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Cat No.	Product Name	Synonyms	Targets
T26559	ACT-462206		OX Receptor
	ACT-462206 is an orally available Orexin 1/Orexin 2 receptor antagonist that crosses the blood-brain barrier.ACT-462206 is highly potent and can be used in studies of sleep and anxiety.		OX Receptor
T10242	ACT-389949		Others
	ACT-389949 is a potent and selective agonist of formyl peptide receptor type 2 (FPR2)/Lipoxin A4 receptor (ALX), with an EC50 of 3 nM for FPR2/ALX internalization into monocytes. It has the potential for the treatment of...		Others
T14119	ACT-678689	Compound Example 1.53.4	Hydroxylase
	ACT-678689 (Compound Example 1.53.4) (Compound Example 1.53.4) is a tryptophan hydroxylase (TPH) inhibitor with an IC50 of 8 nM[1].		Hydroxylase
T26557	ACT-209905	ACT 209905,ACT209905
	ACT-209905 is an agonist of S1P1 receptor.
T9149	2BAct	2B-Act,2B Act	PERK
	2BAct is a novel eif2b activator, preventing neurological defects caused by a chronic integrated stress response		PERK
T14924	Cenerimod	ACT-334441	S1P Receptor
	Cenerimod (ACT-334441) is an orally active, selective, and potent sphingosine 1-phosphate receptor (S1P1) agonist (EC50: 1 nM).Cenerimod inhibits multiple S1P isoforms and can be used to study murine experimental autoimm...		S1P Receptor
T3258	Ponesimod	ACT-128800	S1P Receptor , LPL Receptor
	Ponesimod (ACT-128800) is an orally available sphingosine-1-phosphate receptor 1 (S1PR1, S1P1) agonist with potential immunomodulating activity.		S1P Receptor , LPL Receptor
T4020	Cadazolid	ACT-179811	Antibacterial , Antibiotic
	Cadazolid (ACT-179811) is an oxazolidinone-type antibiotic, with activity against gram-positive bacteria, including Clostridium difficile.		Antibacterial , Antibiotic
T2058	Palosuran	ACT-058362	GPR
	Palosuran (ACT-058362) (ACT-058362) is a new potent and specific antagonist of the human UT receptor.		GPR
T35623	ACT-373898
	ACT-373898 is a metabolite of the endothelin (ET) receptor type A (ETA) and ETBdual antagonist macitentan .1 1.Dingemanse, J., Sidharta, P.N., Maddrey, W.C., et al.Efficacy, safety and clinical pharmacology of macitentan...
T2561	Macitentan	ACT-064992	Apoptosis , Endothelin Receptor
	Macitentan (ACT-064992) is an endothelin receptor antagonist that is used in the therapy of pulmonary arterial hypertension (PAH).		Apoptosis , Endothelin Receptor
T40542	Sinbaglustat	ACT-519276,Sinbaglustat,OGT2378	Transferase
	Sinbaglustat (OGT2378) (OGT2378) is a dual inhibitor of glucose ceramide synthetase (GCS) and non-lysosomal glucose ceramidase (GBA2).Sinbaglustat is an orally administered N-alkyl iminosugar that crosses the blood-brain...		Transferase
T7817	Aprocitentan	ACT-132577	Endothelin Receptor
	Aprocitentan (ACT-132577) is ETA and ETB antagonist .		Endothelin Receptor
T2613	Almorexant	ACT 078573	OX Receptor
	Almorexant (ACT 078573) is a potent and competitive dual orexin 1 receptor (OX1)/orexin 2 receptor (OX2) antagonist with Ki values of 1.3 and 0.17 nM for OX1 and OX2, respectively.		OX Receptor
T14120	ACT-709478		Others
	ACT-709478 is a potent, selective T-type calcium channel blocker that is orally active and capable of penetrating the brain. It is currently utilized in research focusing on generalized epilepsies[1].		Others
T4689	Palosuran hydrochloride 540769-28-6(free base）	ACT-058362 hydrochloride	GPR
	Palosuran hydrochloride 540769-28-6(free base)(ACT-058362 hydrochloride) is a new potent and specific antagonist of the human UT receptor with an IC50 of 3.6±0.2 nM.		GPR
T70616	ACT-672125
	ACT-672125 is a Potent CXCR3 Antagonist with Therapeutic Potential in Autoimmune Diseases. ACT-672125 showed good physicochemical properties and safety profile. In a proof-of-mechanism model of lung inflammation, ACT-672...
T70475	ACT-280778
	ACT-280778 is a potent L/T calcium channel blocker.
T3216	Selexipag	NS-304,ACT-293987,Uptravi	Others , Prostaglandin Receptor
	Selexipag (ACT-293987)(NS-304) is prostacyclin receptor agonist that causes vasodilation in pulmonary vasculature and is used in the therapy of pulmonary arterial hypertension (PAH).		Others , Prostaglandin Receptor
T39665	ACT-1004-1239
	ACT-1004-1239 is a highly potent and selective antagonist of CXCR7, which can be administered orally. It exhibits an impressive inhibitory concentration (IC50) value of 3.2 nM.
T14123	ACT 178882		RAAS
	ACT 178882 is a new Renin inhibitor (IC50: 1.4 nM).		RAAS
T21850	ACT 335827
	ACT-335827 is an orally available, brain-penetrant orexin type 1 receptor selective antagonist. ACT-33582 acts on OXR1 and OXR2 with IC 50 values of 6 nM and 417 nM, respectively. ACT-33582 can be used in studies related...
T3520	Setipiprant	KYTH-105,ACT-129968	GPR , Prostaglandin Receptor
	Setipiprant (ACT-129968) is an orally available, selective CRTH2 antagonist (IC50: 6.0 nM). CRTH2 is a G protein-coupled receptor for prostaglandin (PGD2). PGD2 is produced by the mast cells and is a key mediator in vari...		GPR , Prostaglandin Receptor
T26558	ACT-387042	ACT387042
	ACT-387042 is a Bacterial Topoisomerase Inhibitor, it has broad-spectrum activity against Gram-positive and Gram-negative bacteria.
