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Cat No. | Product Name | Synonyms | Targets |
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T13241 | UB 165 fumarate | UB-165 fumarate,UB165 fumarate | AChR |
UB 165 fumarate is an agonist of the nAChR, a partial agonist of the α4β2 subtype, and a full agonist of the α3β2 subtype, with a Ki value of 0.27 nM for binding to [3H]-nicotine measured in rat brain. | |||
T23485 | UB 165 | Others | |
Subtype-selective nicotinic agonist | |||
T4469 | Nemorubicin | Methoxymorpholinyldoxorubicin,PNU-152243A,PNU 152243 | Others |
Nemorubicin (PNU 152243) is a doxorubicin derivative that differs significantly from its parent drug in terms of spectrum of antitumor activity, metabolism and toxicity profile. The drug is active on tumors resistant to ... | |||
T5200 | Indirubin-3'-monoxime | Indirubin-3'-oxime | GSK-3 , Lipoxygenase , CDK |
Indirubin-3'-monoxime (Indirubin-3'-oxime) is a potent inhibitor of GSK3β (IC50: 22 nM) and also inhibits CDKs ( (IC50s: 100/180/250 nM for Cdk5/p35, Cdk1/cyclin B, Cdk2/cyclin E). | |||
T7011 | Verubecestat | MK-8931 | Beta-Secretase , BACE |
Verubecestat (MK-8931) (MK-8931) is an effective and specific β-secretase inhibitor and β-site APP-cleaving enzyme 1 inhibitor or BACE1 protein inhibitor. | |||
T17192 | Ubiquitin Isopeptidase Inhibitor I, G5 | NSC144303 | Apoptosis |
Ubiquitin Isopeptidase Inhibitor I, G5 is a caspase-independent inducer of cell necrosis that induces cell death via the death receptor pathway (IC50 of 1.76 and 1.6 μM in E1A and E1A/C9DN cells, respectively). | |||
T12166 | Nacubactam | OP0595 free acid | Antibacterial |
Nacubactam (OP0595 free acid) is a potent inhibitor of non-β-lactam-β-lactamase with activity against class A and class C β-lactamases. | |||
T6124 | Mubritinib | TAK-165 | EGFR , FGFR , JAK , PDGFR |
Mubritinib (TAK-165) (TAK-165) is a potent inhibitor of HER2/ErbB2 with IC50 of 6 nM. | |||
T7679 | UBCS039 | Sirtuin , Autophagy | |
UBCS039 is the first synthetic Sirt6 activator(EC50 : 38 μM) | |||
T11090L1 | Aldoxorubicin hydrochloride | Aldoxorubicin hydrochloride (1361644-26-9 Free base) | Topoisomerase |
Aldoxorubicin hydrochloride is an albumin-binding prodrug of Doxorubicin, a DNA topoisomerase II inhibitor. Aldoxorubicin hydrochloride is released from albumin under acidic conditions. Aldoxorubicin hydrochloride exhibi... | |||
TP1862L | [Sar9] Substance P acetate(77128-75-7 free base) | Neurokinin receptor | |
[Sar9]-Substance P acetate is one of NK-1 receptor agonist. The action of SP on progesterone metabolism was mimicked by the rNK1-specific agonist [Sar-9,Met(O2)11]-SP. | |||
T13226 | Tubulin inhibitor 8 | Microtubule Associated | |
Tubulin inhibitor 8 is an inhibitor of tubulin and various cancer cell lines and inhibits tubulin polymerisation and K562 cell growth with an IC50 of 0.73 μM and 14 nM respectively. | |||
T38796L | MBP MAPK Substrate acetate | MBP MAPK Substrate acetate(138028-00-9 free base) | MAPK |
MBP MAPK Substrate acetate can be used as an exogenous substrate for MAPK. | |||
TP2205L | DAPK Substrate Peptide acetate | DAPK | |
DAPK Substrate Peptide acetate is a death-associated protein kinase (DAPK, Km = 9 μM) peptide substrate. | |||
T77647 | Tubulin polymerization-IN-43 | Apoptosis , Microtubule Associated | |
Tubulin polymerization-IN-43 is an inhibitor of tubulin polymerisation.Tubulin polymerization-IN-43 has multiple effects, disrupting the cellular microtubule network by targeting the colchicine locus and promoting cell c... | |||
T24918 | UBP710 | UBP-710,UBP 710 | NMDAR |
UBP710 is an effective and selective NMDA receptor modulator. | |||
T17194 | Ubrogepant | MK-1602 | CGRP Receptor |
Ubrogepant (MK-1602) is an antagonist of calcitonin gene-related peptide receptor that can be used in the acute treatment of migraine studies. | |||
T2318 | Sacubitril/Valsartan | Sacubitril mixture with Valsartan,Valsartan,Sacubitril,LCZ696 | Apoptosis , RAAS , Neprilysin |
Sacubitril/Valsartan (LCZ696) is an orally bioavailable, dual angiotensin II receptor and neprilysin inhibitor for the treatment of hypertension and heart failure. | |||
T0009 | Flubendazole | Flumoxanal,Flumoxane,NSC 313680,Fluvermal | Apoptosis , Microtubule Associated , Parasite |
Flubendazole (Flumoxane) is available OTC in Europe that is an anthelmintic using to treat worm infection in humans. | |||
TP1087 | Substance P | Neurokinin P | Endogenous Metabolite , Neurokinin receptor |
Substance P (Neurokinin P) (SP) is an undecapeptide (a peptide composed of a chain of 11 amino acid residues) member of the tachykinin neuropeptide family. | |||
T60167 | Eubulus-A80 | Others | |
Eubulus-A80 is a anti-tumor agent (WO2021/183702, Compound A80). | |||
T9812 | Tubulin inhibitor 24 | Microtubule Associated | |
Tubulin inhibitor 24 is a potent inhibitor that can inhibit tubulin polymerization. | |||
