T3S1612 |
Kuwanon G
|
75629-19-5
|
98%
|
|
1. Kuwanon G (Moracenin B) as dual inhibitors of PTP1B and α-glucosidase enzymes, as well as insulin sensitizers, it may potentially be utilized as an effective ...
|
TP2063 |
α-Conotoxin MII
|
175735-93-0
|
98%
|
|
α-Conotoxin MII is a highly potent and selective competitive antagonist for α3β2 subunit-containing nicotinic receptors (IC50 = 0.5 - 3.5 nM at α3β2 expressed in...
|
T22013 |
8-Aminoadenine
|
28128-33-8
|
98%
|
|
8-Aminoadenine (7H-purine-6,8-diamine) is a ligand for Adenine Receptor with Ki of 0.0341 μM.
|
T14880 |
CB-7921220
|
115453-99-1
|
98%
|
|
CB-7921220 (6-[2-(4-Aminophenyl)vinyl]-2-pyridinecarboxylic acid) is an inhibitor of adenylate cyclase.
|
T8725 |
A 582941 HCl (848591-90-2(free base))
|
T8725
|
98%
|
|
A-582941 is a alpha7 neuronal nicotinic receptor agonist with broad spectrum cognition-enhancing properties
|
T2555 |
Aclidinium bromide
|
320345-99-1
|
98%
|
|
Aclidinium bromide (LAS-W 330) is a synthetic anticholinergic agent that is used as an inhalant for treatment of acute bronchospasm due to chronic bronchitis or ...
|
T12481 |
Pipecuronium bromide
|
52212-02-9
|
98%
|
|
Pipecuronium bromide (RGH-1106) is a selective and potent nAChR antagonist that also acts as a non-depolarising steroidal neuromuscular blocker, causing muscle r...
|
T0401 |
Benzethonium chloride
|
121-54-0
|
98%
|
|
Benzethonium chloride (Quatrachlor) is a synthetic quaternary ammonium salt with surfactant, antiseptic, and broad spectrum antimicrobial properties.
|
T0296 |
Pempidine
|
79-55-0
|
98%
|
|
Pempidine (1,2,2,6,6-Pentamethylpiperidine) is a nicotinic antagonist, has been used as a ganglionic blocker in the treatment of hypertension.
|
T37196 |
5-AAM-2-CP
|
175424-74-5
|
98%
|
|
5-AAM-2-CP is one of the major metabolites of Acetamiprid. Acetamiprid, a nAChR agonist, is a neonicotinoid insecticide used worldwide.
|
T28531 |
Facinicline hydrochloride
|
677305-02-1
|
98%
|
|
Facinicline hydrochloride (RG3487) is both a novel nicotinic alpha-7 receptor (alpha7nAChR) partial agonist (Ki = 6 nM) and an antagonist of 5-HT3(Ki = 1.2 nM). ...
|
T7500 |
Isoxazole
|
288-14-2
|
98%
|
|
Isoxazole (1,2-oxazole) is the inhibitor of acetylcholinesterase (AChE). The ligands of Isoxazole bind to and inhibit the Sxc- antiporter.
|
T23297 |
(S)-(+)-Dimethindene maleate
|
136152-65-3
|
98%
|
|
(S)-(+)-Dimethindene maleate is an orally available, selective muscarinic M2 receptor and histamine H1 receptor antagonist that inhibits muscarinic M1, M3, and M...
|
T4289 |
Mc-Val-Ala-PAB
|
1870916-87-2
|
98%
|
|
Mc-Val-Ala-PAB, an effective linker, is utilized in antibody-drug-conjugate (ADC).
|
T13992 |
CHF5407
|
1004312-94-0
|
98%
|
|
CHF5407(SVT-47060) is a potent and selective muscarinic M3 receptor antagonist with prolonged action at muscarinic receptors.CHF5407 has an effect on bronchospas...
|
T7056 |
Dronedarone
|
141626-36-0
|
98%
|
|
Dronedarone (SR 33589) is an amiodarone analogue which has an effective and promising treatment for Atrial fibrillation.
|
T13385 |
Zamifenacin fumarate
|
127308-98-9
|
98%
|
|
Zamifenacin fumarate (UK-76654 fumarate) is a potent and gut-selective antagonist of muscarinic M3 receptor.
|
T1459 |
Cisatracurium besylate
|
96946-42-8
|
98%
|
|
Cisatracurium besylate (51W89) is a nondepolarizing skeletal muscle relaxant for intravenous administration.
|
T1072 |
Loxeen
|
6856-31-1
|
98%
|
|
Loxeen (Pridinol methanesulfonate) is used as an anticholinergic and as an antiparkinsonian agent.
|
TN1673 |
Garcinone C
|
76996-27-5
|
98%
|
|
Garcinone C is a xanthone derivative extracted from Garcinia oblongifolia Champ with anti-inflammatory, astringency, and granulation-promoting activities. Garcin...
|