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Cat No. | Product Name | Synonyms | Targets |
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TF0046 | TFA | ||
TFA has a wide range of applications in life science related research. | |||
TP1215 | Abaloparatide TFA | BA 058 TFA,Abaloparatide TFA (247062-33-5 free base),BIM 44058 TFA | Others |
Abaloparatide TFA (BIM 44058 TFA) is a parathyroid hormone-related protein (PTHrP) analog drug used to treat osteoporosis like the related drug teriparatide. | |||
T7326 | 6H05 (TFA) | 6H05 TFA,6H05 trifluoroacetate | Ras |
6H05 TFA (6H05 trifluoroacetate) is a selective, and allosteric oncogenic mutant K-Ras(G12C) inhibitor. | |||
T14665L | Motixafortide TFA(664334-36-5,Free) | TF 14016 TFA,BKT140 TFA,BL-8040 TFA,T140 TFA | CXCR |
Motixafortide TFA(664334-36-5,Free) (BKT140 TFA) is an antagonist of CXCR4 with IC50 of ~1 nM. It induces the apoptosis of AML blasts by down-regulating ERK, BCL-2, MCL-1 and cyclin-D1 via altered miR-15a/16-1 expression... | |||
TP1346 | CYN 154806 TFA | CYN 154806 TFA | Somatostatin |
CYN 154806 TFA is a cyclic octapeptide and an effective selective somatostatin sst2 receptor antagonist. For the recombinant sst2, sst1, sst3, sst4 and sst5 receptors, the pIC50 values are 8.58, 5.41, 6.07, 5.76 and 6.48... | |||
T26641L | Apadenoson TFA | BAY 68-4986 TFA,Apadenoson TFA(250386-15-3 Free base),Discontinued TFA | Adenosine Receptor |
Apadenoson TFA is a potent adenosine A2A receptor (A2AR) agonist that can be used to improve survival in patients infected with SARS. | |||
T33876L1 | Panomifene TFA | Panomifene TFA(77599-17-8 Free base),EGIS5650 TFA,GYKl13504 TFA | Estrogen/progestogen Receptor |
Panomifene TFA(GYKl13504 TFA) is a small molecule antagonist of ERs with anticancer activity that can be used to study breast cancer and musculoskeletal diseases. | |||
T8768 | MM-102 TFA | HMTase Inhibitor IX TFA | Histone Methyltransferase |
MM-102 TFA (HMTase Inhibitor IX TFA) is a potent WDR5/MLL interaction inhibitor, achieves IC50 = 2.4 nM. MM-102 compound prevents the interaction between mixed lineage leukemia 1 (MLL1) and WD Trp-Asp repeat domain 5 (WD... | |||
T11237L | Camizestrant TFA | Camizestrant TFA(2222844-89-3 Free base),AZD-9833 TFA | Estrogen Receptor/ERR |
Camizestrant TFA (AZD-9833 TFA) is a potent and orally active antagonist of estrogen receptor (ER). | |||
T5862 | Ezatiostat TFA | TER199(free base),Ezatiostat TFA (free base),Ezatiostat,TLK199 | GST |
Ezatiostat TFA (TLK199) is a liposomal small-molecule glutathione analog inhibitor of glutathione S-transferase (GST) P1-1 with hematopoiesis-stimulating activity. | |||
TP1796 | Albiglutide TFA (782500-75-8 free base) | Albiglutide TFA | Glucagon Receptor |
Albiglutide TFA (782500-75-8 free base) (Albiglutide TFA) is a long acting GLP-1 receptor agonist for the treatment of type 2 diabetes mellitus (T2DM). | |||
T16790L | Rotigaptide TFA(355151-12-1 free base) | Rotigaptide TFA | Gap Junction Protein |
Rotigaptide TFA(355151-12-1 free base) is a novel and specific modulator of Cx43 and is a potent AAP. Rotigaptide TFA(355151-12-1 free base) prevents the uncoupling of Cx43-mediated gap junction communication and normali... | |||
