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Epigenetics Compound Library

Catalog No. L1200
  Library Compound List   Excel SDF

Epigenetics is the study of molecular processes that influence the flow of information between a constant DNA sequence and variable gene expression patterns. This includes investigation of nuclear organization, DNA methylation, histone modification and RNA transcription. Epigenetic processes can result in intergenerational (heritable) effects as well as clonal propagation of cell identity without any mutational change in DNA sequence. Epigenetics has the potential to be a key element in a paradigm change of our understanding of aging, development, cancer, heart disease, psychological disorders, and other diseases. For example, Epigenetic modifications have a considerable effect on cancer. Changes in the pattern of histone modifications in the promoter sequences as epigenetic regulation lead to changes in chromatin structure thus may be the cause of altered gene expression by activation of oncogenes.

The Epigenetics Compound Library by TargetMol, containing 960 compounds related to epigenetic regulation, can be used for research in epigenetics, high throughput screening and high content screening for new drugs in epigenetic modification.

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.
Compound Libraries | TargetMol
Pack Size
1 mg
30 μL * 10 mM (in DMSO)
50 μL * 10 mM (in DMSO)
100 μL * 10 mM (in DMSO)
250 μL * 10 mM (in DMSO)
If the above compound libraries do not match your needs,
please contact our compound library specialist for a customized compound library at inquiry@targetmol.com
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Product Description

  • Quantity: well-chosen 960 compounds related to epigenetic regulation for research in epigenetics, high throughput screening (HTS) and high content screening (HCS) for new drugs;
  • Targets include HDAC, SIRT, HAT, and HMT, etc.;
  • Detailed compound information with structure, target, activity, IC50 value, and biological activity description, providing reference for your experimental design;
  • NMR and LCMS/HPLC validated to ensure high purity and quality.
  • Structurally diverse, medicinally active, and cell permeable;
  • NMR and HPLC validated to ensure high purity and quality;

Library Customization

Targetmol Compound Libraries can be highly customized! Learn More

Packaging And Storage

  • Powder or pre-dissolved DMSO solutions in 96/384 well plate with optional 2D barcode
  • Shipped with blue ice
Request Library Compound List (L1200)

Publications Cited TargetMol Libraries

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Library Composition

Apoptosis (156)
Epigenetic Reader Domain (144)
Histone Methyltransferase (117)
HDAC (111)
Autophagy (100)
JAK (98)
PKC (78)
AMPK (77)
PARP (75)
Sirtuin (58)
Aurora Kinase (53)
HIF/HIF Prolyl-Hydroxylase (49)
HIF (36)
Histone Demethylase (36)
Histone Acetyltransferase (29)
Tyrosine Kinases (27)
CDK (27)
Endogenous Metabolite (25)
FLT (24)
Antibacterial (23)
DNA Methyltransferase (23)
Pim (21)
STAT (20)
HIV Protease (18)
Influenza Virus (16)
PKA (16)
Akt (16)
VEGFR (15)
Mitophagy (15)
Src (15)
Antibiotic (14)
Parasite (13)
Caspase (13)
EGFR (13)
ERK (12)
Wnt/beta-catenin (12)
FGFR (10)
NF-κB (10)
COX (10)
PDGFR (10)
BCL (10)
Reactive Oxygen Species (10)
PPAR (9)
Bcr-Abl (9)
Virus Protease (9)
p38 MAPK (9)
Topoisomerase (8)
c-RET (8)
ROCK (8)
Syk (8)
P450 (7)
PAD (7)
DNA/RNA Synthesis (7)
TNF (7)
MEK (7)
Casein Kinase (7)
PI3K (7)
GSK-3 (7)
IL Receptor (6)
PLK (6)
JNK (6)
Nrf2 (6)
Antifungal (6)
Adenosine Receptor (5)
AChR (5)
PDE (5)
Ferroptosis (5)
Methionine Adenosyltransferase (MAT) (5)
Calcium Channel (5)
Dehydrogenase (5)
S6 Kinase (5)
CaMK (5)
Serine/threonin kinase (5)
HSV (4)
NO Synthase (4)
MAO (4)
IκB/IKK (4)
Chk (4)
p53 (4)
Monoamine Oxidase (3)
IGF-1R (3)
c-Fms (3)
MAPK (3)
HER (3)
MMP (3)
mTOR (3)
GABA Receptor (3)
HBV (3)
DYRK (3)
IFNAR (3)
Trk receptor (3)
RAAS (3)
Histamine Receptor (3)
Nucleoside Antimetabolite/Analog (3)
Potassium Channel (3)
BTK (3)
SGK (3)
Ligand for E3 Ligase (2)
cholecystokinin (2)
MLK (2)
Hippo pathway (2)
ATP Citrate Lyase (2)
TLR (2)
PROTACs (2)
Phosphatase (2)
Sodium Channel (2)
AChE (2)
TGF-beta/Smad (2)
Serine Protease (2)
Antiviral (2)
YAP (2)
Anti-infection (2)
Dopamine Receptor (2)
Carboxypeptidase (2)
DNA Alkylation (2)
Tyrosinase (2)
Ligands for Target Protein for PROTAC (2)
transporter (2)
LDL (2)
Gamma-secretase (2)
5-HT Receptor (2)
Fatty Acid Synthase (2)
Integrin (2)
Microtubule Associated (2)
Myosin (2)
HCV Protease (2)
DUB (2)
Indoleamine 2,3-Dioxygenase (IDO) (2)
c-Kit (2)
Proteasome (1)
ribosome (1)
Phospholipase (1)
Cannabinoid Receptor (1)
DAPK (1)
NADPH-oxidase (1)
NOD (1)
BMI-1 (1)
TAM Receptor (1)
CFTR (1)
PD-1/PD-L1 (1)
Reverse Transcriptase (1)
PTEN (1)
Beta Amyloid (1)
NADPH (1)
SIK (1)
IAP (1)
Adrenergic Receptor (1)
Glucokinase (1)
Antifolate (1)
Estrogen Receptor/ERR (1)
c-Myc (1)
Tie-2 (1)
PERK (1)
BACE (1)
UGT (1)
Antioxidant (1)
c-Met/HGFR (1)
Estrogen/progestogen Receptor (1)
DNA-PK (1)
NPC1L1 (1)
Transferase (1)
Carbonic Anhydrase (1)
NOS (1)
Proton pump (1)
Chloride channel (1)
E1/E2/E3 Enzyme (1)
GRK (1)
GST (1)
Lipoxygenase (1)
Free radical scavengers (1)
LRRK2 (1)
SARS-CoV (1)
HSP (1)
P-gp (1)
Beta-Secretase (1)
SGLT (1)
Telomerase (1)
Interleukin (1)
Androgen Receptor (1)
GluR (1)
Raf (1)
Mdm2 (1)
CCR (1)
Hedgehog/Smoothened (1)
Guanylate cyclase (1)
ROS (1)
Antifection (1)
Mitochondrial Metabolism (1)
DNA gyrase (1)
NMDAR (1)
P2X Receptor (1)
S1P Receptor (1)