T0125 | Epirubicin hydrochloride | Pharmorubicin,4'-epidoxorubicin HCl,Epirubicin HCl,4'-Epidoxorubicin hydrochloride | Apoptosis , DNA/RNA Synthesis , Topoisomerase |
Epirubicin hydrochloride (Pharmorubicin) is an antineoplastic agent which can inhibit Topoisomerase. | |||
TQ0039 | (±)-Zanubrutinib | (±)-BGB-3111 | BTK |
(±)-Zanubrutinib ((±)-BGB-3111) is a potent and orally available Bruton's tyrosine kinase (Btk) inhibitor that demonstrates superior oral bioavailability, achieving higher exposure and more complete target inhibi. | |||
T9995 | Antituberculosis agent-5 | Others | |
Antituberculosis agent-5 is a small molecule used for high-throughput assays. | |||
T11112 | DUB-IN-3 | DUB | |
DUB-IN-3 is a potent deubiquitinase (USP) enzyme inhibitor and the IC50 for USP8 is 0.56 μM. | |||
TP1051L | Protein Kinase C Peptide Substrate acetate | Protein Kinase C Peptide Substrate acetate(120253-69-2 free base) | Others |
Protein Kinase C Peptide Substrate acetate targets specific cell spacers ina manner that is dependent on second messengers and specific adaptor proteins in response to extracellular signals that activate g protein-couple... | |||
T0559 | Dibenzosuberone | Others | |
Dibenzosuberone, pharmaceutical intermediates, is used for the synthesis of drug amitriptyline. | |||
T7604 | Valrubicin | Valstar,AD-32 | Antibiotic , PKC |
Valrubicin (AD-32) (AD 32) inhibits TPA- and PDBu-induced PKC activation (IC50s: 0.85 and 1.25 μM) and has antitumor and anti-inflammatory activity. | |||
T7828 | [Sar9,Met(O2)11]-Substance P | Bhsar-sp,NA | Neurokinin receptor |
[Sar9,Met(O2)11]-Substance P (NA) is an agonist of NK1 receptor. | |||
T77698 | HCYP3A4 Fluorogenic substrate 1 | Others | |
hCYP3A4 Fluorogenic substrate 1 is a phthalimide derivative and shows low activity against COX. | |||
T19673 | Fuberidazole | Antifungal | |
Fuberidazole is a chemical agent. It is used in fungicides. | |||
T6327 | Tubacin | Virus Protease , HDAC | |
Tubacin is a highly potent and selective, reversible, cell-permeable HDAC6 inhibitor with an IC50 of 4 nM, approximately 350-fold selectivity over HDAC1. | |||
T7554 | Substance P (7-11) | Substance P 7-11(TFA) | Others , Neurokinin receptor |
Substance P (7-11) (Substance P 7-11(TFA)) is a C-terminal fragment of Substance P . | |||
T13244 | Ubiquitination-IN-1 | Others | |
Ubiquitination-IN-1 is an inhibitor of ubiquitination and Cksl-Skp2 protein-protein interaction (IC50: 0.17 μM). | |||
T11332 | FUBP1-IN-1 | FUBP1–IN-1 | Others |
FUBP1 - in-1, with an IC50 value of 11.0 M, is an effective FUSE binding protein 1 (FUBP1) inhibitor that can interfere with the binding of FUBP1 to its SINGLE-strand target DNA FUSE sequence. | |||
T11110 | DUB-IN-1 | DUB | |
DUB-IN-1, with an IC50 value of 0.24 for USP8, is an active inhibitor of ubiquitin-specific protease (USPs). | |||
T67935 | Tubulin inhibitor 11 | Apoptosis , Microtubule Associated | |
Tubulin Inhibitor 11 is a potent, orally active agent that inhibits tubulin by targeting the Colchicine binding site. It impedes tubulin polymerization, leading to mitotic blockade and apoptosis. | |||
T13799 | NQO1 substrate | NADPH | |
NQO1 substrate is a highly potent NQO1 substrate with potential antitumor activity for leukemia research. | |||
T13447 | (R)-Zanubrutinib | (R)-BGB-3111 | BTK |
(R)-Zanubrutinib ((R)-BGB-3111) is a selective inhibitor of Bruton tyrosine kinase (BTK). | |||
T72784 | OTUB1/USP8-IN-1 | DUB | |
OTUB1/USP8-IN-1 is a potent OTUB1/USP8 inhibitor with potential anticancer activity, with IC50 values of 0.17 and 0.28 nM for OTUB1 and USP8, respectively.OTUB1/USP8-IN-1 can be used in the study of non-small-cell lung c... | |||
T28974 | Ticolubant | Calcium Channel , LTR | |
Ticolubant is orally active leukotriene B4 antagonist with high affinity for the human neutrophil LTB4 receptor (Ki = 0.78 nM), blocks LTB4-induced Ca2+ migration with an IC50 of 6.6 ± 1.5 nM, and shows topical anti-inf... | |||
T36802L | Bisubstrate Inhibitor 78 HCl | Bisubstrate Inhibitor 78 HCl(2368247-39-4 Free base) | Others |
Bisubstrate Inhibitor 78 HCl is an NNMT inhibitor (IC50 = 1.41 μM) with potential anticancer activity, inhibiting the proliferation of HSC-2 oral cancer cells at 100 μM. | |||
T67966 | Triflubazam | ||
Triflubazam has a wide range of biological activities that can affect sleep and can be used to treat anxiety syndromes and psychological disorders. | |||
TP1483L | Abl Cytosolic Substrate acetate | Abl Cytosolic Substrate acetate(168202-46-8 free base) | Others |
Abl Cytosolic Substrate acetate is a substrate for Abelson tyrosine kinase (Abl ). | |||
T3689 | Ruboxistaurin hydrochloride | Ruboxistaurin,LY333531 HCl,LY 333531 hydrochloride | PKC |
Ruboxistaurin hydrochloride (LY 333531 hydrochloride) is an Isozyme-selective inhibitor of protein kinase C (PKC); competitively and reversibly inhibits PKCβI and PKCβII (IC50 values are 4.7 and 5.9 nM respectively). Sel... | |||