TP1067 | Pam3CSK4 TFA (112208-00-1 free base) | Pam3CSK4 TFA,Pam3Cys-Ser-(Lys)4 TFA | TLR |
Pam3CSK4 TFA (Pam3Cys-Ser-(Lys)4 TFA) is an agonist of toll-like receptor 1/2 (TLR1/2) (EC50 of 0.47 ng/mL for human TLR1/2). | |||
TP1086 | Men 10376 TFA(135306-85-3,free) | Men 10376 TFA,Neurokinin-2 receptor antagonist TFA | Neurokinin receptor |
Men 10376 TFA(135306-85-3,free) (Neurokinin-2 receptor antagonist TFA) is an effective and selective tachykinin nk-2 receptor antagonist with a K I value of 4.4 M for the nk-2 receptor in the small intestine of rats. | |||
TP1291 | Epithalon TFA (307297-39-8 free base) | Epithalon TFA | Others |
Epithalon TFA (307297-39-8 free base) (Epithalon TFA) is an anti-aging agent and telomerase activator. | |||
TP2050L | CTAP(TFA) (103429-32-9 free base) | CTAP(TFA) | Opioid Receptor |
CTAP(TFA) (103429-32-9 free base) is a potent, highly selective, and brain-penetrant antagonist of the μ-opioid receptor with IC50 of 3.5 nM. It displays over 1200-fold selectivity over δ opioid (IC50=4500 nM) and somato... | |||
T27250L | Elarofiban TFA | Elarofiban TFA(198958-88-2 Free base),RWJ-53308 TFA | Integrin |
Elarofiban TFA (RWJ-53308 TFA) is a novel and orally active and selective GPIIb/IIIa antagonist for the study of cardiovascular disease. | |||
T30191L | Atecegatran TFA | Atecegatran TFA(917904-13-3 Free base),AR-H067637 TFA | Others |
Atecegatran TFA is often used as an anticoagulant and can be used to treat cardiovascular disease. | |||
TP1348 | FC131 TFA (606968-52-9 free base) | FC131 TFA | HIV Protease , CXCR |
FC131 TFA (606968-52-9 free base) (FC131 TFA) is an antagonist of CXCR4 that inhibits the binding of [125I] -sdf-1 to CXCR4(IC50 : 4.5 nM ), and has anti-hiv activity. | |||
T68023L | Tolnapersine TFA | Tolnapersine TFA(70312-00-4 Free base) | Dopamine Receptor , Adrenergic Receptor |
Tolnapersine TFA is a mixed dopamine agonist and alpha adrenergic receptor antagonist. | |||
T61345L | Orbofiban TFA | Orbofiban TFA(163250-90-6 Free base) | Integrin |
Orbofiban TFA is an orally active GPIIb/IIIa platelet receptor antagonist with inhibitory effects on platelet aggregation for the study of unstable coronary syndromes. | |||
TP1430 | DTP3 TFA (1809784-29-9 free base) | DTP3 TFA | Others |
DTP3 TFA (1809784-29-9 free base) (DTP3 TFA) is a potent and selective GADD45β/MKK7 (growth arrest and DNA-damage-inducible β/mitogen-activated protein kinase kinase 7) inhibitor. | |||
TP1300 | GsMTx4 TFA (1209500-46-8 free base) | GsMTx4 TFA | Piezo Channel |
GsMTx4 TFA (1209500-46-8 free base) (GsMTx4 TFA) is a spider venom peptide that selectively inhibits cationic permeable mechanically-sensitive channels (MSCs) belonging to the Piezo and TRP channel families. | |||
TP1254 | [Met5]-Enkephalin, amide TFA | 5-Methionine-enkephalin amide (TFA) | Opioid Receptor |
[Met5]-Enkephalin, amide TFA (5-Methionine-enkephalin amide (TFA)) is a δ opioid receptors agonist as well as putative ζ (zeta) opioid receptors. | |||
T17927 | (S,R,S)-AHPC TFA | VH032-NH2 TFA,VHL ligand 1 TFA | Others , Ligand for E3 Ligase |
