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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T6262 | Evacetrapib | LY2484595 | CETP |
Evacetrapib (LY2484595) (LY2484595) is a potent and selective inhibitor of CETP with IC50 of 5.5 nM, elevates HDL cholesterol without increases in aldosterone or blood pressure. Phase 3. | |||
T8519 | Raphin1 acetate | Phosphatase | |
Raphin1 acetate is a selective and orally bioavailable regulatory phosphatase PPP1R15B (R15B) inhibitor. | |||
T7820 | Raphin1 | Phosphatase | |
Raphin1 is an orally bioavailable, selective inhibitor of the regulatory phosphatase PPP1R15B (R15B). | |||
T38563 | Raptinal | Caspase | |
Raptinal activates caspase-3 directly and initiates intrinsic caspase-dependent apoptosis pathway in multiple cell lines. | |||
T16697 | Pyronaridine tetraphosphate | Topoisomerase | |
Pyronaridine tetraphosphate is an orally active, mannitol-containing inhibitor of DNA topoisomerase 2 and erythrocyte cytokine with antimalarial and antitumour activity.Pyronaridine tetraphosphate treats P. falciparum an... | |||
T12064 | Niraparib (R-enantiomer) | MK 4827 (R-enantiomer),Niraparib R-enantiomer | PARP |
Niraparib R-enantiomer (MK 4827 R-enantiomer) is an inhibitor of PARP1(IC50 of 2.4 nM). | |||
TP2489 | Tetrapeptide-21 Acetate | Tetrapeptide-21 Acetate(960608-17-7 Free base) | Others |
Tetrapeptide-21 Acetate is a novel bioactive and pure tetrapeptide with anti-aging properties based on the skin's own structures for use in skincare formulations. | |||
TP2363L | Acetyl tetrapeptide-2 Acetate | Acetyl tetrapeptide-2 Acetate(757942-88-4 Free base) | Others |
Acetyl tetrapeptide-2 Acetate is most commonly used as a skin conditioner. Acetyl tetrapeptide-2 Acetate is done by compensating for hormone loss in the skin, especially collagen, providing somewhat of a plumping effect ... | |||
T28225 | Obicetrapib | TA8995,AMG899,Obicetrapib (free base),AMG 899,AMG-899,Obicetrapib,TA-8995 | CETP |
Obicetrapib (AMG-899) is an inhibitor of cholesteryl ester transfer protein. | |||
T11824LL | Lanraplenib | GS-9876 | Syk |
Lanraplenib (GS-9876) is a highly selective and orally active SYK inhibitor (IC50=9.5 nM) in development for the treatment of inflammatory diseases. Lanraplenib inhibits SYK activity in platelets via the glycoprotein VI ... | |||
T31204 | Darapladib-impurity | Others | |
Darapladib-impurity is the impurity of Darapladib. Darapladib inhibits lipoprotein-associated phospholipase A2 (Lp-PLA2). | |||
T20656 | Verapamil | NSC 135784,NSC-135784,CP-16533-1,(±)-Verapamil | P450 , Calcium Channel , P-gp |
Verapamil (CP-16533-1) is a calcium channel blocker and an orally active and effective inhibitor of P-gp. Verapamil inhibits CYP3A4 and can be used in studies about the treatment of high blood pressure, heart arrhythmias... | |||
T7013 | Vorapaxar | SCH 530348,MK-5348 | Protease-activated Receptor |
Vorapaxar (MK-5348) (SCH 530348) is an effective and orally active thrombin receptor (PAR-1) antagonist (Ki: 8.1 nM). | |||
TQ0292 | Grapiprant | AAT-007,RQ-00000007,CJ-023423 | Prostaglandin Receptor |
Grapiprant (AAT-007) is a selective EP4 receptor antagonist. Grapiprant displaces [3H]-PGE2 (1 nM) binding to dog recombinant EP4 receptor (IC50: 35 nM, Ki: 24 nM). | |||
T7625 | TRAP-6 | PAR-1 agonist peptide,Thrombin Receptor Activator Peptide 6,TRAP-6(2TFA) | Protease-activated Receptor |
TRAP-6 (Thrombin Receptor Activator Peptide 6)(2TFA) is an agonist of protease-activated receptor 1 (PAR1). | |||
T3407L | Rapastinel acetate | Rapastinel acetate (117928-94-6 Free base) | NMDAR , iGluR |
Rapastinel acetate is a modulator of N-methyl-D-aspartate (NMDA) receptor and a partial agonist of glycine site long-lasting antidepressant effects. | |||
T1595 | Nevirapine | NSC 641530,BI-RG 587,NVP | HIV Protease , Reverse Transcriptase |
Nevirapine (NVP) is a benzodiazepine non-nucleoside reverse transcriptase inhibitor. In combination with other antiretroviral drugs, nevirapine reduces HIV viral loads and increases CD4 counts, thereby retarding or preve... | |||
T3231 | Niraparib | MK-4827 | Apoptosis , Others , PARP |
Niraparib (MK-4827) is a PARP inhibitor that selectively inhibits PARP1 and PARP2 (IC50=3.8/2.1 nM). Niraparib has antitumor activity, inhibits DNA damage repair, and induces apoptosis. | |||
T3353 | Niraparib hydrochloride | MK-4827 hydrochloride,MK-4827 (hydrochloride) | Apoptosis , Others , PARP |
