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Cat No. | Product Name | Synonyms | Targets |
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T9061 | EN4 | EN4 MYC inhibitor | c-Myc |
EN4 (EN4 MYC inhibitor) MYC inhibitor is a covalent ligand that targets cysteine 171 (C171) of MYC. It is selective for c-MYC over N-MYC and L-MYC, and inhibits MYC transcriptional activity, downregulates MYC targets, an... | |||
TP1315 | C-Myc Peptide Trifluoroacetate | Others | |
c-Myc Peptide Trifluoroacetate is a synthetic peptide corresponding to the C-terminal amino acids (410-419) of human c-myc protein. c-Myc Peptide Trifluoroacetate participates in regulation of growth-related gene transcr... | |||
T3048 | 10058-F4 | c-Myc Inhibitor | c-Myc , Autophagy |
10058-F4 (c-Myc Inhibitor) is a cell-permeable thiazolidinone that specifically inhibits the c-Myc-Max interaction and prevents transactivation of c-Myc target gene expression; induces cell-cycle arrest and apoptosis. | |||
TP2311 | C-MYC PEPTIDE EPITOPE TFA | Others | |
C-MYC PEPTIDE EPITOPE TFA, the product of the c-myc proto-oncogene, is a helix-loop-helix leucine zipper phosphoprotein that regulates gene transcription in cell proliferation, cell differentiation and apoptosis. This pe... | |||
T39751 | MYC-IN-2 | ||
MYC-IN-2 is a protein-protein inhibitor targeting the MYC protein, designed for use in cancer research. | |||
T72040 | C-Myc inhibitor 7 | ||
C-Myc Inhibitor 7, serving as both a c-Myc inhibitor and a multi-target protein degrader, effectively degrades proteins c-MYC, CK1α, GSPT1, and IKZF1/2/3 across various tumor cell types. It holds potential for research i... | |||
TP2179 | C-Myc tag Peptide | Others | |
c-Myc Peptide is a useful displacement of c-Myc-tagged fusion proteins bound to anti-c-Myc antibodies in immunoassays. The successful inhibition of antibody binding by c-Myc peptide demonstrates binding is specific. c-My... | |||
T3686 | 10074-G5 | c-Myc , Autophagy | |
10074-G5 is an inhibitor of c-Myc-Max dimerization. | |||
T4252 | ML327 | c-Myc , Autophagy | |
ML327 is a MYC blocker. ML327 can also de-repress E-cadherin transcription and reverse Epithelial-to-Mesenchymal Transition (EMT). | |||
T15665 | KJ Pyr 9 | c-Myc , Autophagy | |
KJ Pyr 9 is an MYC inhibitor (Kd: 6.5 nM in vitro assay). | |||
T9628 | 10074-A4 | c-Myc | |
10074-A4 is a c-Myc binding compound that associates with c-Myc370–409 and behaves like a “ligand cloud” around a “protein cloud”, with distinct features from that of a non-binding ligand. | |||
T12132 | MYCi361 | NUCC-0196361 | c-Myc |
MYCi361 (NUCC-0196361) is an inhibitor of MYC (binding to MYC with Kd of 3.2 μM). | |||
T4367 | Mycro 3 | Mycro-3 | c-Myc , Autophagy |
Mycro 3 is potent and selective for c-Myc in whole cell assays. | |||
T12134 | MYCMI-6 | NSC354961 | Apoptosis , c-Myc |
MYCMI-6 (NSC-354961) is a potent and selective inhibitor of endogenous MYC:MAX protein interactions,reduces proliferation and induces massive apoptosis in tumor tissue from a MYC-driven xenograft tumor model without seve... | |||
T60019 | VPC-70063 | Thiourea, N-[3,5-bis(trifluoromethyl)phenyl]-N'-(phenylmethyl)- | Apoptosis , PARP , c-Myc |
VPC-70063 (Thiourea, N-[3,5-bis(trifluoromethyl)phenyl]-N'-(phenylmethyl)-) is an inhibitor of c-Myc-MAX. VPC-70063 exhibits Myc-Max transcriptional activity inhibition of 106% with an IC50 of 8.9 μM and Myc-Max/UBE2C do... | |||
T9033 | BTYNB | MDK6620,BTYNB IMP1 Inhibitor | Others , c-Myc , NF-κB |
BTYNB (MDK6620) is an inhibitor of the oncofetal mRNA-binding protein IMP1 (IC50 = 5 μM for IMP1 binding to c-Myc mRNA). MDK6620 downregulates β-TrCP1 mRNA and reduces activation of nuclear transcriptional factors-kappa ... | |||
T78055 | MYC-RIBOTAC | c-Myc | |
MYC-RIBOTAC, a ribonuclease-targeting chimera (RIBOTAC) specific to the MYC internal ribosome entry site (IRES), comprises an MYC mRNA-binding element tethered to a small molecule that recruits and activates RNase L1. Th... | |||
T10352 | APTO-253 | LOR-253,LT-253 | Apoptosis , c-Myc , KLF |
APTO-253 (LOR-253) inhibits c-Myc expression, stabilizes G-quadruplex DNA, and induces cell cycle arrest and apoptosis in acute myeloid leukemia cells. APTO-253 mediates anticancer activity through the induction of the K... | |||
T74460 | C-Myc inhibitor 5 | ||
c-Myc Inhibitor 5 (DA3) is a fluorescent bispurine compound with a long-chain bridge that selectively binds to the c-MYC G-quadruplex, exhibiting a dissociation constant (K D) of 16 μM. Unlike other G4-driven oncogenes, ... | |||
T72619 | C-Myc inhibitor 8 | ||
C-Myc Inhibitor 8 is an effective compound for cancer research, inhibiting cell viability across a range of cancer types and demonstrating growth suppression in human prostate and lung cancers within mouse models. This i... | |||
T9032 | MGH-CP1 | Others | |
MGH-CP1 is a potent and selective inhibitor TEAD palmitoylation. It exhibits dose-dependent and potent inhibition of TEAD2/4 auto-palmitoylation in vitro with IC50 of 710 nM and 672 nM, respectively. | |||