T1966 | Tubastatin A | Tubastatin A BASE | Apoptosis , HDAC , Autophagy |
Tubastatin A (Tubastatin A BASE) is an effective and specific HDAC6 inhibitor (IC50: 15 nM, in a cell-free assay). Its selectivity is 1000-fold against all the other isozymes except HDAC8. | |||
T19114L | Sacubitril-(2S,4S)-Isomer | (2S,4S)-Sacubitril | Others |
Sacubitril-(2S,4S)-Isomer ((2S,4S)-Sacubitril) is the isomer of Sacubitril which is a neprilysin inhibitor. | |||
T60062 | Antitubercular agent-41 | Antibiotic | |
Antitubercular agent-41 is a antibacterial agent. | |||
TP1417L | Sakamototide substrate peptide acetate | Others | |
Sakamototide substrate peptide acetate is a peptide substrate of AMPK kinase family and can be used for the determination of kinase activity. |
Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T8852 | Tubuloside B | Apoptosis , Others | |
The neuroprotective effect of tubuloside B, one of the phenylethanoids isolated from the stems of Cistanche salsa, on tumor necrosis factor-alpha (TNFalpha)-induced apoptosis in SH-SY5Y neuronal cells. | |||
T7004 | Tubercidin | Sparsomycin A,7-Deazaadenosine | Influenza Virus , DNA/RNA Synthesis , Antibacterial , Antibiotic |
Tubercidin (Sparsomycin A), an adenosine analogue, is a nucleoside antibiotic. It is incorporated into DNA and inhibits polymerases, thereby inhibiting DNA replication and RNA and protein synthesis. This agent also exhib... | |||
T5S0281 | Tubuloside A | NOS | |
Tubuloside A ( 8.6 microM) can inhibit D-galactosamine-induced death of hepatocytes. Tubuloside A has NO radical-scavenging activity, which possibly contributes to its anti-inflammatory effects.Tubuloside A shows stronge... | |||
T2715 | Tubeimoside I | Tubeimoside-1,Lobatoside-H | Apoptosis , Others |
Tubeimoside I (Tubeimoside-1)(Lobatoside-H) is an extract from Chinese herbal medicine Bolbostemma paniculatum (MAXIM). | |||
T39049 | Yubeinine | Others | |
Yubeinine is an alkaloid natural product possessing tracheal relaxant effects. | |||
T2934 | Bilirubin | Bilibubin,Principal bile pigment,Hematoidin,Hemetoidin | Endogenous Metabolite |
Bilirubin (Principal bile pigment) is a principal pigment of bile and one of the major end products of hemoglobin decomposition. | |||
TN7249 | Nor-rubrofusarin gentiobioside | ||
Nor-rubrofusarin gentiobioside is a natural product found in the leguminous plant Cassia vulgaris. | |||
T6169 | Indirubin | Indigopurpurin,Indigo red,NSC 105327,Couroupitine B | Apoptosis , Raf , GSK-3 , CDK |
Indirubin (Couroupitine B) is a potent cyclin-dependent kinases and GSK-3β inhibitor with IC50 of about 5 uM and 0.6 uM. | |||
TN2165 | Rubrofusarin gentiobioside | Rubrofusarin-6-O-beta-D-gentiobioside | ERK , NF-κB , TGF-beta/Smad |
Rubrofusarin gentiobioside (Rubrofusarin-6-O-beta-D-gentiobioside) can significantly decrease the expression of TGF-beta1 and fibronectin and NF-kappaB DNA binding activity, suggests that it has potential as a preventive... | |||
T5774 | Demethylsuberosin | 7-demethylsuberosin | Prostaglandin Receptor |
7-Demethylsuberosin (7-demethylsuberosin) is a coumarin compound isolated from Angelica gigas Nakai,and has anti-inflammatory activity,and exhibited inhibitory effects on PGE2 production with the IC50 values of 9.42 μM. | |||
TN1799 | Isorubrofusarin-6-O-β-gentiobioside | Isorubrofusarin 10-gentiobioside | BACE , AChR |
Isorubrofusarin-6-O-β-gentiobioside is derived from from Cassia obtusifolia Linn seeds and shows promising inhibitory activity against AChE and BACE1. | |||
T4237 | Rubiadin-1-methyl ether | Rubiadin 1-methyl ether | Anti-infection , NF-κB |
Rubiadin-1-methyl ether (Rubiadin 1-methyl ether) is a natural product.It inhibits osteoclastic bone resorption via inhibition on the phosphorylation of NF-κB p65 and the degradation of IκBα as well as decrease in the nu... | |||
T3S2027 | Rubusoside | Others | |
1. Rubusoside is a natural sweetener . 2. Rubusoside is a solubilizing agent with antiangiogenic and antiallergic properties. | |||
T6S0084 | Tuberostemonine | Tuberstemonine | Parasite |
1. Tuberostemonine (Tuberstemonine) exhibits relatively higher intestinal permeabilities. 2. Tuberostemonine acts in part as an open-channel blocker at the crayfish neuromuscular junction. | |||
T3782 | Jujuboside A | transporter , GABA Receptor | |
Jujuboside A is a glycoside extracted from Semen Ziziphi Spinosae, having neurophysiological inhibitory effects, used as a potential therapeutic agent for the treatment of Alzheimer s disease. | |||
T4953 | Neotuberostemonine | NOS | |
Neotuberostemonine (NTS) is one of the main antitussive alkaloids in the root of Stemona tuberosa Lour, it has a significant protective effect on bleomycin (BLM)-induced pulmonary fibrosis through suppressing the recruit... | |||
T4S0795 | Berberrubine chloride | 9-Berberoline Chloride,Beroline,Beroline Chloride,Berberrubine,9-Berberoline | IL Receptor |