Niraparib hydrochloride (MK-4827 hydrochloride) is an inhibitor of poly (ADP-ribose) polymerase (PARP) with potential antineoplastic activity. Niraparib hydrochloride inhibits PARP activity, enhancing the accumulation of... | |||
TP1042 | Palmitoyl Tetrapeptide-3 | Rigin | Others |
Palmitoyl Tetrapeptide-3 (Rigin) (Rigin) is a synthetic peptide, corrspending to 341-344 amino acid sequence of IgG human H-chain, with phagocytosis stimulating activity.Palmitoyl Tetrapeptide-3 stimulates expression of ... | |||
T11221 | ERAP1-IN-1 | Others | |
ERAP1-IN-1 is an endoplasmic reticulum aminopeptidase 1 (ERAP1) inhibitor. ERAP1-IN-1 allosterically activates ERAP1’s hydrolysis of fluorogenic and chromogenic amino acid substrates but competitively inhibits its activi... | |||
T7744 | Piperaquine tetraphosphate tetrahydrate | Parasite | |
Piperaquine tetraphosphate tetrahydrate is a potent anti-parasites agent. | |||
T4434 | Tirapazamine | Tirazone,Win59075,SR4233,SR259075 | Others |
Tirapazamine (Win59075) is a potent cytotoxic agent under hypoxic conditions, can induce apoptosis by inducing breaks in single and double-stranded DNA, as well as chromosomal breaks. The compound sensitizes cells to oth... | |||
T2499 | Torcetrapib | CP-529414 | CETP |
Torcetrapib (CP-529414) is a cholesteryl ester transfer protein (CETP) inhibitor that reduces the heterotypic transfer of cholesteryl ester from HDL to LDL and/or VLDL. Torcetrapib failed in phase III trials due to exces... | |||
T68165 | Trapencaine | ||
Trapencaine is a newly synthesized carbamate type local anesthetic that induces conformational changes in sodium channels on hypertrophic cell membranes. | |||
T125901 | 14-Epiandrographolide | ||
14-Epiandrographolide is a compound derived from the above-ground parts of Andrographis paniculata that induces cell differentiation and can be used in the study of multiple sclerosis. | |||
TP2313 | Acetyl Tetrapeptide-5 acetate | Acetyl Tetrapeptide-5 acetate(820959-17-9 free base) | Others |
Acetyl Tetrapeptide-5 acetate helps reduce eye puffiness, improve skin elasticity as well as overall smoothness. | |||
TP2365L | Acetyl tetrapeptide-9 Acetate | Acetyl tetrapeptide-9 Acetate(928006-50-2 Free base) | Others |
Acetyl tetrapeptide-9 Acetate plays a role in the stimulation of basement membrane polysaccharide (lumican) and the synthesis of collagen I. | |||
T6109 | Darapladib | SB-480848 | Phospholipase |
Darapladib (SB-480848)(IC50=0.25 nM) is a substituted pyrimidone with inhibitory activity towards lipoprotein-associated phospholipase-A2 (Lp-PLA2). | |||
T0088 | Urapidil hydrochloride | Urapidil HCl | 5-HT Receptor , Adrenergic Receptor |
Urapidil hydrochloride (Urapidil HCl) is 5-HT1A receptor agonist and an α1-adrenoceptor antagonist. | |||
T6892 | Niraparib tosylate | MK-4827 (tosylate),MK 4827 tosylate,Niraparib (MK-4827) tosylate | Apoptosis , PARP |
Niraparib tosylate (MK-4827 (tosylate))(with IC50 of 3.8 nM/2.1 nM) is a selective PARP1/PARP2 inhibitor. | |||
T3098 | Vorapaxar sulfate | SCH 530348 sulfate,Zontivity,vorapaxar monosulfate | Protease-activated Receptor |
Vorapaxar sulfate (Zontivity) is a potent and orally active thrombin receptor (PAR-1) antagonist. | |||
T69140 | Burapitant | SSR 240600 | Neurokinin receptor |
Burapitant (SSR 240600) is a novel non-peptide tachykinin neurokinin 1 (NK) receptor antagonist with anti-coke oven and antidepressant activity. | |||
T7221 | Satraplatin | BMS182751,JM216,BMY45594 | DNA Alkylator/Crosslinker , DNA Alkylation |
Satraplatin (BMS182751) is an orally available antineoplastic platinum(IV) complex.Satraplatin has a favorable toxicity profile and appears to have clinical activity against a variety of malignancies. | |||
T6048 | Dalcetrapib | JTT-705,RO4607381 | CETP |
Dalcetrapib (RO4607381), a rhCETP inhibitor (IC50=0.2 μM), increases the plasma HDL cholesterol. | |||
T1928 | Anacetrapib | MK-0859 | CETP |
Anacetrapib (MK-0859) (MK0859) is an effective, specific, reversible rhCETP and mutant CETP(C13S) inhibitor (IC50: 7.9 nM and 11.8 nM). Anacetrapib reduces the transfer of cholesteryl ester from HDL to LDL and/or VLDL th... | |||
T10820L1 | Ciraparantag acetate | Ciraparantag acetate(1438492-26-2 Free base) | Others |
Ciraparantag acetate, an anticoagulant reversal agent, is a small molecule specifically designed to bind noncovalently by charge-charge interaction to unfractionated heparin and low-molecular-weight heparin. It shows bin... | |||
T0293 | Metyrapone | NSC-25265,Su-4885 | Others , P450 , Dehydrogenase , Autophagy |
