T0337 |
Prednisolone acetate
|
52-21-1
|
99.55%
|
|
Prednisolone acetate (Omnipred) is the acetate salt form of prednisolone, a synthetic glucocorticoid with anti-inflammatory and immunomodulating properties.
|
T0798 |
Triamcinolone
|
124-94-7
|
99.54%
|
|
Triamcinolone (Aristocort) is a synthetic glucocorticoid with anti-inflammatory and immunomodulating properties. Upon cell entry, triamcinolone binds to and acti...
|
T32114 |
Hydrocortisone aceponate
|
74050-20-7
|
99.53%
|
|
Hydrocortisone aceponate (Hydrocortisone 17-propionate 21-acetate) is an effective topical glucocorticoid used in the form of a cream to treat various skin disea...
|
T37908 |
Glucocorticoid receptor agonist-1
|
2166375-82-0
|
99.51%
|
|
Glucocorticoid receptor agonist-1 is a potent glucocorticoid receptor agonist with an IC50 of 2.8 nM[1].
|
T1168 |
Desonide
|
638-94-8
|
99.5%
|
|
Desonide (Prednacinolone) is a synthetic glucocorticosteroid for topical use, with anti-inflammatory activity. Desonide binds to glucocorticoid receptors in the ...
|
T21395 |
Finerenone
|
1050477-31-0
|
99.45%
|
|
Finerenone (BAY-948862) is a third-generation, selective, and orally available nonsteroidal mineralocorticoid receptor (MR) antagonist with IC50 of 18 nM for the...
|
T1261 |
Medroxyprogesterone Acetate
|
71-58-9
|
99.45%
|
|
Medroxyprogesterone Acetate (Farlutin) is a synthetic progestin that is derived from 17-hydroxyprogesterone. It is a long-acting contraceptive that is effective ...
|
T0083 |
Eplerenone
|
107724-20-9
|
99.44%
|
|
Eplerenone (CGP 30083) is an aldosterone receptor antagonist and potassium-sparing diuretic used in the therapy of hypertension. Eplerenone therapy has been asso...
|
T1127 |
Beclometasone dipropionate
|
5534-09-8
|
99.44%
|
|
Beclometasone dipropionate (Vancenase) is the dipropionate ester of a synthetic glucocorticoid with anti-inflammatory and immunomodulating properties. After cell...
|
T0367 |
Fluocinolone (Acetonide)
|
67-73-2
|
99.42%
|
|
Fluocinolone Acetonide (Flucort-N) is a glucocorticoid derivative used topically in the treatment of various skin disorders. It is usually employed as a cream, g...
|
T22818 |
GSK9027
|
1229096-88-1
|
99.36%
|
|
GSK9027 (GR agonist 23a) is a nonsteroidal glucocorticoid receptor (GR) agonist.GSK9027 is a partial agonist on the 2×GRE reporter gene compared to dexamethasone...
|
T14981 |
Clobetasone butyrate
|
25122-57-0
|
99.35%
|
|
Clobetasone butyrate, a synthetic glucocorticoid with topical anti-inflammatory activity, is effective in treating corticosteroid-responsive dermatoses, such as ...
|
TQ0225 |
Velsecorat
|
1196509-60-0
|
99.11%
|
|
Velsecorat (AZD7594) is an effective and selective nonsteroidal glucocorticoid receptor modulator (IC50: 0.9 nM).
|
T4277 |
Osilodrostat
|
928134-65-0
|
99.10%
|
|
Osilodrostat (LCI699) (LCI699) is an effective inhibitor of human 11β-hydroxylase (IC50: 2.5 nM) and aldosterone synthase (IC50: 0.7 nM).
|
T13881 |
Dicirenone
|
41020-79-5
|
99.1%
|
|
Dicirenone (SC26304) inhibits the Mineralocorticoid receptor (MR), aldosterone regulation of the urinary K+:Na+ ratio, and aldosterone binding to renal cytoplasm...
|
T0094 |
Budesonide
|
51333-22-3
|
99.03%
|
|
Budesonide (Pulmicort), an anti-inflammatory corticosteroid, has shown the effective glucocorticoid activitie and few mineralocorticoid activities. According to ...
|
T0270 |
Hydrocortisone 17-butyrate
|
13609-67-1
|
99.01%
|
|
Hydrocortisone 17-butyrate (Cortisol 17-butyrate) is a synthetic glucocorticoid receptor agonist with antiinflammatory, antipruritic and vasoconstrictive effects...
|
T16727 |
Relacorilant
|
1496510-51-0
|
99%
|
|
Relacorilant is a selective and orally bioavailable antagonist of glucocorticoid receptor(Ki of 7.2 nM in HepG2 TAT assay, and also shows Kis of 12, 81.2, 210 nM...
|
T0181 |
Loteprednol etabonate
|
82034-46-6
|
99%
|
|
Loteprednol etabonate (Lotemax) is an ophthalmic analog of the corticosteroid prednisolone with anti-inflammatory activity.
|
T14377 |
AZD5423
|
1034148-04-3
|
98.94%
|
|
AZD5423 is an inhaled, potent, selective, and non-steroidal modulator of glucocorticoid receptor (GR) and it effectively reduces allergen-induced responses in su...
|