonist of A2B adenosine receptor.
PSB-603
T23203
PSB-603 is a selective antagonist of Adenosine A2B receptor(Ki = 0.553 nM) with anti-inflammatory effects.
Amp579 TFA
T67972L
Amp579 TFA is a novel adenosine A1/A2a receptor agonist that induces acute and delayed preconditioning against myocardial shock in vivo.
MRS1220
T23016
MRS1220, a highly potent and selective human A3 adenosine receptor (hA3AR) antagonist with a Ki of 0.59 nM, has therapeutic potential for the research of disease...
Quercetin-3'-o-phosphate TEA
T68132L
Quercetin-3'-o-phosphate TEA (Quercetin 3'-phosphate TEA) is an adenosine A receptor antagonist that can be used to prevent and treat metabolic disorders.
ZM241385
T7021
ZM-241385 is a high-affinity antagonist ligand selective for the adenosine A2A receptor.
Adenosine A1 receptor activator T62
T14127
Adenosine A1 receptor activator T62 is an allosteric enhancer of adenosine A1 receptor, and it produces antinociception in animal models of acute pain and also r...
Xanthine
T0665
Xanthine (Isoxanthine) is a product on the pathway of purine degradation. Xanthine is subsequently converted to uric acid by the action of the Xanthine oxidase e...
Regadenoson
T2671
Regadenoson (CVT-3146) is an adenosine derivative and selective A2A adenosine receptor agonist with coronary vasodilating activity. Upon administration, regadeno...
LUF6096
T9180
LUF6096 (CF-602) is a potent allosteric enhancer of the adenosine A3 receptor. LUF6096 is able to allosterically enhance agonist binding. LUF6096 shows low ortho...
Adenosine antagonist-1
T10248
Adenosine antagonist-1 acts as an adenosine A3 receptor (AA3R) antagonist.
DPTN dihydrochloride
T72067
DPTN dihydrochloride is a potent and selective A3AR antagonist with Ki values of 1.65, 9.61 and 8.53 nM in human, mouse and rat, respectively.
1-Ethyl-6-aminouracil
T8613
1-Ethyl-6-aminouracil (6-AMINO-1-ETHYL-1H-PYRIMIDINE-2,4-DIONE) is an intermediate in the synthesis of a series of new substituted Xanthines which have high affi...
N6-Cyclopentyladenosine
T16263
N6-Cyclopentyladenosine (CPA) is a selective agonist of the adenosine A1 receptor and can be used to mimic the action of the adenosine A1 receptor, with Ki's of ...
VPC171
T29112
VPC171 is a novel adenosine A1 receptor positive allosteric modulator (PAM).
LAS101057
T15715
LAS101057 is a novel orally available and potent and selective A2B receptor antagonist for the study of asthma.
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TargetMol