Metyrapone (NSC-25265) is an inhibitor of the enzyme STEROID 11-BETA-MONOOXYGENASE. It is used as a test of the feedback hypothalamic-pituitary mechanism in the diagnosis of CUSHING SYNDROME. | |||
TP2364L | Acetyl tetrapeptide-3 Acetate | Acetyl tetrapeptide-3 Acetate(827306-88-7 Free base) | Others |
Acetyl tetrapeptide-3 Acetate is a biomimetic peptide. | |||
T0080 | Trapidil | Rocornal,Trapymine,Avantrin,Trapymin,AR-12008 | PDGFR , PDE |
Trapidil (Avantrin) is a coronary vasodilator agent. It was originally developed as a vasodilator and anti-platelet agent and has been used to treat patients with ischemic coronary heart, liver, and kidney disease. | |||
T34262 | RAPTA-C | Apoptosis | |
RAPTA-C induces EAC cell cycle arrest and apoptosis via the mitochondrial and p53-JNK pathways, and can be used in the study of breast and ovarian cancer. | |||
T3407 | Rapastinel | GLYX-13,Thr-Pro-Pro-Thr-NH2,TPPT-amide | NMDAR , iGluR |
Rapastinel (TPPT-amide) (GLYX-13) is an N-methyl-D-aspartate receptor (NMDAR) modulator. | |||
T38852L | TRAP-6 amide acetate | Protease-activated Receptor | |
TRAP-6 amide acetate is a PAR-1 thrombin receptor agonist peptide[1]. | |||
TP2497 | Myristoyl Tetrapeptide-12 Acetate | Myristoyl Tetrapeptide-12 Acetate(959610-24-3 Free base) | Others |
Myristoyl Tetrapeptide-12 Acetate (Myristoyl Tetrapeptide-12 Acetate (959610-24-3 Free base)) , the reaction product of myristic acid and Tetrapeptide-12, is a peptide stimulating hair and eyelash growth and enhancing th... | |||
TP2498 | Tetrapeptide-30 Acetate | Tetrapeptide-30 Acetate(1036207-61-0 Free base) | Others |
Tetrapeptide-30 Acetate (Tetrapeptide-30 Acetate) is a synthetic peptide containing the amino acids proline, glutamic acid, and lysine. It acts on and within specific targets of skin to reduce factors and interrupt the p... | |||
T20494L | Acetyl tetrapeptide-15 Acetate | Skinasensyl Acetate,Acetyl tetrapeptide-15 Acetate (928007-64-1 Free base) | |
Acetyl tetrapeptide-15 Acetate (Skinasensyl Acetate), a synthetic peptide used in cosmetic products for sensitive skin, is an endomorphin-2 derivative that extends the range of neuronal excitability thresholds in the μ-o... | |||
T1010 | Verapamil hydrochloride | Manidon,(±)-Verapamil hydrochlorid,Verapamil HCl,Calcan hydrochloride | P450 , Calcium Channel , P-gp |
Verapamil hydrochloride (Verapamil HCl) is a calcium channel blocker that is a class IV anti-arrhythmia agent. | |||
T0165 | Urapidil | Mediatensyl,Ebrantil,Eupressyl | 5-HT Receptor , Adrenergic Receptor |
Urapidil (Ebrantil), a sympatholytic antihypertensive drug, acts as a 5-HT1A receptor agonist and as an α1-adrenoceptor antagonist. | |||
T5819 | Rapastinel Trifluoroacetate | Thr-Pro-Pro-Thr-NH2 Trifluoroacetate,GLYX-13 Trifluoroacetate | NMDAR , iGluR |
Rapastinel Trifluoroacetate (GLYX-13 Trifluoroacetate) is an NMDA receptor modulator with glycine-site partial agonist properties. | |||
T9497 | Niraparib tosylate monohyrate | PARP | |
Niraparib, also know as MK-4827, is an inhibitor of poly (ADP-ribose) polymerase (PARP) with potential antineoplastic activity. MK4827 inhibits PARP activity, enhancing the accumulation of DNA strand breaks and promoting... |
Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T8281 | (R)-Sulforaphane | L-Sulforaphane | Nrf2 |
(R)-Sulforaphane (L-Sulforaphane) is a potent inducer of the Keap1/Nrf2/ARE pathway. | |||
T6520 | Grape Seed Extract | Grape Seed P.E. | Apoptosis , Others |
Grape Seed Extract (Grape Seed P.E.) is exudate from seeds of the grape plant Vitis vinifera, composed of oils and secondary plant metabolites (BIOFLAVONOIDS and polyphenols) credited with important medicinal properties. | |||
TQ0218 | Deoxyandrographolide | 14-deoxyandrographolide | IL Receptor , TNF |
Deoxyandrographolide (14-deoxyandrographolide) potentiates NGF-induced neurite outgrowth. Deoxyandrographolide suppresses the production of proinflammatory mediators TNF-α and IL-6. | |||
T9218 | Andrograpanin | 19-HYDROXY-8(17),13-LABDADIEN-16,15-OLIDE | p38 MAPK |
Andrograpanin (19-HYDROXY-8(17),13-LABDADIEN-16,15-OLIDE) is a bioactive compound from Andrographis paniculata. Andrograpanin has anti-inflammatory and anti-infectious properties. | |||
TQ0212 | Glucoraphanin | Antioxidant , Reactive Oxygen Species | |
Glucoraphanin, the precursor of the widely extolled chemopreventive agent sulforaphane found in broccoli, has antioxidant activity. | |||
TN1933 | Mitraphylline | IL Receptor , TNF , NF-κB | |
Mitraphylline has antiproliferative effects on human glioma and neuroblastoma cell lines. It also has anti-inflammatory activity, it inhibits lipopolysaccharide-mediated activation of primary human neutrophils. | |||
