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BD-1047 dihydrobromide

Catalog No. T1740 CAS 138356-21-5

Synonyms: BD1047.2HBr

BD-1047 dihydrobromide (BD1047.2HBr) , a selective functional antagonist of sigma receptors, has antipsychotic activity in animal models predictive of efficacy in schizophrenia.

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BD-1047 dihydrobromide Chemical Structure

BD-1047 dihydrobromide, CAS 138356-21-5

Pack Size	Availability	Price/USD
1 mg	In stock	$ 31.00
2 mg	In stock	$ 41.00
5 mg	In stock	$ 67.00
10 mg	In stock	$ 87.00
25 mg	In stock	$ 171.00
50 mg	In stock	$ 306.00
100 mg	In stock	$ 516.00
1 mL * 10 mM (in DMSO)	In stock	$ 68.00

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Purity: 99.39%

Purity: 98.13%

Biological Description

Chemical Properties

Storage & Solubility Information

Description

BD-1047 dihydrobromide (BD1047.2HBr) , a selective functional antagonist of sigma receptors, has antipsychotic activity in animal models predictive of efficacy in schizophrenia.

Synonyms	BD1047.2HBr
Molecular Weight	437.04
Formula	C13H22Br2Cl2N2
CAS No.	138356-21-5

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year

Solubility Information

DMSO: 50 mg/mL (114.41 mM)

References and Literature

1. Skuza G, et al. Pharmacol Rep. 2006 Sep-Oct;58(5):626-635.

Citations

1. Zhang Z, Zhou H, Gu W, et al.CGI1746 targets σ1R to modulate ferroptosis through mitochondria-associated membranes.Nature Chemical Biology.2024: 1-11.

Related compound libraries

This product is contained In the following compound libraries：

Inhibitor Library GPCR Compound Library Preclinical Compound Library Anti-Obesity Compound Library Bioactive Compound Library Neuronal Signaling Compound Library Bioactive Compounds Library Max NO PAINS Compound Library

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Related compounds with same targets

Amitriptyline hydrochloride Siramesine Siramesine hydrochloride KSK67 S1R agonist 2 S1RA hydrochloride AB21 oxalate Sigma-1 receptor antagonist 2

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Method for preparing DMSO master liquid: mg drug pre-dissolved in μL DMSO (Master liquid concentration mg/mL)，Please contact us first if the concentration exceeds the DMSO solubility of the batch of drug.

Method for preparing in vivo formulation：Take μL DMSO master liquid, next add μL PEG300， mix and clarify, next add μL Tween 80，mix and clarify, next add μL ddH₂O, mix and clarify.

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Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.

Keywords

BD-1047 dihydrobromide 138356-21-5 GPCR/G Protein Sigma receptor BD-1047 Dihydrobromide BD-1047 inhibit Inhibitor BD 1047 dihydrobromide Sigma Receptor BD 1047 Dihydrobromide BD 1047 BD1047 BD1047 Dihydrobromide BD1047.2HBr BD1047 dihydrobromide inhibitor

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