TP1738L |
Kassinin acetate(63968-82-1 free base)
|
TP1738L
|
95.81%
|
|
Kassinin acetate is a peptide derived from the Kassina frog. It belongs to tachykinin family of neuropeptides.
|
T7633 |
Senktide
|
106128-89-6
|
100%
|
|
Senktide is an agonist of tachykinin NK3 receptor.
|
TP1369L |
[Sar9,Met(O2)11]-Substance P acetate
|
TP1369L
|
100%
|
|
[Sar9,Met(O2)11]-Substance P acetate is a tachykinin NK1 receptor selective agonist. [Sar9,Met(O2)11]-Substance P acetate is a selective tachykinin NK1 receptor ...
|
TP1385 |
Neurokinin A(4-10) TFA(97559-35-8 free base)
|
TP1385
|
100%
|
|
Neurokinin A(4-10) TFA(97559-35-8 free base) is a tachykinin NK2 receptor agonist[1].
|
T8235 |
L-732138
|
148451-96-1
|
100%
|
|
L-732138 is a potent and competitive antagonist of neurokinin-1 (NK-1) receptor(IC50 : 2.3 nM)
|
T7828 |
[Sar9,Met(O2)11]-Substance P
|
110880-55-2
|
100%
|
|
[Sar9,Met(O2)11]-Substance P (NA) is an agonist of NK1 receptor.
|
TP1008 |
Neurokinin A
|
86933-74-6
|
100%
|
|
Neurokinin A (NKA), formerly known as Substance K, is a neurologically active peptide translated from the pre-protachykinin gene.
|
TP1883 |
[Lys5,MeLeu9,Nle10]-NKA(4-10)
|
137565-28-7
|
100%
|
|
Highy selective and potent NK2 receptor agonist (IC50 = 6.1 nM). Induces contraction of the rat fundus and bladder (EC50 values are 117 and 10 nM respectively).
|
T12000 |
MEN11467
|
214487-46-4
|
100%
|
|
MEN11467 is a novel, orally available, potent and selective peptidomimetic tachykinin NK 1 receptor antagonist for the study of acute colon cancer.
|
T7554 |
Substance P (7-11)
|
51165-05-0
|
100%
|
|
Substance P (7-11) (Substance P 7-11(TFA)) is a C-terminal fragment of Substance P .
|
T69140 |
Burapitant
|
537034-22-3
|
100%
|
|
Burapitant (SSR 240600) is a novel non-peptide tachykinin neurokinin 1 (NK) receptor antagonist with anti-coke oven and antidepressant activity.
|
TP1086 |
Men 10376 TFA(135306-85-3,free)
|
TP1086
|
|
|
Men 10376 TFA(135306-85-3,free) (Neurokinin-2 receptor antagonist TFA) is an effective and selective tachykinin nk-2 receptor antagonist with a K I value of 4.4 ...
|
T3716 |
Rolapitant
|
552292-08-7
|
98%
|
|
Rolapitant (SCH619734) Hydrochloride is the hydrochloride salt form of rolapitant, an orally bioavailable, centrally-acting, selective, neurokinin 1 receptor (NK...
|
TP1851L |
Scyliorhinin II acetate
|
TP1851L
|
98%
|
|
Scyliorhinin II acetate is a selective agonist of the neurokinin-3 (NK3) receptor (Ki = 2.5 nM) in rat cerebral cortex.
|
T19518L |
Physalaemin acetate
|
|
98%
|
|
Physalaemin acetate is a non-mammalian tachykinin with high affinity when binding selectively to neurokinin-1 (NK1) receptor.
|
T20413L |
Spantide acetate
|
T20413L
|
98%
|
|
Spantide acetate is a selective antagonist of NK1 receptor with Kis of 230 nM and 8150 nM for NK1 and NK2.
|
T24697L |
R 396 acetate
|
|
98%
|
|
R 396 acetate is an NK-2 Tachykinin Receptor
Antagonist.
|
T38144 |
Elinzanetant
|
929046-33-3
|
98%
|
|
Elinzanetant is a dual antagonist of neurokinin (NK) receptors 1 and 3 and modulates reproductive hormone secretion.
|
T17156 |
Tradipitant
|
622370-35-8
|
98%
|
|
Tradipitant (VLY-686) is an antagonist of neurokinin-1.
|
T24446L |
MEN 10207 acetate
|
|
98%
|
|
MEN 10207 acetate is a selective antagonist for NK-2 tachykinin receptor.
|