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Grapiprant

Catalog No. TQ0292    CAS 415903-37-6    Synonyms: CJ-023423, RQ-00000007, AAT-007

Grapiprant (CJ-023423) is a selective EP4 receptor antagonist. Grapiprant displaces [3H]-PGE2 (1 nM) binding to dog recombinant EP4 receptor (IC50: 35 nM, Ki: 24 nM).

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50 mg Inquiry 1149.00
100 mg Inquiry 1701.00
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Biological Activity:

Product Description:

Grapiprant (CJ-023423) is a selective EP4 receptor antagonist. Grapiprant displaces [3H]-PGE2 (1 nM) binding to dog recombinant EP4 receptor (IC50: 35 nM, Ki: 24 nM).

Receptor:

Chemical Information:
Molecular Weight 491.60
Formula C26H29N5O3S
CAS Number 415903-37-6
Solubility

:

DMSO: ≥48mg/mL(97.64 mM)

( < 1 mg/ml refers to the product slightly soluble or insoluble )
Storage store at -80°C
Remark For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20 ℃ for several month.