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Search Result

Search Results for " estrogen "

Targets

Estrogen/progestogen Receptor Estrogen Receptor/ERR Estrogen Receptor/ERR

282

Compounds

78

Natural Products

31

Recombinant Proteins

1

Libraries

Cat No. Product Name Synonyms Targets
T15249 Estrogen receptor modulator 1 Estrogen Receptor/ERR
Estrogen receptor modulator 1 causes regression of Tamoxifen-resistant, hormone-independent xenograft tumors. Estrogen receptor modulator 1 is an orally active and selective estrogen receptor modulator (SERM) (pIC50: 0.4...
T78646 Estrogen receptor antagonist 8 Estrogen Receptor/ERR
Estrogen Receptor Antagonist 8 exhibits potent antagonistic activity against the estrogen receptor (ER), demonstrating effective anti-uterotrophic potential in vivo, with an EC50 value of 4.160 μM.
T11237 Camizestrant Estrogen receptor antagonist 2 Estrogen Receptor/ERR
Camizestrant (Estrogen receptor antagonist 2) is an antagonist of the estrogen receptor and can be used in studies about ER+ HER2-advanced breast cancer[1].
T11236 Giredestrant tartrate Estrogen receptor antagonist 1 Estrogen Receptor/ERR , Others
Giredestrant tartrate (Estrogen receptor antagonist 1) is a novel, orally active, selective and effective non-steroidal estrogen receptor antagonist. Giredestrant tartrate strongly binds to ER, resulting in the failure o...
T40893 Estrogen receptor modulator 6
Estrogen receptor modulator 6 (compound 3a) is a highly specific and potent agonist of the estrogen receptor (ER) β with a remarkable affinity (K i = 0.44 nM). This compound exhibits an impressive 19-fold selectivity for...
T19988 Conjugated Estrogen sodium Conjugated estrogens,Conest,HSDB 3076,Kestrin,Estrogens, conjugated,TAG-39
Conjugated estrogens are medicine that contains a mixture of estrogen hormones. It is used to treat moderate to severe hot flashes, changes in and around the vagina, and other symptoms of menopause or low amounts of estr...
T63277 Estrogen receptor antagonist 2
Estrogen receptor antagonist 2 is a selective down-regulator of estrogen receptor. Estrogen (E2) and estrogen alpha receptor (ERα) are important drivers of breast cancer development. estrogen receptor antagonist 2 has re...
T63914 Estrogen receptor antagonist 3
Estrogen receptor antagonist 3 is a potent degradation agent of the estrogen receptor (ER). Estrogen signalling systems play an important role in the regulation of cell growth, differentiation and apoptosis, and Estrogen...
T63106 Estrogen receptor antagonist 4
Estrogen Receptor Antagonist 4 is a potent inhibitor of the estrogen receptor (ER), crucial for regulating cell growth, differentiation, and apoptosis. This compound holds promise for cancer research[1].
T79109 Estrogen receptor modulator 8 Estrogen Receptor/ERR
Estrogen Receptor Modulator 8 (compound 4) is an orally active inhibitor targeting Estrogen Receptor/ERR α with potent efficacy (IC50 = 0.437 nM in MCF-7 cells) and effectively hampers MCF-7 cell proliferation (IC50 = 0....
T62952 Estrogen receptor antagonist 5
Estrogen receptor antagonist 5 is a potent antagonist of the Estrogen receptor. Estrogen receptor (Estrogen receptor) is a ligand-activated transcriptional regulatory protein that interacts with endogenous estrogens and ...
T63582 Estrogen receptor antagonist 1
Estrogen receptor antagonist 1 is a potent antagonist of the estrogen receptor. Estrogen receptor antagonist 1 has shown research potential in breast cancer disease.
T79064 Estrogen receptor modulator 7 Estrogen Receptor/ERR
Estrogen Receptor Modulator 7 is a potent modulator of estrogen receptors, utilized in cancer research [1].
T60293 Estrogen receptor-IN-1
Estrogen receptor-IN-1 (compound 16) is an effective estrogen receptor (ER) inhibitor with IC 50 s of 13, 5μM for ERα and Erβ, respectively [1].
T62953 Estrogen receptor antagonist 6
Estrogen receptor antagonist 6 is a potent antagonist of the Estrogen receptor. Estrogen receptor is a ligand-activated transcriptional regulatory protein that interacts with endogenous estrogens and mediates the inducti...
T61909 Estrogen receptor antagonist 7
Estrogen Receptor Antagonist 7 (Compound 13) is a potent antagonist of estrogen receptors (ER), demonstrating antiproliferative effects against breast and ovarian cancer cells, along with anticancer and anti-uterotrophic...
T82439 Estrogen receptor modulator 10 Estrogen Receptor/ERR
Compound G-5b, an estrogen receptor modulator 10, functions as an estrogen receptor (ER) antagonist (IC50=6.7 nM) and degrader (DC50=0.4 nM). It has the capability to induce apoptosis and block cells at the G1/G0 phase, ...
T62311 Estrogen receptor β antagonist 2
Estrogen receptor β antagonist 2 is a selective, potent estrogen receptor β (ERβ) antagonist that acts on Erα (IC50: 109.10 μM) and Erβ (IC50: 0.63 μM).
T62764 Estrogen receptor α antagonist 1
Estrogen receptor α antagonist 1 (compound 35) is a highly selective estrogen receptor α antagonist that acts on estrogen receptor α (IC50: 0.02 μM), estrogen receptor β (IC50. Estrogen receptor α antagonist 1 (compound ...
T4388 PHTPP Estrogen Receptor/ERR , Estrogen/progestogen Receptor
PHTPP is a selective ERβ antagonist.
T8984 FLTX1 Estrogen Receptor/ERR , Estrogen/progestogen Receptor
FLTX1 is a fluorescent derivative of Tamoxifen, designed to efficiently target and label intracellular Tamoxifen-binding sites (estrogen receptors) both under permeabilized and non-permeabilized conditions. Additionally,...
T7904 SR 19881 Estrogen/progestogen Receptor
SR 19881 is a full agonist of ERRγ(EC50 value of 0.39 μM in a binding assay and an EC50 value of 4.7 μM in a cell-based assay).
T39710 ARV-471 Vepdegestrant Estrogen Receptor/ERR
ARV-471 (Vepdegestrant) is a orally active Cereblon -based estrogen receptor (ER) PROTAC degrader. ARV-471 is developed for the research of breast cancer.
T16566 Propyl pyrazole triol PPT Estrogen Receptor/ERR , Estrogen/progestogen Receptor
