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Cat No. | Product Name | Synonyms | Targets |
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TP1929L1 | Saralasin acetate(34273-10-4 free base) | RAAS | |
Saralasin acetate is a Non-selective angiotensin II antagonist. | |||
T4049 | Genz-123346 free base | Glucokinase | |
Genz 123346 is an inhibitor of GL1 synthase that blocks the conversion of ceramide to GL1. | |||
TP1035L | Cyclic somatostatin Acetate(38916-34-6(free base)) | Somatostatin (sheep), monoacetate (salt),Somatostatin-14,SRIF-14,monoacetate (salt) | Others |
Cyclic somatostatin Acetate(38916-34-6(free base)) (Somatostatin-14) is a cyclic tetradecapeptide regulating many endocrine and nervous system functions. | |||
T11321 | FR194738 free base | Antifungal | |
FR194738 free base inhibits squalene epoxidase activity in HepG2 cell homogenates with an IC50 of 9.8 nM. | |||
T7407 | Thyrotropin-Releasing Hormone (TRH), Free Acid | TRH-OH | Others |
Thyrotropin-Releasing Hormone (TRH), Free Acid (TRH-OH) (TRH-OH) causes a variety of thyroidal and non-thyroidal effects, the best known being the feedback regulation of thyroid hormone levels. | |||
TP2212L | A-MSH, amide Acetate(581-05-5 free base) | Melanocortin Receptor | |
a-MSH, amide Acetate as an endogenous neuropeptide. It is an endogenous melanocortin receptor 4 (MC4R) agonist with anti-inflammatory and antipyretic activities. α-MSH is a post-translational derivative of pro-opiomelano... | |||
T10468 | Elimusertib hydrochloride(1876467-74-1 free base) | BAY-1895344 hydrochloride | ATM/ATR |
Elimusertib hydrochloride(1876467-74-1 free base) (BAY-1895344 hydrochloride) is a effective, orally available and selective ATR inhibitor with anti-tumor activity. | |||
T10893 | CS-722 Free base | Others | |
CS-722 Free base is a synthetic central muscle relaxant with muscle relaxant activity and inhibitory effect on spinal reflex. CS-722 Free base may inhibit spontaneous inhibitory post-synaptic current and excitatory post-... | |||
T30677L | C15AlkOPP Tetrabutylamine salt(946615-44-7 Free base) | C15AlkOPP Tetrabutylamine salt(946615-44-7 Free base) | Others |
C15AlkOPP Tetrabutylamine salt is a “clickable” alkyne-modified analogs of the lipid substrates farnesyl diphosphate (FPP). | |||
T4696 | BMS202 hydrochloride (1675203-84-5(free base)) | PD-1/PD-L1 inhibitor 2 hydrochloride | PD-1/PD-L1 |
BMS202 hydrochloride (1675203-84-5(free base)) (PD-1/PD-L1 inhibitor 2 hydrochloride) is a small-molecule PD-1/PD-L1 interaction inhibitor (IC50: 18 nM). Biophysical studies demonstrate that BMS202 binds directly to PD-L... | |||
TP1281L1 | Bombesin acetate(31362-50-2 free base) | Bombesin Receptor | |
Bombesin acetate is a 14-amino acid peptide originally isolated from the skin of the European fire-bellied toad (Bombina bombina). It has two known homologs in mammals called neuromedin B and gastrin-releasing peptide. | |||
T7173L | [Leu5]-Enkephalin acetate(58822-25-6 free base) | Leucine enkephalin,Leu-enkephalin,Leucyl-enkephalin | Opioid Receptor , Endogenous Metabolite |
[Leu5]-Enkephalin acetate(58822-25-6 free base) is an endogenous neuropeptide involved in nociception and an agonist of δ-opioid and μ-opioid receptors (Kis = 4.0 and 3.4 nM, respectively) | |||
TP1275 | 3X FLAG peptide TFA (402750-12-3 free base) | 3X FLAG peptide TFA | Others |
3X FLAG peptide TFA (402750-12-3 free base) (3X FLAG peptide TFA) is a synthetic peptide of 23 amino acid residue. The Asp-Tyr-Lys-Xaa-Xaa-Asp motif is repeated three times in the peptide. | |||
