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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T22761 | EIT hydrobromide | 2-Ethyl-2-thiopseudourea hydrobromide,S-Ethylisothiourea hydrobromide | NOS |
EIT hydrobromide (S-Ethylisothiourea hydrobromide) is an iNOS inhibitor. | |||
T78410 | Gly-Pro-AMC hydrobromide | Gly-Pro-AMC HCl | |
Gly-Pro-AMC hydrobromide (Gly-Pro-AMC HCl) is a specific fluorescent dye used in cytofluorescence assays to detect Dipeptidyl peptidase IV (DPP-IV) activity. | |||
T8495 | Alobresib | Vorolanib,GS-5829 | Epigenetic Reader Domain |
Alobresib (Vorolanib) is an inhibitor of BET bromodomain,is an antineoplastic drug candidate. | |||
T5351L | PU-WS13 hydrobromide | PU-WS13 hydrobromide (1454619-14-7 Free base) | GPR |
PU-WS13 hydrobromide is a GRP94 inhibitor with anti-inflammatory activity and inhibits the proliferation of M2-like macrophages in mouse TNBC tumors. | |||
T1534 | Darifenacin hydrobromide | Darifenacin HBr,UK-88525 | AChR |
Darifenacin hydrobromide (UK-88525) is a selective muscarinic receptor antagonist used to treat urinary incontinence and overactive bladder syndrome. | |||
T12172 | NAN-190 hydrobromide | 5-HT Receptor | |
NAN-190 hydrobromide is an antagonist of serotonin receptor 5-HT. | |||
T7208 | AMD 3465 hexahydrobromide | GENZ-644494 (hexahydrobromide) | HIV Protease , CXCR |
AMD 3465 hexahydrobromide (GENZ-644494 (hexahydrobromide)) is a CXCR4 receptor antagonist with potential anticancer and anti-HIV activity. | |||
T3156 | Ciliobrevin A | Hedgehog Pathway Inhibitor 4,HPI-4 | Hedgehog/Smoothened |
Ciliobrevin A (HPI-4) is an inhibitor of hedgehog signaling pathway with an IC50 <10 μM. | |||
T21788 | BD 1008 dihydrobromide | Sigma receptor | |
BD 1008 dihydrobromide is a selective antagonist of the sigma 1 (σ1) receptor (Ki = 2 nM). BD 1008 dihydrobromide have high affinity for sigma1 receptors, moderate affinity for sigma2 receptors. | |||
T2395L | Vortioxetine hydrobromide | Vortioxetine (Lu AA21004) HBr,Vortioxetine HBr,Lu AA21004 hydrobromide | 5-HT Receptor , Serotonin Transporter |
Vortioxetine hydrobromide (Lu AA21004 hydrobromide) is a serotonin (5-HT) modulator and stimulator (SMS), inhibits 5-HT1A/1B/3A/7 receptor and SERT (IC50: 15/33/3.7/19/1.6 nM). | |||
T22864 | Immethridine dihydrobromide | Others | |
Immethridine dihydrobromide is a histamine H3 receptor agonist. | |||
T61151 | Beclobrate | Sgd 24774 | Others |
Beclobrate (Sgd 24774) is a novel orally available fibric acid derivative that has shown significant lipid and cholesterol-lowering activity in rodents and may be used in the study of primary hyperlipoproteinemia. | |||
T10813 | Cilobradine hydrochloride | DK-AH 269 | HCN Channel |
Cilobradine hydrochloride (DK-AH 269) is an HCN Channel blocker and an open channel blocker of neuronal Ih and related cardiac If channels. | |||
T22534 | 8-Hydroxy-DPAT hydrobromide | 8-OH-DPAT hydrobromide | 5-HT Receptor |
8-Hydroxy-DPAT hydrobromide (8-OH-DPAT hydrobromide) (8-OH-DPAT hydrobromide) is a potent and selective 5-HT1A agonist with a pIC50 of 8.19. 8-Hydroxy-DPAT hydrobromide has a selectivity of almost 1000 fold for a subtype... | |||
T77795 | L-DABA hydrobromide | L-2,4-Diaminobutyric acid hydrobromide | Others , Endogenous Metabolite |