T9093 | NY2267 | Acetic acid, 2-[[6-[2-(cyclohexylamino)-1-[[(4-methoxyphenyl)methyl](2-pyridinylcarbonyl)amino]-2-oxoethyl]-2-naphthalenyl]oxy]-, 1,1-dimethylethyl ester | c-Myc |
NY2267 (Acetic acid, 2-[[6-[2-(cyclohexylamino)-1-[[(4-methoxyphenyl)methyl](2-pyridinylcarbonyl)amino]-2-oxoethyl]-2-naphthalenyl]oxy]-, 1,1-dimethylethyl ester) is a disruptor of Myc-Max interaction, with an IC50 of 36... | |||
T63359 | C-Myc inhibitor 4 | ||
c-Myc inhibitor 4 is a potent, orally active c-Myc-reducing compound. c-Myc is an important proto-oncogene, which is closely associated with the development of many tumors. | |||
T79439 | C-Myc inhibitor 12 | c-Myc | |
Compound 67h, also known as c-Myc inhibitor 12, is a potent inhibitor of c-Myc, exhibiting a pEC50 value of 6.4 [1]. | |||
T72620 | C-Myc inhibitor 9 | ||
c-Myc Inhibitor 9 (Compound 332) is an effective c-Myc inhibitor, exhibiting a logEC50 of ≥6, and demonstrating significant tumor growth inhibition in nude mouse models. This compound is utilized in cancer research. | |||
T79438 | C-Myc inhibitor 11 | c-Myc | |
c-Myc inhibitor 11 (Compound 67e), a c-MYC inhibitor (p EC 50 : 6.4), exhibits high clearance, a moderate volume of distribution, and a short half-life in rat pharmacokinetic assays, making it suitable for cancer researc... | |||
T75239 | C-Myc inhibitor 10 | ||
C-Myc Inhibitor 10 (compound 17), exhibiting enhanced cellular potency, benefits from increased permeability due to the methylation of the morpholine nitrogen [1]. | |||
T9370 | DCBP-1 | Epigenetic Reader Domain , Ligand for E3 Ligase | |
dCBP-1 is a chemical degrader of p300/CBP. dCBP-1 hijacks the E3 ubiquitin ligase CRBN for selective degradation of p300/CBP. Degradation of p300/CBP by dCBP-1 leads to effective multiple myeloma cell killing. | |||
T20533 | NNK | Nicotine-derived nitrosamine ketone | Lipoxygenase |
NNK (Nicotine-derived nitrosamine ketone) is a procarcinogen and a major tobacco-specific toxicant. It inhibits the expression of lysyl oxidase which is a tumor suppressor. | |||
T11285 | FIDAS-5 | Others | |
FIDAS-5, a potent and orally active methionine S-adenosyltransferase 2A (MAT2A) inhibitor with an IC50 of 2.1 μM, competitively inhibits S-adenosylmethionine (SAM) binding to MAT2A. It exhibits anticancer activities. | |||
T11284 | FIDAS-3 | Others , Wnt/beta-catenin , Methionine Adenosyltransferase (MAT) | |
FIDAS-3, a stilbene derivative and potent Wnt inhibitor with an IC50 of 4.9 μM for methionine S-adenosyltransferase 2A (MAT2A), exhibits anticancer activities by effectively competing with S-adenosylmethionine (SAM) for ... | |||
T10760 | Ceramides Mixture | Telomerase | |
Ceramides Mixture, an endogenous ceramide, consists of hydroxy and non-hydroxy fatty acid-containing ceramides. It is involved in the regulation of cell cycle arrest, growth inhibition, and modulation of telomerase activ... | |||
T6010 | Idarubicin hydrochloride | Idamycin,4-demethoxydaunorubicin (NSC256439, 4-DMDR) HCl,4-Demethoxydaunorubicin hydrochloride,Idarubicin HCl,Zavedos | Topoisomerase , Antibacterial , Autophagy , Antifungal |
Idarubicin hydrochloride (Zavedos), a hydrochloride salt form of Idarubicin, is a DNA topoisomerase II (topo II) inhibitor for MCF-7 cells ( IC50: 3.3 ng/mL). | |||
T8658 | NEO2734 | EP31670 | Epigenetic Reader Domain , Histone Acetyltransferase |
NEO2734 (EP31670) is an orally active and selective inhibitor of p300/CBP and BET bromodomain(IC50 of <30 nM for both p300/CBP and BET bromodomains). | |||
T10765 | Eragidomide | CC-90009,Cereblon modulator 1 | Apoptosis , Ligand for E3 Ligase , Molecular Glues |
Eragidomide (CC-90009; Cereblon modulator 1) is a cereblon (CRBN) E3 ligase modulator. Eragidomide specifically binds to CRBN, thereby affecting the activity of the ubiquitin E3 ligase complex. | |||
T6203 | Saxagliptin | BMS-477118,Onglyza | Proteasome , DPP-4 |
Saxagliptin (BMS-477118) is a selective and reversible DPP4 inhibitor with IC50 of 26 nM. | |||
T0178 | Saxagliptin hydrate | Onglyza hydrate,BMS-477118 hydrate | Proteasome , DPP-4 |
Saxagliptin hydrate (Onglyza hydrate) is a selective and reversible DPP4 inhibitor (IC50: 26 nM; Ki: 1.3 nM). | |||
T12133 | MYCi975 | NUCC-0200975 | c-Myc |
MYCi975 (NUCC-0200975) is an orally active inhibitor of MYC. | |||
T1142 | Clindamycin phosphate | Clindamycin 2-phosphate,Clindamycin 2-dihydrogen phosphate,NSC 618653,U-28508 | ribosome , Antibacterial , Antibiotic , Parasite |
Clindamycin Phosphate is the phosphate salt form of clindamycin, a semi-synthetic, chlorinated broad-spectrum antibiotic produced by chemical modification of lincomycin. Clindamycin phosphate (Clindamycin 2-dihydrogen ph... | |||
T22297 | Clindamycin hydrochloride monohydrate | Clindamycin alcoholate | Antibiotic |
Clindamycin hydrochloride monohydrate (Clindamycin alcoholate) is a protein synthesis inhibitor used orally, capable of diminishing virulence factor expression in Staphylococcus aureus at sub-minimum inhibitory concentra... | |||
T16684 | Puromycin aminonucleoside | NSC 3056 | Apoptosis , Proteasome , Aminopeptidase , Antibacterial , Antibiotic |
