keep away from moisture
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
[Leu5]-Enkephalin acetate(58822-25-6 free base) is an endogenous neuropeptide involved in nociception and an agonist of δ-opioid and μ-opioid receptors (Kis = 4.0 and 3.4 nM, respectively)
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
10 mg | In stock | $ 51.00 | |
25 mg | In stock | $ 101.00 | |
50 mg | In stock | $ 153.00 | |
100 mg | In stock | $ 230.00 | |
200 mg | In stock | $ 345.00 |
Description | [Leu5]-Enkephalin acetate(58822-25-6 free base) is an endogenous neuropeptide involved in nociception and an agonist of δ-opioid and μ-opioid receptors (Kis = 4.0 and 3.4 nM, respectively) |
Targets&IC50 | μ opioid receptor:3.4 nM(ki), δ opioid receptor:4.0 nM(ki) |
In vivo | [Leu5]-Enkephalin is found in the brain, the brainstem, and the spinal cord as well as in the peripheral nervous system. Leu-Enkephalin (1 mg/kg) decreases the visceromotor response to colon distension in a mouse model of visceral pain induced by colorectal distension[1]. |
Synonyms | Leucine enkephalin, Leu-enkephalin, Leucyl-enkephalin |
Molecular Weight | 555.63 |
Formula | C28H37N5O7 |
CAS No. | T7173L |
keep away from moisture
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
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[Leu5]-Enkephalin acetate(58822-25-6 free base) T7173L Endocrinology/Hormones GPCR/G Protein Metabolism Neuroscience Opioid Receptor Endogenous Metabolite [Leu5] Enkephalin acetate(58822 25 6 free base) [Leu5]Enkephalin acetate(58822256 free base) Leucine enkephalin Leu-enkephalin Leucyl-enkephalin [Leu-5]-Enkephalin acetate(58822-25-6 free base) inhibitor inhibit