L-DABA hydrobromide (L-2,4-Diaminobutyric acid hydrobromide) is a potent GABA transaminase inhibitor with antitumor and anticonvulsant activity for the study of neurological disorders. | |||
T12352L | Oxidopamine hydrobromide | 6-Hydroxydopamine hydrobromide,6-OHDA hydrobromide | Mitophagy , Dopamine Receptor , Autophagy |
Oxidopamine hydrobromide (6-OHDA hydrobromide) is a neurotransmitter dopamine antagonist. | |||
T1986L | Atopaxar Hydrobromide | Protease-activated Receptor | |
Atopaxar, a reversible PAR-1 thrombin receptor antagonist, interferes with platelet signaling. Atopaxar has been investigated for the treatment of Coronary Artery Disease and Acute Coronary Syndrome. | |||
T5956 | VP3.15 dihydrobromide | GSK-3 , PDE | |
VP3.15 dihydrobromide is a potent, orally bioavailable and CNS-penetrant dual phosphodiesterase (PDE7- glycogen synthase kinase (GSK)3 inhibitor(with IC50s of 1.59 μM , 0.88 μM,respectively.) | |||
T13110 | Tedatioxetine hydrobromide | Lu AA 24530 hydrobromide | Dopamine Receptor , 5-HT Receptor , Norepinephrine |
Tedatioxetine hydrobromide (Lu AA 24530 hydrobromide) is a serotonin-norepinephrine-dopamine reuptake inhibitor and an antagonist of 5-HT2A, 5-HT2C, 5-HT3, and α1A-adrenergic receptors, which can be used to treat depress... | |||
T6133 | Remodelin hydrobromide | Remodelin,Remodelin HBR | RAAS , Histone Acetyltransferase |
Remodelin hydrobromide (Remodelin HBR) is a novel potent and selective inhibitor of the acetyl-transferase protein NAT10. | |||
T1483 | Citalopram hydrobromide | Lu 10-171,Nitalapram HBr,Bonitrile HBr,XU-62-320,Lu 10-171 HBr,Citalopram HBr | 5-HT Receptor , Serotonin Transporter , Autophagy |
Citalopram hydrobromide (XU-62-320) , a selective serotonin reuptake inhibitor (SSRI), selectively inhibits the CNS neuronal reuptake of serotonin, thereby potentiating serotonergic activity in the central nervous system... | |||
T8439 | Clobenpropit dihydrobromide | Apoptosis , Histamine Receptor | |
Clobenpropit dihydrobromide is a potent antagonist and inverse agonist of histamine H3R (histamine H3LR,pEC50 of 8.07) | |||
T1740 | BD-1047 dihydrobromide | BD1047.2HBr | Sigma receptor |
BD-1047 dihydrobromide (BD1047.2HBr) , a selective functional antagonist of sigma receptors, has antipsychotic activity in animal models predictive of efficacy in schizophrenia. | |||
T36287 | Pirtobrutinib | BTK | |
Pirtobrutinib (LOXO-305) is an advanced BTK inhibitor that displays high selectivity and operates through a non-covalent mechanism. This compound effectively inhibits various BTK C481 substitution mutations, leading to t... | |||
T14965 | Ciliobrevin D | ATPase , Hedgehog/Smoothened | |
Ciliobrevin D is a AAA+ ATPase motor cytoplasmic dynein inhibitor. Ciliobrevin D inhibits Hedgehog (Hh) signaling and primary cilia formation and it also inhibits dynein-dependent microtubule gliding and ATPase activity ... | |||
T17002 | Tazemetostat hydrobromide | E-7438 hydrobromide,EPZ-6438 hydrobromide | Histone Methyltransferase |
Tazemetostat hydrobromide (E-7438 hydrobromide) is a potent and selective EZH2 inhibitor. Tazemetostat hydrobromide inhibits the activity of human polycomb repressive complex 2 (PRC2)-containing wild-type EZH2 (Ki: 2.5 n... | |||
T4570 | Pipobroman | Vercyte,A-8103,Amedel | Others , DNA Alkylator/Crosslinker |