Puromycin aminonucleoside (NSC-3056) increases podocyte permeability by modulating ZO-1 in an oxidative stress-dependent manner. | |||
T67717L | Questiomycin A derivatives 18 TFA | ||
Questiomycin A derivatives 18 TFA is A Questiomycin A derivative with antibacterial and anticancer activity and inhibition of the expression of the cell-protective ER chaperone protein GRP78. | |||
T67711 | Questiomycin A derivatives 12 | Others | |
Questiomycin A derivatives 12 is a Questiomycin A derivative. | |||
T3097 | Mycophenolic Acid Impurity | 5,7-dihydroxy-4-methylphthalide | Others |
Mycophenolic Acid Impurity (5,7-dihydroxy-4-methylphthalide) is an an immunosuppresant drug and potent anti-proliferative, and can be used in place of the older anti-proliferative azathioprine. It is usually used as part... | |||
T12242 | Norvancomycin hydrochloride | Desmethyl-vancomycin hydrochloride | Antibacterial |
Norvancomycin hydrochloride (Desmethyl-vancomycin hydrochloride) is used as a treatment for endocarditis, osteomyelitis, pneumonia, sepsis, or soft tissue infections caused by Staphylococcus. | |||
T4989 | Fosfomycin Tromethamine | Antibacterial , Antibiotic | |
An antibiotic produced by Streptomyces fradiae. | |||
T6116L | Bleomycin hydrochloride | DNA/RNA Synthesis | |
Bleomycin hydrochloride is a potent antitumor antibiotic that functions as a DNA synthesis inhibitor and DNA damaging agent. | |||
T1434 | Clarithromycin | A-56268 | P450 , ribosome , MRP , Antibacterial , Antibiotic , Autophagy |
Clarithromycin (A-56268) is a Macrolide Antimicrobial. The mechanism of action of clarithromycin is as a Cytochrome P450 3A4 Inhibitor, and Cytochrome P450 3A Inhibitor, and P-Glycoprotein Inhibitor. The chemical classif... | |||
T67713 | Questiomycin A derivatives 14 | Others | |
Questiomycin A derivatives 14 is a Questiomycin A derivative. | |||
T3131 | Fosfomycin calcium | Phosphomycin calcium salt,Fosmicin | Antibacterial , Antibiotic |
Fosfomycin calcium (Phosphomycin calcium salt) is a blood-brain barrier penetrating, broad-spectrum antibiotic by irreversibly inhibiting an early stage in cell wall synthesis. |
Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
TN1892 | Lusianthridin | Others , c-Myc | |
Lusianthridin is a natural product from Dendrobium venustum. Lusianthridin exhibits anti-migratory property at nontoxic concentrations. Lusianthridin enhances c-Myc degradation through the inhibition of Src-STAT3 signali... | |||
T21065 | Artemisitene | Others | |
Artemisitene is the oxidized form of Artemisinin and is an antimalarial agent. Artemisinin precursors are the important basic substances for biosynthesis of Artemisinin, including Artemisinin B, Artemisitene, Artemisini... | |||
T3673 | Mollugin | Rubimaillin | HER , JAK |
Mollugin (Rubimaillin) may be a JAK2 inhibitor and inhibits LPS-induced inflammatory responses by blocking the activation of the JAK-STAT pathway. Mollugin as a candidate for a chemotherapeutic agent in OSCCs via the upr... | |||
T4S1173 | Agrimol B | Sirtuin , PPAR | |
1. Agrimol B is a main active ingredient isolated from Agrimonia pilosa Ledeb. | |||
T2764 | (S)-10-Hydroxycamptothecin | 10-Hydroxycamptothecin,10-HCPT | Apoptosis , Topoisomerase |
(S)-10-Hydroxycamptothecin (10-HCPT) is a DNA topoisomerase I inhibitor, utilized as a clinical therapy agent against hepatoma. | |||
T0060 | Streptomycin sulfate | Plantomycin,Estreptomicina,Phytomycin | ribosome , Antibacterial , Antibiotic |
Streptomycin sulfate (Phytomycin) is a sulfate salt of streptomycin that is a protein synthesis inhibitor. | |||
T12540 | Pristinamycin IA | Mikamycin IA,Mikamycin B | Others , Antibiotic , P-gp |
Pristinamycin IA (Mikamycin B) is a substrate for the P-glycoprotein and a cyclo-peptidic macrolactone antibiotic. | |||
T3629 | Gamithromycin | ML-1709460 | Antibacterial , Antibiotic |
Gamithromycin (ML-1709460) is a macrolide compound with antibacterial activity. | |||
T17143 | Toyocamycin | Vengicide | Apoptosis , Others , IRE1 , Antibiotic , Antifungal |
Toyocamycin (Vengicide) is an adenosine analog produced by Actinomycete, acts as an XBP1 inhibitor, inhibits IRE1α-induced ATP-dependent XBP1 mRNA cleavage (IC50: 80 nM). Toyocamycin induces apoptosis. | |||
T21344 | 1-Deoxynojirimycin hydrochloride | Moranoline,AT2220,Duvoglustat hydrochloride,1-Deoxynojirimycin,DNJ,deoxynojirimycin | PI3K , Antibacterial , Antibiotic , Glucosidase |
1-Deoxynojirimycin hydrochloride (Moranoline) is a potent and selective inhibitor of alpha-glucosidase, most commonly found in mulberry leaves. Duvoglustat is used to suppress the elevation of postprandial hyperglycemia. | |||
T3675 | 1-Deoxynojirimycin | Duvoglustat,Moranoline,moranolin | PI3K , Glucosidase |
1-Deoxynojirimycin (Moranoline) is a potent α-glucosidase inhibitor, suppressing postprandial blood glucose, thereby possibly preventing diabetes mellitus. | |||
T1084 | Apramycin sulfate | Nebramycin II,Ai3-29795 | Antibacterial , Antibiotic |