TP1101 | Nonapeptide-1 acetate salt (158563-45-2 free base) | Melanostatine-5 acetate salt,Nonapeptide-1 acetate salt | Melanocortin Receptor |
Nonapeptide-1 acetate salt (158563-45-2 free base) (Melanostatine-5 acetate salt) , a peptide hormone, is a potent α-Melanocyte-stimulating hormone (α-MSH) antagonist, with an IC50 of 11 nM. Nonapeptide-1 acetate salt (1... | |||
TP1127L1 | Nemifitide acetate(173240-15-8 free base) | INN 00835 acetate | 5-HT Receptor |
Nemifitide acetate(173240-15-8 free base) (INN 00835 acetate) is a synthetic pentapeptide antidepressant with a potential for rapid onset of action. It is a peptide analog of melanocyte-inhibiting factor (MIF). | |||
TP1895L1 | KYL acetate(676657-00-4 free base) | Ephrin Receptor | |
KYL acetate is an EphA4 receptor tyrosine kinase inhibitor (Kd = 0.8 μM); inhibits EphA4-EphrinA5 interactions (IC50 = 6.34 μM). Prevents AβO induced synaptic damage, dendritic spine loss and prevents the blocking of LTP... | |||
T5162 | MRT67307 HCl (1190378-57-4(free base)) | IκB/IKK , AMPK , Autophagy | |
MRT67307 is a kinase inhibitor of TBK1, MARK1-4, IKKε, and NUAK1 (IC50: 19, 27-52, 160, and 230 nM, respectively). | |||
T12111L | MS31 trihydrochloride (2366264-12-0 free base) | MS31 trihydrochloride | Epigenetic Reader Domain |
MS31 trihydrochloride (2366264-12-0 free base) is a potent, highly affinity and selective fragment-like methyllysine reader protein spindlin 1 (SPIN1) inhibitor. | |||
T4418 | GSK2879552 2HCl (1401966-69-5(free base)) | Histone Demethylase | |
GSK2879552 is an orally available, irreversible inhibitor of lysine specific demethylase 1 (LSD1), with potential antineoplastic activity. | |||
TP2165 | Urotensin II, mouse acetate (9047-55-6 free base) | Urotensin II, mouse acetate | GPR |
Urotensin II, mouse acetate (9047-55-6 free base) is an endogenous ligand for the orphan GPR14 or SENR. It is a potent vasoconstrictor. | |||
T15805L | LY2510924 acetate(1088715-84-7 free base) | CXCR | |
Ly2510924 acetate is an potent and selective CXCR4 antagonist. It prevents the binding of SDF-1 to CXCR4 with an IC50 of 0.079 nM. | |||
T7384 | Ocifisertib(CFI-400945 free base) | PLK | |
CFI-400945 is an potent, selective and orally active inhibitor of polo-like kinase 4(PLK4; Ki value of 0.26 nM). | |||
TP2323L | Deslorelin acetate(57773-65-6 free base) | Deslorelin acetate | GNRH Receptor |
Deslorelin acetate(57773-65-6 free base) is a gonadotropin releasing hormone super-agonist (GnRH agonist) | |||
TP1806L | BCMA72-80 acetate(2293841-58-2 free base) | Others | |
BCMA72-80 acetate is a HLA-A2 specific B cell maturation antigen (BCMA) peptide. It is used to study multiple myeloma and tumors, which expresses B cell maturation antigen. | |||
TP1457 | BIO-11006 acetate salt (901117-03-1 free base) | BIO-11006 acetate salt | Others |
BIO-11006 acetate salt (901117-03-1 free base) is a polyglycosylated alanine rich C kinase substrate (MARCKS) inhibitor similar to MANS peptides. | |||
TP1074L | Neuropeptide FF acetate(99566-27-5 free base) | NPFF acetate | Neuropeptide Y Receptor |
Neuropeptide FF acetate(99566-27-5 free base) (NPFF acetate) is an octapeptide belonging to the RF amide family. NPFF interacts with G-protein-coupled receptors NPFF (1) and NPFF (2). | |||
T4324 | PQ401 hydrochloride (196868-63-0(free base)) | IGF-1R | |
PQ401 inhibits autophosphorylation of IGF-1R domain with IC50 of <1 μM. | |||
T10759 | CEP-28122 mesylate salt (1022958-60-6 free base) | CEP-28122 mesylate salt | ALK |
CEP-28122 mesylate salt (1022958-60-6 free base) is a highly selective orally active ALK inhibitor (IC50: 1.9 nM in an enzyme-based TRF assay). | |||