Propyl pyrazole triol (PPT) is a selective agonist of estrogen receptor alpha. The relative binding affinity of Propyl pyrazole triol for ERα (ERα: 49%) around 410 times higher compared with estrogen receptor beta (ERβ: ...
T0593 XCT790 Estrogen Receptor/ERR , Estrogen/progestogen Receptor , Autophagy
XCT790 is a potent, selective and inverse agonist of estrogen-related receptor alpha(ERRα).
T7644 DPN Diarylpropionitrile Apoptosis , Estrogen Receptor/ERR , Estrogen/progestogen Receptor , Autophagy
DPN (Diarylpropionitrile) is an selective agonist of estrogen receptor β (ERβ) .
T15364 G-1 Estrogen Receptor/ERR , GPR
G-1 is a nonsteroidal, high-affinity and selective GPR30 agonist (Ki: 11 nM).
T7389 G15 Estrogen Receptor/ERR
G15 is a cell-permeable non-steroidal antagonist of GPER (Ki = 20 nM)
T3958 WAY-200070 WAY 200070 Estrogen Receptor/ERR , Estrogen/progestogen Receptor
WAY-200070 is a specific agonist of estrogen receptor β (ERRβ, IC50: 2.3 nM).
T14987 CMP8 Estrogen Receptor/ERR , Estrogen/progestogen Receptor
CMP8 is a selective ligand for estrogen receptor. CMP8 binds to the mutant estrogen receptor ligand binding domain (ERLBD). CMP8 has IC50 values of 29 nM , 41 nM, 1100 nM and 2200 nM for MGERα, MGRERα, hERα and hERβ, res...
T3975 AZD9496 Estrogen Receptor/ERR , Estrogen/progestogen Receptor
AZD9496 is an orally available selective estrogen receptor(ERα) antagonist, with potential antineoplastic activity.
T5531 GSK-4716 Estrogen Receptor/ERR
GSK4716 is an ERRβ/γ agonist (IC50 = 2 µM) that can activate the receptor with similar potency as the protein ligand
T6533 Hexestrol Bibenzyl,Hexanoestrol,meso-Hexestrol,Hexestrofen Estrogen Receptor/ERR , Estrogen/progestogen Receptor
Hexestrol (Hexanoestrol) binds to ERα and ERβ with EC50 of 0.07 nM and 0.175 nM, respectively.
T20625 Prochloraz Sporgon,Prelude Estrogen Receptor/ERR , AhR , Androgen Receptor , Antifungal
Prochloraz (Prelude) is a broad-spectrum contact imidazole fungicide. Prochloraz inhibits human placental microsomal aromatase in vitro (IC50 = 40 nM). Prochloraz also acts as an estrogen receptor (IC50s = 25 μM) and and...
T1216 Diethylstilbestrol Stilbestrol,DES Estrogen Receptor/ERR , Estrogen/progestogen Receptor
Diethylstilbestrol (DES) is used in the treatment of menopausal and postmenopausal disorders.
T8370 GSK5182 Estrogen Receptor/ERR , Estrogen/progestogen Receptor , Reactive Oxygen Species
GSK5182 is a highly selective inverse estrogen-related receptor γ agonist (IC50 : 79 nM)
T13443 (R)-Equol (+)-Equol Estrogen/progestogen Receptor
(R)-Equol ((+)-Equol) is an ERα and ERβ agonist with Kis of 27.4 and 15.4 nM, respectively.
T6306 Erteberel LY500307 Estrogen Receptor/ERR , Estrogen/progestogen Receptor
Erteberel (LY500307) is a potent, selective estrogen receptor β agonist with EC50 of 0.66 nM, 32-fold selectivity against estrogen receptor α. Phase 2.
T5633 H3B-5942 Estrogen Receptor/ERR , Estrogen/progestogen Receptor
H3B-5942 belongs to a class of ERα antagonists referred to as selective estrogen receptor covalent antagonists (SERCA).
T6620 Ospemifene FC-1271a Estrogen Receptor/ERR , Estrogen/progestogen Receptor
Ospemifene (FC-1271a) is a new selective non-hormonal estrogen receptor modulator (SERM) that is used for the treatment of moderate to severe dyspareunia, a symptom of vulvar and vaginal atrophy, due to menopause. FDA ap...
T2567 Etonogestrel 3-Oxodesogestrel,3-keto-Desogestrel,Nexplanon,Implanon Estrogen Receptor/ERR , Estrogen/progestogen Receptor , Progesterone Receptor , Endogenous Metabolite
Etonogestrel (Implanon) is a steroidal progestin used as hormonal contraceptives.
T13674 Elacestrant RAD1901 Estrogen Receptor/ERR , Estrogen/progestogen Receptor
Elacestrant (RAD1901) with IC50s of 48 and 870 nM for ERα and ERβ, respectively.Elacestrant  is an orally available selective estrogen receptor degrader .
T0168 Estradiol (cypionate) Depofemin,Estradiol cypionate Estrogen Receptor/ERR , Estrogen/progestogen Receptor
Estradiol cypionate (Depofemin), the 17 β-cyclopentylpropinate ester of estradiol, inhibits ET-1 synthesis via estrogen receptor.
T13507 4,4'-Iminodiphenol Leucoindophenol Estrogen/progestogen Receptor
4,4'-Iminodiphenol (Leucoindophenol) is an inactive estrogen receptor ligand with a diphenylamine backbone.
T0035 Dienestrol Restrol,Dehydrostilbestrol,Dienoestrol,Cycladiene Estrogen Receptor/ERR , Estrogen/progestogen Receptor
Dienestrol (Restrol) is a synthetic and nonsteroidal estrogen, which is an estrogen receptor agonist. Estrogens can increase a normal clear discharge from the vagina and make the vulva and urethra healthy.
T0384 Estradiol benzoate Benzoestrofol,Benzhormovarine,Benovocylin Estrogen Receptor/ERR , Estrogen/progestogen Receptor
Estradiol benzoate (Benzhormovarine) is the synthetic benzoate ester of estradiol, a steroid sex hormone vital to the maintenance of fertility and secondary sexual characteristics in females.
T7556 Fadrozole hydrochloride CGS 16949A Aromatase
Fadrozole hydrochloride (CGS 16949A) is a model aromatase inhibitor that has been shown to suppress estrogen production in the ovaries of fish.
T7313 Enclomiphene citrate Enclomifene citrate,(E)-Clomiphene citrate,trans-Clomiphene citrate Estrogen Receptor/ERR
Enclomiphene citrate (trans-Clomiphene citrate) is a non-steroidal estrogen receptor antagonist,with antioestrogenic property
T4420 4-Hydroxytamoxifen ICI 79280,(Z)-4-hydroxy Tamoxifen,trans-4-Hydroxytamoxifen Estrogen Receptor/ERR , Estrogen/progestogen Receptor
4-Hydroxytamoxifen (ICI 79280) is the active metabolite of Tamoxifen, an estrogen receptor modulator (SERM) with selective and oral potency. 4-Hydroxytamoxifen has antitumor activity and may be used in breast cancer rese...
T11399 Giredestrant GDC-9545 Estrogen Receptor/ERR , Estrogen/progestogen Receptor
Giredestrant (GDC-9545) potently competes with estradiol for binding and induces a conformational change within the ER ligand binding domain. Giredestrant has anti-tumor activity. Giredestrant, a non-steroidal ER ligand,...

