Search Result

Search Results for " hts "

Targets

Compounds

Natural Products

Recombinant Proteins

Libraries

Cat No.	Product Name	Synonyms	Targets
T16275	NB001	HTS 09836	Adenylyl cyclase
	NB001 (HTS 09836) is an inhibitor of adenyl cyclase 1 exhibiting effects on neural and non-neural pain.		Adenylyl cyclase
T2048	LY-364947	LY 364947,HTS466284	MLK , Casein Kinase , TGF-beta/Smad , RIP kinase
	LY-364947 (HTS466284) is a potent ATP-competitive inhibitor of TGFβR-I.		MLK , Casein Kinase , TGF-beta/Smad , RIP kinase
T32453	L 650719	6-HTS,L650719,L-650719
	L 650719 is a bioactive chemical.
T15506	HTS01037		Others
	HTS01037 is an inhibitor of fatty acid-binding. HTS01037 is a competitive antagonist of protein-protein interactions mediated by AFABP/aP2 (Ki: 0.67 μM).		Others
T61316	HTS07545		NADPH
	HTS07545 is a potent sulfide:quinone oxidoreductase inhibitor (IC50: 30 nM).HTS07545 reduces the rate of hydrogen sulfide (H2S) decomposition.HTS07545 has been used in heart failure studies.		NADPH
T34055	Phtstllap
	Phtstllap is a luteinizing hormone-releasing factor
T4178	NSC 80538		Others
	NSC 80538 is an inhibitor of MEK Kinase PB1 Domains in multiplex HTS assays.		Others
T4531	GSK2200150A		Antibacterial
	GSK2200150A is an anti-tuberculosis (TB) agent identified by high-throughput screening (HTS) campaign.		Antibacterial
T9256	N-Cyclohexyl-4-[1-(1-piperazinyl)-2,6-naphthyridin-3-yl]-2-pyridinamine		Serine/threonin kinase , PKC
	N-Cyclohexyl-4-[1-(1-piperazinyl)-2,6-naphthyridin-3-yl]-2-pyridinamine is a novel 2,6-naphthyridine identified by high throughput screen (HTS) as a dual protein kinase C/D (PKC/PKD) inhibitor[1].		Serine/threonin kinase , PKC
T8411	C-215		Others
	C-215 is a novel inhibitor of mycobacterial membrane protein large 3 (MmpL3).		Others
T83800	6-Biotin-17-NAD+ sodium	6-Biotin-17-Nicotinamide adenine dinucleotide,β-Nicotinamide-N6-(2-(6-(6-[biotinyl]aminohexanoyl)aminohexanoyl)aminoethyl)adenine dinucleotide
	6-Biotin-17-NAD+, a biotinylated derivative of the signaling molecule and enzyme cofactor NAD+, is utilized in high-throughput screening (HTS) assays to measure the activity of mitochondrial complex I, also referred to a...

Compounds

NB001

T16275

Synonym: HTS 09836

Target: Adenylyl cyclase

LY-364947

T2048

Synonym: LY 364947,HTS466284

Target: MLK, Casein Kinase, TGF-beta/Smad, RIP kinase

L 650719

T32453

Synonym: 6-HTS,L650719,L-650719

Target: Antibacterial

N-Cyclohexyl-4-[1-(1-piperazinyl)-2,6-naphthyridin-3-yl]-2-pyridinamine

T9256

Synonym:

Target: Serine/threonin kinase, PKC

6-Biotin-17-NAD+ sodium

T83800

Synonym: 6-Biotin-17-Nicotinamide adenine dinucleotide,β-Nicotinamide-N6-(2-(6-(6-[biotinyl]aminohexanoyl)aminohexanoyl)aminoethyl)adenine dinucleotide

Target:

Cat No.	Product Name	Synonyms	Targets
T6808	Coelenterazine	Oplophorus luciferin,Coelenteramine	Others
	Coelenterazine (Coelenteramine) is a luminescent enzyme substrate, used for monitoring reporter genes in BRET, ELISA and HTS techniques.		Others

Natural Products

Coelenterazine

T6808

Synonym: Oplophorus luciferin,Coelenteramine

Target: Others

Recombinant Proteins

Species：

Expression System：

Tag：

Cat No.	Product Name	Species	Expression System
TMPK-00311	APCDD1 Protein, Human, Recombinant (His)	Human	HEK293 Cells
	APCDD1 Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with C-His tag. The predicted molecular weight is 54.4 kDa and the accession number is Q8J025.
TMPK-00989	APCDD1 Protein, Mouse, Recombinant (His)	Mouse	HEK293 Cells
	APCDD1 Protein, Mouse, Recombinant (His) is expressed in HEK293 mammalian cells with C-His tag. The predicted molecular weight is 54.4 kDa and the accession number is Q3U128.
TMPY-03046	APCDD1 Protein, Human, Recombinant (hFc)	Human	HEK293 Cells
	Osteosarcoma (OS) is the most common type of bone tumor in children and adults. The expression of APCDD1, a Wnt antagonist, was reduced in OS tissues and cells compared to adjacent normal tissue and osteoblast cells, res...