T23625	ACT-451840	ACT451840
	ACT-451840 is a drug of antimalarial activity. It has effective activity against sensitive and resistant Plasmodium falciparum strains.
T71363	ACT-281959
	ACT-281959, a prodrug of ACT-246475, is a novel potent and selective P2Y12 Receptor Antagonist with a Wider Therapeutic Window in the Rat Than Clopidogrel. ACT-281959 showed antithrombotic efficacy after oral administr...
T73148	ACT-777991
	ACT-777991 is an orally active, selective CXCR3 antagonist with demonstrated stability in microsomes and hepatocytes across various animal models. This compound effectively inhibits the migration of activated T cells tow...
T63761	ACT-660602
	ACT-660602 is an orally active chemokine receptor CXCR3 antagonist (IC50: 204 nM). ACT-660602 inhibits T cell migration and has shown significant effects in an in vivo model of acute lung injury. ACT-660602 can be used t...
T73100	ACT-606559
	ACT-606559, a metabolite of ACT451840, is a novel chemical compound exhibiting antimalarial properties. It is utilized in malaria research.
T77442	Glenzocimab	ACT017	Others
	Glenzocimab (ACT017) is a Fab fragment of a humanized anti-GPVI monoclonal antibody. Glenzocimab demonstrated inhibition of collagen-induced platelet aggregation in an ischemic stroke model. Glenzocimab has been studied ...		Others
T24478	MK-8141	MK 8141,ACT 077825,ACT077825,ACT-077825
	MK-8141 is a renin inhibitor. It displays some antihypertensive efficacy in hypertensive patients.
T10351	Aprocitentan D4	ACT-132577 D4	Others
	Aprocitentan D4 (ACT-132577 D4) is a deuterium-labeled Aprocitentan. Aprocitentan is a major and pharmacologically active metabolite of Macitentan. Aprocitentan is a dual ETA/ETB antagonist (IC50s: 3.4 nM and 987 nM; pA2...		Others
T11934	Macitentan-d4	Macitentan D4,ACT-064992 D4	Endothelin Receptor
	Macitentan-d4 (ACT-064992 D4) is a deuterated substitute for Macitentan and can be used as a dual antagonist of the non-peptides ETA and ETB (endothelin receptor).Macitentan-d4 is less toxic than Macitentan, has a longer...		Endothelin Receptor
T6155	Almorexant hydrochloride	ACT-078573 hydrochloride,Almorexant HCl	OX Receptor
	Almorexant hydrochloride (ACT-078573 hydrochloride) is a potent and competitive dual orexin 1 receptor (OX1)/orexin 2 receptor (OX2) antagonist with Ki values of 1.3 and 0.17 nM for OX1 and OX2, respectively.		OX Receptor
T70474	Gallamine
	Gallamine is an allosteric antagonist at muscarinic M2 acetylcholine receptors and an inhibitor of acetylcholinesterase.
T70614	SLR080811 HCl
	SLR080811 is a SphK inhibitor. Sphingosine-1-phosphate (S1P) is a ubiquitous, endogenous small molecule that is synthesized by two isoforms of sphingosine kinase (SphK1 and 2). Intervention of the S1P signaling pathway h...
T71361	CHS-828 nicotinate
	CHS-828 nicotinate is a CHS-828 salt with Nicotinic acid.. CHS-828 also known as GMX-1778, is a potent and selective NAMPT inhibitor. CHS-828 inhibits cellular synthesis of NAD. CHS 828 kill tumour cells by inhibiting ...
T7744	Piperaquine tetraphosphate tetrahydrate		Parasite
	Piperaquine tetraphosphate tetrahydrate is a potent anti-parasites agent.		Parasite
T71362	GCC-4401C free base
	GCC-4401C free base is a factor Xa inhibitor similar to rivaroxaban that is currently under development for venous thromboembolic disease (VTE).
T7532	Piperaquine		Parasite
	Piperaquine is a bis-quinoline compound that inhibits the ex vivo growth of P. falciparum isolates from malaria-infected patients with IC50s ranging from 11.8-217.3 nM.		Parasite
TP1240	Adrenocorticotropic Hormone (ACTH) (18-39), human TFA	CLIP (human) (TFA)	Others
	Adrenocorticotropic Hormone (ACTH) (18-39), human TFA (CLIP human TFA) is a corticotropinlike intermediate lobe peptide, it is is produced in the melanotrophs of the intermediate lobe of the pituitary.		Others
T40923	Calcium lactate	Lactic acid calcium,Hemicalcium L-lactate,Lactate calcium,Conclyte calcium	Others
	Calcium lactate (Conclyte calcium) is used by the beverage industry as a source of calcium to fortify fruit juice. Calcium lactate facilitates the growth and phytic acid degradation of soybean sprouts.		Others
T77385	Idactamab	INT-001
	Idactamab (INT-001) is a monoclonal antibody to the human amino acid transport protein ASCT2.
