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Search Result

Search Results for " upa "

64

Compounds

51

Natural Products

21

Recombinant Proteins

Cat No. Product Name Synonyms Targets
T29051 UK-122 TFA salt UK122,uPA Inhibitor II,UK122 TFA salt,UK 122,UK-122,K122 trifloroacetic acid
UK-122 is a potent and selective uPA inhibitor (Ki = 20 nM). The IC(50) of UK122 in a cell-free indirect uPA assay is 0.2 micromol/L. UK122 showed little cytotoxicity against CFPAC-1 cells (IC(50) > 100 micromol/L) but s...
T13408 ZK824190 Others , Serine Protease
ZK824190 is an orally available and selective inhibitor of urokinase plasminogen activator (uPA) as a potential treatment for multiple sclerosis(IC50s of 237, 1600 and 1850 nM for uPA, tPA, and Plasmin, respectively).
T8362 Benzamidine hydrochloride Benzamidine HCl Serine/threonin kinase , Serine Protease
Benzamidine hydrochloride (Benzamidine HCl) is a reversible inhibitor of serine proteases, including trypsin, plasmin, and thrombin (Ki of 35, 350, and 220 μM, respectively).
T13257 Upamostat PAI-1 , Serine/threonin kinase , Serine Protease
Upamostat is an inhibitor of a serine protease and is a urokinase plasminogen activator (uPA) inhibitor.
T61932 Nesuparib JPI-547/OCN-201 PARP , Wnt/beta-catenin
Nesuparib (JPI-547/OCN-201) is a potent PARP inhibitor with inhibitory effects on PARP and TNKS1.Nesuparib has antitumor activity and can be used in the treatment of tumors, endocrine and metabolic disorders, genitourina...
T77566 (3aR,9aR)-Fluparoxan Adrenergic Receptor
(3aR,9aR)-Fluparoxan is a highly selective and potent adrenergic receptor α2B antagonist for the prevention, amelioration or treatment of neurodevelopmental disorders and neurodegenerative diseases.
T1827 Buparlisib BKM120,NVP-BKM120 Apoptosis , PI3K
Buparlisib (BKM120) is an orally bioavailable specific oral inhibitor of the pan-class I PI3K (IC50s: 52/166/116/nM for p110α, p110β, and p110δ).
T7503 Upadacitinib ABT-494 JAK
Upadacitinib (ABT-494) (ABT-494) is a selective Janus kinase (JAK) 1 inhibitor, which is being studied for the treatment of several autoimmune disorders in the IC50 of 43 nM.
T76735 Mupadolimab CPI-006 CD73
Mupadolimab (CPI-006) is a humanized FC-γR binding deficient IgG1 anti-CD73 antibody with potential anticancer activity and activation of CD73POS B cells.
T11122 DUPA(OtBu)-OH Others
DUPA(OtBu)-OH is a DUPA precursor. DUPA is used as the targeting moiety to actively deliver Docetaxel (DTX) for treatment of Prostate-Specific Membrane Antigen (PSMA) expressing prostate cancer. PSMA has a high affinity ...
T19301 DUPA N,N''-Carbonylbis[L-glutamic acid],(2S,2'S)-2,2'-Carbonylbis(Azanediyl)Dipentanedioic Acid Others , Ligands for Target Protein for PROTAC
DUPA (N,N''-Carbonylbis[L-glutamic acid]) is used as the targeting moiety to actively deliver DTX for treatment of Prostate-Specific Membrane Antigen (PSMA) expressing prostate cancer.
T6242 Rupatadine Fumarate Rinialer,Rupafin,Alergoliber PAFR , Autophagy , Histamine Receptor
Rupatadine Fumarate (Rinialer) (UR-12592 Fumarate) is a potent dual PAF/H1 antagonist with Ki of 0.55/0.1 uM.
T77565 Fluparoxan hydrochloride Adrenergic Receptor
Fluparoxan hydrochloride is a highly selective and potent α2-adrenoceptor antagonist for the prevention, amelioration or treatment of neurodevelopmental disorders and neurodegenerative diseases.
T77412 Lupartumab BAY 1112623 Others
Lupartumab (BAY 1112623) is an anti-LYPD3 (C4.4A) monoclonal antibody that can be used to synthesize antibody-active molecular couplers that can be used to study LYPD3-associated tumor diseases.
T4269 Buparvaquone Butalex,BW 720C Antibiotic , Parasite
Buparvaquone (BW 720C) is a hydroxynaphthoquinone antiprotozoal drug related to atovaquone and parvaquone.
T29067L Upacicalcet HCl Upacicalcet HCl(1333218-50-0 Free base) CaSR
Upacicalcet HCl is an intravesical calcium mimetic that inhibits excessive parathyroid hormone (PTH) secretion by directly acting on calcium-sensitive receptors in parathyroid cell membranes, thereby lowering PTH levels ...
T29067 Upacicalcet PLS-240,SK-1403,AJT-240 Calcium Channel
Upacicalcet (AJT-240) is an intraventricular calcium mimetic, a SHPT available for human hemodialysis, that inhibits excessive parathyroid hormone (PTH) secretion by directly acting on parathyroid cell membrane calcium-s...