Compounds

Estrogen receptor modulator 1
T15249
Synonym:
Target: Estrogen Receptor/ERR
Estrogen receptor antagonist 8
T78646
Synonym:
Target: Estrogen Receptor/ERR
Camizestrant
T11237
Synonym: Estrogen receptor antagonist 2
Target: Estrogen Receptor/ERR
Giredestrant tartrate
T11236
Synonym: Estrogen receptor antagonist 1
Target: Estrogen Receptor/ERR, Others
Estrogen receptor modulator 6
T40893
Synonym:
Target:
Conjugated Estrogen sodium
T19988
Synonym: Conjugated estrogens,Conest,HSDB 3076,Kestrin,Estrogens, conjugated,TAG-39
Target:
Estrogen receptor antagonist 2
T63277
Synonym:
Target:
Estrogen receptor antagonist 3
T63914
Synonym:
Target:
Estrogen receptor antagonist 4
T63106
Synonym:
Target:
Estrogen receptor modulator 8
T79109
Synonym:
Target: Estrogen Receptor/ERR
Estrogen receptor antagonist 5
T62952
Synonym:
Target:
Estrogen receptor antagonist 1
T63582
Synonym:
Target:
Estrogen receptor modulator 7
T79064
Synonym:
Target: Estrogen Receptor/ERR
Estrogen receptor-IN-1
T60293
Synonym:
Target:
Estrogen receptor antagonist 6
T62953
Synonym:
Target:
Estrogen receptor antagonist 7
T61909
Synonym:
Target:
Estrogen receptor modulator 10
T82439
Synonym:
Target: Estrogen Receptor/ERR
Estrogen receptor β antagonist 2
T62311
Synonym:
Target:
Estrogen receptor α antagonist 1
T62764
Synonym:
Target:
PHTPP
T4388
Synonym:
Target: Estrogen Receptor/ERR, Estrogen/progestogen Receptor
FLTX1
T8984
Synonym:
Target: Estrogen Receptor/ERR, Estrogen/progestogen Receptor
SR 19881
T7904
Synonym:
Target: Estrogen/progestogen Receptor
ARV-471
T39710
Synonym: Vepdegestrant
Target: Estrogen Receptor/ERR
Propyl pyrazole triol
T16566
Synonym: PPT
Target: Estrogen Receptor/ERR, Estrogen/progestogen Receptor
XCT790
T0593
Synonym:
Target: Estrogen Receptor/ERR, Estrogen/progestogen Receptor, Autophagy
DPN
T7644
Synonym: Diarylpropionitrile
Target: Apoptosis, Estrogen Receptor/ERR, Estrogen/progestogen Receptor, Autophagy
G-1
T15364
Synonym:
Target: Estrogen Receptor/ERR, GPR
G15
T7389
Synonym:
Target: Estrogen Receptor/ERR
WAY-200070
T3958
Synonym: WAY 200070
Target: Estrogen Receptor/ERR, Estrogen/progestogen Receptor
CMP8
T14987
Synonym:
Target: Estrogen Receptor/ERR, Estrogen/progestogen Receptor
AZD9496
T3975
Synonym:
Target: Estrogen Receptor/ERR, Estrogen/progestogen Receptor
GSK-4716
T5531
Synonym:
Target: Estrogen Receptor/ERR
Hexestrol
T6533
Synonym: Bibenzyl,Hexanoestrol,meso-Hexestrol,Hexestrofen
Target: Estrogen Receptor/ERR, Estrogen/progestogen Receptor
Prochloraz
T20625
Synonym: Sporgon,Prelude
Target: Estrogen Receptor/ERR, AhR, Androgen Receptor, Antifungal
Diethylstilbestrol
T1216
Synonym: Stilbestrol,DES
Target: Estrogen Receptor/ERR, Estrogen/progestogen Receptor
GSK5182
T8370
Synonym:
Target: Estrogen Receptor/ERR, Estrogen/progestogen Receptor, Reactive Oxygen Species
(R)-Equol
T13443
Synonym: (+)-Equol
Target: Estrogen/progestogen Receptor
Erteberel
T6306
Synonym: LY500307
Target: Estrogen Receptor/ERR, Estrogen/progestogen Receptor
H3B-5942
T5633
Synonym:
Target: Estrogen Receptor/ERR, Estrogen/progestogen Receptor
Ospemifene
T6620
Synonym: FC-1271a
Target: Estrogen Receptor/ERR, Estrogen/progestogen Receptor
Etonogestrel
T2567
Synonym: 3-Oxodesogestrel,3-keto-Desogestrel,Nexplanon,Implanon
Target: Estrogen Receptor/ERR, Estrogen/progestogen Receptor, Progesterone Receptor, Endogenous Metabolite
Elacestrant
T13674
Synonym: RAD1901
Target: Estrogen Receptor/ERR, Estrogen/progestogen Receptor
Estradiol (cypionate)
T0168
Synonym: Depofemin,Estradiol cypionate
Target: Estrogen Receptor/ERR, Estrogen/progestogen Receptor
4,4'-Iminodiphenol
T13507
Synonym: Leucoindophenol
Target: Estrogen/progestogen Receptor
Dienestrol
T0035
Synonym: Restrol,Dehydrostilbestrol,Dienoestrol,Cycladiene
Target: Estrogen Receptor/ERR, Estrogen/progestogen Receptor
Estradiol benzoate
T0384
Synonym: Benzoestrofol,Benzhormovarine,Benovocylin
Target: Estrogen Receptor/ERR, Estrogen/progestogen Receptor
Fadrozole hydrochloride
T7556
Synonym: CGS 16949A
Target: Aromatase
Enclomiphene citrate
T7313
Synonym: Enclomifene citrate,(E)-Clomiphene citrate,trans-Clomiphene citrate
Target: Estrogen Receptor/ERR
4-Hydroxytamoxifen
T4420
Synonym: ICI 79280,(Z)-4-hydroxy Tamoxifen,trans-4-Hydroxytamoxifen
Target: Estrogen Receptor/ERR, Estrogen/progestogen Receptor
Giredestrant
T11399
Synonym: GDC-9545
Target: Estrogen Receptor/ERR, Estrogen/progestogen Receptor
1 2 3 4 5 6
Cat No. Product Name Synonyms Targets
TN1052 Lindleyin Estrogen Receptor/ERR , Estrogen/progestogen Receptor
Lindleyin is a novel phytoestrogen and might trigger many of the biological responses evoked by the physiological estrogens.
T13768 (+)-Medicarpin Estrogen/progestogen Receptor
(+)-Medicarpin, a pterocarpan, is an isoflavonoid compound derived from multiple medicinal plant species such as Sophora japonica, Zollernia paraensis, Platymiscium yucatamun, Machaerium aristulatum, and Platymiscium flo...
T5S0543 Isocurcumenol Apoptosis , Estrogen Receptor/ERR , Reductase
1. Isocurcumenol inhibits 5α-reductase which converts testosterone to dihydrotestosterone (DHT).
T0301 Ethisterone 17α-Ethynyltestosterone,Pregneninolone Estrogen Receptor/ERR , Estrogen/progestogen Receptor
Ethisterone (17α-Ethynyltestosterone) is a progestogen hormone.
T3665 Tectoridin Shekanin Estrogen Receptor/ERR , Reductase
Tectoridin (Shekanin) possesses an estrogenic and thyroid hormone-like agent by activating estrogen and thyroid hormone receptors. Tectoridin has anti-oxidant, anti-inflammatory and hypoglycemic activities; Tectoridin an...
T3855 Tracheloside Estrogen Receptor/ERR , Phosphorylase
Tracheloside significantly decreases the activity of alkaline phosphatase (IC50: 0.31 μg/ml), a level of inhibition comparable to that of tamoxifen (IC50: 0.43 μg/ml).
TQ0295 Coumestrol Estrogen Receptor/ERR
Coumestrol that existed in soybean products suppresses the proliferation of ES2 cells (IC50: 50 μM). It exhibits activities against neurological disorders, cancers and autoimmune diseases.
