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AChR

An acetylcholine receptor (abbreviated AChR) is an integral membrane protein that responds to the binding of acetylcholine, a neurotransmitter.
Signaling Pathways | Target | TargetMol
Cat. No. Product name CAS No. Purity Chemical Structure
T0322 Fipexide 34161-24-5 99.95%
Fipexide
Fipexide (Attentil, Vigilor), a psychoactive drug of the piperazine chemical class, was developed in Italy in 1983. It was served as a nootropic drug in France a...
T7671 Myosmine 532-12-7 99.95%
Myosmine
Myosmine is a minor tobacco alkaloid that is structurally related to nicotine.
T22448 Tropisetron 89565-68-4 99.95%
Tropisetron
Tropisetron (ICS 205-930) is an α7-nicotinic receptor agonist and 5-HT3 receptor antagonist with Kis of 6.9 nM and 5.3 nM, respectively.
T23348 SEN12333 874450-44-9 99.94%
SEN12333
SEN12333 is an α7 nicotinic acetylcholine receptor (nAChR) agonist
T2198 Arecoline hydrobromide 300-08-3 99.94%
Arecoline hydrobromide
Arecoline hydrobromide (Arecoline HBr) is a muscarinic acetylcholine receptor agonist.
T1069 Metoclopramide hydrochloride 7232-21-5 99.94%
Metoclopramide hydrochloride
Metoclopramide hydrochloride (Metoclopramide HCl) is a selective dopamine D2 receptor antagonist, used as an antiemetic.
T6547 Ipratropium Bromide 22254-24-6 99.94%
Ipratropium Bromide
Ipratropium Bromide (Sch 1000) is a synthetic anticholinergic agent that is used as an inhalant for treatment of acute bronchospasm due to chronic bronchitis and...
T23116 Oxotremorine sesquifumarate 17360-35-9 99.94%
Oxotremorine sesquifumarate
Oxotremorine sesquifumarate is a muscarinic agonist.
T21439 Tacrine 321-64-2 99.94%
Tacrine
Tacrine (CS 12602) is an indirect cholinergic agonist and centrally acting anticholinesterase. It is approved for the treatment of Alzheimer's disease.
T0455 Clozapine 5786-21-0 99.93%
Clozapine
Clozapine (HF 1854) is a tricylic dibenzodiazepine, classified as an atypical antipsychotic agent. It binds several types of central nervous system receptors, an...
T1472 Trospium chloride 10405-02-4 99.93%
Trospium chloride
Trospium chloride (Spasmex) is an antispasmodic and anticholinergic agent used to treat urinary incontinence and overactive bladder syndrome. Trospium chloride h...
T1567 Olanzapine 132539-06-1 99.92%
Olanzapine
Olanzapine (LY170053) is an atypical antipsychotic that is used currently in the treatment of schizophrenia and bipolar illness.
T0103 Dipivefrin hydrochloride 64019-93-8 99.92%
Dipivefrin hydrochloride
Dipivefrin hydrochloride (Dipivefrin HCl) that is available as an ophthalmic solution is a prodrug of adrenaline, which is used to treat glaucoma.
T5051 Isopropamide Iodide 71-81-8 99.91%
Isopropamide Iodide
Isopropamide iodide is a long-acting anticholinergic drug. It is used in the treatment of peptic ulcers and other gastrointestinal disorders. It also acts as a m...
T1636 Paroxetine hydrochloride 78246-49-8 99.91%
Paroxetine hydrochloride
Paroxetine hydrochloride (Paroxetine HCl) is a serotonin uptake inhibitor that is effective in the treatment of depression.
T6684 Succinylcholine Chloride Dihydrate 6101-15-1 99.91%
Succinylcholine Chloride Dihydrate
Succinylcholine Chloride Dihydrate (Succinyldicholine dichloride) is a nicotinic AChR agonist and also acts as a depolarizing neuromuscular blocker.
T1460 Dicyclomine hydrochloride 67-92-5 99.91%
Dicyclomine hydrochloride
Dicyclomine hydrochloride is a muscarinic antagonist used as an antispasmodic and in urinary incontinence.