TP2338L Cenupatide acetate Cenupatide acetate(1006388-38-0 Free base) Others
Cenupatide acetate is an urokinase plasminogen activator receptor (uPAR) inhibitor for treating disorders associated altered cell migration, such as cancer.
TP2338 Cenupatide UPARANT,Cenupatide trifluoroacetic acid salt,Ac-Arg-Aib-Arg-α(Me)Phe-NH2)
Cenupatide is a urokinase plasminogen activator receptor (uPAR) inhibitor. Cenupatide inhibits uPAR binding to the formyl peptide receptors (FPRs) can improve kidney lesions in a rat model of STZ-induced diabetes. Cenupa...
T69648 Inupadenant HCl
Inupadenant, also known as EOS-850, is a highly selective small molecule antagonist of the adenosine A2a receptor, in the adenosine triphosphate adenosine pathway, a key driver of immunosuppression in the tumor microenv...
T39444 Upacicalcet sodium
Upacicalcet (sodium) is an intravenous calcimimetic agent that acts directly on parathyroid cell membrane calcium-sensing receptors to suppress excessive parathyroid hormone (PTH) secretion, thereby lowering blood PTH le...
T32964 Lupanine perchlorate
Lupanine perchlorate is a bioactive chemical.
T32965 Lupanine dihydrochloride, (+/-)-
Lupanine dihydrochloride, (+/-)- is a bioactive chemical.
T80918 Tuparstobart Incagn-02385
Tuparstobart (Incagn-02385) is an IgG1κ monoclonal antibody that targets the immune checkpoint receptor protein LAG-3, which is predominantly expressed on activated T cells, NK cells, B cells, and plasmacytoid dendritic ...
T125919 Eupalinolide H
Eupalinolide H is a useful organic compound for research related to life sciences and the catalog number is T125919.
T36618 Rupatadine
Rupatadine (UR-12592) is a potent dual PAF/H1 antagonist with Ki of 0.55/0.1 uM(rabbit platelet membranes/guinea pig cerebellum membranes).IC50 value:Target: PAF/H1 antagonistin vitro: Rupatadine competitively inhibited ...
T32966 Lupanine, 17-hydroxy-
Lupanine, 17-hydroxy- is a bioactive chemical.
T37014 Inupadenant
Inupadenant is an orally active, highly selective A2A receptor antagonist. Inupadenant is not brain-penetrant. Inupadenant has potent anti-tumor activity[1]. [1]. Laurence Buisseret, et al. Phase 1 trial of the adenosine...
T7503L Upadacitinib tartrate ABT 494,ABT-494,ABT494
Upadacitinib is a potent and selective JAK inhibitor. Upadacitinib is approximately 74 fold selective for Jak1 over Jak2 in cellular assays dependent on specific, relevant cytokines. Upadacitinib demonstrates efficacy in...
T32968 Lupanol 3-beta-diglucoside
Lupanol 3-beta-diglucoside is a bioactive chemcial.
T32967 Lupanine, 17-hydroxy-, monohydrochloride
Lupanine, 17-hydroxy-, monohydrochloride is a drug / Therapeutic Agent.
T125102 Eupatoletin
Eupatoletin is a useful organic compound for research related to life sciences and the catalog number is T125102.
T124623 Eupassopilin
Eupassopilin is a useful organic compound for research related to life sciences. The catalog number is T124623 and the CAS number is 57718-81-7.
T124968 Eupalitin 3-galactoside
Eupalitin 3-galactoside is a useful organic compound for research related to life sciences and the catalog number is T124968.
T131460 3,20,29-Lupanetriol
3,20,29-Lupanetriol is a useful organic compound for research related to life sciences and the catalog number is T131460.
T124791 Alpha-Isolupanine
alpha-Isolupanine is a useful organic compound for research related to life sciences and the catalog number is T124791.
T27340 Fluparoxan HCl GR50360,GR 50360,Fluparoxan hydrochloride,GR-50360A,GR-50360
Fluparoxan is a potent α2-adrenergic receptor antagonist (pKB = 7.9) with excellent α2/α1 selectivity (2630 fold).
T70785 Mefuparib Free Base
Mefuparib Free Base is a potent, highly selective, competitive PARP1/2 inhibitor with IC50 of 3.2/1.9 nM, respectively. Mefuparib (CVL218), has been shown to have promising antiviral activity against the virus that cause...
T11992 Mefuparib hydrochloride MPH PARP
Mefuparib hydrochloride induces apoptosis and possesses prominent anticancer activity in vitro and in vivo. Mefuparib hydrochloride (MPH) is an orally active, substrate-competitive and selective PARP1/2 inhibitor with IC...
T16365 Buparlisib Hydrochloride NVP-BKM120 Hydrochloride,BKM120 Hydrochloride Others
Buparlisib Hydrochloride is an inhibitor of pan-class I PI3K (IC50: 52 nM/166 nM/116 nM/262 nM for p110α/p110β/p110δ/p110γ, respectively).
T80895 Upanovimab SCTA01
Upanovimab (SCTA01) is a monoclonal antibody [1].
T29291L 17-Oxolupanine hydrochloride
17-Oxolupanine hydrochloride is a drug / Therapeutic Agent.