T41287	N-3-Oxo-octanoyl-L-homoserine lactone		Others
	N-3-Oxo-octanoyl-L-homoserine lactone is a quorum-sensing signal molecule and an autoinducer for Agrobacterium.		Others
T60073	Antimycobacterial agent-4	4-nitro-N-[4-(2-pyridyl)thiazol-2-yl]benzamide	Antibacterial
	Antimycobacterial agent-4 (4-nitro-N-[4-(2-pyridyl)thiazol-2-yl]benzamide) has antibacterial activity against Mycobacterium tuberculosis.		Antibacterial
T35795	Lactisole	na-PMP	Taste receptor
	Lactisole (na-PMP) is an inhibitor of the glucose-sensing receptor		Taste receptor
T39924	NF-κΒ activator 2		NF-κB
	NF-κΒ Activator 2 is a potent, orally active compound that efficiently activates NF-κB with an EC50 value of 1.58 μM. By enhancing NF-κB expression and activation, it induces SOD 2 synthesis, rendering it useful for amyo...		NF-κB
T9612	Antibacterial agent 27		Anti-infection
	Antibacterial agent 27 has potent anti-Candida activity.		Anti-infection
T9400	KCNQ2/3 activator-1		Others
	KCNQ2/3 activator-1 is a Kv7.2/Kv7.3 (KCNQ2/3) potassium channel activator.		Others
T38476	Metallo β-lactamase ligand 1		Antibacterial
	Metallo β-lactamase ligand 1 is an inhibitor of class B β-lactamase exhibiting antibacterial activities.		Antibacterial

Cat No.	Product Name	Synonyms	Targets
T3S2007	MRE-269	MRE 269,ACT-333679,MRE269	Prostaglandin Receptor
	MRE-269 (ACT-333679) is an orally available and long-acting prostacyclin receptor agonist prodrug. MRE-269(ACT-333679) is used for the treatment of pulmonary arterial hypertension. MRE-269(ACT-333679) is an active metabo...		Prostaglandin Receptor
T1683	Actriol	Epiestriol	Glucocorticoid Receptor
	Actriol (Epiestriol) is always used as Glucocorticoid Receptor agonist.		Glucocorticoid Receptor
T12045	(-)-Hydroxycitric acid lactone	Garcinia lactone	ATP Citrate Lyase
	(-)-Hydroxycitric acid lactone (Garcinia lactone) is an anti-obesity agent.(-)-Hydroxycitric acid lactone was a potent inhibitor of ATP citrate lyase, which catalyzes the extramitochondrial cleavage of citrate to oxaloac...		ATP Citrate Lyase
TN2539	1beta-Hydroxyalantolactone		IL Receptor , TNF
	1beta-Hydroxyalantolactone is a small molecular compound isolated from the flower head of the medicinal plant giant British flower, which can inhibit the expression of TNF-α, IL-17 and IFN-γ in cells, promote the secreti...		IL Receptor , TNF
TN7212	Acacetin-7-O-beta-D-galactopyranoside		Others
	Acacetin-7-O-beta-D-galactopyranoside is a natural product found in Chrysanthemum indicum.		Others
T2S0410	Euphorbia factor L1	Euphorbiasteroid	Apoptosis , P-gp
	Euphorbia factor L1 (Euphorbiasteroid) can reduce Bcl-2, PI3K, AKT, and mTOR protein and mRNA levels, and up-regulate caspase-9 and caspase-3 protein levels. It induces autophagy and has anti-cancer, anti-adipogenic, ant...		Apoptosis , P-gp
T4455	DL-3-Phenyllactic acid	3-Phenyllactic acid,2-Hydroxy-3-phenylpropanoic acid	Others , Endogenous Metabolite , Antibacterial
	3-Phenyllactic acid (PhLA) is a broad spectrum antimicrobial compound active against bacteria and fungi, DL-3-Phenyllactic acid (3-Phenyllactic acid) is a reagent involved in biological studies of nantioselectivity of li...		Others , Endogenous Metabolite , Antibacterial
TN1106	Cyanidin-3-O-galactoside chloride	Ideain chloride	Antioxidant
	Cyanidin-3-O-galactoside chloride (Ideain chloride), extracted from hawthorn pericarp (EPHF), has antioxidant activity and can be used in obesity research.		Antioxidant
T7995	α-Angelica lactone	Alpha-Angelica Lactone	Others , GST
	α-Angelica lactone has cardiotonic activity, may exert their effects by providing an increased contraction-dependent calcium pool to be released upon systolic depolarization.		Others , GST
T5798	Euphorbia Factor L2	euphorbiafactor L2	Apoptosis , NF-κB
	Euphorbia Factor L2 alleviates lipopolysaccharide-induced acute lung injury and inflammation through inhibits NF-κB activation.		Apoptosis , NF-κB
T8213	Isolinderalactone		NOS , STAT
	Isolinderalactone shows anti-inflammatory and anticancer capacity, and it exhibits moderate iNOS inhibitory activity, with the IC50 value of 0.30 uM.		NOS , STAT
T2833	Dehydrocostus Lactone	Epiligulyl oxide,(-)-Dehydrocostus lactone	IκB/IKK
	Dehydrocostus Lactone ((-)-Dehydrocostus lactone) shows anti-inflammatory, anti-ulcer, immunomodulatory and anti-tumor properties.		IκB/IKK
T5220	D-(-)-Lactic acid sodium	Sodium D-lactate	Others , Endogenous Metabolite
	D-(-)-Lactic acid sodium (Sodium D-lactate) is an organic acid. It is a chiral molecule, consisting of two optical isomers, L-lactic acid and D-lactic acid, with the L-isomer being the most common in living organisms. D-...		Others , Endogenous Metabolite
TQ0284	Hydroxyphenyllactic acid		Endogenous Metabolite , Antifungal
	Hydroxyphenyllactic acid is an antifungal metabolite, fungi such as Lactobacillus sp. SK007.		Endogenous Metabolite , Antifungal
TJO2795	D-Galacturonic acid hydrate	D-(+)-Galacturonic acid	Others , Endogenous Metabolite
	D-Galacturonic acid hydrate is used in the synthesis of N-(D-galacturonoyl) amino acids and dipeptides.		Others , Endogenous Metabolite
T0591	D-Galactose	D-(+)-Galactose,D-Galactopyranose,Alpha-D-galactose	Endogenous Metabolite
	D-Galactose (Alpha-D-galactose) is an aldohexose that exists naturally in the D-form in lactose, cerebrosides, gangliosides, and mucoproteins and is converted enzymatically into D-glucose for metabolism or polysaccharide...		Endogenous Metabolite
T4845	L-Lactic acid	2-HYDROXYPROPIONIC ACID,L-(+)-Lactic acid,(S)-2-Hydroxypropanoic acid	Endogenous Metabolite , Antibacterial , Antibiotic
	L-Lactic acid ((S)-2-Hydroxypropanoic acid) is a natural product produced by the anaerobic glycolysis of pyruvic acid. L-Lactic acid is a sensitive indicator of tissue hypoxia and can be used as a hemodynamic indicator i...		Endogenous Metabolite , Antibacterial , Antibiotic
TN6945	Lactic acid	2-hydroxypropanoic acid	Others
	Lactic acid (2-hydroxypropanoic acid) is a product of glycolysis and is widely found in nature.Lactic acid is produced in the body during hypoxia in contracted skeletal muscle and can be removed under fully aerobic condi...		Others
TQ0118	Britannilactone	Desacetylinulicin	Others
	Britannilactone, extracted from the dried flower of Inula britannica L, significantly reduces melanin production in a dose-dependent manner (IC50: 15.5 uM).		Others
TN1635	Euphorbia factor L8		Others
	Euphorbia factor L8 is a natural product		Others
TN1634	Euphorbia factor L7b		Others
	Euphorbia factor L7b,a natural product obtained from the herbs of Euphorbia pekinensis Rupr.		Others
T2829	Isoalantolactone	(+)-Isoalantolactone,Isohelenin	Apoptosis , Endogenous Metabolite , Antibacterial , Autophagy
	Isoalantolactone (Isohelenin), isolated from Inula spp., can inhibit the growth of several types of Y cells.