1. Berberrubine chloride (9-Berberoline Chloride) has antitumor activity. 2. Berberrubine has antidiabetic activity. 3. Berberrubine dose-dependently inhibits IL-8 and MCP-1 protein levels in the media and mRNA expressio... | |||
T5795 | Suberosin | Others , NF-κB | |
Suberosin exhibits anti-inflammatory, and anticoagulant activities, it also shows biting deterrent activity against Aedes aegypti, it may be useful for use as mosquito larvicidal agent. | |||
T5853 | Rubitecan | RFS 2000,9-Nitrocamptothecin | Topoisomerase |
Rubitecan (9-Nitrocamptothecin) is a DNA topoisomerase I inhibitor. It inhibits DNA topoisomerase I and increases the fraction of supercoiled DNA in a cell-free assay in a concentration-dependent manner.Rubitecan is a se... | |||
T3781 | Jujuboside B | Others | |
Jujuboside B has potent inhibitory effects on collagen-, thrombin-, AA-, and ADP-induced aggregation, and also exhibits superior protection on the thromboembolic model. | |||
T4S1849 | Tubeimoside III | Others | |
Tubeimoside III has anti-inflammatory, anti-tumor, and anti-tumorigenic activities, stronger than those of tubeimoside II. | |||
T4734 | Suberic acid | Octanedioic acid,1,8-Octanedioic acid | Others , Endogenous Metabolite |
Suberic acid (1,8-Octanedioic acid) is present in the urine of patients with fatty acid oxidation disorders. A metabolic breakdown product derived from oleic acid. Elevated levels of this unstaruated dicarboxylic acid ar... | |||
T3416 | Aucubin | Aucuboside,Rhinanthin | IL Receptor , NF-κB , Antibacterial |
Aucubin (Rhinanthin) is an iridoid glycoside with anti-inflammatory, anti-microbial, anti-algesic as well as anti-tumor activities. | |||
T4S1848 | Tubeimoside II | Tubeimoside-B | Others |
Tubeimoside II (also known as Tubeimoside-B), a natural oleanane-type triterpenoid saponin analogue, exhibits anti-inflammatory, antitumor, and antitumor-promoting properties. | |||
TN6795 | 5-Methoxysuberenone | Others | |
5-Methoxysuberenone is a chemical constituent of the root bark of Toddalia asiatica (L.) Lam. (T. aculeata Pers.), Rutaceae. | |||
T4241 | Rubiadin | 1,3-Dihydroxy-2-Methylanthracene-9,10-Dione | Free radical scavengers , PARP , Caspase |
Rubiadin (1,3-Dihydroxy-2-Methylanthracene-9,10-Dione) possesses potent antioxidant property, it can prevent lipid peroxidation induced by FeSO4 and t-butylhydroperoxide (t-BHP) in a dose dependent manner. | |||
T1511 | Daunorubicin hydrochloride | Daunomycin HCl,RP-13057 Hydrochloride,Rubidomycin hydrochloride,Daunorubicin HCl,Daunomycin | Apoptosis , DNA/RNA Synthesis , Topoisomerase , Antibacterial , Antibiotic , Autophagy |
Daunorubicin hydrochloride (Rubidomycin hydrochloride), an anthracycline aminoglycoside antineoplastic, inhibits DNA replication and repair and RNA and protein synthesis. | |||
T1020 | Doxorubicin hydrochloride | Adriamycin,Doxorubicin (Adriamycin) HCl,Hydroxydaunorubicin hydrochloride,NSC 123127 | Apoptosis , Mitophagy , HBV , HIV Protease , Topoisomerase , Antibacterial , Antibiotic , AMPK , Autophagy |
Doxorubicin hydrochloride (Adriamycin) belongs to the anthracycline class of antibiotics and is an inhibitor of human DNA topoisomerase I/II (IC50=0.8/2.67 μM). Doxorubicin hydrochloride exhibits cytotoxicity and antitum... | |||
TN4924 | Rubiprasin A | Others | |
Rubiprasin A is a natural product from Rubia cordifolia var. pratensis. | |||
T13939 | Tubulysin E | Others | |
Tubulysin E is a natural product isolated from the myxobacterial species Archangium geophyra and Angiococcus disciformis, and is a highly cytotoxic peptide. | |||
T26953 | Carubicin hydrochloride | NSC 275649,Karminomycin hydrochloride,Carubicin HCl | |
Carubicin HCl is an anthracycline antineoplastic antibiotic. Through intercalates into DNA and interacts with topoisomerase II, Carubicin inhibits DNA replication and repair and RNA and protein synthesis. | |||
TN4240 | Hydroxytuberosone | Others | |
Hydroxytuberosone is a natural product from Pueraria lobata. | |||
TN2637 | 15-Dihydroepioxylubimin | Others | |
15-Dihydroepioxylubimin is a natural product for research related to life sciences. The catalog number is TN2637 and the CAS number is 129214-59-1. | |||
TN3188 | 6-O-p-Hydroxybenzoylaucubin | Others | |
6-O-p-Hydroxybenzoylaucubin is a natural product of Crescentia, Bignoniaceae. The catalog number is TN3188 and the CAS number is 1016987-87-3. 6-O-p-Hydroxybenzoylaucubin can be used as a reference standard. | |||
TN3993 | Erysubin B | Others | |
Erysubin B is a natural product from Erythrina caffra Thunb. | |||
T75684 | Monascorubrin | ||
Monascorubrin, a compound extracted from the mycelium of Monascus purpureus, exhibits significant antibiotic activity against Bacillus subtilis and Candida pseudotropicalis [1]. | |||
TN1155 | Corytuberine | Others | |
Corytuberine shows proconvulsant effects. The anti-jumping effect of Corytuberine was inhibited only by naloxone. | |||
T13941 | Tubulysin G | Others | |
