Home Tools

Adenosine Receptor

The adenosine receptors are a class of purinergic G protein-coupled receptors with adenosine as the endogenous ligand. There are four known types of adenosine receptors in humans: A1, A2A, A2B and A3; each is encoded by a different gene.

Cat. No.	Product name	CAS No.	Purity
T23201	PSB 1115	152529-79-8	99.24%
T23201	human A2B adenosine receptor antagonist
T16980	Taminadenant	1337962-47-6	99.2%
T16980	Taminadenant is an adenosine receptor antagonist.
T15655	KFM19	133058-72-7	99.18%
T15655	KFM19 is a potent and selective adenosine receptor (A1-receptor) antagonist (IC50 : 50 nM) for the study of neurological disorders.
T0892	Diphylline	479-18-5	99.1%
T0892	Diphylline (Diprophylline) is a xanthine derivative. Diphylline exerts bronchodilator effects and to a lesser extent vasodilator and diuretic properties. Diphyll...
T14506	BAY 60-6583	910487-58-0	98.87%
T14506	BAY 60-6583 is a potent, high-affinity adenosine A2B receptor agonist (EC50 = 3 nM) with affinity for A2B receptors that exceeds that for A1, A2A, and A3 recepto...
TQ0125	Capadenoson	544417-40-5	98.85%
TQ0125	Capadenoson (BAY 68-4986) is a selective adenosine-A1 receptor agonist.
T10058	A2B receptor antagonist 1	531506-36-2	98.83%
T10058	A2B receptor antagonist 1 (EXAMPLE 9B) is a potent A2B adenosine receptor antagonist.
T8551	Nitrobenzylthioinosine	38048-32-7	98.83%
T8551	Nitrobenzylthioinosine (NBMPR) is an inhibitor of ENT1 transporter that binds to ENT1 transporter with high affinity.
T6441	CGS 21680 Hydrochloride	124431-80-7	98.81%
T6441	CGS 21680 Hydrochloride (CGS 21680 HCl)(IC50=22 nM), an adenosine receptor agonist, exhibits 140-fold potency in A2 receptor over A1 receptor.
T27800	LAS38096	851371-22-7	98.71%
T27800	LAS38096 is an A2B adenosine receptor antagonist (Ki : 17 nM) that is potent, selective and efficient .
T22234	Alloxazine	490-59-5	98.68%
T22234	Alloxazine (Isoalloxazine) is an A2 receptor antagonist, which is approximately 10-fold more selective for the A2B receptor than for the A2A receptor.
T5S1895	Norisoboldine	23599-69-1	98.64%
T5S1895	1. Norisoboldine ((+)-Laurelliptine) might be a potential therapeutic agent for rheumatoid arthritis, and it functions through protecting joint destruction as we...
T6552	Istradefylline	155270-99-8	98.57%
T6552	Istradefylline (KW-6002)(Ki of 2.2 nM) is a selective adenosine A2A receptor (A2AR) antagonist, which is under development in Phase 3 trails. It has been used in...
T26641L	Apadenoson TFA		98.40%
T26641L	Apadenoson TFA is a potent adenosine A2A receptor (A2AR) agonist that can be used to improve survival in patients infected with SARS.
T0853L	Adenosine 5'-monophosphate monohydrate	18422-05-4	98.36%
T0853L	Adenosine 5'-monophosphate monohydrate (5'-AMP) , also known as 5'-adenylic acid, is a nucleotide that is used as a monomer in RNA. It is an ester of phosphoric ...
T12160	N6-Cyclohexyladenosine	36396-99-3	98.31%
T12160	N6-Cyclohexyladenosine (CHA) is a selective agonist of A1 receptor with EC50 of 8.2 Nm. N6-Cyclohexyladenosine exerts anticonvulsant effects and protects against...
T7683	Adenosine amine congener	96760-69-9	98.29%
T7683	Adenosine amine congener (ADAC) (ADAC) is an agonist of selective A1 adenosine receptor,.
T6115	Fostamatinib	901119-35-5	98.24%
T6115	Fostamatinib (R788)(IC50 of 41 nM), which is a prodrug of the active metabolite R406, is a Syk inhibitor. It does not work on Lyn.
T22031	ANR 94	634924-89-3	98.21%
T22031	ANR94 is a potent, selective antagonist of the adenosine A2A receptor (AA2AR), exhibiting a K_i value of 46 nM for the human AA2AR (hAA2AR). This compound shows ...
T4290	Preladenant	377727-87-2	98.18%
T4290	Preladenant (SCH-420814) is an orally bioavailable antagonist of the adenosine A2A receptor (Ki: 1.1 nM) and has >1000-fold selectivity over all other adenosine ...