TN1637	Eurycomalactone		Anti-infection , NF-κB
	Eurycomalactone is a natural product isolated from Eurycoma longifolia Jack., acts as a potent NF-κB inhibitor( IC50 of 0.5 μM). Eurycomalactone inhibits protein synthesis, depletes cyclin D1, but does not affect TNFα-in...		Anti-infection , NF-κB
T35709	N-acetyl-D-Lactosamine	N-Acetyllactosamine	Endogenous Metabolite
	N-acetyl-D-Lactosamine (N-Acetyllactosamine) is a disaccharide consisting of galactose and N-acetylglucose, which is an important component of various oligosaccharides and can be used as a starting material for the synth...		Endogenous Metabolite
T8085	(-)-Corey lactone diol	Corey Lactone Diol	Others
	(-)-Corey lactone diol is a pharmaceutical intermediate		Others
T4942	Galactose 1-phosphate Potassium salt	α-D-Galactose-1-phosphate Dipotassium Pentahydrate	Others , Endogenous Metabolite
	Galactose 1-phosphate Potassium salt (α-D-Galactose-1-phosphate Dipotassium Pentahydrate) is an intermediate in the galactose metabolism and nucleotide sugars metabolism pathways.		Others , Endogenous Metabolite
T74862	N-Lactoyl-Phenylalanine	N-Lactoylphenylalanine	Endogenous Metabolite
	N-Lactoyl-Phenylalanine (Lac-Phe) is a peptide coupling of lactic acid and phenylalanine, one of the metabolites in acute exercise, which can be used in the study of obesity and metabolism-related diseases.		Endogenous Metabolite
TN6796	2'-FUCOSYLLACTOSE	2'-Fucosyl-D-lactose	Others
	2'-FUCOSYLLACTOSE (2'-Fucosyl-D-lactose) is a fucose-containing oligosaccharide.		Others
T5968	DL-Homocysteine thiolactone hydrochloride	DL-Homocysteinethiolactone hydrochloride	Endogenous Metabolite
	DL-Homocysteine thiolactone hydrochloride (DL-Homocysteinethiolactone hydrochloride) is a cysteine derivative that binds to and induces conformational changes in various plasma proteins, slowing coagulation and inducing ...		Endogenous Metabolite
T25192	Butyrolactone I	Olomoucin	CDK
	Butyrolactone I (Olomoucin) is an ATP-competitive inhibitor of CDK and cdc2 kinase family. Butyrolactone I shows antitumor effects in non-small cell lung, small cell lung, and prostate cancer cell lines.		CDK
T125211	Deoxy euphorbia factor L1		Others
	Deoxy euphorbia factor L1 is a natural product found in the seeds of Euphorbia lathyris L		Others
T5663	α-Lactose	Lactose	Others
	α-Lactose is the major sugar present in milk and the main source of energy supplied to the newborn mammalian in its mother's milk. Lactose is also an important osmotic regulator of lactation.		Others
T5578	L-Gulono-1,4-lactone		Others , Endogenous Metabolite
	L-Gulono-1,4-lactone is a substrate of L-gulono-1,4-lactone oxidoreductase, which catalyzes the last step of the biosynthesis of L-ascorbic (Vitamin) C.		Others , Endogenous Metabolite
TN1962	Myricetin 3-O-galactoside	Myricetin 3-O-beta-D-galactopyranoside	NOS , Xanthine Oxidase
	Myricetin 3-O-galactoside (Myricetin 3-O-beta-D-galactopyranoside) can inhibit xanthine oxidase (xanthine oxidase; XO) activity, lipid peroxidation and scavenging free radicals. Myricetin 3-O-galactoside has many effects...		NOS , Xanthine Oxidase
T10941	D-Ribonolactone		Endogenous Metabolite , Antibacterial
	D-Ribonolactone is sugar lactone and an inhibitor of β-galactosidase of Escherichia coli (Ki : 26 Mm).		Endogenous Metabolite , Antibacterial
T3902	Atractylenolide III	ICodonolactone,8β-Hydroxyasterolide	Apoptosis
	Atractylenolide III (ICodonolactone) may have therapeutic potential in treating homocysteine-mediated cognitive impairment and neuronal injury. Atractylenolide III is a potential candidate for the treatment of human lung...		Apoptosis
TN1823	Kaempferol 3-O-β-D-galactopyranoside	Kaempferol 3-O-beta-D-galactoside,Kaempferol-3-O-galactoside	Immunology/Inflammation related
	Kaempferol 3-O-β-D-galactopyranoside has antioxidant, anti-inflammatory and antinociceptive activities.		Immunology/Inflammation related
T3S0156	Atractyloside potassium salt	Atractyloside Dipotassium Salt	Others
	1. Atractyloside potassium salt (Atractyloside Dipotassium Salt) inhibits oxidative phosphorylation by blocking the transfer of adenosine nucleotides through the mitochondrial membrane.		Others
T3234	Dihydroactinidiolide	R-(-)Dihydro actinidiolide	Others
	Dihydroactinidiolide (R-(-)Dihydro actinidiolide)is avolatileterpene. It has a sweet,tea-likeodorand is used as a fragrance.		Others
T5742	Isodemethylwedelolactone	Isodemethylwedelolacton	Others
	Isodemethylwedelolactone (Isodemethylwedelolacton) is a natual product,has Clotting activity.		Others
T6528	Gynostemma Extract	Gypenoside IX,Gypenoside,Gynostemma Pentaphyllum,Notoginsenoside Fd,Ginsenoside C-Mx1,Gynosaponin I	Others , Endogenous Metabolite
