Adenosine Receptor

The adenosine receptors are a class of purinergic G protein-coupled receptors with adenosine as the endogenous ligand. There are four known types of adenosine receptors in humans: A1, A2A, A2B and A3; each is encoded by a different gene.

Cat. No.	Product name	CAS No.	Purity
T21519	CCPA	37739-05-2	99.91%
T21519	CCPA (2-chloro-N(6)cyclopentyladenosine) is a potent and selective agonist of adenosine A1 receptor
T23347	SDZ WAG 994	130714-47-5	99.90%
T23347	SDZ WAG 994 is an A1 adenosine receptor agonist.
T9330	MIPS521	1146188-19-3	99.88%
T9330	MIPS521 ({2-Amino-4-[3,5-bis(trifluoromethyl)phenyl]thiophen-3-yl}(4-chlorophenyl)methanone) is a positive allosteric modulator of the A1R.
T8312	Derenofylline	251945-92-3	99.84%
T8312	Derenofylline is a selective and potent adenosine A(1) antagonist in vitro (Ki=1 nM)
T9516	Binodenoson	144348-08-3	99.84%
T9516	Binodenoson (WRC 0470) is a potent and selective A2A adenosine receptor agonist (KD=270 nM). Binodenoson is being developed as a short-acting coronary vasodilato...
T0362	Ticlopidine hydrochloride	53885-35-1	99.82%
T0362	Ticlopidine hydrochloride (Ticlodix) is an effective inhibitor of platelet aggregation commonly used in the placement of STENTS in CORONARY ARTERIES.
T0625	Theobromine	83-67-0	99.82%
T0625	Theobromine (3,7-Dimethylxanthine), a xanthine alkaloid, is used as a bronchodilator and as a vasodilator.
T10212	A2AR-agonist-1	41552-95-8	99.82%
T10212	A2AR-agonist-1 (N-(2-(1H-Indol-3-yl)ethyl)adenosine) is a potent A2AR and ENT1 agonist (Ki: 4.39 and 3.47 for A2AR and ENT1. It targets the Adenosine A2A Recepto...
T1083L	Theophylline monohydrate	5967-84-0	99.79%
T1083L	Theophylline monohydrate (Quibron) appears to inhibit phosphodiesterase and prostaglandin production, regulate calcium flux and intracellular calcium distributio...
T5940	Proxyphylline	603-00-9	99.79%
T5940	Proxyphylline (7-(2-Hydroxypropyl)theophylline) is a dual of adenosine A1/A2a receptor inhibitor and phosphodiesterase (PDE) inhibitor. Proxyphylline acts as a c...
T0437	Inosine	58-63-9	99.78%
T0437	Inosine (NSC-20262) is a purine nucleoside that has hypoxanthine linked by the N9 nitrogen to the C1 carbon of ribose. It has immunomodulatory, neuroprotective, ...
T27439	GS-9667	618380-90-8	99.76%
T27439	GS-9667, a selective and partial agonist of the A(1) adenosine receptor (AR), represents an effective therapy for Type 2 diabetes (T2DM) and dyslipidemia via low...
T27509	GW-493838	253124-46-8	99.76%
T27509	GW-493838 is a potent adenosine A1A receptor agonist for the treatment of dyslipidemia and neuropathic pain, with analgesic effects on post-herpetic neuralgia or...
T17023	Tecadenoson	204512-90-3	99.76%
T17023	Tecadenoson (CVT-510) is a selective agonist of A1 adenosine receptor.
T37792	A2A receptor antagonist 1	443103-97-7	99.76%
T37792	A2A receptor antagonist 1 (CPI-444 analog) is an antagonist of both adenosine A2A receptor and A1 receptor with Kis of 4 and 264 nM, respectively.
T6979	SCH 58261	160098-96-4	99.75%
T6979	SCH 58261 is a potent and selective A2a adenosine receptor antagonist.The Ki =2.3 nM for rat A2a and 2 nM is for bovine A2a.
T1825	Reversine	656820-32-5	99.75%
T1825	Reversine, a small synthetic purine analogue (2, 6-disubstituted purine), is a potent inhibitior of Aurora A/B/C(IC50s=150-500 nM).
T31731	Evodenoson	844873-47-8	99.74%
T31731	Evodenoson (ATL313) is a potent and selective adenosine A2a receptor (A2aR) agonist for the treatment of eye diseases, tumors, and immune system disorders, and m...
TN2247	Swertisin	6991-10-2	99.74%
TN2247	Swertisin, a novel herbal biomolecule, shows a strong antihyperglycemic action. Swertisin is an adenosine A1 receptor antagonist, is known to have antidiabetic, ...
T16378	Ogerin	1309198-71-7	99.7%
T16378	Ogerin is a selective GPR68 positive allosteric modulator (pEC50: 6.83). Ogerin blocks recall in fear conditioning in mice. Ogerin displays inverse agonist and a...