Apramycin sulfate (Nebramycin II) is an aminoglycoside antibiotic. | |||
T1419 | Azithromycin hydrate | CP-62993 dihydrate,Azithromycin dihydrate | ribosome , Antibacterial , Antibiotic , Autophagy |
Azithromycin hydrate (CP-62993 dihydrate) is a semi-synthetic macrolide antibiotic structurally related to ERYTHROMYCIN. It has been used in the treatment of Mycobacterium avium intracellulare infections, toxoplasmosis, ... | |||
T9605 | Sangivamycin | BA-90912,NSC 65346 | Nucleoside Antimetabolite/Analog , PKC |
Sangivamycin (NSC-65346) is an effective inhibitor of protein kinase C (PKC, Ki = 10 μM). Sangivamycin exhibits antiproliferative activity against a variety of human cancers. | |||
T36818 | Questiomycin A | GPR , Antibacterial | |
Questiomycin A is an antibiotic produced in crème fraiche with antibacterial and anticancer activities. Questiomycin A suppresses expression of GRP78, a cell-protective ER chaperone protein. | |||
T0474 | Erythromycin ethylsuccinate | EES | ribosome , HIV Protease , Antibacterial , Antibiotic , Autophagy |
Erythromycin ethylsuccinate (EES) is a macrolide antibiotic, produced by Streptomyces erythreus. | |||
T5003 | Rifamycin sodium | Rifamycin sodium salt | Antibacterial , Antibiotic |
Rifamycin sodium (Rifamycin sodium salt) salt is an antibiotic that inhibits bacterial DNA-dependent RNA polymerase. It is effective against Gram-positive bacteria. | |||
TP1072 | Valinomycin | NSC 122023 | Apoptosis , PTEN , Antibacterial , Antibiotic , Autophagy |
Valinomycin (NSC-122023) is a cyclic depsipeptide antibiotic and a potassium-specific ionophore.Valinomycin induces PINK1 activation and promotes Parkin phosphorylation at Ser65. | |||
T8118 | Bekanamycin | Kanamycin B | Antibacterial , Antibiotic |
Bekanamycin (Kanamycin B) is an aminoglycoside antibiotic. | |||
T0950 | Neomycin sulfate | Framycin sulfate | Phospholipase , ribosome , Antibacterial , Antibiotic |
Neomycin sulfate (Framycin sulfate) is a broad-spectrum aminoglycoside antibiotic that blocks the synthesis of bacterial proteins in order to exert antimicrobial activity. Neomycin sulfate is commonly used to screen prok... | |||
T1335 | Mycophenolic acid | Mycophenolate,RS-61443 | Apoptosis , Dehydrogenase , Endogenous Metabolite , Antibacterial , Antibiotic , UGT , Antifungal |
Mycophenolic acid (Mycophenolate) is an inosine monophosphate dehydrogenase(IMPDH) inhibitor with anti-proliferative activity. | |||
T60104 | Mycophenolic acid-β-D-glucuronide solution | Others | |
Mycophenolic acid glucuronide is the glucuronide metabolite of mycophenolic acid in human plasma. | |||
T21820 | Resistomycin | Geliomycin,Heliomycin | Antibiotic |
Resistomycin (Geliomycin), a pentacyclic polyketide antibiotic, exhibits potent anticancer properties by triggering apoptosis. | |||
T0971 | Dirithromycin | Dirithromycinum,ASE 136,LY237216,Diritromicina,Dirithromycine | ribosome , Antibacterial , Antibiotic |
Dirithromycin (LY237216) is a macrolide glycopeptide antibiotic. It is used to treat many different types of bacterial infections, such as bronchitis, pneumonia, tonsillitis, and even skin infections. | |||
T1235 | Lincomycin hydrochloride monohydrate | Lincomycin hydrochloride hydrate | ribosome , Antibacterial , Antibiotic |
Lincomycin hydrochloride monohydrate (Lincomycin hydrochloride hydrate) is an antibiotic produced by Streptomyces lincolnensis var. lincolnensis. It has been used in the treatment of staphylococcal, streptococcal, and Ba... | |||
T21494 | Oligomycin | HIF | |
Oligomycin is an antifungal antibiotic that is an inhibitor of H+-ATP synthetase. The Oligomycin blocks oxidative phosphorylation and the electron transport chain. Oligomycin inhibited HIF-1alpha expression in hypoxic tu... | |||
T20699 | Daunomycinone | Daunomycinon,Leukaemomycinone C,NSC 109351,NSC-109351,NSC109351 | Antibiotic |
Daunomycinone (NSC-109351) is a glycan of daunomycin, which belongs to the antibiotic class and is a representative glycan of tumour-inhibiting anthracyclines, used in the treatment of cancer and leukaemia. | |||
T1032 | Erythromycin | E-Mycin | ribosome , Antibacterial , Antibiotic |
Erythromycin (E-Mycin) is a Macrolide and Macrolide Antimicrobial. The physiologic effect of erythromycin is by means of Decreased Sebaceous Gland Activity. | |||
T6740 | Bafilomycin A1 | Apoptosis , Proton pump , Antibacterial , Antibiotic , Autophagy | |
Bafilomycin A1 belongs to the macrolide class of antibiotics and is a V-ATPase (IC50=0.44 nM) that is specific and reversible. Bafilomycin A1 is an inhibitor of the late phase of autophagy, blocking the fusion of autopha... | |||
T1381 | Milbemycin oxime | Others , Antibiotic , Parasite | |
Milbemycin oxime is a broad spectrum antiparasitic, used as a veterinary drug. | |||
T2481 | Ascomycin | FK520,Immunomycin,FR-900520 | Phosphatase , Others , Antibiotic , Parasite , Antifungal |
Ascomycin (Immunomycin)(Immunomycin, FR-900520, FK520) is an ethyl analog of tacrolimus (FK506) with strong immunosuppressant properties. | |||
T13229 | Tunicamycin | Influenza Virus , Antibacterial , Antibiotic , Antifungal | |