T68074 Fluparoxan
Fluparoxan is a highly selective and potent alpha 2-adrenoceptor antagonist.
T29291 17-Oxolupanine
17-Oxolupanine is a bioactive chemical.
T61232 (Rac)-Upacicalcet
(Rac)-Upacicalcet is a racemate of Upacicalcet, which serves as an intravenous calcimimetic agent. Upacicalcet acts by directly targeting calcium-sensing receptors on parathyroid cell membranes, effectively suppressing t...
T3442 UK-371804 UK371804 PAI-1 , Serine Protease
UK-371804 is an effective and specific uPA inhibitor. It was selected as a candidate for further preClinicalal evaluation for the treatment of chronic dermal ulcers.
T60248 4-Aminobenzamidine dihydrochloride p-Aminobenzamidine dihydrochloride Serine Protease
4-Aminobenzamidine dihydrochloride (p-Aminobenzamidine dihydrochloride) is a strong trypsin inhibitor and a relatively weak inhibitor of urokinase type plasminogen activator (uPA) (K i =82 μM). 4-Aminobenzamidine can inh...
T26629 Angstrom6 A-6,A 6 peptide,A6,A 6,A6 peptide,A-6 peptide PAI-1
Angstrom6 (A-6 peptide) is an 8 amino acid peptide derived from single chain urokinase fibrinogen activator (scuPA) that interferes with the uPA/uPAR cascade and abrogates the downstream effects.Angstrom6 has antitumor a...
T0175 Amiloride hydrochloride Amiloride HCl,MK-870 hydrochloride Apoptosis , Serine Protease , Sodium Channel , TRP/TRPV Channel
Amiloride hydrochloride (Amiloride HCl) is an effective sodium channel blocker of epithelial.
T13409 ZK824859 Others
ZK824859 is an oral available and selective inhibitor of urokinase plasminogen activator (uPA)(IC50s of 79 nM, 1580 nM and 1330 nM for human uPA, tPA, and plasmin, respectively).

Compounds

UK-122 TFA salt
T29051
Synonym: UK122,uPA Inhibitor II,UK122 TFA salt,UK 122,UK-122,K122 trifloroacetic acid
Target:
ZK824190
T13408
Synonym:
Target: Others, Serine Protease
Benzamidine hydrochloride
T8362
Synonym: Benzamidine HCl
Target: Serine/threonin kinase, Serine Protease
Upamostat
T13257
Synonym:
Target: PAI-1, Serine/threonin kinase, Serine Protease
Nesuparib
T61932
Synonym: JPI-547/OCN-201
Target: PARP, Wnt/beta-catenin
(3aR,9aR)-Fluparoxan
T77566
Synonym:
Target: Adrenergic Receptor
Buparlisib
T1827
Synonym: BKM120,NVP-BKM120
Target: Apoptosis, PI3K
Upadacitinib
T7503
Synonym: ABT-494
Target: JAK
Mupadolimab
T76735
Synonym: CPI-006
Target: CD73
DUPA(OtBu)-OH
T11122
Synonym:
Target: Others
DUPA
T19301
Synonym: N,N''-Carbonylbis[L-glutamic acid],(2S,2'S)-2,2'-Carbonylbis(Azanediyl)Dipentanedioic Acid
Target: Others, Ligands for Target Protein for PROTAC
Rupatadine Fumarate
T6242
Synonym: Rinialer,Rupafin,Alergoliber
Target: PAFR, Autophagy, Histamine Receptor
Fluparoxan hydrochloride
T77565
Synonym:
Target: Adrenergic Receptor
Lupartumab
T77412
Synonym: BAY 1112623
Target: Others
Buparvaquone
T4269
Synonym: Butalex,BW 720C
Target: Antibiotic, Parasite
Upacicalcet HCl
T29067L
Synonym: Upacicalcet HCl(1333218-50-0 Free base)
Target: CaSR
Upacicalcet
T29067
Synonym: PLS-240,SK-1403,AJT-240
Target: Calcium Channel
Cenupatide acetate
TP2338L
Synonym: Cenupatide acetate(1006388-38-0 Free base)
Target: Others
Cenupatide
TP2338
Synonym: UPARANT,Cenupatide trifluoroacetic acid salt,Ac-Arg-Aib-Arg-α(Me)Phe-NH2)
Target:
Inupadenant HCl
T69648
Synonym:
Target:
Upacicalcet sodium
T39444
Synonym:
Target:
Lupanine perchlorate
T32964
Synonym:
Target:
Lupanine dihydrochloride, (+/-)-
T32965
Synonym:
Target:
Tuparstobart
T80918
Synonym: Incagn-02385
Target:
Eupalinolide H
T125919
Synonym:
Target:
Rupatadine
T36618
Synonym:
Target:
Lupanine, 17-hydroxy-
T32966
Synonym:
Target:
Inupadenant
T37014
Synonym:
Target:
Upadacitinib tartrate
T7503L
Synonym: ABT 494,ABT-494,ABT494
Target:
Lupanol 3-beta-diglucoside
T32968
Synonym:
Target:
Lupanine, 17-hydroxy-, monohydrochloride
T32967
Synonym:
Target:
Eupatoletin
T125102
Synonym:
Target:
Eupassopilin
T124623
Synonym:
Target:
Eupalitin 3-galactoside
T124968
Synonym:
Target:
3,20,29-Lupanetriol
T131460
Synonym:
Target:
alpha-Isolupanine
T124791
Synonym:
Target:
Fluparoxan HCl
T27340
Synonym: GR50360,GR 50360,Fluparoxan hydrochloride,GR-50360A,GR-50360
Target:
Mefuparib Free Base
T70785
Synonym:
Target:
Mefuparib hydrochloride
T11992
Synonym: MPH
Target: PARP
Buparlisib Hydrochloride
T16365
Synonym: NVP-BKM120 Hydrochloride,BKM120 Hydrochloride
Target: Others
Upanovimab
T80895
Synonym: SCTA01
Target:
17-Oxolupanine hydrochloride
T29291L
Synonym:
Target:
fluparoxan
T68074
Synonym:
Target:
17-Oxolupanine
T29291
Synonym:
Target:
(Rac)-Upacicalcet
T61232
Synonym:
Target:
UK-371804
T3442
Synonym: UK371804
Target: PAI-1, Serine Protease
4-Aminobenzamidine dihydrochloride
T60248
Synonym: p-Aminobenzamidine dihydrochloride
Target: Serine Protease
Angstrom6
T26629
Synonym: A-6,A 6 peptide,A6,A 6,A6 peptide,A-6 peptide
Target: PAI-1
Amiloride hydrochloride
T0175
Synonym: Amiloride HCl,MK-870 hydrochloride
Target: Apoptosis, Serine Protease, Sodium Channel, TRP/TRPV Channel
ZK824859
T13409
Synonym:
Target: Others
1 2
Cat No. Product Name Synonyms Targets
TN6762 (+)-Cuparene Others
(+)-Cuparene is a bioactive chemical.
T7032 Eupatorin Others , P450
Eupatorin has antiproliferative and antiangiogenic effects. Eupatorin has antiproliferative and cytostatic effects on MDA-MB-468 human breast cancer cells due to CYP1-mediated metabolism. Eupatorin-induced cell death is ...
T6S2238 Eupalinolide B Others
Eupalinolide A has the effects of relieving phlegm and relieving cough, clearing away heat and detoxification, diuretic swelling and reducing blood pressure.
T3362 Eupatilin NSC 122413 PPAR , Autophagy
Eupatilin (NSC-122413), a flavone derived from Artemisia princepsPampanini, is a PPARα agonist, with pharmacological activity.
T5826 Eupalinolide A HSP
Eupalinolide B is a natural product ,and demonstrates potent cytotoxicity against A-549, BGC-823, SMMC-7721, and HL-60 tumour cell lines.
TN3469 Aucuparin 2,6-dimethoxy-4-phenylphenol NADPH-oxidase
Aucuparin (2,6-dimethoxy-4-phenylphenol) is a plant antibiotic with anti-inflammatory activity. Aucuparin inhibited pulmonary fibrosis in mouse models induced by bleomycin (BLM). ABTS and FRAP showed clear scavenging act...
TN3503 Beta-Furoyleupatolide Others
Beta-Furoyleupatolide is a natural product for research related to life sciences. The catalog number is TN3503 and the CAS number is 114437-24-0.
TN4035 Eupalinolide I STAT
Eupalinolide I is a natural product from Eupatorium lindleyanum.
TN2693 2,3-Dihydro-12,13-dihydroxyeuparin Others
2,3-Dihydro-12,13-dihydroxyeuparin is a natural product for research related to life sciences. The catalog number is TN2693 and the CAS number is 135531-75-8.
T82432 Eupatolin
Eupatolin, a natural product, can be isolated from Rudbeckia hirta [1].
T80706 α-Isolupanine
α-Isolupanine, an alkaloid found in Narrow-Leafed Lupin (Lupinus angustifolius L.), can be isolated for the study of anthracnose [1].
T81653 Noraucuparin
Noraucuparin, a biphenyl-type phytoalexin with antifungal properties, can be isolated from the leaves of Sorbus pohuashanensis [1].
TN4038 Eupatolide TNF , NOS , NF-κB , ROS , MAPK , Akt , COX , DNA/RNA Synthesis , Nrf2 , PDGFR , NO Synthase , Prostaglandin Receptor , Autophagy
Eupatolide is isolated from the flowers of Inula japonica with anti-inflammatory activity. Eupatolide can be used in studies about TRAIL resistance in breast cancer cells.
T75644 Lupanine hydrochloride
Lupanine hydrochloride, a natural ketonic derivative of Sparteine ((+)-Sparteine), exhibits ganglioplegic activity and binds to the nicotinic receptor (nAChR) with a K i value of 500 nM [1].
T83452 13β-Hydroxylupanine
13β-Hydroxylupanine, a natural product, is present in Caulophyllum robustum Maxim [1].
TN4039 Eupatorin-5-methylether Others
Eupatorin-5-methylether is a natural product for research related to life sciences. The catalog number is TN4039 and the CAS number is 21764-09-0.
TN2843 2alpha-Hydroxyeupatolide 8-O-angelate Others
2alpha-Hydroxyeupatolide 8-O-angelate is a natural product from Eupatorium chinense var. tozanense.