Pipobroman (Vercyte) is an anti-cancer drug that probably acts as an alkylating agent. Pipobroman has well documented clinical activity in polycythemia vera (PV) and essential thrombocythemia (ET). Pipobroman allows, wit... | |||
T0216 | Eletriptan hydrobromide | Eletriptan HBr,UK-116044 | 5-HT Receptor |
Eletriptan hydrobromide (Eletriptan HBr) is an orally active agonist with specific affinity for the 5-hydroxytriptamine1B/1D receptor. | |||
T2707 | Pifithrin-α hydrobromide | Pifithrin hydrobromide,Pifithrin-α (PFTα) HBr,Pifithrin-α,PFTα,PFTα hydrobromide | Ferroptosis , Aryl Hydrocarbon Receptor , p53 |
Pifithrin-α hydrobromide (Pifithrin-α hydrobromide) is a p53 inhibitor, inhibiting p53-dependent transactivation of p53-responsive genes. | |||
T6999 | Teneligliptin hydrobromide | Teneligliptin hydrobromide anhydrous,MP-513 (hydrobromide) | Others , Proteasome , DPP-4 |
Teneligliptin hydrobromide (MP-513 (hydrobromide)) is a novel, potent, and long-lasting dipeptidyl peptidase-4 inhibitor; competitively inhibited human plasma, rat plasma, and human recombinant DPP-4 in vitro, with IC50 ... | |||
T7206L | 2-Iminobiotin hydrobromide | Guanidinobiotin | NOS , NO Synthase |
2-Iminobiotin hydrobromide (Guanidinobiotin) is a cyclic guanidino analog of biotin that acts as a reversible inhibitor of inducible nitric oxide synthase (iNOS) and neuronal NOS (nNOS; Ki of 21.8 and 37.5 μM for mouse i... | |||
TD0105 | Sulfobromophthalein disodium salt | Others | |
Sulfobromophthalein disodium salt is an organic anion dye, it is used in the study of a variety of membrane carriers expressed in animal tissues and involved in transport of drugs and metabolites. | |||
T40363 | Poly-D-lysine hydrobromide (MW 30000-70000) | Poly-D-lysine HBr (MW 30000-70000) | CaSR |
Poly-D-lysine hydrobromide (MW 30000-70000)(Poly-D-lysine HBr) is an orally available peptide CaSR agonist that removes proteinase K-resistant PrP from prion-infected SN56 neuroblastoma cells. | |||
T6832 | Fatostatin hydrobromide | Fatostatin HBr,Fatostatin A,Fatostatin A HBr,Fatostatin | NPC1L1 , Fatty Acid Synthase |
Fatostatin hydrobromide (Fatostatin A HBr) ia an inhibitor of sterol regulatory element binding protein (SREBP). It impairs the activation of SREBP-1 and SREBP-2. | |||
T3637 | Pifithrin-β hydrobromide | Cyclic PFT-α,PFT-β,Cyclic Pifithrin-α hydrobromide,Pifithrin-β,PFT β (hydrobromide) | Ferroptosis , p53 |
Pifithrin-β hydrobromide (Cyclic PFT-α) is an inhibitor of p53; reversibly blocks p53-dependent transcriptional activation and apoptosis. Protects against neuronal death in models of stroke and neurodegenerative disorder... | |||
T10104 | 3,4-Dihydroxybenzylamine hydrobromide | NSC 263475 hydrobromide | Others , DNA/RNA Synthesis |
3,4-Dihydroxybenzylamine hydrobromide (NSC-263475 hydrobromide) inhibits DNA polymerase activity in melanoma cells and displays growth inhibitory activity in melanoma cell lines with varying degrees of tyrosinase activit... | |||
T4387 | Evobrutinib | MSC2364447C,M2951 | BTK |
Evobrutinib(M2951) , also known as M-2951 and MSC-2364447C, is a highly selective inhibitor of the Bruton's tyrosine kinase (BTK), which is important in the development and functioning of various immune cells including B... | |||
T21685 | CCT 031374 hydrobromide | Wnt/beta-catenin | |
CCT 031374 hydrobromide is a TCF/β-catenin inhibitor with antitumor activities. | |||