(S,R,S)-AHPC TFA (VHL ligand 1 TFA) (VH032-NH2 TFA) is a VH032-based ligand designed for von Hippel-Lindau (VHL) protein recruitment. This compound can be linked to protein ligands (e.g., BCR-ABL1) using a linker to crea... | |||
TP2036L | DPDPE TFA (88373-73-3 free base) | DPDPE TFA | Opioid Receptor |
DPDPE TFA is selective δ-opioid receptor agonist peptide. Inhibits electrically stimulated contraction of mouse vas deferens in vitro (EC50 = 5.2 nM), and is antinociceptive in vivo. | |||
TP2158 | TRV-120027 TFA | TRV-120027 TFA (1234510-46-3 free base) | RAAS , Arrestin |
TRV120027 TFA is a β-arrestin-1-biased agonist of the angiotensin II receptor type 1 (AT1R) and engages ß-arrestins while blocking G-protein signaling. | |||
TP1918L | Lys-[Des-Arg9]Bradykinin,TFA | Lys-[Des-Arg9]Bradykinin,TFA 71800-36-7(fb-tfa) | Bradykinin Receptor |
Lys-[Des-Arg9]Bradykinin,TFA is Endogenous potent and highly selective bradykinin B1 receptor agonist (Ki values are 0.12 and > 30000 nM at human B1 and B2 receptors respectively). Hypotensive agent that reduces peripher... | |||
T34921L1 | Tresperimus TFA | Tresperimus TFA(160677-67-8 Free base) | Others |
Tresperimus TFA can be used as an immune agent and can be used to study retinitis. | |||
T68166L | Traxanox TFA | Traxanox TFA(58712-69-9 Free base) | Others |
Traxanox TFA is an orally available diuretic. Traxanox TFA enhances phagocytosis of yeast granules by mouse peritoneal macrophages or rat peritoneal polymorphonuclear leukocytes in vitro. Traxanox TFA restores inhibition... | |||
TP1079 | (Arg)9 TFA (143413-47-2 free base) | Nona-L-arginine (TFA),(Arg)9 TFA,Peptide R9 (TFA) | Others |
(Arg)9 TFA (Peptide R9 TFA) is a cell-penetrating peptide. (Arg)9 TFA (Nona-L-arginine TFA) exhibits neuroprotective activity with an IC50 of 0.78 μM in the glutamic acid model. | |||
T64133L | Laniquidar TFA | Laniquidar TFA(197509-46-9 Free base),R101933 | P-gp |
Laniquidar TFA (R101933) is a novel orally available non-competitive P-glycoprotein (P-gp) inhibitor with an IC50 value of 0.51 μM.Laniquidar has limited bioavailability and can be used to modulate the multidrug resistan... | |||
TP1065 | PAR-4 Agonist Peptide, amide TFA | PAR-4-AP (TFA),AY-NH2 (TFA) | Protease-activated Receptor |
PAR-4 Agonist Peptide, amide TFA (PAR-4-AP (TFA)), is a selective activator of the proteinase-activated receptor-4 (PAR-4), demonstrating specificity by not influencing PAR-1 or PAR-2, and its activity can be inhibited b... | |||
TP1412 | RNAIII-inhibiting peptide TFA | RNAIII-inhibiting peptide(TFA) | Antibacterial |
RNAIII-inhibiting peptide TFA (RNAIII-inhibiting peptide(TFA))(228544-21-6 free base) inhibits S. aureus, effective in the diseases such as cellulitis, keratitis, septic arthritis, osteomylitis and mastitis. | |||
TP1318 | Antennapedia Peptide TFA(188842-14-0 free base) | Antennapedia Peptide(TFA) | Others |
Antennapedia Peptide TFA (188842-14-0 free base), a peptide of 16 amino acids, is a member of the family of Cell-penetrating peptides, originally derived from the 60 amino acid long homeodomain of the Drosophila transcri... | |||
TP1240 | Adrenocorticotropic Hormone (ACTH) (18-39), human TFA | CLIP (human) (TFA) | Others |