T13542 α-Zearalenol Estrogen Receptor/ERR
α-Zearalenol is one of the major metabolites of Zearalenone. α-Zearalenol has structural analogy to estrogen, thus α-Zearalenol can bind to estrogen receptors (ERs).
T3325 Liquiritigenin 4',7-Dihydroxyflavanone Estrogen Receptor/ERR , Estrogen/progestogen Receptor
Liquiritigenin (4',7-Dihydroxyflavanone), a flavonoid aglycone from licorice, is a highly selective estrogen receptor β (ERβ) agonist.
T3913 Saikosaponin D Estrogen Receptor/ERR , NF-κB , Antibacterial , STAT
Saikosaponin D is a novel SERCA inhibitor by inhibiting NF-κB and STAT3 signaling to protect against acetaminophen-induced hepatotoxicity.
T3846 Bavachin Corylifolin Estrogen Receptor/ERR , Estrogen/progestogen Receptor
Bavachin (Corylifolin) is a phytoestrogen that activates the estrogen receptors ERα and ERβ.
T1590 Letrozole CGS 20267 Aromatase , Autophagy
Letrozole (CGS 20267) is an Aromatase Inhibitor. The mechanism of action of letrozole is as an Aromatase Inhibitor.
T4000 (±)-Equol Equol,(R,S)-Equol Estrogen Receptor/ERR , Estrogen/progestogen Receptor , Drug Metabolite
(±)-Equol ((R,S)-Equol) is a non-steroidal estrogen produced from the metabolism of the isoflavonoid phytoestrogen daidzen by human intestinal microflora. The estrogen receptor (ER) agonist activity of the naturally occu...
TMA1644 Segetalin B Estrogen Receptor/ERR
Segetalin B is a natural product from Vaccaria segetalis (Neck.) Garcke, has estrogen-like activity.
T1009 Estrone Oestrone,Fluoroethyl,Aquacrine Estrogen Receptor/ERR , Estrogen/progestogen Receptor , Endogenous Metabolite
Estrone (Aquacrine) is an aromatized C18 steroid with a 3-hydroxyl group and a 17-ketone, a major mammalian estrogen. It is converted from ANDROSTENEDIONE directly, or from TESTOSTERONE via ESTRADIOL. In humans, it is pr...
T1571 Estriol NSC-12169,Oestriol Estrogen Receptor/ERR , Estrogen/progestogen Receptor , MRP , Endogenous Metabolite
Estriol (Oestriol) is a hydroxylated metabolite of ESTRADIOL or ESTRONE that has a hydroxyl group at C3, 16-alpha, and 17-beta position. Estriol is a major urinary estrogen. During PREGNANCY, a large amount of estriol is...
T3840 Dihydroresveratrol 3,4',5-Trihydroxybibenzyl Estrogen Receptor/ERR , Others
Dihydroresveratrol (3,4',5-Trihydroxybibenzyl) is a major metabolite of resveratrol that is produced by animal-associated bacteria, including the gut microbiota. Dihydroresveratrol and dihydroresveratrol monosulfate are ...
T1048 Estradiol E2,17β-Estradiol,17β-Oestradiol,β-Estradiol Estrogen Receptor/ERR , Estrogen/progestogen Receptor , Endogenous Metabolite
Estradiol (E2) is a naturally occurring steroidal sex hormone that is essential for female fertility and maintenance of secondary sexual characteristics. Estradiol upregulates IL-6 expression through estrogen receptor be...
T3385 Gypenoside XVII GP-17,Gynosaponin S Estrogen Receptor/ERR , GSK-3 , Endogenous Metabolite
Gypenoside XVII (Gynosaponin S) confers protection against Aβ25-35-induced neurotoxicity through estrogen receptor-dependent activation of PI3K/Akt pathways, activation of Nrf2/ARE/HO-1 and inactivation of GSK-3β pathway...
T36857 Estrone sulfate sodium Estrone 3-sulfate (sodium salt),17β-Estrone 3-sulfate Endogenous Metabolite
Estrone sulfate sodium (17β-Estrone 3-sulfate) is an endogenous steroid and an estrogen ester that is biologically inactive. It is converted by steroid sulfatase into estrone . Estrone sulfate sodium has been investigate...
T0760 Cholesterol Cholesterin,Cholesteryl alcohol Estrogen Receptor/ERR , MRP , Endogenous Metabolite , ROR
Cholesterol (cholesteryl alcohol) is a natural product that is the major sterol in mammals and an agonist of estrogen-related receptor α (ERRα). Cholesterol is widely found in the cell membranes of animals and is also us...
T2177 Kaempferol Kempferol,Robigenin Apoptosis , Estrogen Receptor/ERR , Mitophagy , Estrogen/progestogen Receptor , HIV Protease , Endogenous Metabolite , Parasite , Autophagy
Kaempferol (Robigenin) is a natural flavonoid and an inverse agonist of ERRα and ERRγ. Kaempferol has a wide range of antitumor, anti-inflammatory, antioxidant, antibacterial and antiviral activities.
T2837 Chrysin 5, 7-Dihydroxyflavone,NSC 407436,5,7-Dihydroxyflavone Estrogen Receptor/ERR , Antioxidant
Chrysin (5,7-Dihydroxyflavone) exhibits many biological activities and pharmacological effects, including antioxidant, anti-inflammatory, anticancer, and antiviral activities.
T6491 (-)-(S)-Equol (−)-Equol,Equol,4',7-Dihydroxyisoflavan,4',7-Isoflavandiol Estrogen Receptor/ERR , Estrogen/progestogen Receptor , Endogenous Metabolite
(-)-(S)-Equol (4',7-Dihydroxyisoflavan) is an orally bioavailable, non-steroidal estrogen naturally produced by the metabolism of the isoflavonoid daidzein by human intestinal microflora, with potential chemoprotective a...
T1424 Ethynyl estradiol 17α-Ethynylestradiol,Ethinyl Estradiol Estrogen Receptor/ERR , Estrogen/progestogen Receptor , Endogenous Metabolite
Ethynyl estradiol is a semisynthetic alkylated ESTRADIOL with a 17-alpha-ethinyl substitution. It has high estrogenic potency when administered orally, and is often used as the estrogenic component in ORAL CONTRACEPTIVES...
TQ0274 27-Hydroxycholesterol 25(R)-27-hydroxy Cholesterol Estrogen/progestogen Receptor , Liver X Receptor
27-Hydroxycholesterol (25(R)-27-hydroxy Cholesterol) is a selective modulator of estrogen receptor and an agonist of the liver X receptor.
T0345 Estropipate Piperazine estrone sulfate,Pipestrone,Estrone sulfate piperazine salt Estrogen Receptor/ERR , Estrogen/progestogen Receptor
Estropipate (Piperazine estrone sulfate) is a natural estrogenic substance composed of estrone sulfate and piperazine.
T2810 (20S)-Protopanaxatriol 20(S)-APPT,g-PPT Apoptosis , Estrogen Receptor/ERR , Glucocorticoid Receptor , Estrogen/progestogen Receptor , Liver X Receptor
(20S)-Protopanaxatriol (g-PPT)(g-PPT), a metabolite of ginsenoside, could regulate endothelial cell functions through the estrogen receptor and glucocorticoid receptor.