Tubulysin G is a natural product isolated from the myxobacterial species Archangium geophyra and Angiococcus disciformis, and is a highly cytotoxic peptide. Tubulysin G is a cytotoxic activity tubulysin that inhibits tub... | |||
TN1914 | Marrubiin | Others | |
Marrubiin is a natural product | |||
TN5938 | Rubifolic acid | 30-Hydroxyursolic acid | |
Rubifolic acid is a natural product of Galium, Rubiaceae. The catalog number is TN5938 and the CAS number is 80489-65-2. Rubifolic acid can be used as a reference standard. | |||
TN3421 | Anhydrotuberosin | Others | |
Anhydrotuberosin is a natural product of Pueraria, Fabaceae. The catalog number is TN3421 and the CAS number is 41347-49-3. Anhydrotuberosin can be used as a reference standard. | |||
TN4647 | Neotuberostemonone | Others | |
Neotuberostemonone is a natural product from Stemona mairei. | |||
TN4186 | Hebeirubescensin H | Others | |
Hebeirubescensin H is a natural product from Isodon parvifolius. | |||
TN2340 | Quercetin 3-O-sambubioside | Quercetin 3-Sambubioside | Others |
Quercetin 3-Sambubioside has a role as an antioxidant and a plant metabolite. It is a quercetin O-glucoside, a disaccharide derivative and a tetrahydroxyflavone. | |||
TN5568 | Isosalvipuberulin | Isopuberulin | |
Isosalvipuberulin is a natural product of Salvia, Lamiaceae. The catalog number is TN5568 and the CAS number is 115321-32-9. Isosalvipuberulin can be used as a reference standard. | |||
T24744 | Rubone | ||
Rubone is the tumor suppressor miRNA-34a modulator that acts by inhibiting the growth of hepatocellular carcinoma. | |||
T26167 | Rubropunctatin | Rubropunctamine | |
Rubropunctatin is a monascus pigment with very potent cancer cell proliferation inhibitory effects. | |||
TN5192 | Tuberosin | NOS , Glucokinase | |
Tuberosin shows anti-inflammatory and antioxidant activities.It demonstrated a significantly potent inhibition on yeast α-glucosidase in a dose dependent manner. | |||
TN4925 | Rubiprasin B | Others | |
Rubiprasin B is a natural product from Rubia cordifolia var. pratensis. | |||
T32979 | Lushanrubescensin E | ||
Lushanrubescensin E is a bioactive chemical. | |||
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Cat No. | Product Name | Species | Expression System |
---|---|---|---|
TMPJ-00999 | UBE2D1 Protein, Human, Recombinant (GST) | Human | E. coli |
Ubiquitin-conjugating enzyme E2 D1(UBE2D1)belongs to the ubiquitin-conjugating enzyme family. Ubiquitination involves at least three classes of enzymes: ubiquitin-activating enzymes, or E1s, ubiquitin-conjugating enzymes... | |||
TMPY-00065 | Ebola virus EBOV (subtype Bundibugyo, strain Uganda 2007) VP40/Matrix protein VP40 Protein (His) | EBOV | E. coli |
Ebola virus EBOV (subtype Bundibugyo, strain Uganda 2007) VP40/Matrix protein VP40 Protein (His) is expressed in E. coli expression system with His tag. The predicted molecular weight is 34.4 kDa and the accession number... | |||
TMPY-01552 | HIV-1 (group M, subtype B, strain 92418) p24 Protein (His) | HIV | E. coli |
HIV-1 (group M, subtype B, strain 92418) p24 Protein (His) is expressed in E. coli expression system with His tag. The predicted molecular weight is 26.5 kDa and the accession number is B6DRA0. | |||
TMPY-01373 | HIV-1 (group M, subtype CRF07_BC) gp120 Protein (His) | HIV | HEK293 Cells |
HIV-1 (group M, subtype CRF07_BC) gp120 Protein (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 54.8 kDa and the accession number is I6TSC9. | |||
TMPY-04192 | HIV-1 (group M, subtype B, strain HXB2) p24 Protein (His) | HIV | E. coli |
HIV-1 (group M, subtype B, strain HXB2) p24 Protein (His) is expressed in E. coli expression system with His tag. The predicted molecular weight is 26.5 kDa and the accession number is P04591. | |||
TMPY-02882 | HIV-1 (group M, subtype CRF07_BC) gp140 Protein (His) | HIV | HEK293 Cells |
HIV-1 (group M, subtype CRF07_BC) gp140 Protein (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 78.2 kDa. | |||
TMPJ-01035 | UBE2G2 Protein, Human, Recombinant (GST) | Human | E. coli |
Ubiquitin-Conjugating Enzyme E2 G2 (UBE2G2) is an important cellular mechanism for targeting abnormal or short-lived proteins for degradation, which belong to the ubiquitin-conjugating enzyme family. It shares 60% and 10... | |||
TMPY-02842 | UBE2L6 Protein, Human, Recombinant (His) | Human | E. coli |
UBCH8, also known as UBE2L6, belongs to the ubiquitin-conjugating enzyme family. The family of ubiquitin-conjugating (E2) enzymes is characterized by the presence of a highly conserved ubiquitin-conjugating (UBC) domain.... | |||
TMPY-02426 | UBE2D1 Protein, Human, Recombinant (His) | Human | E. coli |
Ubiquitin-conjugating enzyme E2 D1 (UBE2D1), a member of human E2 ubiquitin-conjugating enzymes, is closely related to SFT, which is short for stimulator of iron (Fe) transport. In other words, UbcH5A is significantly up... | |||