TN1889 Lupalbigenin ERK , Akt , Topoisomerase
Lupalbigenin sensitizes detachment-induced cell death in human lung cancer cell through down-regulation of pro-survival proteins.
TN5531 Eupalitin 3,5,4'-Trihydroxy-6,7-dimethoxyflavone
Eupalitin is a natural product for research related to life sciences. The catalog number is TN5531 and the CAS number is 29536-41-2.
TN5362 20-Dehydroeupatoriopicrin semiacetal
20-Dehydroeupatoriopicrin semiacetal is a natural product for research related to life sciences. The catalog number is TN5362 and the CAS number is 94234-24-9.
TN2888 3,4-Secolupa-4(23),20(29)-diene-3,28-dioic acid Others
3,4-Secolupa-4(23),20(29)-diene-3,28-dioic acid exhibits potent inhibition of superoxide-anion generation with 86.9 ± 2.8% inhibition at 1 uM.
TN1628 Eupalinilide B Others
Eupalinilides B demonstrates potent cytotoxicity against P-388 and A-549 tumor cell lines.
TN1212 2-Hydroxyeupatolide Others , TNF , NF-κB
2-Hydroxyeupatolide has anti-inflammatory activity,it may suppress the inflammatory response through inhibiting the activation of NF-κB signaling pathways, and make a contribution to further understanding the pharmaceuti...
TN4037 Eupatarone Others
Eupatarone is a natural product from Eupatorium sternbergianum.
TN1631 Eupalinolide K STAT
Eupalinolide K is a natural product
TN4040 Eupatoriochromene Antifection
Eupatoriochromene retard seed germination , reduced radicle and hypocotyl growth of weed and crop plant seedlings and increased adventitious root formation of mung bean cuttings. Eupatoriochromene has insecticidal activi...
TN6574 13-Hydroxylupanine
13-Hydroxylupanine is a natural product from Cytisus scoparius.
TN4258 Isocuparenal Others
Isocuparenal is a natural product for research related to life sciences. The catalog number is TN4258 and the CAS number is 16982-01-7.
TN4308 Isolupalbigenin Antifection
Isolupalbigenin shows promising cytotoxic effects toward HL-60 cells (IC50 4.3 ± 0.7 to 18.0 ± 1.7 uM), it also shows in vitro inhibitory activity toward human glyoxalase I. Isolupalbigenin shows two different antibacter...
TN4034 Eupaglehnin C Others
Eupaglehnin C shows cytotoxic (2.19 mg/ml) against HeLa-S3.
TN2989 3alpha-Acetoxy-20-oxo-29-norlupane-23,28-dioic acid Others
3alpha-Acetoxy-20-oxo-29-norlupane-23,28-dioic acid is a natural product for research related to life sciences. The catalog number is TN2989 and the CAS number is 262272-76-4.
TN5964 Adiantulupanone
Adiantulupanone is a natural product for research related to life sciences. The catalog number is TN5964 and the CAS number is 51511-05-8.
TN2800 20-Hydroxy-3-oxo-28-lupanoic acid Others
20-Hydroxy-3-oxo-28-lupanoic acid is a natural product for research related to life sciences. The catalog number is TN2800 and the CAS number is 93372-87-3.
TN6563 Eupalinolide O
Eupalinolide O is a natural product for research related to life sciences. The catalog number is TN6563 and the CAS number is 2170228-67-6.
TN1632 Euparin Antifection
Euparin exhibits a moderate antioxidant activity, it also exhibits antifungal activity against Trichophyton mentagrophytes. Euparin has antiviral activity, it exerts its effect during the early events of the replication ...
TN3780 Deacetyleupaserrin Others
Deacetyleupaserrin is an antileukemic sesquiterpene lactone.
TN1629 Eupalinilide C Others
Eupalinilide C is a natural product from Impatiens balsamina L.
TN1630 Eupalinilide D Others
Eupalinilide D is a natural product from Impatiens balsamina L.
T78477 Drupanin
Drupanin, isolated from green propolis, selectively inhibits the AKR1C3 enzyme and shows promise for breast cancer research [1].
TN5160 Trans-2,3-Dihydro-3-ethoxyeuparin Others
trans-2,3-Dihydro-3-ethoxyeuparin is a natural product for research related to life sciences. The catalog number is TN5160 and the CAS number is 1015698-14-2.
TN2596 12-Hydroxy-2,3-dihydroeuparin Others
12-Hydroxy-2,3-dihydroeuparin is a natural product of Eupatorium, Asteraceae. The catalog number is TN2596 and the CAS number is 68776-42-1. 12-Hydroxy-2,3-dihydroeuparin can be used as a reference standard.
TMA0805 Lupanine ATPase , Potassium Channel , Calcium Channel
Lupanine has a weak sedative effect on the central nervous system, interaction with specific drugs used for treatment of the CNS and for analgesic activity. Lupanine improves glucose homeostasis by influencing KATP-chann...
TN5358 Eupahualin C
Eupahualin C shows significant activities against cell lines of human chronic myelogenous leukemia (K562) and human bone cancer (U2OS).