Tunicamycin is a mixture of antibiotics that inhibit N-linked glycosylation by blocking GlcNAc phosphotransferase (GPT). Tunicamycin has antitumor activity, as well as anti-bacterial, anti-fungal, and anti-viral activity... | |||
T1214 | Ribostamycin sulfate | Vistamycin sulfate | Antibacterial , Antibiotic |
Ribostamycin sulfate (Vistamycin sulfate) , an aminoglycoside antibiotic, contains a neutral sugar moiety and is produced by Streptomyces ribosome. | |||
T3607 | Leucomycin | Kitasamycin,Leucomycin V,Turimycin | Antibacterial , Antibiotic |
Leucomycin (Turimycin) is a macrolide antibiotic. | |||
T6402 | Azomycin | 2-Nitroimidazole,Ro 05-9129,Amicin | Antibacterial , Antibiotic |
Azomycin (Ro 05-9129) is an antimicrobial antibiotic produced by a strain of Nocardia mesenterica. | |||
T1255 | Tobramycin | NSC 180514,Nebramycin Factor 6,Deoxykanamycin B | ribosome , Antibacterial , Antibiotic |
Tobramycin (NSC-180514) is an aminoglycoside, broad-spectrum antibiotic produced by Streptomyces tenebrarius. | |||
T11665 | Ionomycin calcium | SQ23377 calcium | Apoptosis , Calcium Channel , Antibacterial , Antibiotic , PKC |
lonomycin calcium is a potent, selective calcium ionophore and an antibiotic produced by Streptomyces conglobatus. also induces the activation of protein kinase C (PKC). Ionomycin calcium (SQ23377 calcium) is highly spec... | |||
T14329 | Ascamycin | Nucleoside Antimetabolite/Analog , Others , Antibacterial , Antibiotic | |
Ascamycin is a 5'-O-sulfonamide ribonucleoside antibiotic produced by Streptomyces spp. It shows selective antibacterial activity against Xanthomonas species and inhibits Xanthomonas citri, Xanthomonas oryzae and phage w... | |||
T8347 | Rifamycin S | Reactive Oxygen Species , ROS , Antibacterial , Antibiotic | |
Rifamycin S is a potent DNA-dependent RNA polymerase inhibitor,is a quinone and an antibiotic agnet against Gram-positive bacteria | |||
T6343 | Geldanamycin | NSC 122750 | HSP , Influenza Virus , Tyrosine Kinases , Antibacterial , Antibiotic |
Geldanamycin, an HSP90 inhibitor (Kd: 1.2 μM), specifically disrupts glucocorticoid receptor (GR)/HSP association. | |||
T6293 | Mycophenolate Mofetil | TM-MMF,RS 61443 | Apoptosis , Dehydrogenase , Drug Metabolite |
Mycophenolate Mofetil (TM-MMF), an immunosuppressive agent, is the 2-morpholinoethyl ester of mycophenolic acid (MPA), and an inhibitor of inosine monophosphate dehydrogenase (IMPDH). | |||
T6401 | Azithromycin | Zithromax,CP 62993,XZ-450 | Others , Antibacterial , Antibiotic , Autophagy |
Azithromycin (CP 62993) is an antibiotic by inhibiting protein synthesis, used for the treatment of bacterial infections. | |||
T7148 | JOSAMYCIN | EN-141 | Antibacterial , Antibiotic |
Josamycin (EN-141) is a macrolide antibiotic exhibiting antimicrobial activity. The dissociation constant Kd from ribosome for Josamycin is 5.5 nM. | |||
T0709 | Natamycin | Pimaricin | Estrogen/progestogen Receptor , Endogenous Metabolite , Antibiotic , Antifungal |
Natamycin (Pimaricin) is a Polyene Antimicrobial. | |||
T6116 | Bleomycin Sulfate | Blenoxane,NSC125066 | DNA/RNA Synthesis , Antibiotic |
Bleomycin Sulfate (Blenoxane) is a glycopeptide antibiotic, an inhibitor of DNA synthesis. Bleomycin Sulfate causes DNA strand breaks but not RNA strand breaks. Bleomycin Sulfate has antitumor activity. | |||
T1022 | Hygromycin B | Hygrovetine | ribosome , Antibacterial , Antibiotic , Antifungal |
Hygromycin B (Hygrovetine) is an aminoglycoside antibiotic that inhibits protein synthesis by interfering with translocation and causing mistranslation of the 70S ribosome. Hygromycin B can be used to screen prokaryotic ... | |||
T1537 | Rapamycin | Sirolimus,AY 22989,NSC-2260804 | Others , Endogenous Metabolite , Antibiotic , mTOR , Autophagy , Antifungal |
Rapamycin (AY 22989) is a natural product of macrolides, an mTOR inhibitor with specificity (HEK293 cells: IC50=0.1 nM). Rapamycin has immunosuppressive activity and induces autophagy. | |||
T5530 | Mithramycin A | Plicamycin | DNA/RNA Synthesis |
Mithramycin A (Plicamycin), a DNA-binding antitumor antibiotic, is a selective specificity protein 1 (Sp1) inhibitor, which inhibits the growth of various cancers by decreasing Sp1 protein. Specificity protein 1 (Sp1) is... | |||
T0906 | Salinomycin | Procoxacin | Wnt/beta-catenin , Antibacterial |
Salinomycin (Procoxacin), a polyether potassium ionophore antibiotic, specifically inhibits the growth of gram-positive bacteria. It acts as a potent inhibitor of Wnt/β-catenin signaling, blocking Wnt-induced LRP6 phosph... | |||
T2762 | Kasugamycin hydrochloride | Kasumin | Antibacterial , Antibiotic , Antifungal |
Kasugamycin hydrochloride (Kasumin) is an aminoglycoside antibiotic that was originally isolated in 1965, from Streptomyces kasugaensis, a Streptomyces strain found near the Kasuga shrine in Nara, Japan. Kasugamycin hydr... | |||
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Cat No. | Product Name | Species | Expression System |
---|---|---|---|
