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TargetMol | Compound Library

Kinase Inhibitor Library

Catalog No. L1600

In biochemistry, a kinase is an enzyme that catalyzes the transfer of phosphate groups from high-energy, phosphate-donating molecules (ATP) to specific substrates. This process is known as phosphorylation. The protein kinases make up the majority of all kinases and are widely studied. A protein kinase modifies other molecules, mostly proteins, by phosphorylation to regulate the majority of cellular pathways, especially those involved in signal transduction. Various other kinases act on small molecules such as lipids, carbohydrates, amino acids, and nucleotides, either for signaling or to prime them for metabolic pathways. TargetMol’s Kinase Inhibitor Library, containing 2720 kinase inhibitors/regulators , can be used for research in chemical genomics, pharmacological study, and drug screening for related diseases.

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.

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Catalog No. L1600

Kinase Inhibitor Library
sizeIn stock
  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
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Product Description Product Description

  • A unique collection of 2720 kinase inhibitors for high throughput screening and high content screening for drug discovery in kinase related diseases;
  • Bioactivity and safety confirmed by pre-clinical research and clinical trials, and some of them are approved by FDA;
  • Targets include MAPK, PI3K, JAK, STAT, CDK, MEK, Insulin/IGF receptors, CaM Kinease II, PKA, JNK, PKC, RAF, EGFR, SAPK, GSK, MLCK, Src-family, IKK, PDGFR, VEGFR, etc;
  • Detailed compound information with structure, target, activity, IC50 value, and biological activity description;
  • Structurally diverse, medicinally active, and cell permeable;
  • NMR and HPLC validated to ensure high purity and quality;

Packaging And Storage | TargetMol Packaging And Storage

  • Powder or pre-dissolved DMSO solutions in 96/384 well plate with optional 2D barcode
  • Shipped with blue ice

Library Customization | TargetMol Library Customization

Compound Library | TargetMol
Targetmol Compound Libraries
can be highly customized!
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Library Customization | TargetMol Library Composition

Apoptosis
Autophagy
CDK
PI3K
EGFR
VEGFR
mTOR
JAK
ERK
Akt
p38 MAPK
FLT
Src
PDGFR
PKC
AMPK
GSK-3
FGFR
Raf
c-Kit
Ras
NF-κB
c-Met/HGFR
Bcr-Abl
ALK
Aurora Kinase
MAPK
BTK
JNK
PKA
MEK
Tyrosine Kinases
ROCK
Casein Kinase
Serine/threonin kinase
Endogenous Metabolite
IGF-1R
Antibacterial
DNA-PK
c-RET
TAM Receptor
Epigenetic Reader Domain
Glucosidase
CaMK
Trk receptor
IκB/IKK
FAK
S6 Kinase
RIP kinase
TGF-beta/Smad
PLK
Glucokinase
ATM/ATR
STAT
HER
c-Fms
TNF
Syk
Parasite
Chk
Pim
PERK
ROR
IRAK
Caspase
DYRK
COX
LRRK2
PDK
Mitophagy
Antibiotic
HIV Protease
PAK
Influenza Virus
Wnt/beta-catenin
Rho
Reactive Oxygen Species
PI4K
IRE1
IL Receptor
DNA/RNA Synthesis
Tyrosinase
Ferroptosis
Calcium Channel
Ephrin Receptor
ROS Kinase
Phosphatase
AChR
Antifungal
PPAR
BCL
MMP
5-HT Receptor
Adrenergic Receptor
CSF-1R
P450
Potassium Channel
Dehydrogenase
PDE
GRK
ROS
MNK
Discoidin Domain Receptor (DDR)
MLK
S1P Receptor
Kinesin
Adenosine Receptor
Serine Protease
HSV
SGK
Microtubule Associated
PKM
NO Synthase
PARP
LIM Kinase
Wee1
Antiviral
SARS-CoV
Beta Amyloid
HDAC
Sodium Channel
Tie-2
Virus Protease
SIK
AAK1 (AP2 associated kinase 1)
Mitochondrial Metabolism
Lipoxygenase
Interleukin
AChE
HCV Protease
Histamine Receptor
Topoisomerase
Drug Metabolite
P-gp
Nrf2
MELK
Dopamine Receptor
Histone Methyltransferase
Integrin
Antioxidant
TOPK
PYK2
LDL
Antifection
ACK
TLR
transporter
ASK
Hippo pathway
Ligand for E3 Ligase
Carbonic Anhydrase
Estrogen/progestogen Receptor
LPL Receptor
GTPase
Myosin
GluR
Carboxypeptidase
DAPK
ATPase
NOS
Transferase
Ligands for Target Protein for PROTAC
YAP
BACE
IFNAR
NADPH
Glutathione Peroxidase
Estrogen Receptor/ERR
HBV
Hck
TRP/TRPV Channel
MAO
Aryl Hydrocarbon Receptor
E1/E2/E3 Enzyme
Haspin Kinase
Hexokinase
DNA Alkylation
Indoleamine 2,3-Dioxygenase (IDO)
HSP
Prostaglandin Receptor
Sirtuin
PAI-1
Phospholipase
cholecystokinin
HIF/HIF Prolyl-Hydroxylase
p53
Chloride channel
PROTACs
RAAS
Serotonin Transporter
Nucleoside Antimetabolite/Analog
FXR
Gamma-secretase
PTEN
cAMP
DUB
BCRP
Beta-Secretase
Histone Acetyltransferase
Reverse Transcriptase
CRISPR/Cas9
GPR
HIF
Cannabinoid Receptor
Anti-infection
NADPH-oxidase
Proteasome
Proton pump
NPC1L1
DHFR
MyD88
Arrestin
RAR/RXR 
Histone Demethylase
CETP
Necroptosis
gp120/CD4
Melatonin Receptor
MRP
Antifolate
cell cycle arrest
Liver X Receptor
NAMPT
Stemness kinase
iGluR
Phosphorylase
P2X Receptor
NMDAR
Monoamine Transporter
Opioid Receptor
PROTAC Linker
Fatty Acid Synthase
Bombesin Receptor
Hedgehog/Smoothened
FAAH
PAD
Thrombopoietin Receptor
Norepinephrine
DNA
Lipid
ATP Citrate Lyase
PGE Synthase
Acyltransferase
Porcupine
STING
Decarboxylase
cGAS
RSV
GPX
Retinoid Receptor
Protease
Aromatase
GABA Receptor
Hydroxylase
RXFP receptor
Gap Junction Protein
Fer/FerT kinase
BMI-1
Sigma receptor
Protease-activated Receptor
p97
AhR
PD-1/PD-L1

Keywords