T5764 |
Alliin
|
556-27-4
|
99.62%
|
|
Alliin ((S)-3-(Allylsulphinyl)-L-alanine) is a garlic organosulfur compound that possesses various pharmacological properties.alliin protected against LPS-induce...
|
T3867 |
Alpinetin
|
36052-37-6
|
99.61%
|
|
Alpinetin ((-)-alpinetin) has antibacterial activity.Alpinetin has anti-inflammatory activity.Alpinetin can enhance the sensitivity of HepG2 hepatoma cells to th...
|
T0705 |
Triflusal
|
322-79-2
|
99.61%
|
|
Triflusal (UR1501) is a 2-acetoxy-4-trifluoromethylbenzoic acid and it is an aspirin chemically-related molecule but not a derivative.
|
T60184 |
TUG-499
|
1206629-08-4
|
99.59%
|
|
TUG-499 is a selective free fatty acid receptor 1 (FFAR1 or GPR40) agonist (EC50: 7.39).TUG-499 has an affinity for FFAR1 or GPR40 over the related receptors FFA...
|
T15581 |
Inolitazone
|
223132-37-4
|
99.58%
|
|
Inolitazone (RS5444) a high-affinity PPARγ agonist. Inolitazone exhibits IC50 for growth inhibition is ~0.8 nM in vitro.
|
T0214 |
Pioglitazone
|
111025-46-8
|
99.57%
|
|
Pioglitazone (U 72107) is an insulin sensitizing agent and thiazolidinedione that is indicated for the treatment of type 2 diabetes. Pioglitazone has been linked...
|
TN3500 |
Beta-Amyrone
|
638-97-1
|
99.55%
|
|
beta-Amyrone (β-Amyron) has antifungal activity against Chikungunya virus replication with an EC50 of 86 uM. beta-Amyrone has anti-inflammatory activity through ...
|
T4408 |
Elafibranor
|
923978-27-2
|
99.55%
|
|
Elafibranor (GFT505) is an agonist of the peroxisome proliferator-activated receptor-α (PPAR-α) and peroxisome proliferator-activated receptor-δ (PPAR-δ) with EC...
|
T0212 |
Seratrodast
|
112665-43-7
|
99.54%
|
|
Seratrodast (ABT-001) (INN), a thromboxane A2 (TXA2) receptor (TP receptor) antagonist, is mainly used in the therapy of asthma. It was the first TP receptor ant...
|
T2413 |
FH535
|
108409-83-2
|
99.5%
|
|
FH535, a Wnt/β-catenin signaling and PPAR inhibitor, exhibits anti-tumor activities.
|
T15049 |
Daltroban
|
79094-20-5
|
99.49%
|
|
Daltroban (SKF 96148) is a specific thromboxane A2 (TXA2) receptor antagonist. Daltroban shows protective effect in reperfusion injury. Daltroban increase intrac...
|
T67933 |
BAY-4931
|
423150-91-8
|
99.47%
|
|
BAY-4931 is a potent, covalent and selective PPARγ inverse-agonist with an IC 50 of 0.17 nM .
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T23389 |
SR1664
|
1338259-05-4
|
99.43%
|
|
SR1664 is a potent and selective PPARγ inhibitor with potential antidiabetic activity. SR1664 binds to PPARγ and potently inhibits Cdk5-mediated PPARγ phosphoryl...
|
T0334 |
Rosiglitazone
|
122320-73-4
|
99.43%
|
|
Rosiglitazone (BRL49653) is a PPARγ agonist, TRPC5 activator, and TRPM3 inhibitor with oral activity. Rosiglitazone is also a hypoglycemic agent and a thiazolidi...
|
T14176 |
Aleglitazar
|
475479-34-6
|
99.42%
|
|
Aleglitazar (R1439) (R1439) is a potent dual PPARα/γ agonist, with IC50s of 38 nM and 19 nM for human PPARa and PPARγ, respectively. Aleglitazar can be used for ...
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T67936 |
BAY-0069
|
420826-65-9
|
99.41%
|
|
BAY-0069 is a potent and selective PPARγ transactivator that inhibits human PPARγ and murine PPARγ with IC50s of 6.3 nM and 24 nM, respectively.BAY-0069 can be u...
|
T12527L |
Mavodelpar free acid hydrochloride
|
|
99.39%
|
|
Mavodelpar free acid hydrochloride (Pparδ agonist HCl) is a potent PPARδ agonist.
|
T6926 |
Palmitoylethanolamide
|
544-31-0
|
99.38%
|
|
Palmitoylethanolamide (Impulsin) is an endogenously fatty acid amide. It has a role as an anti-inflammatory drug, an antihypertensive agent, a neuroprotective ag...
|
T9767 |
CC618
|
1680204-90-3
|
99.37%
|
|
CC618 is a selective PPARβ/δ antagonist with an IC50 of 10.0 μM.
|
T19500 |
Palmitelaidic Acid
|
10030-73-6
|
99.36%
|
|
Palmitelaidic Acid (trans-Palmitoleic acid) is one of the most abundant fatty acids in serum and tissue.
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