TMPH-02791 | C-Myc Protein, Mouse, Recombinant (GST) | Mouse | E. coli |
Transcription factor that binds DNA in a non-specific manner, yet also specifically recognizes the core sequence 5'-CAC[GA]TG-3'. Activates the transcription of growth-related genes. Binds to the VEGFA promoter, promotin... | |||
TMPH-01720 | C-Myc Protein, Human, Recombinant (His) | Human | E. coli |
Transcription factor that binds DNA in a non-specific manner, yet also specifically recognizes the core sequence 5'-CAC[GA]TG-3'. Activates the transcription of growth-related genes. Binds to the VEGFA promoter, promotin... | |||
TMPH-01721 | C-Myc Protein, Human, Recombinant (Avi & His & MBP), Biotinylated | Human | E. coli |
Transcription factor that binds DNA in a non-specific manner, yet also specifically recognizes the core sequence 5'-CAC[GA]TG-3'. Activates the transcription of growth-related genes. Binds to the VEGFA promoter, promotin... | |||
TMPY-02888 | MAX Protein, Human, Recombinant (His & GST) | Human | Baculovirus Insect Cells |
MYC associated factor X contains 1 basic helix-loop-helix (bHLH) domain and belongs to the MAX family. It is highly expressed in the brain, heart, and lung while lower levels are seen in the liver, kidney, and skeletal m... | |||
TMPJ-01040 | MAX Protein, Human, Recombinant (His) | Human | E. coli |
Myc-Associated Factor X (MAX) is a member of the basic helix-loop-helix leucine zipper (bHLHZ) family of transcription factors. It contains 1 basic helix-loop-helix (bHLH) domain. It is found in the brain, heart, and lun... | |||
TMPH-03328 | Mcpt1 Protein, Rat, Recombinant (Myc) | Rat | E. coli |
Major secreted protease of mast cells with suspected roles in vasoactive peptide generation, extracellular matrix degradation, and regulation of gland secretion. May participate in generating perivascular beta-protein wh... | |||
TMPH-01898 | PARL Protein, Human, Recombinant (Myc) | Human | E. coli |
Required for the control of apoptosis during postnatal growth. Essential for proteolytic processing of an antiapoptotic form of OPA1 which prevents the release of mitochondrial cytochrome c in response to intrinsic apopt... | |||
TMPH-02552 | BMP3 Protein, Mouse, Recombinant (Myc) | Mouse | E. coli |
Negatively regulates bone density. Antagonizes the ability of certain osteogenic BMPs to induce osteoprogenitor differentitation and ossification. | |||
TMPH-02825 | ACOX1 Protein, Mouse, Recombinant (Myc) | Mouse | E. coli |
Catalyzes the desaturation of acyl-CoAs to 2-trans-enoyl-CoAs. First enzyme of the fatty acid beta-oxidation pathway.; Shows highest activity against medium-chain fatty acyl-CoAs and activity decreases with increasing ch... | |||
TMPH-01794 | NR2F6 Protein, Human, Recombinant (His & Myc) | Human | HEK293 Cells |
NR2F6 Protein, Human, Recombinant (His & Myc) is expressed in HEK293 mammalian cells with N-6xHis-Myc tag. The predicted molecular weight is 47.0 kDa and the accession number is P10588. | |||
TMPH-02828 | PLAA Protein, Mouse, Recombinant (His & Myc) | Mouse | Baculovirus Insect Cells |
PLAA Protein, Mouse, Recombinant (His & Myc) is expressed in Baculovirus insect cells with N-10xHis and C-Myc tag. The predicted molecular weight is 13.6 kDa and the accession number is P27612. | |||
TMPH-02647 | FAM20C Protein, Mouse, Recombinant (His & Myc) | Mouse | Baculovirus Insect Cells |
FAM20C Protein, Mouse, Recombinant (His & Myc) is expressed in Baculovirus insect cells with N-10xHis and C-Myc tag. The predicted molecular weight is 60.4 kDa and the accession number is Q5MJS3. | |||
TMPH-02692 | PLA2G15 Protein, Mouse, Recombinant (His & Myc) | Mouse | E. coli |
PLA2G15 Protein, Mouse, Recombinant (His & Myc) is expressed in E. coli expression system with N-10xHis and C-Myc tag. The predicted molecular weight is 50.5 kDa and the accession number is Q8VEB4. | |||
TMPH-01783 | NOTCH2NLB Protein, Human, Recombinant (His & Myc) | Human | Baculovirus Insect Cells |
NOTCH2NLB Protein, Human, Recombinant (His & Myc) is expressed in Baculovirus insect cells with N-10xHis and C-Myc tag. The predicted molecular weight is 31.3 kDa and the accession number is P0DPK3. | |||
TMPH-03114 | ITGB1 Protein, Pig, Recombinant (His & Myc) | Sus scrofa (Pig) | E. coli |
ITGB1 Protein, Pig, Recombinant (His & Myc) is expressed in E. coli expression system with N-10xHis and C-Myc tag. The predicted molecular weight is 34.1 kDa and the accession number is Q9GLP0. | |||
TMPH-03249 | ATP5F1B Protein, Rat, Recombinant (His & Myc) | Rat | E. coli |
ATP5F1B Protein, Rat, Recombinant (His & Myc) is expressed in E. coli expression system with N-10xHis and C-Myc tag. The predicted molecular weight is 59.2 kDa and the accession number is P10719. | |||
TMPH-00993 | SLC4A1 Protein, Human, Recombinant (His & Myc) | Human | E. coli |
SLC4A1 Protein, Human, Recombinant (His & Myc) is expressed in E. coli expression system with N-10xHis and C-Myc tag. The predicted molecular weight is 50.3 kDa and the accession number is P02730. | |||
TMPH-02429 | Fukutin Protein, Cynomolgus, Recombinant (His & Myc) | Cynomolgus | E. coli |