TMPJ-01053 | UBE2I Protein, Human, Recombinant (GST) | Human | E. coli |
SUMO-Conjugating Enzyme UBC9 (UBC9) belongs to the ubiquitin-conjugating enzyme family. UBC9 is homologous to ubiquitin-conjugating enzymes (E2s). However, instead of conjugating ubiquitin, UBC9 conjugates a ubiquitin ho... | |||
TMPY-02604 | UBE2D4 Protein, Human, Recombinant (His) | Human | E. coli |
UBE2D4 is a member of the ubiquitin-conjugating E2 family whose members perform the second step in the ubiquitination reaction. Initially identified as the main process for protein degradation, ubiquitination is believed... | |||
TMPY-02718 | Doublecortin/DCX Protein, Human, Recombinant (aa 45-150, GST) | Human | E. coli |
DCX (doublecortin, N-GST chimera)contains 2 doublecortin domains and belongs to the doublecortin family. It is highly expressed in neuronal cells of fetal brain, but not expressed in other fetal tissues. In the adult, it... | |||
TMPY-02606 | UBE2G1 Protein, Human, Recombinant | Human | E. coli |
UBE2G1 is a member of the ubiquitin-conjugating E2 family whose members perform the second step in the ubiquitination reaction. Initially identified as the main process for protein degradation, ubiquitination is believed... | |||
TMPY-02642 | UBE2W Protein, Human, Recombinant (His) | Human | E. coli |
Ubiquitin-conjugating enzymes, also known as UBE2W, E2 enzymes and more rarely as ubiquitin-carrier enzymes, perform the second step of protein ubiquitination. The modification of protein with ubiquitin is an important c... | |||
TMPH-00314 | Lingual antimicrobial peptide Protein, Bubalus bubalis, Recombinant (His & KSI) | Bubalus bubalis | E. coli |
Has bactericidal activity. Lingual antimicrobial peptide Protein, Bubalus bubalis, Recombinant (His & KSI) is expressed in E. coli expression system with N-6xHis-KSI tag. The predicted molecular weight is 19.8 kDa and th... | |||
TMPH-01519 | HIV-1 (group M, subtype C, isolate 92BR025) Protein Vpr (His & Myc) | HIV-1 | E. coli |
HIV-1 (group M, subtype C, isolate 92BR025) Protein Vpr (His & Myc) is expressed in E. coli expression system with N-10xHis and C-Myc tag. The predicted molecular weight is 18.9 kDa and the accession number is O12160. | |||
TMPH-03015 | MPT64 Protein, Mycobacterium tuberculosis, Recombinant (E. coli, His) | Mycobacterium tuberculosis | E. coli |
N/A. MPT64 Protein, Mycobacterium tuberculosis, Recombinant (E. coli, His) is expressed in E. coli expression system with N-6xHis tag. The predicted molecular weight is 26.4 kDa and the accession number is P9WIN9. | |||
TMPH-03013 | HRP1 Protein, Mycobacterium tuberculosis, Recombinant (His & Myc & SUMO) | Mycobacterium tuberculosis | E. coli |
Unlike some other CBS-domain containing proteins does not seem to bind AMP. | |||
TMPH-03017 | CYP51 Protein, Mycobacterium tuberculosis, Recombinant (His & Myc) | Mycobacterium tuberculosis | Baculovirus Insect Cells |
Its precise biological substrate is not known. Catalyzes C14-demethylation of lanosterol, 24,25-dihydrolanosterol and obtusifoliol which is critical for ergosterol biosynthesis. It transforms lanosterol into 4,4'-dimethy... | |||
TMPH-00321 | Snaclec rhodocytin subunit alpha Protein, Calloselasma rhodostoma, Recombinant (His & SUMO) | Calloselasma rhodostoma | E. coli |
Elicits platelet aggregation by the binding to the C-type lectin domain family 1 member B (CLEC1B/CLEC2). Binding leads to tyrosine phosphorylation in the cytoplasmic tail of CLEC1B, which promotes the binding of spleen ... | |||
TMPH-03074 | UBC5A Protein, Japonica rice, Recombinant (His & Myc) | Rice | E. coli |
E2 conjugating enzyme that associates with the E3 ubiquitin-protein ligase EL5 to mediates ubiquitination of target proteins. UBC5A Protein, Japonica rice, Recombinant (His & Myc) is expressed in E. coli expression syste... | |||
TMPJ-00571 | UBE2D3 Protein, Human, Recombinant | Human | E. coli |
UBE2D3 is an enzyme that belongs to the ubiquitin-conjugating enzyme family. Ubiquitination involves at least three classes of enzymes: ubiquitin-activating enzymes, or E1s, ubiquitin-conjugating enzymes, or E2s, and ubi... | |||
TMPY-04871 | HIV-1 (group M, subtype C, strain 92BR025) gp140 Protein (Fc) | HIV | HEK293 Cells |
HIV-1 (group M, subtype C, strain 92BR025) gp140 Protein (Fc) is expressed in HEK293 mammalian cells with Fc tag. The predicted molecular weight is 99.9 kDa and the accession number is O12164. | |||
TMPY-02840 | Ubiquitin Activating Enzyme E1/UBA1 Protein, Human, Recombinant (His & GST) | Human | Baculovirus Insect Cells |
UBE1, also known as UBA1, belongs to the ubiquitin-activating E1 family. UBE1 gene complements an X-linked mouse temperature-sensitive defect in DNA synthesis, and thus may function in DNA repair. It is part of a gene cl... | |||
TMPH-03562 | Leukocidin-F subunit/LukF Protein, S. aureus, Recombinant (His & Myc & SUMO) | Staphylococcus aureus | E. coli |