T10717 | Inobrodib | CBP-IN-1 | Epigenetic Reader Domain |
Inobrodib (CBP-IN-1) is a potent inhibitor of p300/CBP bromodomain. | |||
T7543 | S-(2-aminoethyl) Isothiourea (dihydrobromide) | NOS | |
S-(2-aminoethyl) Isothiourea (dihydrobromide) is a non-selective inhibitor of all NOS isoforms. For human nNOS, eNOS, and iNOS, the Ki values are 1.8, 2.1, and 0.59 µM, respectively | |||
T39814 | Bromo-PEG1-NH2 hydrobromide | Bromo-PEG1-NH2 hydrobromide | |
Bromo-PEG1-NH2 hydrobromide is a polyethylene glycol (PEG)-based linker compound employed in the synthesis of proteolysis-targeting chimeras (PROTACs). | |||
T32227 | Isoquinoline, 5,5'-oxybis(decahydro-2-ethyl-, dihydrobromide | ||
Isoquinoline, 5,5'-oxybis(decahydro-2-ethyl-, dihydrobromide is a bioactive chemical. | |||
T30000 | Amlodipine hydrobromide | Amlodipine HBr | |
Amlodipine hydrobromide is a salt of Amlodipine --- a medication used to lower blood pressure and prevent chest pain. | |||
T24035 | Eptazocine hydrobromide | MCV 4169,ST-2121,MCV-4169,sT 2121, l-,l-ST-2121 | |
Eptazocine hydrobromide is an agonist of the Opioid receptor and is a kappa-Opioid receptor agonist. It is also an Opioid analgesic and an Opioid receptor antagonist. | |||
T24669 | Protheobromine | Pro-Cor,Theocor,Protheobrominum,TEBE,Vascopil | |
Protheobromine is a diuretic drug. | |||
T65237 | Glycine 7-amido-4-methylcoumarin hydrobromide | ||
Glycine 7-amido-4-methylcoumarin hydrobromide is a useful organic compound for research related to life sciences. The catalog number is T65237 and the CAS number is 113728-13-5. | |||
T15565 | Imetit dihydrobromide | VUF 8325 dihydrobromide,SKF 91105 dihydrobromide | Histamine Receptor |
Imetit dihydrobromide is a high affinity and effective agonist of histamine H3 and H4 receptors (Ki: 0.3 and 2.7 nM). Imetit mimics the histamine effect in triggering a shape change in eosinophils (EC50: 25 nM). | |||
T23362 | SKF-83566 hydrobromide | SKF 83566 hydrobromide | Others |
D1-like dopamine receptor antagonist | |||
T61215 | Alinidine hydrobromide | ||
Alinidine hydrobromide, a specific bradycardic agent, diminishes the slope of the diastolic depolarization in sinoatrial tissue and Purkinje fibers [1]. | |||
T61999 | Quinine hydrobromide | ||
Quinidine is a potent, orally active, selective inhibitor of cytochrome P450db. Quinidine hydrobromide is a K + channel blocker (IC 50= 19.9 μM). Quinidine hydrobromide shows antiarrhythmic activity. Quinidine hydrobromi... |
Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T41372 | (22S,23S)-Homobrassinolide | SSHB | Others |
(22S,23S)-Homobrassinolide (SSHB) induces plant growth in various plant bioassay systems. | |||
T6560 | Lappaconitine hydrobromide | Lappaconite HBr,Allapinine | Others |
Lappaconitine hydrobromide (Allapinine) is a kind of alkaloid extracted from Aconitum sinomontanum Nakai. It has anti-inflammatory effects. | |||
T8304 | Anisodamine Hydrobromide | 6-Hydroxyhyoscyamine | Adrenergic Receptor , AChR |
Anisodamine Hydrobromide (6-Hydroxyhyoscyamine) is an anticholinergic and α1-adrenergic receptor antagonist used in the treatment of acute circulatory shock. | |||
T2198 | Arecoline hydrobromide | Arecoline HBr,Arecoline bromide | AChR |
Arecoline hydrobromide (Arecoline HBr) is a muscarinic acetylcholine receptor agonist. | |||