APCDD1 Protein, Human, Recombinant (His)

TMPK-00311

Species: Human

Expression System: HEK293 Cells

APCDD1 Protein, Mouse, Recombinant (His)

TMPK-00989

Species: Mouse

Expression System: HEK293 Cells

APCDD1 Protein, Human, Recombinant (hFc)

TMPY-03046

Species: Human

Expression System: HEK293 Cells

Cat No.	Product Name
L6000	Natural Product Library for HTS	4533 compounds
	A unique collection of 4533 pure natural products and their derivatives with known biological activity for drug discovery, pharmacological study, stem cell differentiation, fingerprint study and quality research, and can...
L7000	Bioactive Lipid Compound Library	385 compounds
	A unique collection of 385 bioactive lipids related compounds for high throughput screening (HTS) and high content screening (HCS), including Agonists & Antagonists, Endocannabinoids, Farnesyl/geranylgeranyl derivates, ...
L1000	Approved Drug Library	2808 compounds
	A unique collection of 2808 approved drugs for high throughput screening (HTS) and high content screening (HCS);
L2530	Mouse Metabolite Compound Library	218 compounds
	A unique collection of 218 mouse metabolites, which can be used for HTS and HCS;
L5610	Golden Scaffold Library	10000 compounds
	Diversity: Selected from 1,600,000 drug-like compounds, 10000compounds representing 5000 scaffolds selected from a large drug-like chemical source；
L5700	Featured Fragment Library	246 compounds
	A unique collection of 246 fragment-like small molecules for FBDD;
LF1000	Pre-plated Diversity Sets	50000 compounds
	For your convenience, there are Diversity Sets of 5,000, 10,000, 15,000, and 20,000 compounds with no structure overlap.
L3410	Preclinical Compound Library	701 compounds
	A unique collection of 701 preclinical compounds for high throughput screening (HTS) and high content screening (HCS);
L6100	Polyphenolic Natural Product Library	635 compounds
	A unique collection of 635 natural polyphenolic compounds for high throughput screening (HTS) and high content screening (HCS);
L3900	DNA Damage & Repair Compound Library	910 compounds
	A unique collection of 910 DNA Damage & Repair related compounds for high throughput screening (HTS) and high content screening (HCS);
L5500	Toxic Compound Library	262 compounds
	A unique collection of 262 toxic substances for high throughput screening (HTS) and high content screening (HCS);
L8800	Drug-Fragment Library	1119 compounds
	1119 drug fragments，a must-have tool for FBDD;
L9200	Drug Repurposing Compound Library	4541 compounds
	A unique collection of 4541 approved and clinical drugs for high throughput screening (HTS) and high content screening (HCS);
L3980	DNA Damage and Repair Compound Library Plus	667 compounds
	Well-chosen 667 compounds with unique structures targeting DNA damage & repair;
L1010	FDA-Approved & Pharmacopeia Drug Library	3157 compounds
	3157 compounds from marketed drugs for high throughput screening (HTS) and high content screening (HCS);
L4200	FDA-Approved Drug Library	1729 compounds
	A unique collection of 1729 FDA approved drugs for high throughput screening (HTS) and high content screening (HCS);
L5200	Anti-Metabolism Disease Compound Library	1544 compounds
	A unique collection of 1544 metabolism diseases related compounds for high throughput screening (HTS) and high content screening (HCS);
L3400	Clinical Compound Library	3404 compounds
	A unique collection of 3404 compounds in clinical trial phases for high throughput screening (HTS) and high content screening (HCS);
L6700	Anti-Tumor Natural Product Library	1772 compounds
	A unique collection of 1772 natural products with known anti-cancer activity for high throughput screening (HTS) and high content screening (HCS);
L6010	Natural Product Library	3840 compounds
	A unique collection of 3840 natural products for high throughput screening (HTS) and high content screening (HCS);
L5800	Drug Metabolite/Impurity Library	197 compounds
	A unique collection of 197 drug isomers/metabolites for high throughput screening (HTS) and high content screening (HCS);
L2620	Anti-Neurodegenerative Disease Compound Library	2154 compounds
	A unique collection of 2154 compounds related to neurodegenerative diseases can be used for HTS or HCS；
L6160	RO5 Drug-like Natural Product Library	2703 compounds
	A unique collection of 2703 natural product monomers that meet the "Lipinski's Rule of Five", a powerful tool for HTS and HCS screening;
L9820	Beta-Lactam Compound Library	97 compounds