Leukocidin causes cytotoxic changes in polymorphonuclear leukocytes. Gamma-hemolysin causes hemolysis in red blood cells. Leukocidin-F subunit/LukF Protein, S. aureus, Recombinant (His & Myc & SUMO) is expressed in E. co... | |||
TMPH-00383 | Tubulin beta-1 chain Protein, Chicken, Recombinant (His) | Chicken | E. coli |
Tubulin is the major constituent of microtubules. It binds two moles of GTP, one at an exchangeable site on the beta chain and one at a non-exchangeable site on the alpha chain. Tubulin beta-1 chain Protein, Chicken, Rec... | |||
TMPH-00815 | HBV-A subtype adw2 (isolate Germany/991/1990) Capsid protein (His & Myc) | HBV-A | E. coli |
HBV-A subtype adw2 (isolate Germany/991/1990) Capsid protein (His & Myc) is expressed in E. coli expression system with N-10xHis and C-Myc tag. The predicted molecular weight is 28.9 kDa and the accession number is P0C69... | |||
TMPH-03006 | Ag85B Protein, Mycobacterium tuberculosis, Recombinant (His) | Mycobacterium tuberculosis | P. pastoris (Yeast) |
Ag85B Protein, Mycobacterium tuberculosis, Recombinant (His) is expressed in yeast with N-6xHis tag. The predicted molecular weight is 32.7 kDa and the accession number is P9WQP0. | |||
TMPH-03427 | Rubella virus (strain RA27/3 vaccine) Structural polyprotein (His) | RUBV | Baculovirus Insect Cells |
Rubella virus (strain RA27/3 vaccine) Structural polyprotein (His) is expressed in Baculovirus insect cells with C-6xHis tag. The predicted molecular weight is 53.4 kDa and the accession number is P19725. | |||
TMPH-00172 | Subtilisin E Protein, Bacillus subtilis, Recombinant (His & SUMO) | Bacillus subtilis | E. coli |
Subtilisin is an extracellular alkaline serine protease, it catalyzes the hydrolysis of proteins and peptide amides. Subtilisin E Protein, Bacillus subtilis, Recombinant (His & SUMO) is expressed in E. coli expression sy... | |||
TMPY-02260 | HEXA Protein, Human, Recombinant (Subunit A, His) | Human | Baculovirus Insect Cells |
HEXA Protein, Human, Recombinant (Subunit A, His) is expressed in Baculovirus insect cells with His tag. The predicted molecular weight is 59.7 kDa and the accession number is AAD13932.1. | |||
TMPY-02313 | Influenza A H5N1 (A/Hubei/1/2010) Hemagglutinin/HA Protein (His) | H5N1 | HEK293 Cells |
Influenza A H5N1 (A/Hubei/1/2010) Hemagglutinin/HA Protein (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 60.1 kDa. | |||
TMPY-00255 | Ebola virus EBOV (subtype Zaire, strain H.sapiens-wt/GIN/2014/Kissidougou-C15) GP2/Glycoprotein Protein (Fc) | EBOV | HEK293 Cells |
Ebola virus EBOV (subtype Zaire, strain H.sapiens-wt/GIN/2014/Kissidougou-C15) GP2/Glycoprotein Protein (Fc) is expressed in HEK293 mammalian cells with Fc tag. The predicted molecular weight is 43.4 kDa and the accessio... | |||
TMPY-00216 | Ebola virus EBOV (subtype Sudan, strain Gulu) VP40/Matrix protein VP40 Protein (His) | EBOV | E. coli |
Ebola virus EBOV (subtype Sudan, strain Gulu) VP40/Matrix protein VP40 Protein (His) is expressed in E. coli expression system with His tag. The predicted molecular weight is 34.5 kDa and the accession number is B0LPL6. | |||
TMPY-03970 | TMUB2 Protein, Human, Recombinant (His) | Human | HEK293 Cells |
TMUB2 Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 24 kDa and the accession number is Q71RG4-2. | |||
TMPH-00315 | BUsg_347 Protein, Buchnera aphidicola subsp., Recombinant (His & Myc & SUMO) | Buchnera aphidicola | E. coli |
Forms pores that allow passive diffusion of small molecules across the membrane. BUsg_347 Protein, Buchnera aphidicola subsp., Recombinant (His & Myc & SUMO) is expressed in E. coli expression system with N-10xHis-SUMO a... | |||
TMPH-03021 | PstP Protein, Mycobacterium tuberculosis, Recombinant (His) | Mycobacterium tuberculosis | E. coli |
Plays an important role in regulating cell division and growth by reversible phosphorylation signaling. May play important roles in regulating cellular metabolism and signaling pathways, which could mediate the growth an... | |||
TMPH-00671 | Major curlin subunit Protein, E. coli O157:H7, Recombinant (His) | E. coli | P. pastoris (Yeast) |
Curlin is the structural subunit of the curli. Curli are coiled surface structures that assemble preferentially at growth temperatures below 37 degrees Celsius. Curli can bind to fibronectin. Major curlin subunit Protein... | |||
TMPY-00302 | HIV-1 (group M, subtype A, isolate 92RW020) gp160 (gp120 subunit) Protein (His) | HIV | HEK293 Cells |
HIV-1 (group M, subtype A, isolate 92RW020) gp160 (gp120 subunit) Protein (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 52.2 kDa and the accession number is Q6BC58. | |||
TMPH-00168 | Levanase Protein, Bacillus subtilis, Recombinant (His) | Bacillus subtilis | E. coli |
Exo-fructosidase that can hydrolyze both levan and inulin, leading to the production of free fructose. Is also able to hydrolyze sucrose and to a small extent raffinose, but not melezitose, stachylose, cellobiose, maltos... | |||
