Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Ticolubant is orally active leukotriene B4 antagonist with high affinity for the human neutrophil LTB4 receptor (Ki = 0.78 nM), blocks LTB4-induced Ca2+ migration with an IC50 of 6.6 ± 1.5 nM, and shows topical anti-inflammatory activity in a mouse model of skin inflammation.
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
1 mg | In stock | $ 210.00 | |
5 mg | In stock | $ 530.00 | |
10 mg | In stock | $ 766.00 | |
25 mg | In stock | $ 1,180.00 | |
50 mg | In stock | $ 1,590.00 | |
100 mg | In stock | $ 2,150.00 | |
500 mg | In stock | $ 4,290.00 |
Description | Ticolubant is orally active leukotriene B4 antagonist with high affinity for the human neutrophil LTB4 receptor (Ki = 0.78 nM), blocks LTB4-induced Ca2+ migration with an IC50 of 6.6 ± 1.5 nM, and shows topical anti-inflammatory activity in a mouse model of skin inflammation. |
Molecular Weight | 460.37 |
Formula | C23H19Cl2NO3S |
CAS No. | 154413-61-3 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 50 mg/mL (108.61 mM)
You can also refer to dose conversion for different animals. More
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Ticolubant 154413-61-3 Immunology/Inflammation Membrane transporter/Ion channel Metabolism LTR Calcium Channel inhibitor inhibit