Library Information Sample

Empty 1000025-07-9 1000413-72-8 229005-80-5 1000787-75-6 946387-07-1 1000998-59-3 1175526-27-8 1001288-58-9 1001350-96-4 1001404-83-6 Empty
Vadadustat TAK875 TAK-779 Tegobuvir RN-1734 BMS-687453 AM211 FT011 BMS754807 AAI101
Empty 1001625-82-6 1001645-58-4 1001753-24-7 1001908-89-9 1002304-34-8 1002-84-2 100291-86-9 100299-08-9 10030-52-1 10040-45-6 Empty
RPW-24 SRT1720 hydrochloride INH6 SRT 2183 AMG208 Pentadecanoic acid Apiopaeonoside Pemirolast potassium L-Anserine nitrate salt Sodium Picosulfate
Empty 100427-26-7 1004316-88-4 10045-45-1 100462-37-1 1004990-28-6 100-51-6 1005-24-9 1005264-47-0 1005334-57-5 1005342-46-0 Empty
Lercanidipine Cobicistat 1-Ethyl-2-benzimidazolinone ROSIRIDIN PF-AKT400 Benzyl alcohol 1-Methylnicotinamide chloride MX69 CVT-10216 LCL161
Empty 1005491-05-3 100-55-0 1005504-62-0 1005883-72-6 100643-71-8 1007207-67-1 10075-50-0 1007647-73-5 100784-20-1 10083-24-6 Empty
Tirasemtiv Roniacol Rg3039 Z433927330 Desloratadine CH5132799 5-Bromoindole Smurf1-IN-A01 Halosulfuron-methyl Piceatannol
Empty 100872-83-1 100874-08-6 1009119-64-5 1009119-65-6 100929-71-3 1009298-09-2 1009298-59-2 100929-99-5 1009734-33-1 10097-84-4 Empty
ML346 SB 4 Daclatasvir Daclatasvir dihydrochloride NADPH (tetracyclohexanamine) AZD8055 Vistusertib PAβN dihydrochloride HZ1157 Rotundine
Empty 1009816-48-1 1009817-63-3 1009820-21-6 100986-85-4 101001-34-7 1010411-21-8 1010-60-2 1011244-68-0 1011301-27-1 1011529-10-4 Empty
Thiamet G B-AP15 Silmitasertib Levofloxacin Pamicogrel GSK369796 Dihydrochloride 2-Chloronaphthoquinone TFAP Tenovin3 Azvudine
Empty 101152-94-7 101155-02-6 1011557-82-6 1011-74-1 101-20-2 1012054-59-9 101-21-3 101-26-8 101303-98-4 1013101-36-4 Empty
Milnacipran hydrochloride BW-A78U Tenovin-6 DL-Normetanephrine hydrochloride Triclocarban CUDC101 Chlorpropham Mestinon Zacopride hydrochloride PF04691502
Empty 101-31-5 1013-69-0 1013750-77-0 1013753-99-5 10138-52-0 1013920-15-4 1013937-63-7 1014691-61-2 101477-54-7 101494-95-5 Empty
L-Hyoscyamine Noreugenin ML-030 BC-1382 Gadolinium chloride Vorolanib VTP-27999 TFA GSK0660 Lomerizine hydrochloride 8-CHLOROQUINAZOLIN-4(1H)-ONE
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