T3884 | Neoandrographolide | Neoandrographiside | NOS , COX |
Neoandrographolide (Neoandrographiside) has potent hypolipidemic effect and protects the cardiovascular without significant liver damage.Neoandrographolide has anti-inflammatory effect, might result from inhibition of iN... | |||
TQ0207 | Sulforaphane | Apoptosis , Nrf2 , HDAC | |
Sulforaphane is derived from the consumption of cruciferous vegetables, such as broccoli. It has shown anticancer and cardioprotective activities. | |||
T2738 | Dehydroandrographolide | NOS , Influenza Virus | |
Dehydroandrographolide is a natural compound extracted from herbal medicine Andrographis paniculata (Burm f) Nees. | |||
T37009 | Oxychlororaphine | phenazine-1-carboxamide | Antibacterial |
Oxychlororaphine (phenazine-1-carboxamide) inhibits strongly the growth of Streptomyces sp. 441. | |||
TN4893 | Rapanone | 2,5-Dihydroxy-3-tridecyl-[1,4]benzoquinone,2,5-Dihydroxy-3-tridecylcyclohexa-2,5-diene-1,4-dione | Apoptosis , Phospholipase , Antibacterial , Parasite |
Rapanone (2,5-Dihydroxy-3-tridecyl-[1,4]benzoquinone) is a natural benzoquinone that is a potent and selective inhibitor of human synovial PLA2. | |||
T3667 | Kalii Dehydrographolidi Succinas | Ddhads,Dehydroandrographolide Succinate Potasium Salt | Others |
Kalii Dehydrographolidi Succinas (Dehydroandrographolide Succinate Potasium Salt) is a natural compound with anti-virus infection activity. | |||
T8288 | 14-Deoxyandrographolide | Apoptosis , Others | |
14-Deoxyandrographolide is a bioactive compound of Andrographis paniculata with hepatoprotective efficacy. It desensitizes hepatocytes to TNF-α-mediated apoptosis through the release of TNFRSF1A release. | |||
T2898 | Andrographolide | Andrographis | SARS-CoV , Influenza Virus , NF-κB , Autophagy |
Andrographolide (Andrographis)(Andrographis), an irreversible antagonist of NF-κB, has anti-inflammatory and anti-platelet aggregation activities and potential antineoplastic. | |||
T2S0257 | Dehydroandrographolide succinate | Others , Influenza Virus | |
Dehydroandrographolide Succinate is a traditional Chinese medicine used in the treatment of pneumonia, respiratory tract infection. | |||
TQ0185 | 14-Deoxy-11,12-didehydroandrographolide | AP10,14-dehydro Andrographolide | NF-κB |
14-Deoxy-11,12-didehydroandrographolide (AP10) has hypotensive, anti-inflammatory, anti-asthma, and anti-cancer actions. It can inhibit NF-κB activation. | |||
T4115 | Auraptene | 7-geranyloxycoumarin | MMP , BACE |
Auraptene is a coumarin derived from citrus plants that bears a geranyloxyl moiety at its C-7. It has anti-inflammatory, anti-carcinogenic, anti-bacterial, neuroprotective, and hepatoprotective activities. It inhibits le... | |||
TL0016 | Sulforaphene | Apoptosis , ERK , EGFR , NF-κB | |
Sulforaphene is a natural product isolated from radish seeds, exhibits an ED50 against velvetleaf seedlings approximately 2 x 10 -4 M. Sulforaphene promotes cancer cells apoptosis and inhibits migration via inhibiting EG... | |||
T1537 | Rapamycin | Sirolimus,AY 22989,NSC-2260804 | Others , Endogenous Metabolite , Antibiotic , mTOR , Autophagy , Antifungal |
Rapamycin (AY 22989) is a natural product of macrolides, an mTOR inhibitor with specificity (HEK293 cells: IC50=0.1 nM). Rapamycin has immunosuppressive activity and induces autophagy. | |||
TN3530 | Borapetoside B | Others | |
Borapetoside B is a natural product of Tinospora, Menispermaceae. The catalog number is TN3530 and the CAS number is 104901-05-5. Borapetoside B can be used as a reference standard. | |||
TN5336 | 9-Oxo-10,11-dehydroageraphorone | 4,7(11)-Cadinadiene-3,8-dione,DTD,7,11-Dehydro-8-oxoageraphorone | |
9-Oxo-10,11-dehydroageraphorone has acaricidal activity. It induces hepatotoxicity and cholestasis in rats. 9-Oxo-10,11-dehydroageraphorone also effectively inhibits the proliferation of HeLa cells by arresting the cell ... | |||
TN5586 | 14-Deoxy-12-hydroxyandrographolide | ||
14-Deoxy-12-hydroxyandrographolide is a natural product of Andrographis, Acanthaceae. The catalog number is TN5586 and the CAS number is 219721-33-2. 14-Deoxy-12-hydroxyandrographolide can be used as a reference standard... | |||
TN6029 | Rauvotetraphylline E | ||
Rauvotetraphylline E is a natural product from Rauvolfia tetraphylla. | |||
T25305 | Demethoxyrapamycin | AY 24668,AY24668,AY-24668 | |
Demethoxyrapamycin is a new antifungal antibiotic agent which is co-produced with rapamycin by Streptomyces hygroscopicus. | |||