T3806 Kaempferide Kaempferol 4'-O-methyl ether,Kaempferol 4'-methyl ether,4'-Methylkaempferol,4'-O-Methylkaempferol Estrogen Receptor/ERR , Estrogen/progestogen Receptor , Influenza Virus , Antibacterial , Autophagy
kaempferide (4'-Methylkaempferol) inhibits the proliferation of native and estrogen receptor beta overexpressing colon cancer cells through a mechanism not mediated by ligand binding dependent estrogen receptor activatio...
T1549 Raloxifene hydrochloride LY156758 hydrochloride,Raloxifene HCl,LY139481 hydrochloride,Keoxifene hydrochloride,LY156758 (Keoxifene) HCl Estrogen Receptor/ERR , Others , MAO , Estrogen/progestogen Receptor , Autophagy
Raloxifene hydrochloride (LY156758 hydrochloride) is a second generation selective estrogen receptor modulator (SERM) used to prevent osteoporosis in postmenopausal women. It has estrogen agonist effects on bone and chol...
T2882 Genistin Genistoside,Genistein glucoside,Genistein 7-glucoside,Genistine,Genistein 7-O-β-D-glucopyranoside Apoptosis , Estrogen Receptor/ERR , Others
Genistin (Genistoside) is the major isoflavonoid of soybeans and soy products.It has been reported to possess various therapeutic effects, including anti-inflammatory and anticancer activities
T7299 β-Estradiol 17-acetate beta-estradiol 17-acetate,1,3,5(10)-Estratriene-3,17β-diol 17-acetate Estrogen Receptor/ERR , Others
β-Estradiol 17-acetate (1,3,5(10)-Estratriene-3,17β-diol 17-acetate) is a metabolite of estradiol.
TN1719 Gymnestrogenin Liver X Receptor
Gymnestrogenin has a dual LXRα±/α2 antagonistic profile.
T0419 Testosterone propionate Others , Androgen Receptor , Transferase
Testosterone Propionate is a short acting oil-based injectable formulation of testosterone. Testosterone inhibits gonadotropin secretion from the pituitary gland and ablates estrogen production in the ovaries, thereby de...
T13481 2-Methoxyestrone Endogenous Metabolite
2-Methoxyestrone is a methoxylated catechol estrogen and metabolite of estrone (pKa: 10.81).
T36857L Premarin Estrone 3-sulfate,Estrone sulfate Estrogen Receptor/ERR
Premarin (Estrone 3-sulfate) is an an estrogen sulfate with neuroprotective actions during traumatic brain injury.
T15248 Estetrol Donesta Estrogen Receptor/ERR , Endogenous Metabolite
Estetrol(Donesta) is an orally available, selective modulator of the estrogen receptor, a naturally occurring estrogen synthesized by the human fetal liver during pregnancy.Estetrol has effects on the endometrium or cent...
TN2197 Secoisolariciresinol TNF
Secoisolariciresinol is an enterolignan precursor, it has antioxidant, and estrogen-like activities, it can significantly suppress triglyceride (TG) accumulation in 3T3-L1 adipocytes.
T3378 Alpha-Estradiol Alfatradiol,17α-Estradiol,Epiestrol,Epiestradiol Estrogen/progestogen Receptor , Reductase , Endogenous Metabolite
Alpha-Estradiol (Epiestradiol) is an estrogen that inhibits 5alpha-reductase and has potential in the study of androgenetic alopecia.
T73772 Estrone sulfate potassium Endogenous Metabolite
Estrone sulfate potassium is an estrogen ester and conjugate, a natural endogenous steroid.
TN1148 Isopsoralenoside Estrogen Receptor/ERR , Estrogen/progestogen Receptor , Antibacterial
Isopsoralenoside shows estrogen-like, osteoblastic proliferation accelerating, antitumor, and antibacterial effects.
T16338 Norgestimate metabolite Norelgestromin 17-Deacetyl norgestimate,17-Deacylnorgestimate Drug Metabolite
Norgestimate metabolite Norelgestromin (17-Deacylnorgestimate) is one of the active metabolites of norgestimate.It is a steroidal progestin used in contraceptive patches, where it is combined with the estrogen ethinyl es...
T16525 PhIP Others
PhIP is a heterocyclic aromatic amine (HAA) from cooked meat. It belongs to pyridine heterocyclic amine and is a 2B carcinogen with estrogen activity. PhIP forms adducts with DNA that promote cancer.
TN1008 Psoralenoside CaMK , Calcium Channel , Histamine Receptor
Psoralenoside is a natural product isolated from the fruits of Psoralea corylifolia, shows estrogen-like activity, osteoblastic proliferation accelerating activity, antitumor effects and antibacterial activity.
T2777 Ginsenoside Rg1 Sanchinoside C1,Panaxoside Rg1,Sanchinoside Rg1,Panaxoside A,Ginsenoside A2 Apoptosis , Beta Amyloid , NF-κB
Ginsenoside Rg1 (Panaxoside Rg1) is a class of steroid glycosides, and triterpene saponins found exclusively in the plant genus Panax (ginseng). It improves spatial learning and increase hippocampal synaptophysin level i...
TN1702 Glycycoumarin P450 , JNK , AMPK , Autophagy
Glycycoumarin is an estrogen agonist, it shows moderate inhibitory effects against CYP1A2 and CYP2B6.
TN1918 Medicarpin Apoptosis , BCL , ROS , JNK
Medicarpin, a legume phytoalexin, acts as an estrogen receptor (ER) agonist, can stimulate osteoblast differentiation likely via ERα², promote achievement of peak bone mass, and is devoid of uterine estrogenicity; in add...
T3717 Hinokitiol 4-Isopropyltropolone,β-thujaplicin DNA Methyltransferase , Virus Protease , Estrogen/progestogen Receptor , Nrf2
Hinokitiol (4-Isopropyltropolone) can inhibit ultraviolet B-induced apoptosis in keratinocytes and strongly suggest that the inhibitory mechanism is due to the antioxidant activity of metallothionein induced by the agent...
T3923 Calycosin Cyclosin,3'-Hydroxyformononetin Apoptosis , Tyrosinase
Calycosin (Cyclosin) acts as a selective estrogen receptor modulator. Calycosin induces apoptosis in human ovarian cancer SKOV3 cells by activating caspases and Bcl-2 family proteins. Calycosin suppresses breast cancer c...
T1660 Silibinin Silibinin A,Silybin,Silymarin I Reactive Oxygen Species , Autophagy
Silibinin (Silybin) is the major active constituent of silymarin, a standardized extract of the milk thistle seeds, containing a mixture of flavonolignans consisting of silibinin, isosilibinin, silicristin, silidianin an...
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Natural Products