Adrenocorticotropic Hormone (ACTH) (18-39), human TFA (CLIP human TFA) is a corticotropinlike intermediate lobe peptide, it is is produced in the melanotrophs of the intermediate lobe of the pituitary. | |||
T33836L | Oxamisole TFA | Oxamisole TFA(99258-56-7 Free base) | Antiviral |
Oxamisole TFA is an orally available T-cell immune repair agent. | |||
T36201L | AZD5582 TFA | AZD5582 TFA(1258392-53-8 free base) | Apoptosis , IAP |
AZD5582 TFA is a potent IAP antagonist that binds to the BIR3 domain of cIAP1, cIAP2, and XIAP with IC50 values of 15, 21, and 15 nM, respectively.AZD5582 TFA induces apoptosis. | |||
T67972L | Amp579 TFA | Amp579 TFA(213453-89-5 Free base) | Adenosine Receptor |
Amp579 TFA is a novel adenosine A1/A2a receptor agonist that induces acute and delayed preconditioning against myocardial shock in vivo. | |||
TP1947L | P110 TFA | Others | |
P110 TFA is a dynamin-related protein 1 (Drp1) inhibitor, inhibits Drp1 GTPase activity. | |||
T7760 | Thalidomide-O-amido-C3-NH2 TFA | Cereblon Ligand-Linker Conjugates 16 TFA,E3 Ligase Ligand-Linker Conjugates 52 TFA | E3 Ligase Ligand-Linker Conjugate , Ligand for E3 Ligase |
Thalidomide-O-amido-C3-NH2 TFA (Cereblon Ligand-Linker Conjugates 16 TFA) is a synthesized E3 ligase ligand-linker conjugate. Thalidomide-O-amido-C3-NH2 TFA incorporates the Thalidomide based cereblon ligand and a linker... | |||
TP1200 | CGRP (83-119), rat TFA | Calcitonin Gene Related Peptide(83-119), rat TFA | Others |
CGRP (83-119), rat TFA (Calcitonin Gene Related Peptide(83-119), rat TFA) is a 37 amino acid calcitonin family of neuropeptide, acts through calcitonin receptor-like receptor. | |||
T7666 | Valorphin TFA(144313-54-2(free base)) | Valorphin TFA(144313-54-2(free bas)) | Others |
Valorphin TFA(144313-54-2(free base)) is a semisynthetic derivative of dihydrovaltrate with opioid analgesic activity | |||
TP1275 | 3X FLAG peptide TFA (402750-12-3 free base) | 3X FLAG peptide TFA | Others |
3X FLAG peptide TFA (402750-12-3 free base) (3X FLAG peptide TFA) is a synthetic peptide of 23 amino acid residue. The Asp-Tyr-Lys-Xaa-Xaa-Asp motif is repeated three times in the peptide. | |||
T28072L | MLN-3897 TFA | MLN-3897 TFA(1010731-97-1 Free base) | CCR |
MLN-3897 TFA is a potent CCR1 antagonist that inhibits the binding of 125I-MIP-1α to THP-1 cell membranes. | |||
TP1622 | DX600 TFA | RAAS | |
DX600 TFA is a specific inhibitor of ACE2 and does not cross-react with ACE. | |||
TP1433 | CMD178 TFA | STAT | |
CMD178 (TFA) is a lead peptide that consistently reduces the expression of Foxp3 and STAT5 induced by IL-2/s IL-2Rα signaling. | |||
TP1216 | CaM kinase II inhibitor TFA salt | Autocamtide-2-related inhibitory peptide (TFA) | CaMK |
CaM kinase II inhibitor TFA salt (Autocamtide-2-related inhibitory peptide (TFA)) is a highly specific and potent inhibitor of CaMKII with an IC50 of 40 nM. | |||
TP1351L | Kemptide TFA | Others | |
Kemptide TFA is a synthetic heptapeptide, acting as a substrate for cAMP-dependent protein kinase (PK). | |||
T37496L | Alamandine TFA | RAAS | |
Alamandine TFA , a member of the renin-angiotensin system (RAS), a vasoactive peptide, is an endogenous ligand of the G protein-coupled receptor MrgD. Alamandine TFA targets to protect the kidney and heart through anti-h... |