T72580 | Isoandrographolide | ||
Isoandrographolide, a compound known for its cell differentiation-inducing and hepatoprotective effects, also inhibits NLRP3 inflammasome activation and mitigates silicosis in mice. | |||
TN3411 | Andrographidine C | Others | |
Andrographidine C is a natural product of Andrographis, Acanthaceae. The catalog number is TN3411 and the CAS number is 113963-39-6. Andrographidine C can be used as a reference standard. | |||
TN6038 | 1,2-Methylenedioxy-3,10,11-trimethoxynoraporphine | ||
1,2-Methylenedioxy-3,10,11-trimethoxyaporphine exerts moderate vessel-relaxing activities with the IC 50 value from 16.50 to 32.81 microM at the test concentrations. | |||
TN3533 | Borapetoside F | Others | |
Borapetoside F is a natural product of Tinospora, Menispermaceae. The catalog number is TN3533 and the CAS number is 151200-50-9. Borapetoside F can be used as a reference standard. | |||
T13582 | Bisandrographolide C | Others | |
Bisandrographolide C is identified from Andrographis paniculata. Bisandrographolide C activates TRPV1 and TRPV3 channels (Kds: 289 and 341 μM) and protects cardiomyocytes from hypoxia-reoxygenation injury. | |||
TN2623 | 14-Deoxy-17-hydroxyandrographolide | Antifection | |
14-Deoxy-17-hydroxyandrographolide is a natural product of Andrographis, Acanthaceae. The catalog number is TN2623 and the CAS number is 869384-82-7. 14-Deoxy-17-hydroxyandrographolide can be used as a reference standard... | |||
TN5585 | 14-Deoxy-11-hydroxyandrographolide | ||
14-Deoxy-11-hydroxyandrographolide shows potent cell differentiation-inducing activity towards mouse myeloid leukemia (M1) cells. | |||
TN5636 | Caraphenol A | ||
Caraphenol A is a natural product of Caragana, Fabaceae. The catalog number is TN5636 and the CAS number is 354553-35-8. Caraphenol A can be used as a reference standard. | |||
TN3795 | Dehydroborapetoside B | Others | |
Dehydroborapetoside B is a natural product for research related to life sciences. The catalog number is TN3795 and the CAS number is 1221178-16-0. | |||
TN2463 | 14-Deoxy-11-oxoandrographolide | Others | |
14-Deoxy-11-oxoandrographolide is a natural product from Andrographis paniculata | |||
TN6599 | Andrographidine A | ||
Andrographidine A is a natural product for research related to life sciences. The catalog number is TN6599 and the CAS number is 113963-37-4. | |||
TN3412 | Andrographiside | Others | |
Andrographiside shows protective effects on hepatotoxicity induced in mice by carbon tetrachloride or tert-butylhydroperoxide (tBHP) intoxication, the effects could be due to its glucoside groups which may act as strong ... | |||
TN2622 | 14-Deoxy-11,12-didehydroandrographiside | Others | |
14-Deoxy-11,12-didehydroandrographiside is a natural product of Andrographis, Acanthaceae. The catalog number is TN2622 and the CAS number is 141973-41-3. 14-Deoxy-11,12-didehydroandrographiside can be used as a referenc... | |||
TN4269 | Isocarapanaubine | Others | |
Isocarapanaubine and reserpiline are cytotoxic constituents from the barks of Ochrosia elliptica. | |||
TN3532 | Borapetoside E | Others | |
Borapetoside E has anti-hyperglycemic activity, it can significantly reduce serum glucose levels at dose-dependent manners in alloxan-induced hyperglycemic mice and db/db type 2 diabetic mice. | |||
TN4896 | Rauvotetraphylline B | Others | |
Rauvotetraphylline B is a natural product from Rauvolfia tetraphylla. | |||
TN3329 | 9-Oxoageraphorone | Others | |
9-Oxoageraphorone has strong acaricidal activity against P. cuniculi in vitro, it also exhibits high insecticidal effects. | |||
TN3531 | Borapetoside D | Others | |
Borapetoside D is a natural product of Tinospora, Menispermaceae. The catalog number is TN3531 and the CAS number is 151200-48-5. Borapetoside D can be used as a reference standard. | |||
TN3518 | Bisandrographolide A | Others | |
Bisandrographolide A activates TRPV4 channels, could play a role in some of the effects of Andrographis extract described in traditional medicine. | |||
TN4895 | Rauvotetraphylline A | Others | |
Rauvotetraphylline A is a natural product from Rauvolfia tetraphylla. | |||
TN4897 | Rauvotetraphylline C | Others | |
Rauvotetraphylline C is a natural product from Rauvolfia tetraphylla. | |||
TN4311 | Isomitraphylline | Others | |
Isomitraphylline and pteropodine are the most suitable for standardization of medical cat's claw preparations. Isomitraphylline can inhibit proliferation of acute lymphoblastic leukaemia cells. | |||
