Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Upamostat is an inhibitor of a serine protease and is a urokinase plasminogen activator (uPA) inhibitor.
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
1 mg | In stock | $ 97.00 | |
5 mg | In stock | $ 247.00 | |
10 mg | In stock | $ 397.00 | |
25 mg | In stock | $ 663.00 | |
50 mg | In stock | $ 945.00 | |
100 mg | In stock | $ 1,280.00 | |
1 mL * 10 mM (in DMSO) | In stock | $ 343.00 |
Description | Upamostat is an inhibitor of a serine protease and is a urokinase plasminogen activator (uPA) inhibitor. |
In vitro | Upamostat is an inhibitor of urokinase plasminogen activator (uPA). Upamostat is the oral prodrug of the active metabolite WX-UK1, a novel inhibitor of uPA [1]. Upamostat inhibits the urokinase-type plasminogen activator (uPA) system, and plays a major role in tumor invasion and metastasis. Upamostat is the orally available amidoxime- (i.e. hydroxyamidine-) prodrug of the pharmacologically active form, WX-UK1 [2]. |
Molecular Weight | 629.81 |
Formula | C32H47N5O6S |
CAS No. | 590368-25-5 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 250 mg/mL (396.95 mM)
You can also refer to dose conversion for different animals. More
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Upamostat 590368-25-5 Cell Cycle/Checkpoint Metabolism Proteases/Proteasome PAI-1 Serine/threonin kinase Serine Protease inhibit Threonine proteases WX 671 Inhibitor Ser/Thr Protease Plasminogen activator inhibitor-1 Serine endopeptidases WX-671 WX671 Serine proteases inhibitor