T79718 |
CaMKIIα-PHOTAC
|
|
98%
|
|
CaMKIIα-PHOTAC is a photochemically targeted chimera (PHOTAC) that specifically targets Ca2+/calmodulin-dependent protein kinase II α (CaMKIIα). This molecule fa...
|
T80269 |
AC3-I, myristoylated
|
|
98%
|
|
Myristoylated AC3-I is a biologically active peptide and a myristoylated variant of the Autocamtide-3-Derived Inhibitory Peptide (AC3-I). It acts as a highly spe...
|
T80549 |
Calmodulin Kinase IINtide, Myristoylated
|
|
98%
|
|
Myristoylated Calmodulin Kinase IINtide (Myr-CaMKIINtide) serves as a selective and noncompetitive inhibitor of CaMKII [1].
|
T16752 |
Rimacalib
|
215174-50-8
|
98%
|
|
Rimacalib is an inhibitor of Ca2+/calmodulin-dependent protein kinase II (IC50s: ~1 μM for CaMKIIα and ~30 μM for CaMKIIγ).
|
T2606 |
KN-93 Phosphate
|
1913269-12-1
|
99.97%
|
|
KN-93 phosphate is a novel membrane-permeant synthetic inhibitor of purified neuronal CaMK-II with K i of 370 nM. KN-93 phosphate inhibits serum-induced fibrobla...
|
T2946 |
Tanshinone IIA sulfonate sodium
|
69659-80-9
|
99.9%
|
|
Tanshinone IIA sulfonate sodium (Tanshinone IIA sodium sulfonate) is a water-soluble derivative of tanshinone IIA extracted from Savia miltiorrhiza; a potent neg...
|
T23523 |
W-5 hydrochloride
|
61714-25-8
|
99.88%
|
|
W-5 hydrochloride (N-(6-Aminohexyl)-1-naphthalenesulfonamide HCl) is a potent calmodulin antagonist.
|
T14069 |
A-3 hydrochloride
|
78957-85-4
|
99.79%
|
|
A-3 hydrochloride is a potent, cell-permeable, reversible, ATP-competitive non-selective antagonist of various kinases. A-3 hydrochloride also inhibits PKC and c...
|
T20792 |
W-7 hydrochloride
|
61714-27-0
|
99.75%
|
|
W-7 hydrochloride (W-7 HCl), a calmodulin antagonist, inhibits Ca2+-calmodulin-dependent myosin light chain kinase and phosphodiesterase, W-7 hydrochloride induc...
|
T68048 |
Cloxacepride
|
65569-29-1
|
99.72%
|
|
cloxacepride is a CaM antagonist that is used to treat asthma disease.
|
T8543 |
KN-92 hydrochloride
|
1431698-47-3
|
99.71%
|
|
KN-92 hydrochloride is an inactive derivative of KN-93. KN-93 is a selective Ca2+/calmodulin-dependent kinase II (CaMKII) inhibitor, competitively blocking CaM b...
|
T3S0807 |
Berbamine
|
478-61-5
|
99.64%
|
|
Berbamine is a natural product extracted from Phellodendron amurense. It acts as a calcium channel blocker and possesses anti-tumor, immunomodulatory, and cardio...
|
T0364 |
Dibucaine
|
85-79-0
|
99.64%
|
|
Dibucaine (Cinchocaine), a local anesthetic of the amide type, is now usually used for surface anesthesia.
|
TP1910L1 |
CALP1 acetate
|
TP1910L1
|
99.63%
|
|
CALP1 acetate is a calmodulin (CaM) agonist (Kd of 88 µM) that binds to the CaM EF-hand/Ca2+-binding site. CALP1 blocks calcium influx and apoptosis (IC50 of 44....
|
T1090 |
Perphenazine
|
58-39-9
|
99.63%
|
|
Perphenazine (Trilafon) is a phenothiazine derivative and a dopamine antagonist with antiemetic and antipsychotic properties.
|
T22538 |
A-7 hydrochloride
|
79127-24-5
|
99.54%
|
|
A-7 hydrochloride is a calmodulin antagonist and causes alterations in the subpopulation of CD44+CD24- in MDA-MB-231 cells.
|
T13384L |
Y-33075 dihydrochloride
|
173897-44-4
|
99.43%
|
|
Y-33075 dihydrochloride is a selective inhibitor of ROCK(IC50 of 3.6 nM).
|
T4530 |
KN-92 phosphate
|
1135280-28-2
|
99.39%
|
|
KN-92 phosphate (KN92-H3PO4) is an inactive derivative of KN-93. KN-93 is a selective inhibitor of Ca2+/calmodulin-dependent kinase II (CaMKII), competitively bl...
|
T1146 |
Nifedipine
|
21829-25-4
|
99.30%
|
|
Nifedipine (Procardia) is a dihydropyridine calcium channel blocking agent. Nifedipine inhibits the transmembrane influx of extracellular calcium ions into myoca...
|
T0445 |
Promethazine
|
60-87-7
|
99.11%
|
|
Promethazine (Proazamine) is an analogue of anti-glaucoma prostaglandin (PG) .
|