Fukutin Protein, Cynomolgus, Recombinant (His & Myc) is expressed in E. coli expression system with N-10xHis and C-Myc tag. The predicted molecular weight is 58.0 kDa and the accession number is Q60HG0. | |||
TMPH-02930 | TREX1 Protein, Mouse, Recombinant (His & Myc) | Mouse | E. coli |
TREX1 Protein, Mouse, Recombinant (His & Myc) is expressed in E. coli expression system with N-10xHis and C-Myc tag. The predicted molecular weight is 41.1 kDa and the accession number is Q91XB0. | |||
TMPH-02916 | SULT1A1 Protein, Mouse, Recombinant (His & Myc) | Mouse | E. coli |
SULT1A1 Protein, Mouse, Recombinant (His & Myc) is expressed in E. coli expression system with N-10xHis and C-Myc tag. The predicted molecular weight is 39.0 kDa and the accession number is P52840. | |||
TMPH-01606 | BAG6 Protein, Human, Recombinant (His & Myc) | Human | Baculovirus Insect Cells |
BAG6 Protein, Human, Recombinant (His & Myc) is expressed in Baculovirus insect cells with N-10xHis and C-Myc tag. The predicted molecular weight is 38.7 kDa and the accession number is P46379. | |||
TMPH-02920 | SMN1 Protein, Mouse, Recombinant (His & Myc) | Mouse | HEK293 Cells |
SMN1 Protein, Mouse, Recombinant (His & Myc) is expressed in HEK293 mammalian cells with N-10xHis and C-Myc tag. The predicted molecular weight is 35.3 kDa and the accession number is P97801. | |||
TMPH-02950 | HADHB Protein, Mouse, Recombinant (His & Myc) | Mouse | E. coli |
HADHB Protein, Mouse, Recombinant (His & Myc) is expressed in E. coli expression system with N-10xHis and C-Myc tag. The predicted molecular weight is 54.6 kDa and the accession number is Q99JY0. | |||
TMPH-01892 | ATP4A Protein, Human, Recombinant (His & Myc) | Human | E. coli |
ATP4A Protein, Human, Recombinant (His & Myc) is expressed in E. coli expression system with N-10xHis and C-Myc tag. The predicted molecular weight is 54.6 kDa and the accession number is P20648. | |||
TMPH-02949 | HADHA Protein, Mouse, Recombinant (His & Myc) | Mouse | E. coli |
HADHA Protein, Mouse, Recombinant (His & Myc) is expressed in E. coli expression system with N-10xHis and C-Myc tag. The predicted molecular weight is 52.1 kDa and the accession number is Q8BMS1. | |||
TMPH-03372 | Sharpin Protein, Rat, Recombinant (His & Myc) | Rat | E. coli |
Sharpin Protein, Rat, Recombinant (His & Myc) is expressed in E. coli expression system with N-10xHis and C-Myc tag. The predicted molecular weight is 47.7 kDa and the accession number is Q9EQL9. | |||
TMPH-01086 | CSPG4 Protein, Human, Recombinant (His & Myc) | Human | HEK293 Cells |
CSPG4 Protein, Human, Recombinant (His & Myc) is expressed in HEK293 mammalian cells with N-10xHis and C-Myc tag. The predicted molecular weight is 73.2 kDa and the accession number is Q6UVK1. | |||
TMPH-01255 | DNM1L Protein, Human, Recombinant (His & Myc) | Human | E. coli |
DNM1L Protein, Human, Recombinant (His & Myc) is expressed in E. coli expression system with N-10xHis and C-Myc tag. The predicted molecular weight is 84.4 kDa and the accession number is O00429. | |||
TMPH-03747 | CCDC112 Protein, Human, Recombinant (His & Myc) | Human | E. coli |
CCDC112 Protein, Human, Recombinant (His & Myc) is expressed in E. coli expression system with N-10xHis and C-Myc tag. The predicted molecular weight is 61.0 kDa and the accession number is Q8NEF3. | |||
TMPH-01392 | GRIA2 Protein, Human, Recombinant (His & Myc) | Human | E. coli |
GRIA2 Protein, Human, Recombinant (His & Myc) is expressed in E. coli expression system with N-10xHis and C-Myc tag. The predicted molecular weight is 63.3 kDa and the accession number is P42262. | |||
TMPH-02224 | TEAD4 Protein, Human, Recombinant (His & Myc) | Human | Baculovirus Insect Cells |
TEAD4 Protein, Human, Recombinant (His & Myc) is expressed in Baculovirus insect cells with N-10xHis and C-Myc tag. The predicted molecular weight is 44.5 kDa and the accession number is Q15561. | |||
TMPH-00968 | ATP5C1 Protein, Human, Recombinant (His & Myc) | Human | E. coli |
ATP5C1 Protein, Human, Recombinant (His & Myc) is expressed in E. coli expression system with N-10xHis and C-Myc tag. The predicted molecular weight is 37.6 kDa and the accession number is P36542. | |||
TMPH-03389 | TRPA1 Protein, Rat, Recombinant (His & Myc) | Rat | E. coli |
TRPA1 Protein, Rat, Recombinant (His & Myc) is expressed in E. coli expression system with N-10xHis and C-Myc tag. The predicted molecular weight is 27.3 kDa and the accession number is Q6RI86. | |||
TMPH-02793 | Myocilin Protein, Mouse, Recombinant (His & Myc) | Mouse | Baculovirus Insect Cells |
Myocilin Protein, Mouse, Recombinant (His & Myc) is expressed in Baculovirus insect cells with N-10xHis and C-Myc tag. The predicted molecular weight is 35.2 kDa and the accession number is O70624. | |||
TMPH-02292 | B3GNT7 Protein, Human, Recombinant (His & Myc) | Human | E. coli |
B3GNT7 Protein, Human, Recombinant (His & Myc) is expressed in E. coli expression system with N-10xHis and C-Myc tag. The predicted molecular weight is 50.5 kDa and the accession number is Q8NFL0. | |||