	Gynostemma Extract (Gypenoside IX) is a saponins extract derived from the Gynostemma pentaphyllum.		Others , Endogenous Metabolite
T3666	Atractylodin	Atractydin	Lipid
	Atractylodin (Atractydin) has high lipase inhibitory activity (IC5:39.12 μM); Atractylodin possesses strong repellency activities against T. castaneum adults (LD50: 1.83 μg/cm). The repellency of Atractylodin (0.63 μg/cm...		Lipid
T0434	D-Glucuronic acid lactone	Glucuronolactone,D-Glucurone,Dicurone	Others , Endogenous Metabolite
	D-Glucuronic acid lactone (Dicurone) is a naturally occurring chemical that is an important structural component of nearly all connective tissues. Glucuronolactone is also found in many plant gums.		Others , Endogenous Metabolite
T5S0689	Demethylwedelolactone		Serine Protease
	Demethylwedelolactone is a natural product isolated from Eclipta alba, has trypsin inhibitory effect an IC50 of 3.0 μM. it exerts anti-invasive growth effect on breast cancer cells.		Serine Protease
T3999	D(+)-Galactosamine hydrochloride	D-Galactosamine HCl	Others
	D(+)-Galactosamine hydrochloride (D-Galactosamine HCl) hepatotoxicity is associated with endotoxin sensitivity and mediated by lymphoreticular cells in mice.		Others
T5S0168	Atractylenolide II	2-Atractylenolide,Asterolide	Apoptosis , ERK , p38 MAPK , Akt , STAT
	1. Atractylenolide II (2-Atractylenolide) has antimelanoma effect by inhibiting STAT3 signalling. 2. Atractylenolide II has cytotoxic/apoptotic effects may via p38 activation , ERK and Akt inactivation, p53 dependent.		Apoptosis , ERK , p38 MAPK , Akt , STAT
T8064	Lactobionic acid		Others , Antibacterial
	Lactobionic acid with antioxidant, antimicrobial and moisturizing propertie		Others , Antibacterial
T1353	DL-Mevalonolactone	Mevalonolactone	Others , Endogenous Metabolite
	DL-Mevalonolactone (Mevalonolactone) is very soluble in water and polar organic solvents. It exists in equilibrium with its lactone form, called mevalonolactone, that is formed by internal condensation of its terminal al...		Others , Endogenous Metabolite
T5274	D-(+)-Phenyllactic acid	D-3-Phenyllactic acid	Endogenous Metabolite , Antibacterial
	D-(+)-Phenyllactic acid (D-3-Phenyllactic acid), an antibacterial compound produced by Geotrichum candidum, effectively inhibits various Gram-positive and Gram-negative bacteria originating from humans and food products[...		Endogenous Metabolite , Antibacterial
T8098	γ-Hexalactone	γ-caprolactone	Others
	γ-Hexalactone (γ-caprolactone) belongs to the class of organic compounds known as gamma butyrolactones. Gamma butyrolactones are compounds containing a gamma butyrolactone moiety, which consists of an aliphatic five-memb...		Others
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Cat No.	Product Name	Species	Expression System
TMPY-06668	Act d 8 Protein, Actinidia deliciosa, Recombinant	Actinidia deliciosa	P. pastoris (Yeast)
	Act d 8 Protein, Actinidia deliciosa, Recombinant is expressed in P. pastoris yeast expression system. The predicted molecular weight is 26.7 kDa.
TMPK-00464	OX40/TNFRSF4 Protein, Mouse, Recombinant (His & Avi), Biotinylated	Mouse	HEK293 Cells
	Tumor necrosis factor receptor superfamily, member 4 (TNFRSF4), also known as CD134 and OX40 receptor. OX40 is a secondary co-stimulatory immune checkpoint molecule, expressed after 24 to 72 hours following activation; i...
TMPK-00168	OX40/TNFRSF4 Protein, Human, Recombinant (aa 29-216, His & Avi), Biotinylated	Human	HEK293 Cells
	Tumor necrosis factor receptor superfamily, member 4 (TNFRSF4), also known as CD134 and OX40 receptor. OX40 is a secondary co-stimulatory immune checkpoint molecule, expressed after 24 to 72 hours following activation; i...
TMPY-01423	OX40/TNFRSF4 Protein, Human, Recombinant (His)	Human	HEK293 Cells
	OX40/TNFRSF4 Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 21.7 kDa and the accession number is P43489.
TMPK-00169	OX40/TNFRSF4 Protein (Primary Amine Labeling), Human, Recombinant (hFc), Biotinylated	Human	HEK293 Cells
	Tumor necrosis factor receptor superfamily, member 4 (TNFRSF4), also known as CD134 and OX40 receptor. OX40 is a secondary co-stimulatory immune checkpoint molecule, expressed after 24 to 72 hours following activation; i...
TMPK-00167	OX40/TNFRSF4 Protein, Human, Recombinant (His & Avi)	Human	HEK293 Cells
	Tumor necrosis factor receptor superfamily, member 4 (TNFRSF4), also known as CD134 and OX40 receptor. OX40 is a secondary co-stimulatory immune checkpoint molecule, expressed after 24 to 72 hours following activation; i...