TN1415 | Auraptenol | 5-HT Receptor | |
Auraptenol possesses robust antidepressant-like efficacy in mice. |
Cat No. | Product Name | Species | Expression System |
---|---|---|---|
TMPY-00992 | ERAP2 Protein, Human, Recombinant (His) | Human | HEK293 Cells |
Leukocyte-derived arginine aminopeptidase (LRAP), also known as endoplasmic reticulum-aminopeptidase 2 (ERAP2), is the second identified aminopeptidase localized in the in the lumenal side of endoplasmic reticulum ... | |||
TMPY-01732 | LRPAP1 Protein, Mouse, Recombinant (His) | Mouse | HEK293 Cells |
LRPAP1 Protein, Mouse, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 40.4 kDa and the accession number is P55302. | |||
TMPY-01233 | LRPAP1 Protein, Human, Recombinant (His) | Human | HEK293 Cells |
LRPAP1 Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 39.2 kDa and the accession number is P30533. | |||
TMPY-01446 | IL-18R beta/IL-18RAP Protein, Human, Recombinant (His) | Human | HEK293 Cells |
IL-18R beta/IL-18RAP Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 40 kDa and the accession number is O95256-1. | |||
TMPY-04580 | IL-1RAP/IL-1RAcP Protein, Mouse, Recombinant (His) | Mouse | HEK293 Cells |
IL-1RAP/IL-1RAcP Protein, Mouse, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 39.7 kDa and the accession number is Q3UEL3. | |||
TMPY-03102 | IL-18R beta/IL-18RAP Protein, Rhesus, Recombinant (hFc) | Rhesus | HEK293 Cells |
IL-18R beta/IL-18RAP Protein, Rhesus, Recombinant (hFc) is expressed in HEK293 mammalian cells with hFc tag. The predicted molecular weight is 65.4 kDa and the accession number is XP_001108108.1. | |||
TMPY-05593 | IL-1RAP/IL-1RAcP Protein, Human, Recombinant (His & Avi), Biotinylated | Human | HEK293 Cells |
IL-1RAP/IL-1RAcP Protein, Human, Recombinant (His & Avi), Biotinylated is expressed in HEK293 mammalian cells with His and Avi tag. The predicted molecular weight is 42.4 kDa and the accession number is Q9NPH3-1. | |||
TMPY-05840 | IL-1RAP/IL-1RAcP Protein, Cynomolgus, Recombinant (His) | Cynomolgus | HEK293 Cells |
IL-1RAP/IL-1RAcP Protein, Cynomolgus, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 40.56 kDa and the accession number is P59822-1. | |||
TMPK-00330 | IL-1RAP/IL-1RAcP Protein, Human, Recombinant (His & Avi) | Human | HEK293 Cells |
IL-1RAP/IL-1RAcP Protein, Human, Recombinant (His & Avi) is expressed in HEK293 mammalian cells with C-His-Avi tag. The predicted molecular weight is 42 kDa and the accession number is Q9NPH3-1. | |||
TMPY-03048 | PRAP1 Protein, Human, Recombinant (mFc) | Human | HEK293 Cells |
PRAP1 Protein, Human, Recombinant (mFc) is expressed in HEK293 mammalian cells with mFc tag. The predicted molecular weight is 41.4 kDa and the accession number is AAL16670.1. | |||
TMPK-01029 | IL-1RAP/IL-1RAcP Protein, Mouse, Recombinant (aa 21-367, His) | Mouse | HEK293 Cells |
Interleukin (IL)-1R3 is the co-receptor in three signaling pathways that involve six cytokines of the IL-1 family (IL-1α, IL-1β, IL-33, IL-36α, IL-36β and IL-36γ). In many diseases, multiple cytokines contribute to disea... | |||
TMPY-02117 | Marapsin Protein, Human, Recombinant (His) | Human | HEK293 Cells |
The name "Pancreasin" because it is transcribed strongly in the pancreas. This secreted, tryptic serine protease, also known as Marapsin or PRSS27 (Protease, serine, 27), is a member of the peptidase S1 family. Pancreasi... | |||
TMPY-03076 | PRAP1 Protein, Human, Recombinant (His) | Human | HEK293 Cells |
PRAP1 Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 16.4 kDa and the accession number is AAL16670.1. | |||
TMPH-03231 | AFP2 Protein, Raphanus sativus, Recombinant (His & SUMO) | Raphanus sativus | E. coli |
Possesses antifungal activity sensitive to inorganic cations. Induces potential changes in fungal membranes and increased K(+) efflux and Ca(2+) uptake. AFP2 Protein, Raphanus sativus, Recombinant (His & SUMO) is express... | |||
TMPY-05392 | IL-1RAP/IL-1RAcP Protein, Human, Recombinant (hFc) | Human | HEK293 Cells |
IL-1RAP/IL-1RAcP Protein, Human, Recombinant (hFc) is expressed in HEK293 mammalian cells with hFc tag. The predicted molecular weight is 65.8 kDa and the accession number is Q9NPH3-1. | |||
TMPY-06761 | IL-18R beta/IL-18RAP Protein, Rat, Recombinant (His) | Rat | HEK293 Cells |
IL-18R beta/IL-18RAP Protein, Rat, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 40.28 kDa and the accession number is A0A0G2K2K7. | |||
TMPK-00514 | IL-18RAP Protein, Cynomolgus, Recombinant (His) | Cynomolgus | HEK293 Cells |
