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Cat No. | Product Name | Synonyms | Targets |
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TP1286 | Carcinoembryonic Antigen CEA | Others | |
Carcinoembryonic antigen (CEA) is a protein that is present in certain tissues of a developing baby (fetus) | |||
T2711 | Chembridge-5861528 | TCS 5861528 | TRP/TRPV Channel |
Chembridge-5861528 (TCS 5861528) is a TRPA1 channel blocker that antagonizes AITC- and 4-HNE-evoked calcium influx with IC50 values of 14.3 and 18.7 μM, respectively. | |||
T60093 | CHEMBL1380345 | N,N'-(Ethane-1,2-diyl)bis(3-methylbenzenesulfonamide) | Antibacterial |
CHEMBL1380345 exhibits antibacterial activity against Staphylococcus aureus, Bacillus cereus, and Escherichia coli with pMIC values of 3.64, 3.56, and 3.70, respectively. | |||
T74178 | Glembatumumab vedotin | CR011-vcMMAE,CR 011 ADC,CDX-011 | Microtubule Associated |
Glembatumumab vedotin (CDX-011) is an antibody-activated small molecule coupling, Glembatumumab vedotin has potent anticancer effects and can be used in the study of triple negative breast cancer (TNBC). | |||
T3071 | Olverembatinib | GZD 824 | Bcr-Abl |
Olverembatinib (GZD 824) is an orally bioavailable Bcr-Abl inhibitor for Bcr-Abl(WT, IC50: 0.34 nM) and Bcr-Abl(T315I, IC50: 0.68 nM). | |||
T27112 | Cytembena | DNA/RNA Synthesis | |
Cytembena is a cytostatic and a carcinogenic compound that may increase the incidence of fibroadenomas.Cytembena broadly inhibits DNA biosynthesis. | |||
T28750 | Sembragiline | RG-1577,EVT-302,RO-4602522,RO4602522,RG1577,EVT302 | MAO |
Sembragiline (EVT-302) is a selective MAO-B inhibitor for the study of Alzheimer's disease (AD). | |||
T8598 | CHEMBL241987 | 2-PHENYL-2,5-DIHYDRO-4H-PYRAZOLO[3,4-C]QUINOLIN-4-ONE | Adenosine Receptor |
CHEMBL241987 targets the Adenosine receptor A3 (human) | |||
T2429 | Olverembatinib dimesylate | GZD824 Dimesylate,HQP1351 | Bcr-Abl |
Olverembatinib dimesylate (GZD824 Dimesylate) is a novel orally bioavailable Bcr-Abl inhibitor for Bcr-Abl(WT) and Bcr-Abl(T315I). | |||
T67988 | Embeconazole | R 120758,CS 758 | Antifungal |
Embeconazole (R 120758) is a triazole antifungal agent.Embeconazole has strong in vitro activity against clinically important fungi such as Candida, Aspergillus and Cryptococcus neoformans. | |||
T9908 | Pembrolizumab | PD-1/PD-L1 | |
Pembrolizumab is a humanized monoclonal antibody inhibiting the PD-1 receptor and the first in the class of agents called the HER2 dimerization inhibitors that impairs the ability of HER2 to bind to other members of the ... | |||
T77439 | Glembatumumab | Others | |
Glembatumumab is a fully human IgG2 monoclonal antibody targeting the extracellular structural domain of GPNMB expressed in human breast cancer and melanoma.Glembatumumab is a naked antibody to Glembatumumab vedotin and ... | |||
T60092 | CHEMBL1276927 | N-[3-(1H-benzimidazol-2-yl)phenyl]-3-methylbenzamide,N-(3-(1H-benzo[d]imidazol-2-yl)phenyl)-3-methylbenzamide | Antibacterial , Parasite |
CHEMBL1276927 (N-(3-(1H-benzo[d]imidazol-2-yl)phenyl)-3-methylbenzamide) shows antibacterial and antiparasitic activities against Chlamydia pneumoniae and Leishmania donovani. | |||
TP2417 | Tidembersat | Others | |
Tidembersat is a small molecule compound used to treat and/or prevent degenerative diseases such as Huntington's chorea, schizophrenia, neurological. | |||
T124967 | D7-Mesembrenone | ||
D7-Mesembrenone is a useful organic compound for research related to life sciences. The catalog number is T124967 and the CAS number is 35714-44-4. | |||
T124052 | Calophymembranside B | ||