TP1699L | SEB Domain 144-153 acetate(210229-94-0 free base) | Others | |
SEB Domain 144-153 acetate(210229-94-0 free base) is amino acid residues 163-172 of the staphylococcal enterotoxin B domain. SEB Domain 144-153 acetate(210229-94-0 free base) has been shown to inhibit the transcytosis of... | |||
T4680L | HC067047 Hydrochloride(883031-03-6 free base) | TRP/TRPV Channel | |
HC-067047 hydrochloride is a potent and selective TRPV4 antagonist. HC-067047 hydrochloride reversibly inhibited currents through the human, rat, and mouse TRPV4 orthologs with IC50 values of 486 nM, 133nM, and 17 nM, re... | |||
T8761L | [Leu15]-Gastrin I human acetate(39024-57-2 Free base) | ||
[Leu15]-Gastrin I human acetate(39024-57-2 Free base) is a useful organic compound for research related to life sciences and the catalog number is T8761L. | |||
TP2268L | Lys-Bradykinin acetate(342-10-9 free base) | Bradykinin Receptor | |
Lys-Bradykinin acetate is an endogenous bradykinin receptor agonist. | |||
TP1886L1 | NoxA1ds acetate(1435893-78-9 free base) | NADPH-oxidase | |
NoxA1ds acetate is a potent and selective NADPH oxidase 1 (NOX1) inhibitor (IC50 : 20 nM). Exhibits selectivity for NOX1 over NOX2, NOX4, NOX5 and xanthine oxidase. Inhibits NOX1-derived O2- production in HT-29 human col... | |||
TP1199L | Urotensin I acetate (83930-33-0 Free base) | CRFR | |
Urotensin I acetate, a CRF-like neuropeptide, acts as an agonist of CRF receptor with pEC50s of 11.46, 9.36 and 9.85 for human CRF1, human CRF2 and rat CRF2α receptors in CHO cells, and Kis of 0.4, 1.8, and 5.7 nM for hC... | |||
TP1930L1 | Spexin acetate(1370290-58-6 free base) | Neuropeptide Y Receptor | |
Spexin acetate is a potent galanin receptor 2/3 (GAL2/GAL3) agonist (EC50 values are 45.7 and 112.2 nM, respectively). Exhibits no significant activity at galanin receptor 1. Endogenous satiety-inducing peptide; inhibits... | |||
TP1938L | RS09 2TFA (1449566-36-2 free base) | RS09 2TFA 1449566-36-2(free base) | TLR |
RS09 2TFA (1449566-36-2 free base) is a TLR4 agonist. Promotes NF-κB nuclear translocation and induces inflammatory cytokine secretion in RAW264.7 macrophages in vitro. It acts as an adjuvant in vivo and enhances X-15 sp... | |||
TP1897L1 | JIP-1 (153-163) acetate(438567-88-5 free base) | JNK | |
JIP-1 (153-163) acetate(438567-88-5 free base) is a peptide inhibitor of c-Jun N-terminal kinase (JNK), based on residues 153-163 of JNK-interacting protein-1 (JIP-1). JIP-1 (153-163) acetate(438567-88-5 free base) binds... | |||
TP1933 | R715 TFA(185052-09-9 free base) | R 715 | Bradykinin Receptor |
R715 TFA(185052-09-9 free base) is a potent and selective bradykinin B1 receptor antagonist (pA2 = 8.49). Displays no activity at B2 receptors. Reduces mechanical hypernociception in a mouse model of neuropathic pain. Me... | |||
T9690L | LYS006 hydrochloride (1799681-85-8 Free base) | ||
LYS006 hydrochloride (1799681-85-8 Free base) is a useful organic compound for research related to life sciences and the catalog number is T9690L. | |||
T4419 | UNC2025 2HCl (1429881-91-3(free base)) | FLT , TAM Receptor | |
UNC2025 is a potent and orally bioavailable Mer/Flt3 dual inhibitor with IC50 of 0.8/0.74 nM for Mer/Flt3. | |||
TP1112L | LH-RH, salmon acetate(86073-88-3 free base) | Luteinizing Hormone Releasing Hormone (LH-RH), salmon acetate | Others |
LH-RH, salmon acetate(86073-88-3 free base) (Luteinizing Hormone Releasing Hormone (LH-RH), salmon acetate) is a pituitary Hormone synthesized in the hypothalamus and plays a crucial role in the control of reproductive f... | |||