IL-18RAP, also known as IL-18Rβ or IL-1R7, is component of IL-18 receptor complex and its interactions with IL-18R1 mediate signal transduction initiated by IL-18 although it does not directly bind IL-18 in vitro. | |||
TMPH-03316 | IL-1RAP/IL-1RAcP Protein, Rat, Recombinant (His & Myc) | Rat | E. coli |
IL-1RAP/IL-1RAcP Protein, Rat, Recombinant (His & Myc) is expressed in E. coli expression system with N-10xHis and C-Myc tag. The predicted molecular weight is 47.5 kDa and the accession number is Q63621. | |||
TMPY-00985 | IL-1RAPL1 Protein, Human, Recombinant (hFc) | Human | HEK293 Cells |
IL-1RAPL1 Protein, Human, Recombinant (hFc) is expressed in HEK293 mammalian cells with hFc tag. The predicted molecular weight is 65 kDa and the accession number is Q9NZN1. | |||
TMPH-02267 | AGTRAP Protein, Human, Recombinant (His & Myc & SUMO) | Human | E. coli |
Appears to be a negative regulator of type-1 angiotensin II receptor-mediated signaling by regulating receptor internalization as well as mechanism of receptor desensitization such as phosphorylation. Induces also a decr... | |||
TMPY-01200 | IL-18R beta/IL-18RAP Protein, Human, Recombinant (hFc) | Human | HEK293 Cells |
IL-18R beta/IL-18RAP Protein, Human, Recombinant (hFc) is expressed in HEK293 mammalian cells with hFc tag. The predicted molecular weight is 65.2 kDa and the accession number is O95256-1. | |||
TMPY-00587 | GABARAP Protein, Human, Recombinant (His & MBP) | Human | E. coli |
The Atg8/LC3/GABARAP family of proteins, a group that has structural homology with ubiquitin, connects with a large set of binding partners to function in macroautophagy (hereafter autophagy). GABARAP in tumorigenesis in... | |||
TMPY-01251 | IL-1RAP/IL-1RAcP Protein, Human, Recombinant (His) | Human | HEK293 Cells |
IL-1RAP/IL-1RAcP Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 40.7 kDa and the accession number is Q9NPH3-1. | |||
TMPK-00331 | IL-1RAP/IL-1RAcP Protein, Human, Recombinant (aa 21-359, His & Avi), Biotinylated | Human | HEK293 Cells |
IL-1RAP/IL-1RAcP Protein, Human, Recombinant (aa 21-359, His & Avi), Biotinylated is expressed in HEK293 mammalian cells with C-His-Avi tag. The predicted molecular weight is 42 kDa and the accession number is Q9NPH3-1. | |||
TMPY-03268 | GABARAPL1 Protein, Human, Recombinant (His) | Human | E. coli |
ATG8, also known as GABARAPL1, is a ubiquitin-like protein that has a crystal structure. ATG8 consists of a 5-stranded β-sheet, which is enclosed by two α-helices at one side and one α-helix at the other side and exhibit... | |||
TMPK-00654 | IL-1RAP/IL-1RAcP Protein, Cynomolgus, Recombinant (aa 21-362, His) | Cynomolgus | HEK293 Cells |
IL-1RAP/IL-1RAcP Protein, Cynomolgus, Recombinant (aa 21-362, His) is expressed in HEK293 mammalian cells with C-His tag. The predicted molecular weight is 40.49 kDa and the accession number is G7NYP7. | |||
TMPY-01117 | MRAP Protein, Human, Recombinant (hFc) | Human | HEK293 Cells |
MRAP (Melanocortin 2 Receptor Accessory Protein) is a Protein Coding gene. This gene encodes a melanocortin receptor-interacting protein. It belongs to the MRAP family. MRAP, which contains a single transmembrane domain,... | |||
TMPH-02819 | Otoraplin Protein, Mouse, Recombinant (His) | Mouse | P. pastoris (Yeast) |
Otoraplin Protein, Mouse, Recombinant (His) is expressed in yeast with C-6xHis tag. The predicted molecular weight is 14.0 kDa and the accession number is Q9JIE3. | |||
TMPJ-00015 | GABARAP Protein, Human, Recombinant (His & hFc) | Human | E. coli |
GABARAP Protein, Human, Recombinant (His & hFc) is expressed in E. coli expression system with N-6xHis and C-Fc tag. The predicted molecular weight is 50 KDa and the accession number is Q6IAW1. | |||
TMPY-06316 | IL-18R beta/IL-18RAP Protein, Human, Recombinant (hFc & Avi), Biotinylated | Human | HEK293 Cells |
IL-18R beta/IL-18RAP Protein, Human, Recombinant (hFc & Avi), Biotinylated is expressed in HEK293 mammalian cells with hFc and Avi tag. The predicted molecular weight is 67.04 kDa and the accession number is NP_003844.1. | |||
TMPJ-00344 | IL-18RAP Protein, Human, Recombinant (hFc & His) | Human | HEK293 Cells |
IL-18RAP is a single-pass type I membrane protein and contains two Ig-like C2-type domains and one TIR domain, IL18RAP can be induced by IFN-alpha and IL12 in nature killer cells and T-cells. The coexpression of IL18R1 a... | |||
TMPJ-01347 | IL-1RAP/IL-1RAcP Protein, Human, Recombinant (aa 21-356, His) | Human | HEK293 Cells |