TMPK-00463	OX40/TNFRSF4 Protein, Mouse, Recombinant (His & Avi)	Mouse	HEK293 Cells
	Tumor necrosis factor receptor superfamily, member 4 (TNFRSF4), also known as CD134 and OX40 receptor. OX40 is a secondary co-stimulatory immune checkpoint molecule, expressed after 24 to 72 hours following activation; i...
TMPY-01303	Serpin A3 Protein, Human, Recombinant (His)	Human	HEK293 Cells
	SerpinA3, also known as Alpha 1-antichymotrypsin (AACT), is a plasma alpha globulin glycoprotein, and is a member of serpin superfamily of the serine protease inhibitors consisting of at least 35 members. SerpinA3 has be...
TMPH-02567	CCL4 Protein, Mouse, Recombinant (His)	Mouse	E. coli
	Monokine with inflammatory and chemokinetic properties.
TMPY-04993	OX40/TNFRSF4 Protein, Mouse, Recombinant (rFc)	Mouse	HEK293 Cells
	OX40/TNFRSF4 Protein, Mouse, Recombinant (rFc) is expressed in HEK293 mammalian cells with rFc tag. The predicted molecular weight is 47.3 kDa and the accession number is B1ASL3.
TMPY-05020	OX40/TNFRSF4 Protein, Mouse, Recombinant	Mouse	HEK293 Cells
	OX40/TNFRSF4 Protein, Mouse, Recombinant is expressed in HEK293 mammalian cells. The predicted molecular weight is 22.1 kDa and the accession number is B1ASL3.
TMPY-02368	OX40/TNFRSF4 Protein, Mouse, Recombinant (hFc)	Mouse	HEK293 Cells
	OX40/TNFRSF4 Protein, Mouse, Recombinant (hFc) is expressed in HEK293 mammalian cells with hFc tag. The predicted molecular weight is 48.3 kDa and the accession number is B1ASL3.
TMPY-06875	OX40/TNFRSF4 Protein, Human, Recombinant (hFc & Avi), Biotinylated	Human	HEK293 Cells
	OX40/TNFRSF4 Protein, Human, Recombinant (hFc & Avi), Biotinylated is expressed in HEK293 mammalian cells with hFc and Avi tag. The predicted molecular weight is 48.69 kDa and the accession number is NP_003318.1.
TMPY-05339	OX40/TNFRSF4 Protein, Human, Recombinant (hFc)	Human	HEK293 Cells
	OX40/TNFRSF4 Protein, Human, Recombinant (hFc) is expressed in HEK293 mammalian cells with hFc tag. The predicted molecular weight is 46.9 kDa and the accession number is P43489.
TMPY-06906	OX40/TNFRSF4 Protein, Human, Recombinant (His & Avi), Biotinylated	Human	HEK293 Cells
	OX40/TNFRSF4 Protein, Human, Recombinant (His & Avi), Biotinylated is expressed in HEK293 mammalian cells with His and Avi tag. The predicted molecular weight is 23.34 kDa and the accession number is NP_003318.1.
TMPY-00646	CCL4 Protein, Human, Recombinant (His)	Human	P. pastoris (Yeast)
	CCL4 Protein, Human, Recombinant (His) is expressed in yeast with His tag. The predicted molecular weight is 9.2 kDa and the accession number is P13236.
TMPY-05094	Tissue Factor Protein, Cynomolgus, Recombinant (His)	Cynomolgus	HEK293 Cells
	Tissue Factor Protein, Cynomolgus, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 26.4 kDa and the accession number is XP_005542723.1.
TMPY-04778	Prolactin Protein, Human, Recombinant (His)	Human	Baculovirus Insect Cells
	Prolactin Protein, Human, Recombinant (His) is expressed in Baculovirus insect cells with His tag. The predicted molecular weight is 24.3 kDa and the accession number is P01236.
TMPY-01727	GLA/alpha-Galactosidase A Protein, Human, Recombinant (His)	Human	HEK293 Cells
	GLA/alpha-Galactosidase A Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 46.8 kDa and the accession number is P06280.
TMPY-02047	C-Reactive Protein Protein, Rat, Recombinant (His)	Rat	HEK293 Cells
	C-Reactive Protein Protein, Rat, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 24.6 kDa and the accession number is H6X2V1.
TMPY-01053	Prolactin Receptor Protein, Human, Recombinant (His)	Human	HEK293 Cells
	Prolactin Receptor Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 26 kDa and the accession number is P16471-1.
TMPY-00720	Contactin 1 Protein, Human, Recombinant (His)	Human	HEK293 Cells
	Contactin 1 Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 110 kDa and the accession number is A0A024R104.
TMPY-02530	Tissue Factor Protein, Human, Recombinant (His)	Human	HEK293 Cells
	Tissue Factor Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 26.2 kDa and the accession number is P13726.
TMPY-01104	Coagulation factor XI/F11 Protein, Human, Recombinant (His)	Human	HEK293 Cells
	Factor XI (plasma thromboplastin antecedent) is a plasma glycoprotein, and a zymogen acting as a serine protease which participates in blood coagulation as a catalyst in the conversion of factor IX to factor IXa in the p...
TMPY-02185	Coagulation factor XIII B/F13B Protein, Human, Recombinant (His)	Human	HEK293 Cells
	Coagulation factor XIII B chain, also known as Fibrin-stabilizing factor B subunit, Protein-glutamine gamma-glutamyltransferase B chain, Transglutaminase B chain and F13B, is a secreted protein which contains 1 Sushi ...
TMPY-03363	C-Reactive Protein Protein, Human, Recombinant	Human	HEK293 Cells
	C-Reactive Protein Protein, Human, Recombinant is expressed in HEK293 mammalian cells. The predicted molecular weight is 23 kDa and the accession number is P02741-1.
TMPK-00114	C-Reactive Protein /CRP Protein, Human, Recombinant (His)	Human	HEK293 Cells
	C-reactive protein (CRP) is a polypeptide molecule belonging to the family of pentraxins. CRP is synthesized primarily by the liver in response to certain pro-inflammatory cytokines. It plays an important role in innate ...