Lindleyin
TN1052
Synonym:
Target: Estrogen Receptor/ERR, Estrogen/progestogen Receptor
(+)-Medicarpin
T13768
Synonym:
Target: Estrogen/progestogen Receptor
Isocurcumenol
T5S0543
Synonym:
Target: Apoptosis, Estrogen Receptor/ERR, Reductase
Ethisterone
T0301
Synonym: 17α-Ethynyltestosterone,Pregneninolone
Target: Estrogen Receptor/ERR, Estrogen/progestogen Receptor
Tectoridin
T3665
Synonym: Shekanin
Target: Estrogen Receptor/ERR, Reductase
Tracheloside
T3855
Synonym:
Target: Estrogen Receptor/ERR, Phosphorylase
Coumestrol
TQ0295
Synonym:
Target: Estrogen Receptor/ERR
α-Zearalenol
T13542
Synonym:
Target: Estrogen Receptor/ERR
Liquiritigenin
T3325
Synonym: 4',7-Dihydroxyflavanone
Target: Estrogen Receptor/ERR, Estrogen/progestogen Receptor
Saikosaponin D
T3913
Synonym:
Target: Estrogen Receptor/ERR, NF-κB, Antibacterial, STAT
Bavachin
T3846
Synonym: Corylifolin
Target: Estrogen Receptor/ERR, Estrogen/progestogen Receptor
Letrozole
T1590
Synonym: CGS 20267
Target: Aromatase, Autophagy
(±)-Equol
T4000
Synonym: Equol,(R,S)-Equol
Target: Estrogen Receptor/ERR, Estrogen/progestogen Receptor, Drug Metabolite
Segetalin B
TMA1644
Synonym:
Target: Estrogen Receptor/ERR
Estrone
T1009
Synonym: Oestrone,Fluoroethyl,Aquacrine
Target: Estrogen Receptor/ERR, Estrogen/progestogen Receptor, Endogenous Metabolite
Estriol
T1571
Synonym: NSC-12169,Oestriol
Target: Estrogen Receptor/ERR, Estrogen/progestogen Receptor, MRP, Endogenous Metabolite
Dihydroresveratrol
T3840
Synonym: 3,4',5-Trihydroxybibenzyl
Target: Estrogen Receptor/ERR, Others
Estradiol
T1048
Synonym: E2,17β-Estradiol,17β-Oestradiol,β-Estradiol
Target: Estrogen Receptor/ERR, Estrogen/progestogen Receptor, Endogenous Metabolite
Gypenoside XVII
T3385
Synonym: GP-17,Gynosaponin S
Target: Estrogen Receptor/ERR, GSK-3, Endogenous Metabolite
Estrone sulfate sodium
T36857
Synonym: Estrone 3-sulfate (sodium salt),17β-Estrone 3-sulfate
Target: Endogenous Metabolite
Cholesterol
T0760
Synonym: Cholesterin,Cholesteryl alcohol
Target: Estrogen Receptor/ERR, MRP, Endogenous Metabolite, ROR
Kaempferol
T2177
Synonym: Kempferol,Robigenin
Target: Apoptosis, Estrogen Receptor/ERR, Mitophagy, Estrogen/progestogen Receptor, HIV Protease, Endogenous Metabolite, Parasite, Autophagy
Chrysin
T2837
Synonym: 5, 7-Dihydroxyflavone,NSC 407436,5,7-Dihydroxyflavone
Target: Estrogen Receptor/ERR, Antioxidant
(-)-(S)-Equol
T6491
Synonym: (−)-Equol,Equol,4',7-Dihydroxyisoflavan,4',7-Isoflavandiol
Target: Estrogen Receptor/ERR, Estrogen/progestogen Receptor, Endogenous Metabolite
Ethynyl estradiol
T1424
Synonym: 17α-Ethynylestradiol,Ethinyl Estradiol
Target: Estrogen Receptor/ERR, Estrogen/progestogen Receptor, Endogenous Metabolite
27-Hydroxycholesterol
TQ0274
Synonym: 25(R)-27-hydroxy Cholesterol
Target: Estrogen/progestogen Receptor, Liver X Receptor
Estropipate
T0345
Synonym: Piperazine estrone sulfate,Pipestrone,Estrone sulfate piperazine salt
Target: Estrogen Receptor/ERR, Estrogen/progestogen Receptor
(20S)-Protopanaxatriol
T2810
Synonym: 20(S)-APPT,g-PPT
Target: Apoptosis, Estrogen Receptor/ERR, Glucocorticoid Receptor, Estrogen/progestogen Receptor, Liver X Receptor
kaempferide
T3806
Synonym: Kaempferol 4'-O-methyl ether,Kaempferol 4'-methyl ether,4'-Methylkaempferol,4'-O-Methylkaempferol
Target: Estrogen Receptor/ERR, Estrogen/progestogen Receptor, Influenza Virus, Antibacterial, Autophagy
Raloxifene hydrochloride
T1549
Synonym: LY156758 hydrochloride,Raloxifene HCl,LY139481 hydrochloride,Keoxifene hydrochloride,LY156758 (Keoxifene) HCl
Target: Estrogen Receptor/ERR, Others, MAO, Estrogen/progestogen Receptor, Autophagy
Genistin
T2882
Synonym: Genistoside,Genistein glucoside,Genistein 7-glucoside,Genistine,Genistein 7-O-β-D-glucopyranoside
Target: Apoptosis, Estrogen Receptor/ERR, Others
β-Estradiol 17-acetate
T7299
Synonym: beta-estradiol 17-acetate,1,3,5(10)-Estratriene-3,17β-diol 17-acetate
Target: Estrogen Receptor/ERR, Others
Gymnestrogenin
TN1719
Synonym:
Target: Liver X Receptor
Testosterone propionate
T0419
Synonym:
Target: Others, Androgen Receptor, Transferase
2-Methoxyestrone
T13481
Synonym:
Target: Endogenous Metabolite
Premarin
T36857L
Synonym: Estrone 3-sulfate,Estrone sulfate
Target: Estrogen Receptor/ERR
Estetrol
T15248
Synonym: Donesta
Target: Estrogen Receptor/ERR, Endogenous Metabolite
Secoisolariciresinol
TN2197
Synonym:
Target: TNF
Alpha-Estradiol
T3378
Synonym: Alfatradiol,17α-Estradiol,Epiestrol,Epiestradiol
Target: Estrogen/progestogen Receptor, Reductase, Endogenous Metabolite
Estrone sulfate potassium
T73772
Synonym:
Target: Endogenous Metabolite
Isopsoralenoside
TN1148
Synonym:
Target: Estrogen Receptor/ERR, Estrogen/progestogen Receptor, Antibacterial
Norgestimate metabolite Norelgestromin
T16338
Synonym: 17-Deacetyl norgestimate,17-Deacylnorgestimate
Target: Drug Metabolite
PhIP
T16525
Synonym:
Target: Others
Psoralenoside
TN1008
Synonym:
Target: CaMK, Calcium Channel, Histamine Receptor
Ginsenoside Rg1
T2777
Synonym: Sanchinoside C1,Panaxoside Rg1,Sanchinoside Rg1,Panaxoside A,Ginsenoside A2
Target: Apoptosis, Beta Amyloid, NF-κB
Glycycoumarin
TN1702
Synonym:
Target: P450, JNK, AMPK, Autophagy
Medicarpin
TN1918
Synonym:
Target: Apoptosis, BCL, ROS, JNK
Hinokitiol
T3717
Synonym: 4-Isopropyltropolone,β-thujaplicin
Target: DNA Methyltransferase, Virus Protease, Estrogen/progestogen Receptor, Nrf2
Calycosin
T3923
Synonym: Cyclosin,3'-Hydroxyformononetin
Target: Apoptosis, Tyrosinase
Silibinin
T1660
Synonym: Silibinin A,Silybin,Silymarin I
Target: Reactive Oxygen Species, Autophagy
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Recombinant Proteins