TN4041 Eupatoriopicrin Others
Eupatoriopicrin shows anti-trypanosomal activity and cytotoxicity against Trypanosoma brucei rhodesiense. Eupatoriopicrin-induced DNA damage may play a role in the observed cytotoxicity, it shows a weak sensitizing capac...
TN5161 Trans-2,3-Dihydro-3-hydroxyeuparin Others
trans-2,3-Dihydro-3-hydroxyeuparin is a natural product for research related to life sciences. The catalog number is TN5161 and the CAS number is 64185-57-5.
TN3899 Drupacine Others
Drupacine and a crude alkaloid extract suppress nematode hatch, activity of mixed life stages, and population numbers on plant roots.
T83454 13-Hydroxylupanine hydrochloride Hydroxylupanine hydrochloride
13-Hydroxylupanine, a characteristic alkaloid of sweet lupins, inhibits ganglionic transmission, reduces cardiac contractility, and induces contraction of uterine smooth muscle [1].
TN4036 Euparone Others
Euparone is a benzofuran from Ruscus aculeatus L..
TN1664 Ganoderic acid H NF-κB , DNA/RNA Synthesis , CDK
Ganoderic acid H is a potent antitumour agent, it mediates its biological effects through the inhibition of transcription factors AP-1 and NF-kappaB, resulting in the down-regulation of expression of Cdk4.
T5740 25(R,S)-Ruscogenin (25RS)-Ruscogenin Others , HIF
25(R,S)-Ruscogenin is a natual product.
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Natural Products

(+)-Cuparene
TN6762
Synonym:
Target: Others
Eupatorin
T7032
Synonym:
Target: Others, P450
Eupalinolide B
T6S2238
Synonym:
Target: Others
Eupatilin
T3362
Synonym: NSC 122413
Target: PPAR, Autophagy
Eupalinolide A
T5826
Synonym:
Target: HSP
Aucuparin
TN3469
Synonym: 2,6-dimethoxy-4-phenylphenol
Target: NADPH-oxidase
Beta-Furoyleupatolide
TN3503
Synonym:
Target: Others
Eupalinolide I
TN4035
Synonym:
Target: STAT
2,3-Dihydro-12,13-dihydroxyeuparin
TN2693
Synonym:
Target: Others
Eupatolin
T82432
Synonym:
Target:
α-Isolupanine
T80706
Synonym:
Target:
Noraucuparin
T81653
Synonym:
Target:
Eupatolide
TN4038
Synonym:
Target: TNF, NOS, NF-κB, ROS, MAPK, Akt, COX, DNA/RNA Synthesis, Nrf2, PDGFR, NO Synthase, Prostaglandin Receptor, Autophagy
Lupanine hydrochloride
T75644
Synonym:
Target:
13β-Hydroxylupanine
T83452
Synonym:
Target:
Eupatorin-5-methylether
TN4039
Synonym:
Target: Others
2alpha-Hydroxyeupatolide 8-O-angelate
TN2843
Synonym:
Target: Others
Lupalbigenin
TN1889
Synonym:
Target: ERK, Akt, Topoisomerase
Eupalitin
TN5531
Synonym: 3,5,4'-Trihydroxy-6,7-dimethoxyflavone
Target:
20-Dehydroeupatoriopicrin semiacetal
TN5362
Synonym:
Target:
3,4-Secolupa-4(23),20(29)-diene-3,28-dioic acid
TN2888
Synonym:
Target: Others
Eupalinilide B
TN1628
Synonym:
Target: Others
2-Hydroxyeupatolide
TN1212
Synonym:
Target: Others, TNF, NF-κB
Eupatarone
TN4037
Synonym:
Target: Others
Eupalinolide K
TN1631
Synonym:
Target: STAT
Eupatoriochromene
TN4040
Synonym:
Target: Antifection
13-Hydroxylupanine
TN6574
Synonym:
Target:
Isocuparenal
TN4258
Synonym:
Target: Others
Isolupalbigenin
TN4308
Synonym:
Target: Antifection
Eupaglehnin C
TN4034
Synonym:
Target: Others
3alpha-Acetoxy-20-oxo-29-norlupane-23,28-dioic acid
TN2989
Synonym:
Target: Others
Adiantulupanone
TN5964
Synonym:
Target:
20-Hydroxy-3-oxo-28-lupanoic acid
TN2800
Synonym:
Target: Others
Eupalinolide O
TN6563
Synonym:
Target:
Euparin
TN1632
Synonym:
Target: Antifection
Deacetyleupaserrin
TN3780
Synonym:
Target: Others
Eupalinilide C
TN1629
Synonym:
Target: Others
Eupalinilide D
TN1630
Synonym:
Target: Others
Drupanin
T78477
Synonym:
Target:
trans-2,3-Dihydro-3-ethoxyeuparin
TN5160
Synonym:
Target: Others
12-Hydroxy-2,3-dihydroeuparin
TN2596
Synonym:
Target: Others
Lupanine
TMA0805
Synonym:
Target: ATPase, Potassium Channel, Calcium Channel
Eupahualin C
TN5358
Synonym:
Target:
Eupatoriopicrin
TN4041
Synonym:
Target: Others
trans-2,3-Dihydro-3-hydroxyeuparin
TN5161
Synonym:
Target: Others
Drupacine
TN3899
Synonym:
Target: Others
13-Hydroxylupanine hydrochloride
T83454
Synonym: Hydroxylupanine hydrochloride
Target:
Euparone
TN4036
Synonym:
Target: Others
Ganoderic acid H
TN1664
Synonym:
Target: NF-κB, DNA/RNA Synthesis, CDK
25(R,S)-Ruscogenin
T5740
Synonym: (25RS)-Ruscogenin
Target: Others, HIF
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Recombinant Proteins

Species：
Human (10)
Mouse (7)
Cynomolgus (2)
Rat (2)
Expression System：
HEK293 Cells (18)
E. coli (3)
Tag：
C-His-Avi (7)
C-His (4)
His (3)
C-6xHis (1)
C-hFc (1)
C-mFc (1)
His, hFc (1)
N-10xHis, C-Myc (1)
N-6xHis (1)
N-6xHis-SUMO (1)
Cat No. Product Name Species Expression System
TMPK-00782 PLAU/uPA Protein, Mouse, Recombinant (His & Avi) Mouse HEK293 Cells
Plasminogen activator, urokinase (uPA) is a secreted serine protease whose Dysregulation is often accompanied by various cancers. PLAU inhibition could suppress tumor growth. Collectively, PLAU is necessary for tumor pro...