Calophymembranside B is a useful organic compound for research related to life sciences. The catalog number is T124052 and the CAS number is 869285-60-9. | |||
T31373 | Dembrexine HCl | Dembroxol | |
Dembrexine is a bioactive agent. | |||
T70261 | Amitriptyline Embonate | ||
Amitriptyline Embonate is an inhibitor of the re-uptake of norepinephrine and serotonin, thereby inhibiting N-methyl-D-aspartate (NMDA) receptors. | |||
TP2198 | Platelet Membrane Glycoprotein IIB Peptide (296-306) | Others | |
GPllb is composed of a 125 Kd heavy chain that is disulfide-linked to a 23 Kd light chain. Hydropathicity analysis of the cDNA sequence indicates that GPllb is anchored to the platelet through a single transmembrane doma... | |||
T81824 | Membrane-Permeable Sequence, MPS | ||
Membrane-Permeable Sequence (MPS) is a cell-penetrating peptide (CPP) utilized in the investigation of membrane crossing mechanisms [1]. | |||
T80209 | Human membrane-bound PD-L1 polypeptide | PD-1/PD-L1 | |
Human membrane-bound PD-L1 polypeptide serves as an antigen for inducing the production of PD-L1 antibodies [1]. | |||
T71902 | CHEMBL94431 | ||
CHEMBL94431 is an inhibitor of the epidermal growth factor receptor (EGFR) tyrosine kinase. | |||
T11180 | Embramine | Others | |
Embramine, used as an antihistamine and anticholinergic, is a monoethanolamine. | |||
T131462 | Embelin Dimethyl ether | ||
Embelin Dimethyl ether is a useful organic compound for research related to life sciences and the catalog number is T131462. | |||
T70054 | Novembichin | ||
Novembichin is a nitrogen mustard agent that crosslinks with DNA, causing inhibition of DNA synthesis. | |||
T69405 | Metformin embonate | ||
Metformin embonate is an AMP-activated protein kinase (AMPK) activator that improves glycemic control by improving insulin sensitivity and decreasing intestinal absorption of glucose. | |||
T131083 | Cembratetraene-16,2:19,6-diolide | ||
Cembratetraene-16,2:19,6-diolide is a useful organic compound for research related to life sciences and the catalog number is T131083. | |||
T35434 | β-Cembrenediol | ||
β-Cembrenediol (β-CBT) is a natural product from tobacco plants that is found in cigarette smoke condensate. β-CBT inhibits induction of the early antigen of Epstein-Barr virus (EA-EBV) by 12-O-tetradecanoylphorbol-13-ac... | |||
T82476 | Embramine hydrochloride | ||
Embramine hydrochloride is a monoethanolamine derivative utilized for its antihistaminic and anticholinergic properties [1]. | |||
T68384 | SCHEMBL12616233 | ||
SCHEMBL12616233 is a novel inhibitor of SARS-CoV-2 main protease (MPro). | |||
T31619 | Embusartan | UNII-4MY73645XA,Bay 10-6734 | |
Embusartan (BAY 10-6734) is a potent, orally active angiotensin II receptor antagonist used as an antihypertensive agent. | |||
T124625 | α-Cembrenediol | ||
α-Cembrenediol is a useful organic compound for research related to life sciences and the catalog number is T124625. | |||
T28749 | SEMBL | ||
SEMBL, a novel inhibitor of DNA binding of NF-kappaB component p65 in vitro, inhibits NF-kappaB and cellular invasion in ovarian carcinoma ES-2 cells. | |||
T76916 | Bafisontamab | ||
Bafisontamab (EMB-01) is a bispecific antibody that targets EGFR and cMET, displaying antitumor activity [1]. | |||
T37880 | OPC-167832 | ||
OPC-167832 is a potent and orally active dprE1 Inhibitor with an IC50 of 0.258 μM. OPC-167832 has antituberculosis activity and can be used for the research of tuberculosis caused by Mycobacterium tuberculosis[1]. OPC-16... |
Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T0810 | Ethambutol dihydrochloride | Ethambutol 2HCl,Emb dihydrochloride,CL40881 | Antibacterial , Antibiotic , Antifungal |
