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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T15243 | Ertiprotafib | PTP 112 | Phosphatase , PPAR |
Ertiprotafib is a PTP1B, IkB kinase β (IKK-β), and a dual PPARα and PPARβ agonist inhibitor ( IC50s: 1.6 μM for PTP1B, 400 nM for IKK-β, an EC50 of ~1 μM for PPARα/PPARβ). |