Adenosine Receptor

The adenosine receptors are a class of purinergic G protein-coupled receptors with adenosine as the endogenous ligand. There are four known types of adenosine receptors in humans: A1, A2A, A2B and A3; each is encoded by a different gene.

Cat. No.	Product name	CAS No.	Purity
T27323	FK-453	121524-18-3	99.69%
T27323	FK-453 is a potent antagonist of non-xanthine adenosine A1 receptor with diuretic and renal vasodilatory activity.
T1083	Theophylline	58-55-9	99.65%
T1083	Theophylline (1,3-Dimethylxanthine) is a methyl xanthine derivative from tea with diuretic, smooth muscle relaxant, bronchial dilation, cardiac and central nervo...
T28881	Sulmazole	73384-60-8	99.64%
T28881	Sulmazole (AR-L 115-BS) is a small molecule Sulmazole is a small molecule cGMP-PDE inhibitor.Sulmazole is a competitive inhibitor of A1 adenosine receptors.Sulma...
T28861	ST-1535	496955-42-1	99.63%
T28861	ST 1535 is a potent and orally active antagonist of A2A adenosine receptor with antiparkinsonian activity and antitremorigenic effects. ST 1535 exhibits the pote...
T14944	CGS 15943	104615-18-1	99.63%
T14944	CGS 15943 is an orally bioavailable non-xanthine antagonist of Adenosine Receptor. In transfected CHO cells, its Ki for human A1, A2A, A2B, and A3 Adenosine Rec...
T4265	AZD4635	1321514-06-0	99.61%
T4265	AZD4635 (HTL1071) is a new-type adenosine 2A receptor (A2AR) inhibitor(Ki=1.7 nM).
T12159	APNEA	89705-21-5	99.58%
T12159	APNEA ((2R,3R,4S,5R)-2-[6-[2-(4-aminophenyl)ethylamino]purin-9-yl]-5-(hydroxymethyl)oxolane-3,4-diol) is a non-selective agonist of adenosine A3 receptor.
T10822	Cirsimarin	13020-19-4	99.55%
T10822	Cirsimarin (Cirsitakaoside) is a flavonoid isolated from Microtea debilis. It shows a potent antilipogenic effect and decreases adipose tissue deposition in mice...
T17117	Tonapofylline	340021-17-2	99.52%
T17117	Tonapofylline is an orally active and selective antagonist of the A1 adenosine receptor (Ki: 7.4 nM for human A1). Tonapofylline can be used in studies about hea...
T4006	Pentostatin	53910-25-1	99.47%
T4006	Pentostatin (CI-825) is an extremely effective and irreversible inhibitor of adenosine deaminase (Ki: 2.5 pM).
T6884	Namodenoson	163042-96-4	99.4%
T6884	Namodenoson (2-Cl-IB-MECA) is an adenosine A3 receptor agonist.
T28748	Selodenoson	110299-05-3	99.33%
T28748	Selodenoson (RG-14202) is a selective adenosine A1 receptor agonist used to slow the heart rate in patients with atrial fibrillation and to treat arrhythmias.
T7736	2-Chloroadenosine	146-77-0	99.24%
T7736	2-Chloroadenosine (CADO) is a metabolically stable analog of adenosine that binds to adenosine A1, A2A, and A3 receptors( Ki:300, 80, and 1,900 nM, respectively)...
T23201	PSB 1115	152529-79-8	99.24%
T23201	human A2B adenosine receptor antagonist
T16980	Taminadenant	1337962-47-6	99.2%
T16980	Taminadenant is an adenosine receptor antagonist.
T15655	KFM19	133058-72-7	99.18%
T15655	KFM19 is a potent and selective adenosine receptor (A1-receptor) antagonist (IC50 : 50 nM) for the study of neurological disorders.
T0892	Diphylline	479-18-5	99.1%
T0892	Diphylline (Diprophylline) is a xanthine derivative. Diphylline exerts bronchodilator effects and to a lesser extent vasodilator and diuretic properties. Diphyll...
T14506	BAY 60-6583	910487-58-0	98.87%
T14506	BAY 60-6583 is a potent, high-affinity adenosine A2B receptor agonist (EC50 = 3 nM) with affinity for A2B receptors that exceeds that for A1, A2A, and A3 recepto...
TQ0125	Capadenoson	544417-40-5	98.85%
TQ0125	Capadenoson (BAY 68-4986) is a selective adenosine-A1 receptor agonist.
T10058	A2B receptor antagonist 1	531506-36-2	98.83%
T10058	A2B receptor antagonist 1 (EXAMPLE 9B) is a potent A2B adenosine receptor antagonist.