T3524 | Halofuginone hydrobromide | Tempostatin,RU-19110 (hydrobromide),Stenorol | Others , Calcium Channel , DNA/RNA Synthesis , Sodium Channel , Parasite , TGF-beta/Smad |
Halofuginone specifically inhibits collagen type I gene expression and matrix metalloproteinase 2 (MMP-2) gene expression, which may result in the suppression of angiogenesis, tumor stromal cell development, and tumor ce... | |||
T1255 | Tobramycin | NSC 180514,Nebramycin Factor 6,Deoxykanamycin B | ribosome , Antibacterial , Antibiotic |
Tobramycin (NSC-180514) is an aminoglycoside, broad-spectrum antibiotic produced by Streptomyces tenebrarius. | |||
T0625 | Theobromine | 3, 7-Dimethylxanthine,3,7-Dimethylxanthine | Endogenous Metabolite , PDE , Adenosine Receptor |
Theobromine (3,7-Dimethylxanthine), a xanthine alkaloid, is used as a bronchodilator and as a vasodilator. | |||
T0086 | Galanthamine hydrobromide | Galantamine hydrobromide,Galanthamine HBr | AChR , AChE |
Galanthamine hydrobromide (Galantamine hydrobromide), a long-acting and centrally active AChE inhibitor (IC50:410 nM), is an allosteric potentiator at neuronal nicotinic ACh receptors. | |||
TN3796 | Dehydrobruceantinol | Others | |
Dehydrobruceantinol shows bitter taste and has antileukemic activity. | |||
TN3051 | 4-Methoxyglucobrassicin | Others | |
4-Methoxyglucobrassicin is a natural product for research related to life sciences. The catalog number is TN3051 and the CAS number is 83327-21-3. | |||
T11041 | Dihydro-β-erythroidine hydrobromide | DHβE hydrobromide | Others |
Dihydro-β-erythroidine hydrobromide(DHβE) is a potent, oral active and competitive antagonist of neuronal nicotinic acetylcholine receptors (nAChRs). Dihydro-β-carotene hydrobromide showed selectivity to α4β4 and α4β2nAC... | |||
T80014 | Guvacine hydrobromide | GABA Receptor | |
Guvacine hydrobromide, an alkaloid derived from the Areca catechu nut, serves as a potent inhibitor of GABA (GABA uptakp) uptake. It effectively inhibits rat GABA transporter isoforms GAT-1, GAT-2, and GAT-3, with respec... | |||
TN6072 | 14-Dehydrobrowniine | ||
14-Dehydrobrowniine is a natural product of Delphinium, Ranunculaceae. The catalog number is TN6072 and the CAS number is 4829-56-5. 14-Dehydrobrowniine can be used as a reference standard. | |||
T1255L | Tobramycin Sulfate | Dartobcin,Nebcine,Tobraneg,Tobrasix | |
Tobramycin Sulfate is a broad-spectrum antibiotic. It is effective against gram-negative bacteria. It especially potent against the Pseudomonas species. | |||
TN4636 | Neoglucobrassicin | Others | |
Neoglucobrassicin is a natural product for research related to life sciences. The catalog number is TN4636 and the CAS number is 5187-84-8. | |||
T82304 | Glucobrassicanapin potassium | 4-Pentenylglucosinolate potassium | |
Glucobrassicanapin (4-Pentenylglucosinolate) potassium, an aliphatic glucosinolate, is found in Brassica rapa vegetable crops [1]. | |||
T80013 | Arecaidine hydrobromide | GABA Receptor | |
Arecaidine hydrobromide, a pyridine alkaloid, functions as a potent GABA uptake inhibitor and acts as a substrate for the H+-coupled amino acid transporter 1 (PAT1, SLC36A1), where it competitively inhibits L-proline upt... | |||
TN1899L | Lycoramine hydrobromide | Lycoramine HBr | |
Lycoramine is a natural alkaloid isolated from Lycoris chinensis. | |||