TMPY-00904 Urokinase/uPA Protein, Human, Recombinant (His) Human HEK293 Cells
Urokinase/uPA Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 46 kDa and the accession number is A0A024QZM9.
TMPK-00783 PLAU/uPA Protein, Mouse, Recombinant (His & Avi), Biotinylated Mouse HEK293 Cells
Plasminogen activator, urokinase (uPA) is a secreted serine protease whose Dysregulation is often accompanied by various cancers. PLAU inhibition could suppress tumor growth. Collectively, PLAU is necessary for tumor pro...
TMPK-00539 PLAU/uPA Protein (active form), Cynomolgus, Recombinant (His) Cynomolgus HEK293 Cells
Plasminogen activator, urokinase (uPA) is a secreted serine protease whose Dysregulation is often accompanied by various cancers. PLAU inhibition could suppress tumor growth. Collectively, PLAU is necessary for tumor pro...
TMPK-00274 PLAU/uPA Protein (active form), Human, Recombinant (His & Avi), Biotinylated Human HEK293 Cells
Plasminogen activator, urokinase (uPA) is a secreted serine protease whose Dysregulation is often accompanied by various cancers. PLAU inhibition could suppress tumor growth. Collectively, PLAU is necessary for tumor pro...
TMPY-03048 PRAP1 Protein, Human, Recombinant (mFc) Human HEK293 Cells
PRAP1 Protein, Human, Recombinant (mFc) is expressed in HEK293 mammalian cells with mFc tag. The predicted molecular weight is 41.4 kDa and the accession number is AAL16670.1.
TMPY-03076 PRAP1 Protein, Human, Recombinant (His) Human HEK293 Cells
PRAP1 Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 16.4 kDa and the accession number is AAL16670.1.
TMPY-04504 Urokinase/uPA Protein, Rat, Recombinant (His) Rat HEK293 Cells
Urokinase/uPA Protein, Rat, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 47.3 kDa and the accession number is A6KKR2.
TMPY-01257 uPAR/PLAUR Protein, Mouse, Recombinant (His) Mouse HEK293 Cells
uPAR/PLAUR Protein, Mouse, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 31.4 kDa and the accession number is P35456-1.
TMPY-02141 uPAR/PLAUR Protein, Human, Recombinant (His) Human HEK293 Cells
uPAR/PLAUR Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 32.8 kDa and the accession number is Q03405-1.
TMPY-01017 uPAR/PLAUR Protein, Mouse, Recombinant (His & hFc) Mouse HEK293 Cells
uPAR/PLAUR Protein, Mouse, Recombinant (His & hFc) is expressed in HEK293 mammalian cells with His and hFc tag. The predicted molecular weight is 58 kDa and the accession number is P35456-1.
TMPK-00227 uPAR/PLAUR Protein, Human, Recombinant (His & Avi), Biotinylated Human HEK293 Cells
The receptor (u-PAR) for urokinase plasminogen activator (u-PA) is a three-domain protein, GPI-anchored to the cell surface, which focuses the enzymatic activity of u-PA, and allows the cell surface activation of plasmin...
TMPK-00216 uPAR/PLAUR Protein, Mouse, Recombinant (His & Avi), Biotinylated Mouse HEK293 Cells
The receptor (u-PAR) for urokinase plasminogen activator (u-PA) is a three-domain protein, GPI-anchored to the cell surface, which focuses the enzymatic activity of u-PA, and allows the cell surface activation of plasmin...
TMPK-00226 uPAR/PLAUR Protein, Human, Recombinant (His & Avi) Human HEK293 Cells
The receptor (u-PAR) for urokinase plasminogen activator (u-PA) is a three-domain protein, GPI-anchored to the cell surface, which focuses the enzymatic activity of u-PA, and allows the cell surface activation of plasmin...
TMPK-00215 uPAR/PLAUR isoform 1 Protein, Mouse, Recombinant (His & Avi) Mouse HEK293 Cells
The receptor (u-PAR) for urokinase plasminogen activator (u-PA) is a three-domain protein, GPI-anchored to the cell surface, which focuses the enzymatic activity of u-PA, and allows the cell surface activation of plasmin...
