T3407 |
Rapastinel
|
117928-94-6
|
99.67%
|
|
Rapastinel (TPPT-amide) (GLYX-13) is an N-methyl-D-aspartate receptor (NMDAR) modulator.
|
T2362 |
QNZ46
|
1237744-13-6
|
99.64%
|
|
QNZ46 is a NR2C/NR2D-selective NMDA receptor non-competitive antagonist.
|
T13480 |
(S)-(-)-5-Fluorowillardiine
|
140187-23-1
|
99.60%
|
|
(S)-(-)-5-Fluorowillardiine ((S)-5-Fluorowillardiine) is an AMPA receptor-specific agonist
|
T3407L |
Rapastinel acetate
|
491872-39-0
|
99.6%
|
|
Rapastinel acetate is a modulator of N-methyl-D-aspartate (NMDA) receptor and a partial agonist of glycine site long-lasting antidepressant effects.
|
T16963 |
SYM 2081
|
31137-74-3
|
99.59%
|
|
SYM 2081 is a specific kainate receptor agonist with an IC50 value of 35 nM for [3H]-kainate binding. SYM 2081 depolarizes the muscle and reduces the EPSP amplit...
|
T9177 |
BPAM344
|
1204572-55-3
|
99.57%
|
|
BPAM344 is a potent positive allosteric modulator (PAM) of the KAR subunits GluK1b, GluK2a, and GluK3a.
|
T1308 |
Orphenadrine hydrochloride
|
341-69-5
|
99.54%
|
|
Orphenadrine hydrochloride (Mephenamin) is a muscarinic antagonist used to treat drug-induced parkinsonism and to relieve pain from muscle spasm.
|
T2O2728 |
Glycine
|
56-40-6
|
99.54%
|
|
glycine (2-Aminoacetic acid) is a non-essential amino acid. It is found primarily in gelatin and silk fibroin and used therapeutically as a nutrient. It is also ...
|
T17179 |
Tulrampator
|
1038984-31-4
|
99.51%
|
|
Tulrampator (S-47445) is an orally bioavailable positive AMPAR with antidepressant effects.
|
T3377 |
L-Phenylalanine
|
63-91-2
|
99.49%
|
|
L-Phenylalanine (3-Phenyl-L-alanine) is an essential amino acid and the precursor of the amino acid tyrosine, acts as an antagonist at α2δ calcium channels.
|
T4113 |
NBQX
|
118876-58-7
|
99.42%
|
|
NBQX (FG9202) is a potent, selective and competitive AMPA receptor antagonist. Neuroprotective and anticonvulsant; active in vivo.
|
T34609 |
Selurampanel
|
912574-69-7
|
99.41%
|
|
Selurampanel (BGG492) is an orally active and selective competitive AMPA glutamate receptor antagonist, a quinazoline-dione sulfonamide. selurampanel is used in ...
|
T5819 |
Rapastinel Trifluoroacetate
|
1435786-04-1
|
99.37%
|
|
Rapastinel Trifluoroacetate (GLYX-13 Trifluoroacetate) is an NMDA receptor modulator with glycine-site partial agonist properties.
|
T7304 |
DNQX
|
2379-57-9
|
99.32%
|
|
DNQX (FG 9041) is a competitive, non-NMDA glutamate receptor antagonist (IC50s = 0.5 and 0.1 μM for AMPA and kainate receptors, respectively)
|
T0324 |
Isoxsuprine hydrochloride
|
579-56-6
|
99.31%
|
|
Isoxsuprine hydrochloride (Isolait) is a beta-adrenergic agonist that causes direct relaxation of uterine and vascular smooth muscle.
|
T8920 |
Sepimostat
|
103926-64-3
|
99.3%
|
|
Sepimostat exhibits neuroprotective activity via NR2B N-methyl-D-aspartate receptor antagonism at the Ifenprodil-binding site of the NR2B subunit. Sepimostat dim...
|
T1884 |
CX516
|
154235-83-3
|
99.29%
|
|
CX516 (Ampalex), an ampakine and nootropic, acts as an AMPA receptor positive allosteric modulator as a therapy for Alzheimer's disease, schizophrenia and mild c...
|
TQ0027 |
Transcrocetinate disodium
|
591230-99-8
|
99.22%
|
|
Transcrocetinate disodium (Disodium trans-crocetinate), extracted from saffron (Crocus sativus L.), is a high-affinity antagonist of NMDA receptor.
|
T4S0171 |
Transcrocetin
|
27876-94-4
|
99.2%
|
|
Transcrocetin (8,8'-Diapocarotenedioic Acid) is a singlet oxygen quencher.
|
T61518 |
TAK-653
|
1358751-06-0
|
99.18%
|
|
TAK-653, a selective positive allosteric modulator (PAM) of AMPA receptors exhibiting minimal agonistic activity, elicits an antidepressant-like response while m...
|