TMPY-02424	Prolactin Protein, Mouse, Recombinant (His)	Mouse	Baculovirus Insect Cells
	Prolactin Protein, Mouse, Recombinant (His) is expressed in Baculovirus insect cells with His tag. The predicted molecular weight is 23.8 kDa and the accession number is Q9CPQ2.
TMPJ-01471	Activin A Protein, Human, Mouse, Rat, Cynomolgus, Rhesus, Recombinant	Human/Mouse/Rat	HEK293 Cells
	Activin and inhibin are two closely related protein complexes that have almost directly opposite biological effects. Activins, members of the TGF-beta superfamily, are disulfide-linked dimeric proteins originally purifi...
TMPY-03221	Intrinsic Factor Protein, Human, Recombinant (His)	Human	HEK293 Cells
	Gastric intrinsic factor, also known as GIF, belongs to the of the cobalamin transport protein family. It is a glycoprotein produced by the parietal cells of the stomach. Gastric intrinsic factor plays a key role in the ...
TMPY-03014	Osteoactivin/GPNMB Protein, Mouse, Recombinant (His)	Mouse	HEK293 Cells
	Osteoactivin/GPNMB Protein, Mouse, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 54.9 kDa and the accession number is Q99P91.
TMPY-01101	Coagulation factor X/F10 Protein, Human, Recombinant (His)	Human	Baculovirus Insect Cells
	Coagulation factor X, also known as FX, F10, Eponym Stuart-Prower factor, and thrombokinase, is an enzyme of the coagulation cascade. It is one of the vitamin K-dependent serine proteases, and plays a crucial role in the...
TMPY-01075	Von Willebrand Factor/vWF Protein, Human, Recombinant (His)	Human	CHO Cells
	Von Willebrand Factor (VWF) is a multimeric glycoprotein involved in hemostasis in blood, binds receptors on the surface of platelets and in connective tissue, thereby mediating the adhesion of platelets to sites of vasc...
TMPY-04921	Complement factor B/CFB Protein, Human, Recombinant (His)	Human	HEK293 Cells
	Complement factor B/CFB Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 84.5 kDa and the accession number is AAH04143.1.
TMPY-02215	Coagulation factor IX/F9 Protein, Human, Recombinant (His)	Human	HEK293 Cells
	Coagulation factor IX/F9 Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 50 kDa and the accession number is AAB59620.1.
TMPH-00758	EspK Protein, Mycobacterium tuberculosis, Recombinant (His & Myc)	Mycobacterium tuberculosis	E. coli
	May act as a chaperone that facilitates EspB secretion through an interaction with EccCb1.
TMPH-00802	VacA Protein, Helicobacter pylori, Recombinant (His & SUMO)	Helicobacter pylori	E. coli
	Induces vacuolation of eukaryotic cells. Causes ulceration and gastric lesions. vacA Protein, Helicobacter pylori, Recombinant (His & SUMO) is expressed in E. coli expression system with N-6xHis-SUMO tag. The predicted m...
TMPH-00798	HP-0175 Protein, Helicobacter pylori, Recombinant (GST)	Helicobacter pylori	E. coli
	N/A. HP-0175 Protein, Helicobacter pylori, Recombinant (GST) is expressed in E. coli expression system with N-GST tag. The predicted molecular weight is 58.8 kDa and the accession number is P56112.
TMPH-00800	UreA Protein, Helicobacter pylori, Recombinant (His)	Helicobacter pylori	P. pastoris (Yeast)
	Ammonia produced by ureolysis increases the gastric pH thereby providing an environment permissive for colonization of the stomach.
TMPH-00019	BlaNDM-1 Protein, Acinetobacter baumannii, Recombinant (His & SUMO)	Acinetobacter baumannii	E. coli
	BlaNDM-1 Protein, Acinetobacter baumannii, Recombinant (His & SUMO) is expressed in E. coli with N-terminal 6xHis-SUMO tag. The predicted molecular weight is 22.0 kDa. Accession number: F8UNN7
TMPH-03015	MPT64 Protein, Mycobacterium tuberculosis, Recombinant (E. coli, His)	Mycobacterium tuberculosis	E. coli
	N/A. MPT64 Protein, Mycobacterium tuberculosis, Recombinant (E. coli, His) is expressed in E. coli expression system with N-6xHis tag. The predicted molecular weight is 26.4 kDa and the accession number is P9WIN9.
TMPH-03013	HRP1 Protein, Mycobacterium tuberculosis, Recombinant (His & Myc & SUMO)	Mycobacterium tuberculosis	E. coli
	Unlike some other CBS-domain containing proteins does not seem to bind AMP.
TMPH-03017	CYP51 Protein, Mycobacterium tuberculosis, Recombinant (His & Myc)	Mycobacterium tuberculosis	Baculovirus Insect Cells
	Its precise biological substrate is not known. Catalyzes C14-demethylation of lanosterol, 24,25-dihydrolanosterol and obtusifoliol which is critical for ergosterol biosynthesis. It transforms lanosterol into 4,4'-dimethy...
TMPH-00006	Actin-1 Protein, Absidia glauca, Recombinant (His & Myc)	Absidia glauca	E. coli
	Actins are highly conserved proteins that are involved in various types of cell motility and are ubiquitously expressed in all eukaryotic cells.
TMPH-00018	29 kDa outer membrane Protein, Acinetobacter baumannii, Recombinant (His & Myc & SUMO)	Acinetobacter baumannii	E. coli
	May be involved in transporting molecules across the outer membrane.
TMPH-03122	Prolactin Protein, Pig, Recombinant (His & SUMO)	Sus scrofa (Pig)	E. coli
	Prolactin acts primarily on the mammary gland by promoting lactation. Prolactin Protein, Pig, Recombinant (His & SUMO) is expressed in E. coli expression system with N-6xHis-SUMO tag. The predicted molecular weight is 39...
