TN3243 |
7-O-Methyleriodictyol
|
51857-11-5
|
99.38%
|
|
7-O-Methyleriodictyol is a flavanone isolated from Artemisia monosperma and shows biological effects on rat isolated smooth muscles.
|
T68599 |
Orphenadrine
|
83-98-7
|
99.38%
|
|
Orphenadrine is a noncompetitive N-methyl-D-aspartate (NMDA) receptor antagonist that inhibits clonal HERG channels in a concentration-dependent manner, producin...
|
T0130 |
Physostigmine Salicylate
|
57-64-7
|
99.36%
|
|
Physostigmine, a parasympathomimetic alkaloid, is a reversible cholinesterase inhibitor. It extracts from the Calabar bean.
|
T1266 |
Terfenadine
|
50679-08-8
|
99.36%
|
|
Terfenadine ((±)-Terfenadine) is a prodrug that is metabolized by intestinal CYP3A4 to the active form fexofenadine, a selective histamine H1-receptor antagonist...
|
T0786 |
Clidinium bromide
|
3485-62-9
|
99.36%
|
|
Clidinium bromide (Ro 2-3773) , a synthetic anticholinergic agent, has been shown in experimental and clinical researchers to have a pronounced antisecretory and...
|
T7695 |
PNU-282987 S enantiomer free base
|
737727-12-7
|
99.35%
|
|
PNU-282987 S enantiomer free base is an agonist of α7 nicotinic acetylcholine receptor (α7 nAChR).
|
T14065 |
9-Ethyladenine
|
2715-68-6
|
99.35%
|
|
9-Ethyladenine (6-Amino-9-ethylpurine) is a partially potent APRT (adenine phosphoribosyltransferase) inhibitor [1].
|
T68154 |
TC-2216
|
646055-67-6
|
99.33%
|
|
TC-2216 is a partial agonist at the neural nicotinic acetylcholine receptor and is used to treat anxiety and depression.
|
T8448 |
ZSET1446
|
887603-94-3
|
99.32%
|
|
ZSET1446 (ST-101) is a T-type calcium channel activator potentially for the treatment of learning deficits in various types of Alzheimer disease (AD) models.
|
T0804 |
Pilocarpine Hydrochloride
|
54-71-7
|
99.29%
|
|
Pilocarpine Hydrochloride (NSC 5746 HCl) , a nonselective muscarinic acetylcholine receptor agonist, is utilized to produce an experimental model of epilepsy.
|
TP2058L |
Catestatin acetate
|
TP2058L
|
99.28%
|
|
Catestatin acetate is a non-competitive antagonist of nAChR and inhibits catecholamine release. Catestatin acetate regulates cardiac function and blood pressure....
|
T68953 |
Arecoline
|
63-75-2
|
99.28%
|
|
Arecoline is a natural alkaloid derived from areca nut in the palm family and is a potent nicotine and partial agonist of muscarinic acetylcholine receptors. Are...
|
T7224 |
Anabasine
|
494-52-0
|
99.27%
|
|
Anabasine ((S)-Anabasine) is an alkaloid extracted from tobacco. Anabasine is a full agonist of nicotinic acetylcholine receptors (nAChRs) with insecticidal acti...
|
T0166 |
Pancuronium dibromide
|
15500-66-0
|
99.27%
|
|
Pancuronium dibromide (Pavulon), a competitive AChR antagonist (IC50 = 5.5 nM), acts as a skeletal muscle relaxant. Pancuronium dibromide(Pancuronium bromide) bl...
|
T9018 |
JHU37160
|
2369979-68-8
|
99.25%
|
|
JHU37160 (JHU 37160) is a Designer Receptors Exclusively Activated by Designer Drug (DREADD) agonist with Ki of 1.9 nM and 3.6 nM for human muscarinic acetylchol...
|
T29123 |
VU0152099
|
612514-42-8
|
99.24%
|
|
VU0152099 is a potent and selective M4 mAChR allosteric potentiator(EC50 = 380 ± 93 nM).
|
T7052 |
Gnetol
|
86361-55-9
|
99.21%
|
|
Gnetol competitivity inhibits butyrylcholinesterase (IC50: 1.3 uM). Gnetol has a strong inhibitory effect on murine tyrosinase activity. Gnetol significantly sup...
|
T4246 |
Varenicline dihydrochloride
|
866823-63-4
|
99.21%
|
|
Varenicline dihydrochloride is a Selective α4β2 nicotinic acetylcholine receptor partial agonist.
|
T0794 |
Mepenzolate Bromide
|
76-90-4
|
99.21%
|
|
Mepenzolate Bromide (Colibantil) is a muscarinic antagonist used to treat gastrointestinal conditions.
|
T0086 |
Galanthamine hydrobromide
|
1953-04-4
|
99.19%
|
|
Galanthamine hydrobromide (Galantamine hydrobromide), a long-acting and centrally active AChE inhibitor (IC50:410 nM), is an allosteric potentiator at neuronal n...
|