Cat No. | Product Name | Synonyms | Targets |
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T78500 | α-Factor Mating Pheromone, yeast TFA | Mating Factor α TFA | |
α-Factor Mating Pheromone (yeast TFA) is a tridecapeptide secreted by Saccharomyces cerevisiae α cells and interacts with the Ste2p receptor [1]. | |||
T36295 | Echistatin TFA | ||
Echistatin TFA, the smallest active RGD protein belonging to the family of disintegrins that are derived from snake venoms, is a potent inhibitor of platelet aggregation. Echistatin is a potent inhibitor of bone resorpti... | |||
T35401 | γ-Glu-Gly TFA | ||
γ-Glu-Gly TFA, a γ-glutamyl dipeptide, is a human lipid metabolite with a structure resembling GABA (γ-aminobutyric acid). It serves as an excitatory amino acid antagonist [1][2][3]. | |||
T75967 | Bactenecin TFA | ||
Bactenecin TFA (Bactenecin, bovine TFA), a potent 12-aa looped antimicrobial peptide derived from bovine neutrophils, effectively inhibits bacterial and yeast growth and eradicates Trichophyton rubrum fungus. It enhances... | |||
T75722 | Chlorotoxin TFA | ||
Chlorotoxin TFA, a peptide derived from the Leiurus quinquestriatus scorpion venom, functions as a chloride channel blocker [1] and exhibits anti-cancer activity [2]. | |||
T75767 | Parasin I TFA | ||
Parasin I (TFA), a peptide derived from the 19 amino acids of histone H2A and isolated from catfish skin, exhibits antimicrobial activity [1]. | |||
T73764 | L-Palmitoylcarnitine TFA | ||
L-Palmitoylcarnitine TFA, a long-chain acylcarnitine and fatty acid metabolite, accumulates in the sarcolemma, disrupting the membrane lipid environment during ischemia. It inhibits K ATP channel activity by interacting ... | |||
T83693 | Magainin 2 TFA | MG2 | |
Magainin 2, a cationic peptide derived from the African clawed frog (X. laevis) skin, exhibits host defense and antimicrobial properties. This compound effectively inhibits a range of pathogens, including E. coli, K. pne... | |||
T75753 | Magainin 1 TFA | ||
Magainin 1 TFA (Magainin I TFA), an antimicrobial and amphipathic peptide derived from Xenopus laevis skin, demonstrates antibiotic efficacy against a broad range of Gram-negative and Gram-positive bacteria [1] [2] [3]. | |||
T75974 | Cecropin A TFA | ||
Cecropin A TFA, a linear 37-residue antimicrobial polypeptide derived from Hyalaphora cecropia pupae, exhibits anti-bacterial, anti-inflammatory [1], and anti-cancer activities [2]. | |||
T75890 | Conantokin G TFA | ||
Conantokin G TFA, a 17-amino-acid peptide, serves as a potent, selective, and competitive antagonist of N-Methyl-D-Aspartate (NMDA) receptors, effectively inhibiting NMDA-evoked currents in murine cortical neurons at an ... | |||
T75743 | HA Peptide TFA | ||
HA Peptide (TFA), a nine amino acid sequence derived from human influenza hemagglutinin (HA), is widely employed in cell biology and biochemistry for the isolation, purification, detection, and tracking of target protein... | |||
T76027 | β-Endorphin, equine TFA | ||
β-Endorphin, equine TFA, an endogenous opioid peptide, demonstrates high affinity binding to μ/δ opioid receptors and possesses analgesic properties [1] [2] [3] [4]. | |||
