T13478 |
β-glycosidase-IN-1
|
176485-27-1
|
98%
|
|
β-glycosidase-IN-1 is a piperidine derivative, and is an inhibitor of β-glycosidase. It has hypoglycemic activity.
|
T29089 |
Valategrast hydrochloride
|
828271-96-1
|
98%
|
|
Valategrast hydrochloride (R411), a dual antagonist of integrin α4β1 (VLA-4), is used for the potential treatment of asthma.
|
T16100 |
Balamapimod
|
863029-99-6
|
98%
|
|
Balamapimod is a reversible inhibitor of Ras/Raf/MEK. It also has a potential anti-tumor activity.
|
T6806 |
Cilengitide TFA
|
199807-35-7
|
98%
|
|
Cilengitide is a potent integrin inhibitor for αvβ3 receptor and αvβ5 receptor with IC50 of 4.1 nM and 79 nM in cell-free assays, respectively; ~10-fold selectiv...
|
T40960 |
Fibronectin
|
86088-83-7
|
98%
|
|
Fibronectin is a macromolecular glycoprotein found in blood, connective tissue, and cell surfaces that serves as a biomarker for tissue damage.Fibronectin is rec...
|
T14573 |
Bimosiamose disodium
|
187269-60-9
|
98%
|
|
Bimosiamose disodium has anti-inflammatory effects[1]. Bimosiamose disodium (TBC-1269Z) is a nonoligosaccharide pan-selectin inhibitor with IC50s of 88 μM, 20 μM...
|
T6657 |
SB273005
|
205678-31-5
|
98%
|
|
SB273005 is a potent integrin inhibitor with Ki of 1.2 nM and 0.3 nM for αvβ3 receptor and αvβ5 receptor, respectively.
|
T14574 |
Bimosiamose
|
187269-40-5
|
98%
|
|
Bimosiamose has anti-inflammatory effects[1]. Bimosiamose (TBC-1269) is a nonoligosaccharide pan-selectin antagonist with IC50s of 88 μM, 20 μM, and 86 μM for E-...
|
T3881 |
Vaccarin
|
53452-16-7
|
99.97%
|
|
Vaccarin is a major flavonoid glycoside in Vaccariae semen, its biotransformation pathways involves methylation, hydroxylation, glycosylation and deglycosylation...
|
T41151L |
K34c hydrochloride
|
|
99.95%
|
|
K34c hydrochloride is an alpha5β1 integrin antagonist for glioblastoma study.
|
T27250 |
Elarofiban
|
198958-88-2
|
99.94%
|
|
Elarofiban(RWJ-53308) is a novel and orally active GPIIb/IIIa antagonist.
|
T8523 |
ILK-IN-3
|
6975-75-3
|
99.88%
|
|
ILK-IN-3 is an inhibitor of integrin linked kinase, and with antitumor activity.
|
T6182 |
Tirofiban
|
144494-65-5
|
99.87%
|
|
Tirofiban (L700462) (MK-383) is a selective palate GPIIb/IIIa antagonist which inhibits platelet aggregation with IC50 of 9 nM.
|
TN1244 |
3'-Demethylnobiletin
|
112448-39-2
|
99.87%
|
|
3'-Demethylnobiletin has chemopreventive effects on colon carcinogenesis, it can significantly inhibit the growth of human colon cancer cells, cause cell-cycle a...
|
T2537 |
Tirofiban hydrochloride monohydrate
|
150915-40-5
|
99.86%
|
|
Tirofiban hydrochloride monohydrate (MK-383 Hydrochloride) is a potent non-peptide, glycoprotein IIb/IIIa (integrins alphaIIbbetaIII) antagonist.
|
T6812 |
Cyclo(-RGDfK)
|
161552-03-0
|
99.83%
|
|
Cyclo(-RGDfK) (Cyclo (-RGDfK)) is an effective and specific αvβ3 integrin inhibitor.
|
TP1459L |
Gly-Arg-Gly-Asp-Ser acetate(96426-21-0 free base)
|
TP1459L
|
99.81%
|
|
Gly-Arg-Gly-Asp-Ser (GRGDS) acetate is a cell binding protein domain derived from the cell-binding region of fibronectin.
|
T5310 |
TR-14035
|
232271-19-1
|
99.81%
|
|
TR-14035 (MDK-1191) is a dual antagonist of α4β7/α4β1 integrins (IC50s: 7/87nM).
|
T2494 |
Cilengitide
|
188968-51-6
|
99.8%
|
|
Cilengitide (EMD 121974) is a potent integrin inhibitor for the αvβ3/5 receptor (IC50: 4.1/79 nM, in cell-free assays); ~10-fold selectivity against gpIIbIIIa.
|
TP1290 |
GRGDSP acetate(91037-75-1 free base)
|
TP1290
|
99.77%
|
|
GRGDSP acetate(91037-75-1 free base) is a synthetic linear RGD peptide and is an integrin inhibitor.
|