T1540 Doxepin hydrochloride 1229-29-4 99.91%
Doxepin hydrochloride
Doxepin hydrochloride (Aponal) is a dibenzoxepin tricyclic compound. It displays a range of pharmacological actions including maintaining adrenergic innervation....
T23588 9-CP-Ade Mesylate 189639-09-6 99.91%
9-CP-Ade Mesylate
9-CP-Ade Mesylate (9 CP Ade Mesylate) is a cell-permeable, stable and non-competitive inhibitor of adenylate cyclase.
T1612 Neostigmine methyl sulfate 51-60-5 99.90%
Neostigmine methyl sulfate
Neostigmine methyl sulfate (Syntostigmin) is a reversible inhibitor of acetylcholinesterase, can not cross the blood-brain barrier, used in the treatment of myas...
Fipexide
T0322
Fipexide (Attentil, Vigilor), a psychoactive drug of the piperazine chemical class, was developed in Italy in 1983. It was served as a nootropic drug in France a...
Myosmine
T7671
Myosmine is a minor tobacco alkaloid that is structurally related to nicotine.
Tropisetron
T22448
Tropisetron (ICS 205-930) is an α7-nicotinic receptor agonist and 5-HT3 receptor antagonist with Kis of 6.9 nM and 5.3 nM, respectively.
SEN12333
T23348
SEN12333 is an α7 nicotinic acetylcholine receptor (nAChR) agonist
Arecoline hydrobromide
T2198
Arecoline hydrobromide (Arecoline HBr) is a muscarinic acetylcholine receptor agonist.
Metoclopramide hydrochloride
T1069
Metoclopramide hydrochloride (Metoclopramide HCl) is a selective dopamine D2 receptor antagonist, used as an antiemetic.
Ipratropium Bromide
T6547
Ipratropium Bromide (Sch 1000) is a synthetic anticholinergic agent that is used as an inhalant for treatment of acute bronchospasm due to chronic bronchitis and...
Oxotremorine sesquifumarate
T23116
Oxotremorine sesquifumarate is a muscarinic agonist.
Tacrine
T21439
Tacrine (CS 12602) is an indirect cholinergic agonist and centrally acting anticholinesterase. It is approved for the treatment of Alzheimer's disease.
Clozapine
T0455
Clozapine (HF 1854) is a tricylic dibenzodiazepine, classified as an atypical antipsychotic agent. It binds several types of central nervous system receptors, an...
Trospium chloride
T1472
Trospium chloride (Spasmex) is an antispasmodic and anticholinergic agent used to treat urinary incontinence and overactive bladder syndrome. Trospium chloride h...
Olanzapine
T1567
Olanzapine (LY170053) is an atypical antipsychotic that is used currently in the treatment of schizophrenia and bipolar illness.
Dipivefrin hydrochloride
T0103
Dipivefrin hydrochloride (Dipivefrin HCl) that is available as an ophthalmic solution is a prodrug of adrenaline, which is used to treat glaucoma.
Isopropamide Iodide
T5051
Isopropamide iodide is a long-acting anticholinergic drug. It is used in the treatment of peptic ulcers and other gastrointestinal disorders. It also acts as a m...
Paroxetine hydrochloride
T1636
Paroxetine hydrochloride (Paroxetine HCl) is a serotonin uptake inhibitor that is effective in the treatment of depression.
Succinylcholine Chloride Dihydrate
T6684
Succinylcholine Chloride Dihydrate (Succinyldicholine dichloride) is a nicotinic AChR agonist and also acts as a depolarizing neuromuscular blocker.
Dicyclomine hydrochloride
T1460
Dicyclomine hydrochloride is a muscarinic antagonist used as an antispasmodic and in urinary incontinence.
Doxepin hydrochloride
T1540
Doxepin hydrochloride (Aponal) is a dibenzoxepin tricyclic compound. It displays a range of pharmacological actions including maintaining adrenergic innervation....
9-CP-Ade Mesylate
T23588
9-CP-Ade Mesylate (9 CP Ade Mesylate) is a cell-permeable, stable and non-competitive inhibitor of adenylate cyclase.
Neostigmine methyl sulfate
T1612
Neostigmine methyl sulfate (Syntostigmin) is a reversible inhibitor of acetylcholinesterase, can not cross the blood-brain barrier, used in the treatment of myas...
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TargetMol