TMPH-02962 | Lyn Protein, Mouse, Recombinant (His & Myc) | Mouse | E. coli |
Lyn Protein, Mouse, Recombinant (His & Myc) is expressed in E. coli expression system with N-10xHis and C-Myc tag. The predicted molecular weight is 63.7 kDa and the accession number is P25911. | |||
TMPH-02948 | TRIB3 Protein, Mouse, Recombinant (His & Myc) | Mouse | E. coli |
TRIB3 Protein, Mouse, Recombinant (His & Myc) is expressed in E. coli expression system with N-10xHis and C-Myc tag. The predicted molecular weight is 46.5 kDa and the accession number is Q8K4K2. | |||
TMPH-03366 | RUNX1 Protein, Rat, Recombinant (His & Myc) | Rat | Baculovirus Insect Cells |
RUNX1 Protein, Rat, Recombinant (His & Myc) is expressed in Baculovirus insect cells with N-10xHis and C-Myc tag. The predicted molecular weight is 52.4 kDa and the accession number is Q63046. | |||
TMPH-02170 | TRBC1 Protein, Human, Recombinant (His & Myc) | Human | E. coli |
TRBC1 Protein, Human, Recombinant (His & Myc) is expressed in E. coli expression system with N-10xHis and C-Myc tag. The predicted molecular weight is 19.7 kDa and the accession number is P01850. | |||
TMPH-00856 | RPSA Protein, Human, Recombinant (His & Myc) | Human | E. coli |
RPSA Protein, Human, Recombinant (His & Myc) is expressed in E. coli expression system with N-10xHis and C-Myc tag. The predicted molecular weight is 37.7 kDa and the accession number is P08865. | |||
TMPH-02589 | COL26A1 Protein, Mouse, Recombinant (His & Myc) | Mouse | Baculovirus Insect Cells |
N/A. COL26A1 Protein, Mouse, Recombinant (His & Myc) is expressed in Baculovirus insect cells with N-10xHis and C-Myc tag. The predicted molecular weight is 47.7 kDa and the accession number is Q91VF6. | |||
TMPH-01901 | DDX53 Protein, Human, Recombinant (His & Myc) | Human | E. coli |
N/A. DDX53 Protein, Human, Recombinant (His & Myc) is expressed in E. coli expression system with N-10xHis and C-Myc tag. The predicted molecular weight is 76.2 kDa and the accession number is Q86TM3. | |||
TMPH-01030 | CAPN14 Protein, Human, Recombinant (His & Myc) | Human | Baculovirus Insect Cells |
Calcium-regulated non-lysosomal thiol-protease. CAPN14 Protein, Human, Recombinant (His & Myc) is expressed in Baculovirus insect cells with N-10xHis and C-Myc tag. The predicted molecular weight is 78.6 kDa and the acce... | |||
TMPH-03387 | TSHB Protein, Rat, Recombinant (His & Myc) | Rat | P. pastoris (Yeast) |
Indispensable for the control of thyroid structure and metabolism. TSHB Protein, Rat, Recombinant (His & Myc) is expressed in yeast with N-6xHis and C-Myc tag. The predicted molecular weight is 16.4 kDa and the accession... | |||
TMPH-02795 | Myoglobin Protein, Mouse, Recombinant (His & Myc) | Mouse | HEK293 Cells |
Serves as a reserve supply of oxygen and facilitates the movement of oxygen within muscles. Myoglobin Protein, Mouse, Recombinant (His & Myc) is expressed in HEK293 mammalian cells with N-10xHis and C-Myc tag. The predic... | |||
TMPH-02495 | APMAP Protein, Mouse, Recombinant (His & Myc) | Mouse | E. coli |
Exhibits strong arylesterase activity with beta-naphthyl acetate and phenyl acetate. May play a role in adipocyte differentiation. APMAP Protein, Mouse, Recombinant (His & Myc) is expressed in E. coli expression system w... | |||
TMPH-03120 | OBP Protein, Pig, Recombinant (His & Myc) | Sus scrofa (Pig) | E. coli |
This protein is found in nasal epithelium and it binds a wide variety of chemical odorants. OBP Protein, Pig, Recombinant (His & Myc) is expressed in E. coli expression system with N-10xHis and C-Myc tag. The predicted m... | |||
TMPH-00891 | ADAMTSL5 Protein, Human, Recombinant (His & Myc) | Human | E. coli |
May play a role in modulation of fibrillin microfibrils in the extracellular matrix (ECM). ADAMTSL5 Protein, Human, Recombinant (His & Myc) is expressed in E. coli expression system with N-10xHis and C-Myc tag. The predi... | |||
TMPH-02708 | HNMT Protein, Mouse, Recombinant (His & Myc) | Mouse | E. coli |
Inactivates histamine by N-methylation. Plays an important role in degrading histamine and in regulating the airway response to histamine. HNMT Protein, Mouse, Recombinant (His & Myc) is expressed in E. coli expression s... | |||
TMPH-01203 | DCAF16 Protein, Human, Recombinant (His & Myc) | Human | E. coli |
Functions as a substrate recognition component for CUL4-DDB1 E3 ubiquitin-protein ligase complex, which mediates ubiquitination and proteasome-dependent degradation of nuclear proteins. DCAF16 Protein, Human, Recombinant... | |||
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A unique collection of 1268 cancer cellular metabolism related compounds for cancer research and high throughput screening (HTS) and high content screening (HCS); | |||
L2550 | Glutamine Metabolism Compound Library | 565 compounds | |
A unique collection of 565 glutamine metabolism related compounds can be used for high throughput screening (HTS) and high content screening (HCS), and also is an effective tool for research in glutamine metabolism and ... |