	A unique collection of 97 beta-lactam compounds, can be used in HTS and HCS;
L2000	Inhibitor Library	8328 compounds
	A unique collection of 8328 inhibitors for research in cell signaling, high throughput screening (HTS) and high content screening (HCS) for new drugs;
L6610	Anti-infective Natural Product Library	1060 compounds
	A unique collection of 1060 species of natural products with anti-infective activity for high throughput screening (HTS) and high content screening (HCS);
L2150	Anti-Cancer Drug Library	3080 compounds
	A unique collection of 3080 anticancer drugs for high throughput screening (HTS) and high content screening (HCS);
L6900	Rare Natural Product Library	693 compounds
	A unique collection of 693 rare natural products, which can be used for high throughput screening (HTS) and high content screening (HCS);
L3200	Autophagy Compound Library	1248 compounds
	A unique collection of 1248 compounds with defined autophagy-inducing or -inhibitory activity for research in autophagy, high throughput screening (HTS) and high content screening (HCS) for new drugs;
L3500	Histone Modification Compound Library	469 compounds
	A unique collection of 469 histone modification related compounds for high throughput screening (HTS) and high content screening (HCS);
L2400	Endocrinology-Hormone Compound Library	784 compounds
	A unique collection of 784 compounds targeting endocrine system for high throughput screening (HTS) and high content screening (HCS) for new drugs;
L9810	Anti-Fibrosis Compound Library	1180 compounds
	A unique collection of 1180 potential anti-fibrosis compounds, can be used in HTS and HCS;
L5900	CNS-Penetrant Compound Library	509 compounds
	A unique collection of 509 CNS-Penetrant compounds for high throughput screening (HTS) and high content screening (HCS);
L4800	Angiogenesis related Compound Library	1353 compounds
	A unique collection of 1353 proangiogenic and antiangiogenic compounds for new targets identification, research in mechanisms of angiogenesis, and high throughput screening (HTS) and high content screening (HCS);
L1200	Epigenetics Compound Library	953 compounds
	Well-chosen 953 compounds related to epigenetic regulation for research in epigenetics, high throughput screening (HTS) and high content screening (HCS) for new drugs;
L2160	Anti-Cancer Active Compound Library	3188 compounds
	A unique collection of 3188 compounds with known anti-cancer activity for high throughput screening (HTS) and high content screening (HCS);
L2192	Anti-Pancreatic Cancer Compound Library	2238 compounds
	A unique collection of 2238 pancreatic cancer related compounds can be used in HTS and HCS;
L5400	Anti-Cardiovascular Disease Compound Library	1408 compounds
	A unique collection of 1408 cardiovascular diseases related compounds for high throughput screening (HTS) and high content screening (HCS);
L2100	Anti-Cancer Compound Library	7234 compounds
	A unique collection of 7234 compounds with anti-cancer activity for high throughput screening (HTS) and high content screening (HCS);
L2120	Anti-Cancer Clinical Compound Library	2545 compounds
	A unique collection of 2545 anti-cancer compounds for high throughput screening (HTS) and high content screening (HCS);
L6620	Antiparasitic Natural Product Library	253 compounds
	A unique collection of 253 natural products with antiparasitic activity, a powerful tool for high throughput screening (HTS) and high content screening (HCS);
L6600	Anti-Gastroenteritis Natural Product Library	219 compounds
	A unique collection of 219 natural products related to gastroenteritis for high throughput screening (HTS) and high content screening (HCS);
L8200	Anti-Aging Compound Library	3279 compounds
	A unique collection of 3279 anti-aging compounds for high throughput screening (HTS) and high content screening (HCS);
L8300	Chromatin Modification Compound Library	250 compounds
	A unique collection of 250 compounds targeting chromatin remodeling pathway for high throughput screening (HTS) and high content screening (HCS);
L8100	Cell Cycle Compound Library	677 compounds
	A unique collection of 677 cell cycle related compounds for high throughput screening (HTS) and high content screening (HCS);
L6140	Saccharide and Glycoside Natural Product Library	362 compounds
	A unique collection of 362 saccharides and glycosides compounds can be used for HTS and HCS；
L8400	Hematonosis Compound Library	514 compounds