Ethambutol dihydrochloride (CL40881) is a bacteriostatic antimycobacterial agent, which obstructs the formation of cell wall by inhibiting arabinosyl transferases. | |||
T13514 | 5-MethoxyPinocembroside | Others | |
5-MethoxyPinocembroside is a flavonoid isolated from leaves of Moringa oleifera. | |||
T2992 | Pinocembrin | 5,7-Dihydroxyflavanone,Dihydrochrysin,Galangin flavanone | NF-κB , Reactive Oxygen Species , Antibacterial , Autophagy |
Pinocembrin (5,7-Dihydroxyflavanone) is a flavanone, a type of flavonoid. It is an antioxidant found in damiana, honey, fingerroot, and propolis. | |||
TN2078 | Pinocembrin chalcone | 2',4',6'-Trihydroxychalcone,Pinocembrinchalcone | Calcium Channel , Tyrosinase , Antibacterial , Antifection |
Pinocembrin chalcone is an inhibitor of tyrosinase with antimutagenic effects. Pinocembrin chalcone can be used in studies about the prevention of gastric ulcers. | |||
T5710 | Pinocembrin-7-O-β-D-glucopyranoside | Pinocembrin 7-O-beta-D-glucoside | Others |
Pinocembrin-7-O-β-D-glucopyranoside (Pinocembrin 7-O-beta-D-glucoside) is a natual product isolated from Penthorum chinense Pursh. | |||
TN2077 | (+/-)-Pinocembrin | NSC 43318,(±)-5,7-Dihydroxyflavanone | GPR , Others |
(+/-)-Pinocembrin (NSC-43318), a natural product from axillary pines, is a GPR120 ligand that promotes wound healing in the HaCaT cell line. | |||
T2S1682 | Pinocembrin 7-O-[3''-O-galloyl-4'',6''-hexahydroxydiphenoyl]-β-D-glucoside | Pinocembrin 7-O-(3''-galloyl-4'',6''-(S)-hexahydroxydiphenoyl)-beta-D-glucose,pinocembrin-7-o-3-o-galloyl-4-6-hexahydroxydiphenoyl-beta-d-glucoside | Amylase |
Pinocembrin 7-O-[3''-O-galloyl-4'',6''-hexahydroxydiphenoyl]-β-D-glucoside can moderately inhibit α-amylase activity, with the IC50 value of 0.03 umol/ml. | |||
TN4221 | Homoembelin | 2,5-dihydroxy-3-nonyl-1,4-benzoquinone | Antibacterial |
Homoembelin (2,5-dihydroxy-3-nonyl-1,4-benzoquinone) is a pigment from E. ribes and C. monocarpus that has antibacterial effects and can be used to study multidrug-resistant bacterial infections. | |||
T6485 | Embelin | NSC 91874,Emberine,Embelic acid | Apoptosis , NF-κB , Lipoxygenase , IAP , Prostaglandin Receptor , Autophagy |
Embelin (Embelic acid), isolated from the Japanese Ardisia herb, is an inhibitor of the X-linked inhibitor of apoptosis (IC50: 4.1 uM). | |||
T28019 | (-)-Mesembrine | Mesembrin,Mesembrine,Mesembranone | |
Mesembrine is a serotonin reuptake inhibitor and is also a weak inhibitor of the enzyme phosphodiesterase 4 (PDE4). | |||
TN6319 | Embinin | ||
Embinin is a natural product for research related to life sciences. The catalog number is TN6319 and the CAS number is 52589-13-6. | |||
T73857 | Mesembrine | ||
Mesembrine ((+)-Mesembrine), a primary alkaloid distinguished by its aryloctahydroindole structure, acts as a potent 5-HT transporter inhibitor with an inhibition constant (K i) of 1.4 nM. Additionally, it demonstrates i... | |||
T83379 | 2-Hydroxypinocembrin | ||
2-Hydroxypinocembrin, a member of the 2-hydroxyflavanones, serves as a substrate for flavonoid C-glycosyltransferases [1]. | |||
T19772 | Mesembrenone | (+)-Mesembrenone | |
Mesembrenone is a selective the serotonin transporter (SERT) inhibitor. Mesembrenone is the main alkaloid of Sceletium tortuosum. | |||
TN4792 | Pinocembrin diacetate | Others | |
Pinocembrin diacetate is a natural product for research related to life sciences. The catalog number is TN4792 and the CAS number is 111441-88-4. | |||
T77289 | 5-O-Methylembelin | ||
5-O-Methylembelin is a natural isocoumarin that inhibits PCSK9 , low-density lipoprotein receptor (IDOL) , and sterol regulatory element binding protein 2 (SREBP2) mRNA expression [1] . | |||
