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DPDPE TFA (88373-73-3 free base)

Catalog No. TP2036L CAS 172888-59-4

Synonyms: DPDPE TFA

DPDPE TFA is selective δ-opioid receptor agonist peptide. Inhibits electrically stimulated contraction of mouse vas deferens in vitro (EC50 = 5.2 nM), and is antinociceptive in vivo.

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DPDPE TFA (88373-73-3 free base) Chemical Structure

DPDPE TFA (88373-73-3 free base), CAS 172888-59-4

Pack Size	Availability	Price/USD
1 mg	In stock	$ 113.00
5 mg	In stock	$ 272.00
10 mg	In stock	$ 413.00
25 mg	In stock	$ 676.00
50 mg	In stock	$ 943.00
100 mg	In stock	$ 1,270.00

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Purity: 99.39%

Biological Description

Chemical Properties

Storage & Solubility Information

Description

DPDPE TFA is selective δ-opioid receptor agonist peptide. Inhibits electrically stimulated contraction of mouse vas deferens in vitro (EC50 = 5.2 nM), and is antinociceptive in vivo.

Synonyms	DPDPE TFA
Molecular Weight	759.81
Formula	C32H40F3N5O9S2
CAS No.	172888-59-4

Storage

keep away from moisture

Powder: -20°C for 3 years | In solvent: -80°C for 1 year

Solubility Information

DMSO: 10 mM

References and Literature

1. Chandrakumar et al (1992) Analogs of the δ opioid receptor selective cyclic peptide [2-D-penicillamine,5-D-penicillamine]-enkephalin: 2',6'-dimethyltyrosine and Gly3-Phe4 amide bond isostere substitutions. J.Med.Chem. 35 2928 PMID: 2. Clark et al (1986) [D-Pen2,D-Pen5]enkephalin (DPDPE): a δ-selective enkephalin with low affinity for μ1 opiate binding sites. Eur.J.Pharmacol. 128 303 PMID: 3. Fraser et al (2000) Supraspinal antinociceptive response to [D-Pen2,5]-enkephalin (DPDPE) is pharmacologically distince from that to other δ-agonists in the rat. J.Pharmacol.Exp.Ther. 295 1135 PMID:

Related compound libraries

This product is contained In the following compound libraries：

Membrane Protein-targeted Compound Library Peptide Compound Library GPCR Compound Library Anti-Neurodegenerative Disease Compound Library Anti-Parkinson's Disease Compound Library Neuronal Signaling Compound Library Bioactive Compound Library NO PAINS Compound Library Covalent Inhibitor Library Neurotransmitter Receptor Compound Library

Related Products

Related compounds with same targets

μ opioid receptor agonist 3 difelikefalin acetate(1024828-77-0 Free base) Loperamide hydrochloride [Leu5]-Enkephalin, amide acetate Deltorphin acetate GR 89696 fumarate Difelikefalin acetate Docusate sodium

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Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.

Keywords

DPDPE TFA (88373-73-3 free base) 172888-59-4 Endocrinology/Hormones GPCR/G Protein Neuroscience Opioid Receptor DOR Inhibitor DPDPE inhibit 88373-73-3 DPDPE TFA (88373733 free base) anticonvulsant DPDPE TFA (88373 73 3 free base) DPDPE TFA agonist 88373-73-3 free base inhibitor

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