Species：
Human (24)
Bovine (2)
Mouse (2)
Canine (1)
Cynomolgus (1)
Rhesus (1)
Expression System：
E. coli (13)
HEK293 (10)
Human Cells (3)
Yeast (3)
Baculovirus-Insect Cells (2)
Tag：
His (8)
N-terminal 6xHis-tagged (5)
Tag Free (5)
hFc (3)
C-6His (2)
C-10His (1)
C-6His,N-T7 tag (1)
C-terminal mFc-tagged (1)
GST (1)
N-6His (1)
Cat No. Product Name Species Expression System
TMPJ-00762 ER alpha Protein, Human, Recombinant (His) Human E. coli
Estrogen Receptor is a major ligand-activated transcription factor belonging to the nuclear hormone receptor superfamily. Estrogen Receptor is composed of several domains important for hormone binding, DNA binding, and a...
TMPY-03496 EBAG9 Protein, Human, Recombinant (His) Human E. coli
RCAS1, also known as EBAG9, is a tumor-associated antigen that is expressed at high frequency in a variety of cancers. RCAS1 gene was identified as an estrogen-responsive gene. Regulation of transcription by estrogen ...
TMPH-00956 Aromatase/CYP19A1 Protein, Human, Recombinant (His) Human E. coli
Aromatase/CYP19A1 Protein, Human, Recombinant (His) is expressed in E. coli.
TMPY-04396 C-ABL/ABL1 Protein, Human, Recombinant (GST) Human Baculovirus-Insect Cells
c-Abl belongs to the class of tyrosine kinases and is the prototype of a subfamily which includes two members, c-Abl and Arg (Abl-related gene). Both proteins are localized at the cell membrane, actin cytoskeleton and cy...
TMPY-00472 IL-8/CXCL8 Protein, Human, Recombinant (aa 28-99) Human E. coli
Interleukin 8 (IL-8), also known as CXCL8, which is a chemokine with a defining CXC amino acid motif that was initially characterized for its leukocyte chemotactic activity, is now known to possess tumorigenic and proang...
TMPY-04726 IL-8/CXCL8 Protein, Human, Recombinant (His) Human Yeast
Interleukin 8 (IL-8), also known as CXCL8, which is a chemokine with a defining CXC amino acid motif that was initially characterized for its leukocyte chemotactic activity, is now known to possess tumorigenic and proang...
TMPY-00754 IL-8/CXCL8 Protein, Human, Recombinant (aa 23-99) Human HEK293
Interleukin 8 (IL-8), also known as CXCL8, which is a chemokine with a defining CXC amino acid motif that was initially characterized for its leukocyte chemotactic activity, is now known to possess tumorigenic and proang...
TMPJ-01192 ELAPOR1 Protein, Human, Recombinant (His) Human Human Cells
Endosome/lysosome-associated apoptosis and autophagy regulator (ELAPOR1), also known as EIG121 protein, is a type I transmembrane protein induced by estrogen. The estrogen-induced gene 121 (EIG121) has been associated wi...
TMPY-01660 SULT1E1 Protein, Human, Recombinant (His) Human E. coli
Estrogen sulfotransferase, also known as Sulfotransferase, estrogen-preferring, Sulfotransferase 1E1, SULT1E1 and ST1E1, is a cytoplasm enzyme that belongs to the sulfotransferase 1 family. Sulfotransferase enzymes catal...
TMPH-01305 ER beta Protein, Human, Recombinant (His) Human Yeast
Nuclear hormone receptor. Binds estrogens with an affinity similar to that of ESR1/ER-alpha, and activates expression of reporter genes containing estrogen response elements (ERE) in an estrogen-dependent manner.; Lacks ...
TMPH-01304 ER beta Protein, Human, Recombinant (E. coli, His) Human E. coli
Nuclear hormone receptor. Binds estrogens with an affinity similar to that of ESR1/ER-alpha, and activates expression of reporter genes containing estrogen response elements (ERE) in an estrogen-dependent manner.; Lacks ...
TMPH-01302 HSD17B1 Protein, Human, Recombinant (His & Myc) Human E. coli
Favors the reduction of estrogens and androgens. Converts estrone (E1) to a more potent estrogen, 17beta-estradiol (E2). Also has 20-alpha-HSD activity. Uses preferentially NADH.
TMPH-02851 PDIA2 Protein, Mouse, Recombinant (His & SUMO) Mouse E. coli
Acts as an intracellular estrogen-binding protein. May be involved in modulating cellular levels and biological functions of estrogens in the pancreas. May act as a chaperone that inhibits aggregation of misfolded protei...
TMPH-00279 Interferon tau-1/IFNT1 Protein, Bovine, Recombinant (His) Bovine Yeast
Paracrine hormone primarily responsible for maternal recognition of pregnancy. Interacts with endometrial receptors, probably type I interferon receptors, and blocks estrogen receptor expression, preventing the estrogen-...
TMPH-00278 Interferon tau-1/IFNT1 Protein, Bovine, Recombinant (E. coli, His) Bovine E. coli
Paracrine hormone primarily responsible for maternal recognition of pregnancy. Interacts with endometrial receptors, probably type I interferon receptors, and blocks estrogen receptor expression, preventing the estrogen-...
TMPY-04780 VMO1 Protein, Human, Recombinant Human HEK293
Vitelline membrane outer layer protein 1 (VMO1), a basic protein present in the outer layer of the vitelline membrane of eggs, plays essential roles in separating the yolk from the egg white and preventing infection from...
TMPY-00375 VMO1 Protein, Human, Recombinant (mFc) Human HEK293
Vitelline membrane outer layer protein 1 (VMO1), a basic protein present in the outer layer of the vitelline membrane of eggs, plays essential roles in separating the yolk from the egg white and preventing infection from...
TMPJ-00705 BCAS2 Protein, Human, Recombinant (His, T7) Human E. coli
Breast Carcinoma-Amplified Sequence 2 (BCAS2) is a member of the SPF27 family. BCAS2 is a nuclear protein and widely expressed in many rtissues. BCAS2 is identified as being overexpressed in various breast cancer cell li...
TMPY-06226 SLC39A6/LIV-1 Protein, Cynomolgus, Recombinant (His) Cynomolgus HEK293
Along with the SLC30 family, SLC39 family members regulate zinc movement in cells. SLC39 metal ion transporters accumulate zinc into the cytosol. SLC39A6, also known as LIV-1, belongs to a new subfamily of Zrt, Irt-like ...
TMPY-01826 Relaxin 1/RLN1 Protein, Human, Recombinant (His) Human HEK293
Relaxin-1, also known as Prorelaxin H1 and RLN1, is a secreted protein that belongs to the insulin family. It is a peptide hormone that was first described in 1926 by Frederick Hisaw. Since its discovery as a reproductiv...
TMPJ-00056 AG-2 Protein, Human, Recombinant (His) Human Human Cells
Anterior Gradient 2 (AGR2) is an 18-21 kDa member of the PDI family of enzymes. AGR2 is widely expressed in secretory cells, such as small intestine goblet, prostate epithelium, enteroendocrine cells, and multiple carcin...
