Opioid Receptor

Opioid receptors belong to the large superfamily of seven transmembrane-spanning (7TM) G protein-coupled receptors (GPCRs). As a class, GPCRs are of fundamental physiological importance mediating the actions of the majority of known neurotransmitters and hormones.

Cat. No.	Product name	CAS No.	Purity
T15799	LY2940094	1307245-86-8	99.6%
T15799	LY2940094 (LY-2940094) decreases ethanol self-administration in animal models. LY2940094 is an effective, selective, and orally available nociceptin receptor ant...
T4386	PZM21	1997387-43-5	99.59%
T4386	PZM21 is an effective and selective μ opioid receptor agonist (EC50: 1.8 nM).
TP2501	Difelikefalin acetate		99.55%
TP2501	Difelikefalin acetate (CR 845 acetate) is a peripherally restricted kappa opioid receptor agonist. CR845 exhibit low P450 CYP inhibition and low penetration into...
T31081L	CP 866087	519052-02-9	99.52%
T31081L	CP 866087 is an opioid receptor antagonist for the study of female sexual dysfunction.
T22849	ICI 199,441 hydrochloride	115199-84-3	99.46%
T22849	ICI 199,441 hydrochloride is a potent, selective agonist of κ-opioid receptor.
T31081	CP-866087	519052-04-1	99.44%
T31081	CP-866087 is a novel, potent and selective mu-opioid receptor antagonist for the study of female sexual dysfunction.
T29663	ADL-5747	850176-30-6	99.44%
T29663	ADL-5747 (ADL-5747 (free base)) (free base) is a delta opioid receptor agonist used in the treatment of neurological disorders, skin and musculoskeletal disorder...
TP1113L	[Leu5]-Enkephalin, amide acetate	TP1113L	99.36%
TP1113L	[Leu5]-Enkephalin, amide acetate is a δ opioid receptor agonist.
T5S0581	Sec-O-Glucosylhamaudol	80681-44-3	99.35%
T5S0581	Sec-O-Glucosylhamaudol (Hamaudol 3-glucoside) has anti-inflammatory effect through regulation of p38 Mitogen-Activated Protein Kinase in Lipopolysaccharide-stimu...
TP1071	Nociceptin	170713-75-4	99.35%
TP1071	Nociceptin (Orphanin FQ) is a 17-amino-acid polypeptide that is structurally related to the opioid peptide dynorphin A.
T0137	Mirtazapine	85650-52-8	99.3%
T0137	Mirtazapine (6-Azamianserin) is a tetracyclic antidepressant with a somewhat unique mechanism of action. Mirtazapine therapy can be associated with transient asy...
T7173L	[Leu5]-Enkephalin acetate(58822-25-6 free base)	T7173L	99.28%
T7173L	[Leu5]-Enkephalin acetate(58822-25-6 free base) is an endogenous neuropeptide involved in nociception and an agonist of δ-opioid and μ-opioid receptors (Kis = 4....
T6553	JTC-801	244218-51-7	99.27%
T6553	JTC-801 is a selective opioid receptor-like1 (ORL1) receptor antagonist with IC50 of 94 nM, weakly inhibits receptors δ, κ, and μ.
T28453L	Propiram fumarate HCl	945013-73-0	99.25%
T28453L	Propiram fumarate HClis an orally available Opioid receptors agonist with analgesic activity for the study of musculoskeletal pain.
T3417	Amentoflavone	1617-53-4	99.22%
T3417	Amentoflavone (3',8''-Biapigenin), as a potent inhibitor of CYP3A4 and CYP2C9, can interact with many other medications. CYP3A4 and CYP2C9 are proteins used for ...
T8991	BMS986187	684238-37-7	99.19%
T8991	BMS986187 is a novel Potent and Selective Positive Allosteric Modulators of the delta-Opioid Receptor.
T22810	GR 89696 fumarate	126766-32-3	99.19%
T22810	GR 89696 fumarate is a highly selective κ2 opioid receptor agonist (IC50 = 0.04nM) with anti-pruritchy, anti-injury and neuroprotective effects.
TP1179L	Porcine dynorphin A(1-13) acetate	TP1179L	99.14%
TP1179L	Porcine dynorphin A(1-13) acetate (Dynorphin A Porcine Fragment 1-13 acetate) is a potent, endogenous κ opioid receptor agonist and is antinociceptive at physiol...
T31750	Faxeladol	433265-65-7	99.13%
T31750	Faxeladol, a potent adrenergic absorption inhibitor and serotonin reuptake inhibitor, is a small-molecule Opioid receptor agonist that can be used to study neuro...
T23335	SCH 221510	322473-89-2	99.10%
T23335	SCH 221510 is an orally available, selective and potent NOP agonist with an EC50 of 12 nM and a Ki of 0.3 nM.SCH 221510 has anxiolytic activity and can be used t...