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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T5158 | N-Desmethylclozapine | Desmethylclozapine,Normethylclozapine,Norclozapine | Virus Protease , Dopamine Receptor , 5-HT Receptor , Opioid Receptor , AChR , Drug Metabolite |
N-Desmethylclozapine (Desmethylclozapine) is an antagonist of serotonin (5-HT) receptor subtype 5-HT2C (IC50: 7.1 nM). It also is an antagonist at dopamine D4 receptors, an agonist at δ-opioid receptors. |