T5677 | SAR125884 hydrochlorid (1116743-46-4(free base)) | c-Met/HGFR | |
SAR125844 is a potent and selective MET kinase inhibitor with a favorable preclinical toxicity profile,(IC50=4.2 nM). | |||
T12942L | SN50 acetate (213546-53-3 free base) | NF-κB | |
SN50 acetate is a cell permeable inhibitor of NF-κB translocation. | |||
TP1215L | Abaloparatide acetate(247062-33-5 free base) | Others | |
Abaloparatide acetate is a parathyroid hormone receptor 1 PTHR1 analogue and an effective and selective activator of the PTHR1 signaling pathway. | |||
TP1796 | Albiglutide TFA (782500-75-8 free base) | Albiglutide TFA | Glucagon Receptor |
Albiglutide TFA (782500-75-8 free base) (Albiglutide TFA) is a long acting GLP-1 receptor agonist for the treatment of type 2 diabetes mellitus (T2DM). | |||
TP1730L | β-catenin peptide acetate(265669-37-2 free base) | Others | |
β-catenin peptide(βCATp) acetate is a naturally occurring self-peptide presented by Kb that very efficiently mediates positive selection of the OT-I thymocytes. | |||
T5146 | Eptifibatide acetate (148031-34-9 free base) | Eptifibatide acetate | Others |
Eptifibatide acetate (148031-34-9 free base) (Eptifibatide acetate) , an antiplatelet drug of the glycoprotein IIb/IIIa inhibitor class, is a cyclic heptapeptide constructed from 6 amino acids and a mercaptopropionyl res... | |||
TP2328L | CJC-1295 acetate(863288-34-0 free base) | DAC:GRF acetate | GHSR |
CJC-1295 acetate(863288-34-0 free base) (DAC:GRF acetate) is a synthetic analogue of growth hormone-releasing hormone (GHRH) (also known as growth hormone-releasing factor (GRF)) and a growth hormone secretagogue (GHS) | |||
TP1775L | LL-37, Human acetate(154947-66-7 free base) | Antibacterial | |
LL-37, Human acetate is a 37-residue, amphipathic, cathelicidin-derived antimicrobial peptide, which exhibits a broad spectrum of antimicrobial activity. | |||
T7567L | Adrenorphin 3TFA(88377-68-8(free base)) | Metorphamide | Opioid Receptor |
Adrenorphin 3TFA(88377-68-8(free base)) (Metorphamide) is an agonist of μ-opioid receptor(Ki :12 nM). |
Cat No. | Product Name | Synonyms | Targets |
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TQ0296L | N-Nornuciferine hydrochloride(4846-19-9 free base) | N-Nornuciferine hydrochloride | P450 |
N-Nornuciferine hydrochloride(4846-19-9 free base) (N-Nornuciferine hydrochloride) is an aporphine alkaloid in lotus leaf, significantly inhibits CYP2D6 (IC50: 3.76 μM, Ki: 2.34 μM). | |||
T20604L | Litorin acetate(55749-97-8 Free base) | Bombesin Receptor | |
Litorin acetate, an amphibian bombesin peptide derivative, is an bombesin receptor agonist. It stimulates the contraction of smooth muscle, stimulates gastrin, gastric acid, and pancreatic secretion, and suppresses the n... | |||
T2782L | Catharanthine Tartrate(2468-21-5(free base)) | Calcium Channel | |
Catharanthine Tartrate is a natural product isolated from Madagascar periwinkle, Catharanthine Tartrate inhibits voltage-operated L-type Ca2+ channel, with anti-cancer and blood pressure-lowering activity | |||
TP1232L | Amylin, amide, rat acetate(124447-81-0,free base) | Amylin Receptor | |
Amylin, amide, rat acetate is a potent and high affinity ligand of AMY1 and AMY3 receptors and variably of AMY2 receptors. | |||
TN7062L | Bufotenidine hydrochloride(487-91-2 Free base) | ||
Bufotenidine hydrochloride(487-91-2 Free base) is a natural product for research related to life sciences. The catalog number is TN7062L and the CAS number is 40581-89-3. | |||
T5143 | Corynoxine hydrochloride(6877-32-3(free base)) | Autophagy | |