TN3797 | Dehydrobruceine A | Antifection | |
Dehydrobruceine A shows strong antitrypanosomal activities with IC(50) values in the range of 2.9-17.8nM. | |||
T75485 | Dehydrobruceine B | ||
Dehydrobruceine B, a quassinoid isolated from Brucea javanica, demonstrates a synergistic effect with Cisplatin in inducing apoptosis through the mitochondrial pathway. It enhances the expression of apoptosis-inducing fa... | |||
TN4237 | Hydrocotarnine hydrobromide | Others | |
Hydrocotarnine hydrobromide is a natural product for research related to life sciences. The catalog number is TN4237 and the CAS number is 5985-00-2. | |||
TN5614 | Dehydrobruceantin | ||
Dehydrobruceantin has anti-tuberculosis activity. |
Cat No. | Product Name | Species | Expression System |
---|---|---|---|
TMPY-01725 | Leptin Receptor Protein, Human, Recombinant (His) | Human | HEK293 Cells |
Leptin Receptor Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 95 kDa and the accession number is P48357-1. | |||
TMPY-00874 | Leptin Receptor Protein, Human, Recombinant (His & hFc) | Human | HEK293 Cells |
Leptin Receptor Protein, Human, Recombinant (His & hFc) is expressed in HEK293 mammalian cells with His and hFc tag. The predicted molecular weight is 121.4 kDa and the accession number is P48357-1. | |||
TMPJ-00411 | LEPR Protein, Human, Recombinant (hFc) | Human | HEK293 Cells |
LEPR Protein, Human, Recombinant (hFc) is expressed in HEK293 mammalian cells with C-Fc tag. The predicted molecular weight is 150-180 KDa and the accession number is P48357. | |||
TMPJ-00976 | LEPR Protein, Mouse, Recombinant (His) | Mouse | HEK293 Cells |
LEPR Protein, Mouse, Recombinant (His) is expressed in HEK293 mammalian cells with C-10His tag. The predicted molecular weight is 120-150 KDa and the accession number is P48356. | |||
TMPJ-00977 | LEPR Protein, Mouse, Recombinant (mFc) | Mouse | HEK293 Cells |
LEPR Protein, Mouse, Recombinant (mFc) is expressed in HEK293 mammalian cells with C-mFc tag. The predicted molecular weight is 130-190 KDa and the accession number is P48356. | |||
TMPJ-00975 | LEPR Protein, Mouse, Recombinant (hFc) | Mouse | HEK293 Cells |
LEPR Protein, Mouse, Recombinant (hFc) is expressed in HEK293 mammalian cells with C-Fc tag. The predicted molecular weight is 130-190 KDa and the accession number is P48356. | |||
TMPH-00031 | Aerolysin Protein, Aeromonas sobria, Recombinant (His & Myc) | Aeromonas sobria | E. coli |
Secreted, cytolytic toxin that forms pores in host membranes after proteolytic removal of a C-terminal propeptide, leading to destruction of the membrane permeability barrier and cell death. The pores are formed by trans... | |||
TMPH-03037 | Alpha-cobratoxin Protein, Naja kaouthia, Recombinant (GST & His & Myc) | Naja kaouthia | E. coli |
Monomer: binds with high affinity to muscular (alpha-1-beta-1-gamma-delta/CHRNA1-CHRNB1-CHRNG-CHRND) nAChR (tested on Torpedo californica, Kd=0.2-4.5 nM) and neuronal alpha-7/CHRNA7 nicotinic acetylcholine receptors (Kd=... | |||
TMPH-03038 | Cobra venom factor Protein, Naja kaouthia, Recombinant (His & SUMO) | Naja kaouthia | E. coli |
Complement-activating protein in cobra venom. It is a structural and functional analog of complement component C3b, the activated form of C3. It binds factor B (CFB), which is subsequently cleaved by factor D (CFD) to fo... |