IL-1RAP/IL-1RAcP Protein, Human, Recombinant (aa 21-356, His) is expressed in HEK293 mammalian cells with C-6xHis tag. The predicted molecular weight is 50-70 KDa and the accession number is Q9NPH3-2. | |||
TMPY-06750 | IL-18R beta/IL-18RAP Protein, Rabbit, Recombinant (His) | Rabbit | HEK293 Cells |
IL-18R beta/IL-18RAP Protein, Rabbit, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 40.22 kDa and the accession number is G1SQ92. | |||
TMPY-01036 | IL-1RAPL1 Protein, Human, Recombinant (His) | Human | HEK293 Cells |
IL-1RAPL1 Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 40 kDa and the accession number is Q9NZN1. | |||
TMPY-06312 | IL-18R beta/IL-18RAP Protein, Human, Recombinant (His & Avi), Biotinylated | Human | HEK293 Cells |
IL-18R beta/IL-18RAP Protein, Human, Recombinant (His & Avi), Biotinylated is expressed in HEK293 mammalian cells with His and Avi tag. The predicted molecular weight is 41.76 kDa and the accession number is NP_003844.1. | |||
TMPY-00609 | IL-18R beta/IL-18RAP Protein, Mouse, Recombinant (His) | Mouse | Baculovirus Insect Cells |
IL-18R beta/IL-18RAP Protein, Mouse, Recombinant (His) is expressed in Baculovirus insect cells with His tag. The predicted molecular weight is 40.1 kDa and the accession number is Q0VBK3. | |||
TMPJ-00016 | GABARAP Protein, Human, Recombinant (GST) | Human | E. coli |
GABARAP Protein, Human, Recombinant (GST) is expressed in E. coli expression system with N-GST tag. The predicted molecular weight is 37 KDa and the accession number is Q6IAW1. | |||
TMPH-00818 | Delta-theraphotoxin-Hm1a Protein, Heteroscodra maculata, Recombinant (His & Myc & SUMO) | Heteroscodra maculata | E. coli |
Delta-theraphotoxin-Hm1a Protein, Heteroscodra maculata, Recombinant (His & Myc & SUMO) is expressed in E. coli expression system with N-6xHis-SUMO and C-Myc tag. The predicted molecular weight is 21.5 kDa and the access... | |||
TMPY-05839 | IL-1RAP/IL-1RAcP Protein, Cynomolgus, Recombinant (hFc) | Cynomolgus | HEK293 Cells |
IL-1RAP/IL-1RAcP Protein, Cynomolgus, Recombinant (hFc) is expressed in HEK293 mammalian cells with hFc tag. The predicted molecular weight is 65.84 kDa and the accession number is P59822-1. | |||
TMPH-00062 | Icarapin Protein, Apis mellifera carnica, Recombinant (His & Myc) | Apis mellifera carnica | E. coli |
Icarapin Protein, Apis mellifera carnica, Recombinant (His & Myc) is expressed in E. coli expression system with N-10xHis and C-Myc tag. The predicted molecular weight is 27.7 kDa and the accession number is Q5EF78. | |||
TMPY-03103 | IL-18R beta/IL-18RAP Protein, Rhesus, Recombinant (His) | Rhesus | HEK293 Cells |
IL-18R beta/IL-18RAP Protein, Rhesus, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 39.85 kDa and the accession number is XP_001108108.1. | |||
TMPH-01428 | TRAP1 Protein, Human, Recombinant (GST) | Human | E. coli |
Chaperone that expresses an ATPase activity. Involved in maintaining mitochondrial function and polarization, downstream of PINK1 and mitochondrial complex I. Is a negative regulator of mitochondrial respiration able to ... | |||
TMPY-03461 | GABARAPL2 Protein, Human, Recombinant (His) | Human | E. coli |
GATE-16, also known as ATG8, belongs to the MAP1 LC3 family. It is expressed at high levels in the brain, heart, prostate, ovary, spleen and skeletal muscle. GATE-16 is expressed at very low levels in lung, thymus and... | |||
TMPY-02547 | IL-1RAPL1 Protein, Mouse, Recombinant (hFc) | Mouse | HEK293 Cells |
IL-1RAPL1 Protein, Mouse, Recombinant (hFc) is expressed in HEK293 mammalian cells with hFc tag. The predicted molecular weight is 65 kDa and the accession number is P59823. | |||
TMPY-04579 | IL-1RAP/IL-1RAcP Protein, Mouse, Recombinant (hFc) | Mouse | HEK293 Cells |
IL-1RAP/IL-1RAcP Protein, Mouse, Recombinant (hFc) is expressed in HEK293 mammalian cells with hFc tag. The predicted molecular weight is 65 kDa and the accession number is Q3UEL3. | |||
TMPJ-01346 | IL-1RAP/IL-1RAcP Protein, Human, Recombinant (hFc & His) | Human | HEK293 Cells |
IL-1RAP/IL-1RAcP Protein, Human, Recombinant (hFc & His) is expressed in HEK293 mammalian cells with C-Fc-6xHis tag. The predicted molecular weight is 80-100 KDa and the accession number is Q9NPH3-2. |
Cat No. | Product Name | ||
---|---|---|---|
L2151 | Chemotherapy Drug Library | 48 compounds | |
48 Chemotherapeutic drugs that can be used for high-throughput and high-content screening. | |||
L2152 | Targeted Therapy Drug Library | 119 compounds | |
119 tumor-targeted drugs that can be used for high-throughput and high-content screening. |