	A unique collection of 514 compounds related to hematologic diseases for high throughput screening (HTS) and high content screening (HCS);
L4000	Bioactive Compound Library	14439 compounds
	A collection of 14439 small molecule compounds with validated activity for high throughput screening (HTS), high content screening (HCS), cell induction, and target identification;
L2110	Anti-Cancer Approved Drug Library	1779 compounds
	A unique collection of 1779 approved anti-cancer drugs for high throughput screening (HTS) and high content screening (HCS);
L7500	Coagulation and Anticoagulation Compound Library	144 compounds
	A unique collection of 144 procoagulation and anticoagulation related compounds for high throughput screening (HTS) and high content screening (HCS);
L2600	Neuronal Signaling Compound Library	2540 compounds
	A unique collection of 2540 compounds targeting CNS signaling for high throughput screening (HTS) and high content screening (HCS) for new drugs;
L3300	Histamine & Melatonin Receptor-Targeted Compound Library	153 compounds
	A unique collection of 153 compounds targeting histaminergic receptor and melatonin receptor for high throughput screening (HTS) and high content screening (HCS) for new drugs;
L9700	Endoplasmic Reticulum Stress Compound Library	193 compounds
	A unique collection of 193 endoplasmic reticulum stress (ER stress) related compounds used for high throughput screening (HTS) and high content screening (HCS);
L5100	Fluorochemical Library	574 compounds
	A unique collection of 574 fluorochemicals that can be used for high through-put screening (HTS) and high content screening (HCS);
L1110	Microtubule-Targeted Compound Library	142 compounds
	A unique collection of 142 microtubule-targeted compounds can be used in HTS and HCS;
L2130	Anti-Cancer Metabolism Compound Library	1268 compounds
	A unique collection of 1268 cancer cellular metabolism related compounds for cancer research and high throughput screening (HTS) and high content screening (HCS);
L2520	Glycometabolism Compound Library	702 compounds
	702 glycometabolism-related comounds, can be used for HTS and HCT;
L2510	Lipid Metabolism Compound Library	492 compounds
	A unique collection of 492 compounds targeting lipid metabolism, can be used for high-throughput screening (HTS) and high-content screening (HCS).
L2540	Gut Microbial Metabolite Library	607 compounds
	A unique collection of 607 gut microbial metabolites which can be used for HTS and HCS;
L5510	Drug-induced Liver Injury (DILI) Compound Library	1001 compounds
	A unique collection of 1001 hepatotoxicity causing compounds, a powerful tool for drug toxicity study, can be used for HTS and HCS screening；
L4600	Selected Plant-Sourced Compound Library	3048 compounds
	A unique collection of 3048 plant-sourced compounds that derived from 277 plant species for high throughput screening (HTS) and high content screening (HCS);
L2610	Neurotransmitter Receptor Compound Library	1513 compounds
	A unique collection of 1513 neurotransmitter receptor compounds, can be used for HTS and HCS screening；
L1310	Cytoskeletal Signaling Pathway Compound Library	759 compounds
	A unique collection of 759 cytoskeleton-related compounds, can be used for HTS and HCS；
L9830	Anti-Parkinson's Disease Compound Library	857 compounds
	A unique collection of 857 compounds with anti-PD activities or acting on main drug targets of PD can be used for HTS and HCS.
L6400	Marine Natural Product Library	144 compounds
	A unique collection of 144 marine natural products for high throughput screening (HTS) and high content screening (HCS);
L6500	Microbial Natural Product Library	550 compounds
	A unique collection of 550 microbial natural products for high throughput screening (HTS) and high content screening (HCS);
L6720	Anti-COVID-19 Traditional Chinese Medicine Compound Library	1147 compounds
	A unique collection of 1147 monomers from 60 TCM plants, a powerful tool for anti-COVID-19 drug discovery, can be used for HTS and HCS screening；
L9840	Anti-Alzheimer's Disease Compound Library	986 compounds
	A unique collection of 986 compounds with anti-AD activities or acting on main drug targets of AD can be used for HTS and HCS.
L2550	Glutamine Metabolism Compound Library	565 compounds
	A unique collection of 565 glutamine metabolism related compounds can be used for high throughput screening (HTS) and high content screening (HCS), and also is an effective tool for research in glutamine metabolism and ...