Corynoxine hydrochloride is a natural oxindole alkaloid and induces autophagy in different neuronal cell lines, including N2a and SHSY-5Y cells. |
Cat No. | Product Name | Species | Expression System |
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TMPY-03847 | FRZB Protein, Human, Recombinant (His) | Human | HEK293 Cells |
FRZB also known as sFRP-3, is a secreted protein containing a domain similar to the putative Wnt-binding region of the frizzled family of transmembrane receptors. FRZB is widely expressed in adult mammalian tissues. In t... | |||
TMPH-01101 | Claudin-3 Protein, Human, Recombinant (Cell-Free, His) | Human | E. coli |
Plays a major role in tight junction-specific obliteration of the intercellular space, through calcium-independent cell-adhesion activity. Claudin-3 Protein, Human, Recombinant (Cell-Free, His) is expressed in E. coli ex... | |||
TMPH-01931 | Cereblon/CRBN Protein, Human, Recombinant (Cell-Free, His) | Human | E. coli |
Cereblon/CRBN Protein, Human, Recombinant (Cell-Free, His) is expressed in in vitro E. coli expression system. | |||
TMPH-02536 | BNIP3 Protein, Mouse, Recombinant (Cell-Free, His) | Mouse | E. coli |
Apoptosis-inducing protein that can overcome BCL2 suppression. May play a role in repartitioning calcium between the two major intracellular calcium stores in association with BCL2. Involved in mitochondrial quality cont... | |||
TMPH-00400 | DHAK Protein, Citrobacter freundii, Recombinant (His & SUMO) | Citrobacter freundii | E. coli |
Catalyzes the phosphorylation of dihydroxyacetone. DHAK Protein, Citrobacter freundii, Recombinant (His & SUMO) is expressed in E. coli expression system with N-6xHis-SUMO tag. The predicted molecular weight is 35.9 kDa ... | |||
TMPH-02235 | TMPRSS2 Protein, Human, Recombinant (Cell-Free, His) | Human | E. coli |
TMPRSS2 Protein, Human, Recombinant (Cell-Free, His) is expressed in E. coli expression system with N-6xHis tag. The predicted molecular weight is 46.9 kDa and the accession number is O15393. | |||
TMPK-00836 | HLA-G Free Heavy Chain Protein, Human, Recombinant (His & Avi) | Human | E. coli |
HLA-G is a molecule that was first known to confer protection to the fetus from destruction by the immune system of its mother, thus critically contributing to fetal-maternal tolerance. The first functional finding const... | |||
TMPH-01798 | Nucleolar transcription factor 1 Protein, Human, Recombinant (Cell-Free, His & SUMO) | Human | E. coli |
Recognizes the ribosomal RNA gene promoter and activates transcription mediated by RNA polymerase I through cooperative interactions with the transcription factor SL1/TIF-IB complex. It binds specifically to the upstream... | |||
TMPH-01023 | C5AR1 Protein, Human, Recombinant (Cell-Free, His) | Human | E. coli |
Receptor for the chemotactic and inflammatory peptide anaphylatoxin C5a. The ligand interacts with at least two sites on the receptor: a high-affinity site on the extracellular N-terminus, and a second site in the transm... | |||
TMPH-00596 | Colicin-E1 Protein, E. coli, Recombinant (Cell-Free, His & Myc) | E. coli | E. coli |
This colicin is a channel-forming colicin. This class of transmembrane toxins depolarize the cytoplasmic membrane, leading to dissipation of cellular energy.; Colicins are polypeptide toxins produced by and active agains... | |||
TMPH-01745 | NOX4 Protein, Human, Recombinant (Cell-Free, His) | Human | E. coli |
NOX4 Protein, Human, Recombinant (Cell-Free, His) is expressed in E. coli expression system with N-10xHis tag. The predicted molecular weight is 69.8?kDa and the accession number is Q9NPH5. |