TMPJ-00253 OPG Protein, Mouse, Recombinant (His) Mouse Human Cells
Osteoprotegerin (OPG, Tnfrsf11b) is a secreted protein that regulates bone density. OPG is widely expressed and constitutively released as a homodimer by mesenchymal stem cells, fibroblasts and endothelial cells. Regulat...
TMPY-02843 GPX7 Protein, Human, Recombinant (hFc) Human HEK293
GPX7 gene contains 3 distinct gt-ag introns. Transcription produces 4 different mRNAs, 3 alternatively spliced variants, and 1 unspliced form. There are 5 validated alternative polyadenylation sites. The mRNAs appear to ...
TMPY-04828 TFF3 Protein, Human, Recombinant (His) Human HEK293
Trefoil factor family (TFF) peptides are involved in the maintenance of epithelial integrity and epithelial restitution. Trefoil factor-3 (TFF3) is an estrogen-regulated gene associated with prognosis in different types ...
TMPY-04422 Casein Kinase 1 gamma 2 Protein, Human, Recombinant (His) Human Baculovirus-Insect Cells
Casein kinase I gamma 2 isoform (CSNK1G2), a member of the large casein kinase I (CKI) subfamily, protein kinase superfamily. It may affect the development of brain, and associate with vesicular trafficking and neurotran...
TMPY-02214 OTUB1 Protein, Human, Recombinant (His) Human E. coli
Ubiquitin thioesterase OTUB1, also known as Deubiquitinating enzyme OTUB1, OTU domain-containing ubiquitin aldehyde-binding protein 1, Otubain-1, Ubiquitin-specific-processing protease OTUB1, OTUB1 and OTB1, is a cytopla...
TMPH-01616 LRP2 Protein, Human, Recombinant (mFc) Human HEK293
Multiligand endocytic receptor. Acts together with CUBN to mediate endocytosis of high-density lipoproteins. Mediates receptor-mediated uptake of polybasic drugs such as aprotinin, aminoglycosides and polymyxin B. In the...
TMPY-03022 IL-8/CXCL8 Protein, Canine, Recombinant Canine E. coli
Interleukin 8 (IL-8), also known as CXCL8, which is a chemokine with a defining CXC amino acid motif that was initially characterized for its leukocyte chemotactic activity, is now known to possess tumorigenic and proang...
TMPY-00755 IL-8/CXCL8 Protein, Human, Recombinant (aa 28-99, hFc) Human HEK293
Interleukin 8 (IL-8), also known as CXCL8, which is a chemokine with a defining CXC amino acid motif that was initially characterized for its leukocyte chemotactic activity, is now known to possess tumorigenic and proang...
TMPY-03480 IL-8/CXCL8 Protein, Rhesus, Recombinant Rhesus E. coli
Interleukin 8 (IL-8), also known as CXCL8, which is a chemokine with a defining CXC amino acid motif that was initially characterized for its leukocyte chemotactic activity, is now known to possess tumorigenic and proang...
TMPY-00753 IL-8/CXCL8 Protein, Human, Recombinant (aa 23-99, hFc) Human HEK293
Interleukin 8 (IL-8), also known as CXCL8, which is a chemokine with a defining CXC amino acid motif that was initially characterized for its leukocyte chemotactic activity, is now known to possess tumorigenic and proang...
ER alpha Protein, Human, Recombinant (His)
TMPJ-00762
Species: Human
Expression System: E. coli
EBAG9 Protein, Human, Recombinant (His)
TMPY-03496
Species: Human
Expression System: E. coli
Aromatase/CYP19A1 Protein, Human, Recombinant (His)
TMPH-00956
Species: Human
Expression System: E. coli
C-ABL/ABL1 Protein, Human, Recombinant (GST)
TMPY-04396
Species: Human
Expression System: Baculovirus-Insect Cells
IL-8/CXCL8 Protein, Human, Recombinant (aa 28-99)
TMPY-00472
Species: Human
Expression System: E. coli
IL-8/CXCL8 Protein, Human, Recombinant (His)
TMPY-04726
Species: Human
Expression System: Yeast
IL-8/CXCL8 Protein, Human, Recombinant (aa 23-99)
TMPY-00754
Species: Human
Expression System: HEK293
ELAPOR1 Protein, Human, Recombinant (His)
TMPJ-01192
Species: Human
Expression System: Human Cells
SULT1E1 Protein, Human, Recombinant (His)
TMPY-01660
Species: Human
Expression System: E. coli
ER beta Protein, Human, Recombinant (His)
TMPH-01305
Species: Human
Expression System: Yeast
ER beta Protein, Human, Recombinant (E. coli, His)
TMPH-01304
Species: Human
Expression System: E. coli
HSD17B1 Protein, Human, Recombinant (His & Myc)
TMPH-01302
Species: Human
Expression System: E. coli
PDIA2 Protein, Mouse, Recombinant (His & SUMO)
TMPH-02851
Species: Mouse
Expression System: E. coli
Interferon tau-1/IFNT1 Protein, Bovine, Recombinant (His)
TMPH-00279
Species: Bovine
Expression System: Yeast
Interferon tau-1/IFNT1 Protein, Bovine, Recombinant (E. coli, His)
TMPH-00278
Species: Bovine
Expression System: E. coli
VMO1 Protein, Human, Recombinant
TMPY-04780
Species: Human
Expression System: HEK293
VMO1 Protein, Human, Recombinant (mFc)
TMPY-00375
Species: Human
Expression System: HEK293
BCAS2 Protein, Human, Recombinant (His, T7)
TMPJ-00705
Species: Human
Expression System: E. coli
SLC39A6/LIV-1 Protein, Cynomolgus, Recombinant (His)
TMPY-06226
Species: Cynomolgus
Expression System: HEK293
Relaxin 1/RLN1 Protein, Human, Recombinant (His)
TMPY-01826
Species: Human
Expression System: HEK293
AG-2 Protein, Human, Recombinant (His)
TMPJ-00056
Species: Human
Expression System: Human Cells
OPG Protein, Mouse, Recombinant (His)
TMPJ-00253
Species: Mouse
Expression System: Human Cells
GPX7 Protein, Human, Recombinant (hFc)
TMPY-02843
Species: Human
Expression System: HEK293
TFF3 Protein, Human, Recombinant (His)
TMPY-04828
Species: Human
Expression System: HEK293
Casein Kinase 1 gamma 2 Protein, Human, Recombinant (His)
TMPY-04422
Species: Human
Expression System: Baculovirus-Insect Cells
OTUB1 Protein, Human, Recombinant (His)
TMPY-02214
Species: Human
Expression System: E. coli
LRP2 Protein, Human, Recombinant (mFc)
TMPH-01616
Species: Human
Expression System: HEK293
IL-8/CXCL8 Protein, Canine, Recombinant
TMPY-03022
Species: Canine
Expression System: E. coli
IL-8/CXCL8 Protein, Human, Recombinant (aa 28-99, hFc)
TMPY-00755
Species: Human
Expression System: HEK293
IL-8/CXCL8 Protein, Rhesus, Recombinant
TMPY-03480
Species: Rhesus
Expression System: E. coli
IL-8/CXCL8 Protein, Human, Recombinant (aa 23-99, hFc)
TMPY-00753
Species: Human
Expression System: HEK293
Cat No. Product Name
L2191 Anti-Breast Cancer Compound Library

1965 compounds
A unique collection of 1965 compounds with anti-breast cancer therapeutic activity or targeting breast cancer’s major signaling pathways, can be used for anti-breast cancer drug discovery and mechanism study；

Libraries

Anti-Breast Cancer Compound Library
L2191
Compounds: 1965
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