TMPJ-01386 | STUB1 Protein, Human, Recombinant | Human | E. coli |
E3 Ubiquitin-Protein Ligase CHIP is a cytoplasmic protein. CHIP is highly expressed in skeletal muscle, heart, pancreas, brain and placenta. CHIP interacts with the molecular chaperones Hsc70-Hsp70 and Hsp90 through its ... | |||
TMPY-00245 | Ebola virus EBOV (subtype Zaire, strain H.sapiens-wt/GIN/2014/Makona-Kissidougou-C15) GP/Glycoprotein Protein (His) | EBOV | HEK293 Cells |
Ebola virus EBOV (subtype Zaire, strain H.sapiens-wt/GIN/2014/Makona-Kissidougou-C15) GP/Glycoprotein Protein (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 69.3 kDa and the ... | |||
TMPH-03003 | Ag85A Protein, Mycobacterium tuberculosis, Recombinant (His & SUMO) | Mycobacterium tuberculosis | E. coli |
Ag85A Protein, Mycobacterium tuberculosis, Recombinant (His & SUMO) is expressed in E. coli expression system with N-6xHis-SUMO tag. The predicted molecular weight is 44.6 kDa and the accession number is P9WQP2. | |||
TMPH-02994 | MAP_1030 Protein, Mycobacterium paratuberculosis, Recombinant (E. coli, His) | Mycobacterium paratuberculosis | E. coli |
MAP_1030 Protein, Mycobacterium paratuberculosis, Recombinant (E. coli, His) is expressed in E. coli expression system with N-10xHis tag. The predicted molecular weight is 32.8 kDa and the accession number is P62039. | |||
TMPY-04196 | HIV-1 (group M, subtype D, strain NDK) p24 Protein (His) | HIV | E. coli |
HIV-1 (group M, subtype D, strain NDK) p24 Protein (His) is expressed in E. coli expression system with His tag. The predicted molecular weight is 26.6 kDa and the accession number is P18800. | |||
TMPH-00322 | Snaclec rhodocytin subunit beta Protein, Calloselasma rhodostoma, Recombinant (His) | Calloselasma rhodostoma | P. pastoris (Yeast) |
Elicits platelet aggregation by the binding to the C-type lectin domain family 1 member B (CLEC1B/CLEC2). Binding leads to tyrosine phosphorylation in the cytoplasmic tail of CLEC1B, which promotes the binding of spleen ... | |||
TMPH-03007 | Ag85C Protein, Mycobacterium tuberculosis, Recombinant (His) | Mycobacterium tuberculosis | E. coli |
Ag85C Protein, Mycobacterium tuberculosis, Recombinant (His) is expressed in E. coli expression system with N-6xHis tag. The predicted molecular weight is 36.1 kDa and the accession number is P9WQN8. | |||
TMPH-01522 | HIV-2 (subtype A, isolate ROD) Protein Vpx (His) | HIV-2 | P. pastoris (Yeast) |
Plays a role in nuclear translocation of the viral pre-integration complex (PIC), thus is required for the virus to infect non-dividing cells. Targets specific host proteins for degradation by the 26S proteasome. Acts by... | |||
TMPJ-00985 | UBE2A Protein, Human, Recombinant (GST, His) | Human | E. coli |
Ubiquitin-Conjugating Enzyme E2 (UBE2A) is a member of the E2 Ubiquitin-Conjugating Enzyme family. The modification of proteins with ubiquitin is an important cellular mechanism for targeting abnormal or short-lived prot... | |||
TMPY-00041 | Ebola virus EBOV (subtype Zaire, strain H.sapiens-wt/GIN/2014/Kissidougou-C15) Glycoprotein/GP1 Protein (His) | EBOV | Baculovirus Insect Cells |
Ebola virus EBOV (subtype Zaire, strain H.sapiens-wt/GIN/2014/Kissidougou-C15) Glycoprotein/GP1 Protein (His) is expressed in Baculovirus insect cells with His tag. The predicted molecular weight is 52.3 kDa and the acce... | |||
------------------------ More ------------------------ |
Cat No. | Product Name | ||
---|---|---|---|
L7810 | High Solubility Polyfunctional Group Fragment Library | 1159 compounds | |
Highly soluble multifunctional fragment library contains 1159 kinds of fragment molecules. | |||
L1110 | Microtubule-Targeted Compound Library | 142 compounds | |
A unique collection of 142 microtubule-targeted compounds can be used in HTS and HCS; | |||
L8600 | Ubiquitination Compound Library | 210 compounds | |
A unique collection of 210 ubiquitination related small chemicals can be used for high throughput and high content screening; | |||
L7820 | High Solubility Micro Fragment Library | 1081 compounds | |
The compound library of highly soluble micro-fragments consists of 1081 low-molecular-weight fragments. | |||
L7840 | High Solubility FragLite Fragment Library | 796 compounds | |
The highly soluble halogenated fragment library contains 796 halogenated fragment compounds. | |||
L7830 | High Solubility Pharmacophore Fragment Library | 985 compounds | |
High Solubility Pharmacophore Fragment library contains 985 fragment small molecules. | |||
L7850 | High Solubility 3D Diversity Fragment Library | 1079 compounds | |
The library of highly soluble 3D structural diversity fragments contains 1079 compounds. | |||
L7800 | High Solubility Fragment Library | 2728 compounds | |
Structurally diverse, medicinally active, and unique chemistry (strong IP potential); | |||
L7870 | Carboxylic Acid Fragment Library With Solubility | 1806 compounds | |