T72742 | (-)-Pinocembrin | ||
(-)-Pinocembrin demonstrates anti-mycobacterial activity against Mycobacterium tuberculosis H37Ra, presenting IC 50 values of 1.11 mg/mL in the dormant phase and 1.21 mg/mL in the active phase. Additionally, this compoun... | |||
TN4791 | Pinocembrin 7-acetate | Others | |
Pinocembrin 7-acetate has antitumor activity. | |||
TN5509 | (2S)-Pinocembrin 7-O-[2''-O-(5'''-O-trans-cinnamoyl)-β-D-apiofuranosyl]-β-D-glucoside | (2S)-Pinocembrin 7-O-[cinnamoyl(1→5)-β-D-apiosyl(1→2)]-β-D-glucoside | |
(2S)-Pinocembrin 7-O-[2''-O-(5'''-O-trans-cinnamoyl)-β-D-apiofuranosyl]-β-D-glucoside is a natural product for research related to life sciences. The catalog number is TN5509 and the CAS number is 773899-29-9. | |||
T72856 | (+)-Cembrene A | ||
(+)-Cembrene A, a nontoxic α-glucosidase inhibitor to human normal hepatocyte (LO2) cells, exhibits an IC50 value of 30.31 μM. |
Cat No. | Product Name | Species | Expression System |
---|---|---|---|
TMPH-02637 | Embigin Protein, Mouse, Recombinant (His) | Mouse | in vitro E. coli expression system |
Plays a role in targeting the monocarboxylate transporters SLC16A1 and SLC16A7 to the cell membrane. Plays a role in the outgrowth of motoneurons and in the formation of neuromuscular junctions. Following muscle denervat... | |||
TMPH-00023 | Outer membrane protein Omp38, Acinetobacter baumannii, Recombinant (His & Myc) | Acinetobacter baumannii | E. coli |
Functions as a porin. Induces apoptosis in human cell lines through caspase-dependent and AIF-dependent pathways. Purified Omp38 enters host cell and localizes to the mitochondria, which presumably leads to a release of ... | |||
TMPH-01138 | Human coronavirus 229E Membrane protein (His) | HCoV-229E | E. coli |
Human coronavirus 229E Membrane protein (His) is expressed in E. coli. | |||
TMPH-00022 | Outer membrane protein Omp38, Acinetobacter baumannii, Recombinant (His & SUMO) | Acinetobacter baumannii | E. coli |
Porin. Induces apoptosis in human cells through caspases-dependent and AIF-dependent pathways. Purified Omp38 enters the cells and localizes to the mitochondria, which leads to a release of proapoptotic molecules such as... | |||
TMPY-04904 | Zika virus (ZIKV) (strain Zika SPH2015) M/Membrane protein (Fc) | ZIKV | HEK293 |
Zika virus (ZIKV) infection causes microcephaly and has been linked to other brain abnormalities. ZIKV has a more selective and larger impact on the expression of genes involved in DNA replication and repair. P53 inhibit... | |||
TMPH-00021 | Outer membrane protein Omp38, Acinetobacter baumannii, Recombinant (His) | Acinetobacter baumannii | Yeast |
Porin. Induces apoptosis in human cells through caspases-dependent and AIF-dependent pathways. Purified Omp38 enters the cells and localizes to the mitochondria, which leads to a release of proapoptotic molecules such as... | |||
TMPH-01151 | Human coronavirus NL63 Membrane protein (His) | HCoV-NL63 | in vitro E. coli expression system |
Human coronavirus NL63 Membrane protein (His) is expressed in in vitro E. coli expression system. | |||
TMPH-03640 | 34 kDa membrane antigen Protein, Treponema pallidum, Recombinant (His & Myc) | Treponema pallidum | E. coli |
34 kDa membrane antigen Protein, Treponema pallidum, Recombinant (His & Myc) is expressed in E. coli. | |||
TMPH-00018 | 29 kDa outer membrane Protein, Acinetobacter baumannii, Recombinant (His & Myc & SUMO) | Acinetobacter baumannii | E. coli |
May be involved in transporting molecules across the outer membrane. |
Cat No. | Product Name | ||
---|---|---|---|
L1520 | Membrane Protein-targeted Compound Library | 4229 compounds | |