T61171 | Cyclo(his-pro) TFA | ||
Cyclo(his-pro) TFA, an orally active cyclic dipeptide structurally related to tyreotropin-releasing hormone, has shown inhibitory effects on NF-κB nuclear accumulation. Additionally, it possesses the ability to cross the... | |||
T4643 | TFAP | N-(5-Aminopyridin-2-yl)-4-(trifluoromethyl)benzamide | COX , Endogenous Metabolite |
TFAP (N-(5-Aminopyridin-2-yl)-4-(trifluoromethyl)benzamide) is a selective cyclooxygenase-1 (COX-1) inhibitor | |||
T19316 | Ethyl oleate | Others | |
Ethyl oleate, a fatty acid ester produced through the condensation of oleic acid and ethanol, serves as the liquid lipid component in nanostructured lipid carriers (NLCs). These NLCs represent a pioneering approach for t... |
Cat No. | Product Name | Species | Expression System |
---|---|---|---|
TMPY-02530 | Tissue Factor Protein, Human, Recombinant (His) | Human | HEK293 Cells |
Tissue Factor Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 26.2 kDa and the accession number is P13726. | |||
TMPK-00993 | Coagulation Factor III/Tissue Factor Protein, Canine, Recombinant (His) | Canine | HEK293 Cells |
Tissue factor (also named Coagulation Factor III) is a cell surface glycoprotein responsible for initiating the extrinsic pathway of coagulation.Tissue factor is the primary cellular initiator of blood coagulation via in... | |||
TMPY-06957 | Tissue Factor Protein, Human, Recombinant (hFc & Avi), Biotinylated | Human | HEK293 Cells |
Tissue Factor Protein, Human, Recombinant (hFc & Avi), Biotinylated is expressed in HEK293 mammalian cells with hFc and Avi tag. The predicted molecular weight is 53.34 kDa and the accession number is P13726. | |||
TMPY-05083 | Tissue Factor Protein, Human, Recombinant (aa 1-295, His) | Human | Baculovirus Insect Cells |
Tissue Factor Protein, Human, Recombinant (aa 1-295, His) is expressed in Baculovirus insect cells with His tag. The predicted molecular weight is 31 kDa and the accession number is P13726-1. | |||
TMPY-02537 | Tissue Factor Protein, Human, Recombinant (hFc) | Human | HEK293 Cells |
Tissue Factor Protein, Human, Recombinant (hFc) is expressed in HEK293 mammalian cells with hFc tag. The predicted molecular weight is 51.8 kDa and the accession number is P13726. | |||
TMPH-01724 | MRTFA Protein, Human, Recombinant (His & KSI) | Human | E. coli |
MRTFA Protein, Human, Recombinant (His & KSI) is expressed in E. coli expression system with N-6xHis-KSI tag. The predicted molecular weight is 25.4 kDa and the accession number is Q969V6. | |||
TMPH-02939 | TFAM Protein, Mouse, Recombinant (His & Myc) | Mouse | E. coli |
TFAM Protein, Mouse, Recombinant (His & Myc) is expressed in E. coli expression system with N-10xHis and C-Myc tag. The predicted molecular weight is 30.9 kDa and the accession number is P40630. | |||
TMPY-02949 | AP2 Gamma/TFAP2C Protein, Human, Recombinant (His) | Human | E. coli |
TFAP2C, also known as AP2-GAMMA, is a member of the activating protein 2 family of transcription factors. AP-2 factors bind to the consensus sequence 5'-GCCNNNGGC-3' and activate genes involved in a large spectrum of imp... |