AChR

An acetylcholine receptor (abbreviated AChR) is an integral membrane protein that responds to the binding of acetylcholine, a neurotransmitter.

Cat. No.	Product name	CAS No.	Purity
T1540	Doxepin hydrochloride	1229-29-4	99.91%
T1540	Doxepin hydrochloride (Aponal) is a dibenzoxepin tricyclic compound. It displays a range of pharmacological actions including maintaining adrenergic innervation....
T23588	9-CP-Ade Mesylate	189639-09-6	99.91%
T23588	9-CP-Ade Mesylate (9 CP Ade Mesylate) is a cell-permeable, stable and non-competitive inhibitor of adenylate cyclase.
T8147	Solifenacin	242478-37-1	99.91%
T8147	Solifenacin (YM905 free base) (YM905 free base) is a novel muscarinic receptor antagonist, its pKis for M1, M2 and M3 receptors is of 7.6, 6.9 and 8.0, respectiv...
T1612	Neostigmine methyl sulfate	51-60-5	99.90%
T1612	Neostigmine methyl sulfate (Syntostigmin) is a reversible inhibitor of acetylcholinesterase, can not cross the blood-brain barrier, used in the treatment of myas...
T3619	VU0357017 hydrochloride	1135242-13-5	99.9%
T3619	VU0357017 hydrochloride (ML071 hydrochloride) is highly selective M1 agonists act at an allosteric site to activate the receptor (EC50: 477 ± 172 nM; Pec50: 6.37...
T10961	Darenzepine	84629-61-8	99.9%
T10961	Darenzepine is a muscarinic receptor inhibitor.
T1657	Varenicline Tartrate	375815-87-5	99.9%
T1657	Varenicline Tartrate (CP 526555-18) is a benzazepine derivative that functions as an ALPHA4/BETA2 NICOTINIC RECEPTOR partial agonist. It is used for SMOKING CESS...
T1039	Choline chloride	67-48-1	99.89%
T1039	Choline chloride (Biocoline) is a basic constituent of lecithin that is found in many plants and animal organs. It is important as a precursor of acetylcholine, ...
T6478	Donepezil Hydrochloride	120011-70-3	99.89%
T6478	Donepezil HCl(Aricept) is a selective and effective AChE inhibitor for bAChE and hAChE (IC50: 8.12/11.6 nM).
T2191	Tacrine hydrochloride (hydrate)	206658-92-6	99.89%
T2191	Tacrine hydrochloride hydrate (Tetrahydroaminacrine) is a cholinesterase inhibitor that crosses the blood-brain barrier. Tacrine has been used to counter the eff...
T0944	Levamisole hydrochloride	16595-80-5	99.89%
T0944	Levamisole hydrochloride ((-)-Tetramisole hydrochloride) is an antihelminthic drug that has been tried experimentally in rheumatic disorders where it apparently ...
T2984	Scopoletin	92-61-5	99.88%
T2984	Scopoletin (Esculetin 6-methyl ether) is a plant growth factor derived from the root of Scopolia carniolica, inhibits of acetylcholinesterase (AChE).
TQ0304	Metixene hydrochloride hydrate	7081-40-5	99.88%
TQ0304	Metixene hydrochloride hydrate has potential anticholinergic activity and inhibits the binding of quinine ring benzoate (QNB) to muscarine receptors, with IC50 a...
T1215	Nicardipine hydrochloride	54527-84-3	99.87%
T1215	Nicardipine hydrochloride (YC-93 Hydrochloride) is the hydrochloride salt form of nicardipine, a synthetic derivative of nitrophenyl-pyridine and potent calcium ...
T19940	Sulfoxaflor	946578-00-3	99.87%
T19940	Sulfoxaflor (GF 2032), an agonist of nAChR1 and nAChR2 subtypes, is a systemic insecticide that acts on the central nervous system of insects. Sulfoxaflor is use...
T3026	(-)-Huperzine A	102518-79-6	99.87%
T3026	(-)-Huperzine A (HupA) , an active Lycopodium alkaloid extracted from the traditional Chinese herb, is a potent, selective and reversible acetylcholinesterase (A...
T0678	Amitriptyline hydrochloride	549-18-8	99.87%
T0678	Amitriptyline hydrochloride (Annoyltin) is the hydrochloride salt of the tricyclic dibenzocycloheptadiene amitriptyline with antidepressant and antinociceptive ...
T0287	Hexamethonium Bromide	55-97-0	99.87%
T0287	Hexamethonium Bromide (Hexamethonium Dibromide), a specific antagonist of neuronal-type nicotinic AChR in ganglia, is poorly absorbed from the gastrointestinal t...
T14333	Asoxime dichloride	34433-31-3	99.86%
T14333	Asoxime dichloride (Tert-Butyl2-(2-hydroxyethyl)-1-pyrrolidinecarboxylate) is an antagonist to acetylcholine receptors (AChRs) including the nicotinic receptor, ...
T2387	Glycopyrrolate	596-51-0	99.86%
T2387	Glycopyrrolate (Glycopyrrolate bromide) is a muscarinic antagonist used as an antispasmodic, in some disorders of the gastrointestinal tract, and to reduce saliv...