TMPK-00228 uPAR/PLAUR Protein, Human, Recombinant (hFc) Human HEK293 Cells
The receptor (u-PAR) for urokinase plasminogen activator (u-PA) is a three-domain protein, GPI-anchored to the cell surface, which focuses the enzymatic activity of u-PA, and allows the cell surface activation of plasmin...
TMPK-01175 uPAR/PLAUR Protein, Cynomolgus, Recombinant (His) Cynomolgus HEK293 Cells
The receptor (u-PAR) for urokinase plasminogen activator (u-PA) is a three-domain protein, GPI-anchored to the cell surface, which focuses the enzymatic activity of u-PA, and allows the cell surface activation of plasmin...
TMPH-03397 uPAR/PLAUR Protein, Rat, Recombinant (His) Rat E. coli
Acts as a receptor for urokinase plasminogen activator. Plays a role in localizing and promoting plasmin formation. Mediates the proteolysis-independent signal transduction activation effects of U-PA. uPAR/PLAUR Protein,...
TMPH-02945 TMPRSS4 Protein, Mouse, Recombinant (His & SUMO) Mouse E. coli
Plasma membrane-anchored serine protease that directly induces processing of pro-uPA/PLAU into the active form through proteolytic activity. Seems to be capable of activating ENaC. TMPRSS4 Protein, Mouse, Recombinant (Hi...
TMPH-02239 TMPRSS4 Protein, Human, Recombinant (His & Myc) Human E. coli
Plasma membrane-anchored serine protease that directly induces processing of pro-uPA/PLAU into the active form through proteolytic activity. Seems to be capable of activating ENaC.; (Microbial infection) In gut epithelia...
TMPJ-00490 Serpin A5 Protein, Human, Recombinant (His) Human HEK293 Cells
Serpin A5 is a member of the human Serpin superfamily consists of at least 35 members. It is synthesized in the liver and has been detected in saliva, cerebral spinal fluid, amniotic fluid, tears and semen. As a potent i...
PLAU/uPA Protein, Mouse, Recombinant (His & Avi)
TMPK-00782
Species: Mouse
Expression System: HEK293 Cells
Urokinase/uPA Protein, Human, Recombinant (His)
TMPY-00904
Species: Human
Expression System: HEK293 Cells
PLAU/uPA Protein, Mouse, Recombinant (His & Avi), Biotinylated
TMPK-00783
Species: Mouse
Expression System: HEK293 Cells
PLAU/uPA Protein (active form), Cynomolgus, Recombinant (His)
TMPK-00539
Species: Cynomolgus
Expression System: HEK293 Cells
PLAU/uPA Protein (active form), Human, Recombinant (His & Avi), Biotinylated
TMPK-00274
Species: Human
Expression System: HEK293 Cells
PRAP1 Protein, Human, Recombinant (mFc)
TMPY-03048
Species: Human
Expression System: HEK293 Cells
PRAP1 Protein, Human, Recombinant (His)
TMPY-03076
Species: Human
Expression System: HEK293 Cells
Urokinase/uPA Protein, Rat, Recombinant (His)
TMPY-04504
Species: Rat
Expression System: HEK293 Cells
uPAR/PLAUR Protein, Mouse, Recombinant (His)
TMPY-01257
Species: Mouse
Expression System: HEK293 Cells
uPAR/PLAUR Protein, Human, Recombinant (His)
TMPY-02141
Species: Human
Expression System: HEK293 Cells
uPAR/PLAUR Protein, Mouse, Recombinant (His & hFc)
TMPY-01017
Species: Mouse
Expression System: HEK293 Cells
uPAR/PLAUR Protein, Human, Recombinant (His & Avi), Biotinylated
TMPK-00227
Species: Human
Expression System: HEK293 Cells
uPAR/PLAUR Protein, Mouse, Recombinant (His & Avi), Biotinylated
TMPK-00216
Species: Mouse
Expression System: HEK293 Cells
uPAR/PLAUR Protein, Human, Recombinant (His & Avi)
TMPK-00226
Species: Human
Expression System: HEK293 Cells
uPAR/PLAUR isoform 1 Protein, Mouse, Recombinant (His & Avi)
TMPK-00215
Species: Mouse
Expression System: HEK293 Cells
uPAR/PLAUR Protein, Human, Recombinant (hFc)
TMPK-00228
Species: Human
Expression System: HEK293 Cells
uPAR/PLAUR Protein, Cynomolgus, Recombinant (His)
TMPK-01175
Species: Cynomolgus
Expression System: HEK293 Cells
uPAR/PLAUR Protein, Rat, Recombinant (His)
TMPH-03397
Species: Rat
Expression System: E. coli
TMPRSS4 Protein, Mouse, Recombinant (His & SUMO)
TMPH-02945
Species: Mouse
Expression System: E. coli
TMPRSS4 Protein, Human, Recombinant (His & Myc)
TMPH-02239
Species: Human
Expression System: E. coli
Serpin A5 Protein, Human, Recombinant (His)
TMPJ-00490
Species: Human
Expression System: HEK293 Cells
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