TMPY-02840	Ubiquitin Activating Enzyme E1/UBA1 Protein, Human, Recombinant (His & GST)	Human	Baculovirus Insect Cells
	UBE1, also known as UBA1, belongs to the ubiquitin-activating E1 family. UBE1 gene complements an X-linked mouse temperature-sensitive defect in DNA synthesis, and thus may function in DNA repair. It is part of a gene cl...
TMPH-00328	Flagellin B(flaB) Protein, Campylobacter jejuni, Recombinant (His)	Campylobacter jejuni	E. coli
	Flagellin is the subunit protein which polymerizes to form the filaments of bacterial flagella. Flagellin B(flaB) Protein, Campylobacter jejuni, Recombinant (His) is expressed in E. coli expression system with C-6xHis ta...
TMPH-00525	DsDNA-binding protein A Protein, Enterobacteria phage T4, Recombinant (His & Myc)	Enterobacteria phage T4	E. coli
	May play a role in transcription of several T4 genes. Binds double-stranded DNA and interacts preferentially with T4 late promoter regions. DsDNA-binding protein A Protein, Enterobacteria phage T4, Recombinant (His & Myc...
TMPH-02974	Von Willebrand Factor/vWF Protein, Mouse, Recombinant (His & Myc)	Mouse	E. coli
	Important in the maintenance of hemostasis, it promotes adhesion of platelets to the sites of vascular injury by forming a molecular bridge between sub-endothelial collagen matrix and platelet-surface receptor complex GP...
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L7000	Bioactive Lipid Compound Library	385 compounds
	A unique collection of 385 bioactive lipids related compounds for high throughput screening (HTS) and high content screening (HCS), including Agonists & Antagonists, Endocannabinoids, Farnesyl/geranylgeranyl derivates, ...
L1380	Transcription Factor-Targeted Compound Library	695 compounds
	Well-chosen 695 compounds with unique structures targeting transcription factor;
L4000	Bioactive Compound Library	14439 compounds
	A collection of 14439 small molecule compounds with validated activity for high throughput screening (HTS), high content screening (HCS), cell induction, and target identification;
L2160	Anti-Cancer Active Compound Library	3188 compounds
	A unique collection of 3188 compounds with known anti-cancer activity for high throughput screening (HTS) and high content screening (HCS);
L4150	Featured Novel Bioactive Compound Library	989 compounds
	It is well-selected from Bioactive compound library Plus (D7800), from which 1-15 compounds with the highest scores (activity value, pharmacological properties, structure-diversity, etc.) were chosen. This library consis...
L9850	Orally Active Compound Library	2427 compounds
	A unique collection of 2427 of orally active compounds for high-throughput screening and high-content screening.
L9820	Beta-Lactam Compound Library	97 compounds
	A unique collection of 97 beta-lactam compounds, can be used in HTS and HCS;
L4520	Anti-Bacterial Compound Library	904 compounds
	A unique collection of 904 antibacterial bioactive compounds, a powerful tool for antibacterial drug development;
L9900	Inactive Ingredient Library	182 compounds
	A Collection of 182 inactive ingredients from FDA-approved drugs.
L4010	Bioactive Compounds Library Max	22555 compounds
	A collection of 22555 bioactive compounds for high-throughput screening, high-content screening, cell induction and target identification.
L7300	Potassium Channel Blocker Library	152 compounds
	A unique collection of 152 potassium channel blockers and agonists for high throughput and high content screening;
L6610	Anti-infective Natural Product Library	1060 compounds
	A unique collection of 1060 species of natural products with anti-infective activity for high throughput screening (HTS) and high content screening (HCS);
L4710	Nonsteroidal Anti-Inflammatory Compound Library	521 compounds
	521 non-steroidal anti-inflammatory compounds for high-throughput and high-content screening.
L3500	Histone Modification Compound Library	469 compounds
	A unique collection of 469 histone modification related compounds for high throughput screening (HTS) and high content screening (HCS);
L1600	Kinase Inhibitor Library	2700 compounds
	A unique collection of 2700 kinase inhibitors/regulators for high throughput screening and high content screening for drug discovery in kinase related diseases;
L1610	FDA-Approved Kinase Inhibitor Library	263 compounds
	A unique collection of 263 kinase inhibitors/regulators for specific targeting of kinases, ready for high-throughput screening and high-content screening.
L3600	Cytokine Inhibitor Library	604 compounds
	A unique collection of 604 compounds targeting cytokine signaling for high throughput screening and high content screening for drug discovery;
L1110	Microtubule-Targeted Compound Library	142 compounds
	A unique collection of 142 microtubule-targeted compounds can be used in HTS and HCS;
L6730	Anti-virus Traditional Chinese Medicine Monomer Library	268 compounds
	A collection of 268 TCM monomers with anti-virus activity. An effective tool for drug development and pharmacological studies.
L5300	Mitochondria-Targeted Compound Library	812 compounds
	A unique collection of 812 promising or approved mitochondria-targeted compounds including Idebenone, the only approved drug targeting mitochondria, for research in mitochondrial medicine;
L9830	Anti-Parkinson's Disease Compound Library	857 compounds
	A unique collection of 857 compounds with anti-PD activities or acting on main drug targets of PD can be used for HTS and HCS.
L2610	Neurotransmitter Receptor Compound Library	1513 compounds
	A unique collection of 1513 neurotransmitter receptor compounds, can be used for HTS and HCS screening；
L2010	Highly Selective Inhibitor Library	575 compounds
	A collection of 575 highly selective inhibitors
L4020	NO PAINS Compound Library	9384 compounds
	TargetMol created the L4020 NO-PAINS Compound Library that applied the PAINS filter, remaining 9384 small molecules that are suitable for new drug development, signaling pathway research, drug repurposing and other resea...
L2170	Immuno-Oncology Compound Library	449 compounds
	A unique collection of 449 compounds acting on immune-oncology therapeutic targets can be used for high throughput and high content screening；
L7110	Anti-Hypertension Compound Library	678 compounds
	678 hypertension-related small molecules for high-throughput and high-content screening.

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