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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T15675 | Tirbanibulin Mesylate | KX2-391 Mesylate,KX01 Mesylate | Microtubule Associated , Src |
Tirbanibulin Mesylate (KX01 Mesylate) is an inhibitor of Src that targets the peptide substrate site of Src (GI50: 9-60 nM in cancer cell lines). | |||
T11578L | Encequidar mesylate | HM30181 mesylate,HM30181A mesylate | P-gp |
Encequidar mesylate (HM30181A mesylate) is a competitive P-glycoprotein inhibitor. | |||
T7212 | Delavirdine mesylate | U 90152 (mesylate),BHAP-U 90152 (mesylate),Delavirdine (mesylate) | HIV Protease , Reverse Transcriptase |
Delavirdine mesylate (BHAP-U 90152 (mesylate)) is a non-nucleoside reverse transcriptase inhibitor (NNRTI). | |||
T2346L | Enasidenib mesylate | AG221 mesylate,AG 221 mesylate,AG-221 mesylate | Dehydrogenase |
Enasidenib mesylate (AG-221 mesylate) is a potent and selective IDH2 mutase inhibitor that promotes differentiation of leukemia myeloid cells for the treatment of acute myeloid leukemia. | |||
T4342 | PF-04929113 Mesylate | PF-04929113 (Mesylate),SNX-5422 Mesylate | HSP , HER |
PF-04929113 Mesylate (SNX-5422 Mesylate), a prodrug of SNX-2112, is an orally available Hsp90 inhibitor (Kd: 41 nM) and also induces Her-2 degradation (IC50: 37 nM). | |||
T13687 | Eribulin mesylate | B1939 mesylate,ER-086526 mesylate,E7389 mesylate | Apoptosis , Others , Microtubule Associated |
Eribulin mesylate (E7389 mesylate) (E7389 mesylate) inhibits the proliferation of cancer cells by binding microtubule proteins and microtubules. Eribulin mesylate (E7389 mesylate) is a microtubule targeting agent that is... | |||
T7547 | Ralfinamide mesylate | FCE-26742A (mesylate) | Sodium Channel |
Ralfinamide mesylate (FCE-26742A (mesylate)) is an orally available Na+ channel blocker. | |||
T11949 | Masupirdine mesylate | SUVN-502 mesylate,SVN-502 mesylate | 5-HT Receptor |
Masupirdine mesylate (SUVN-502 mesylate) is a selective 5-HT6 receptor antagonist that crosses the blood-brain barrier.Masupirdine mesylate is used in the study of neurological disorders such as Alzheimer's disease and d... | |||
T10960L | Darbufelone mesylate | CI-1004 mesylate | Prostaglandin Receptor , LTR |
Darbufelone mesylate (CI-1004 mesylate) inhibited PGF2α and LTB4 in cells. Darbufelone mesylate inhibited PGHS-2 with IC50 value of 0.19 μM and PGHS-1 with IC50 value of 20 μM. | |||
T12059L | Mitoquinone mesylate | MitoQ mesylate,MitoQ10 mesylate | Reactive Oxygen Species |
Mitoquinone mesylate (MitoQ10 mesylate) is a TPP-based, mitochondrially targeted antioxidant to protect against oxidative damage. | |||
T0425 | Pefloxacin Mesylate | Pefloxacinium mesylate | Topoisomerase , Antibacterial , Antibiotic |
Pefloxacin Mesylate (Pefloxacinium mesylate) is a synthetic broad-spectrum fluoroquinolone antibacterial agent active against most gram-negative and gram-positive bacteria. | |||
T2545 | Lomitapide Mesylate | BMS-201038 mesylate,AEGR-733 mesylate | CETP |
Lomitapide Mesylate (BMS-201038 mesylate) is a methanesulfonic acid form of lomitapide, a small molecule inhibitor of microsomal triglyceride transfer protein. | |||
T28978 | Tirilazad mesylate | U-74006 mesylate,U74006 mesylate,U 74006 mesylate,U 74006F mesylate,U-74006F mesylate,U74006F mesylate | Antiviral |
Tirilazad mesylate (U 74006F) is a non-glucocorticoid, lipid peroxidation inhibitor with antiviral activity and neuroprotective activity.Tirilazad mesylate confines intracellular intramembranous foci, attenuates spinal c... | |||
T3634 | Osimertinib mesylate | Mereletinib mesylate,AZD-9291 mesylate | EGFR |
Osimertinib mesylate (Mereletinib mesylate) is an irreversible and mutant selective EGFR inhibitor (IC50s: 12/1 nM for EGFR(L858R) and EGFR(L858R/T790M)). | |||
T2190 | Methiothepin mesylate | Ro 8-6837 mesylate,Metitepine mesylate | Dopamine Receptor , 5-HT Receptor |
Methiothepin mesylate (Metitepine mesylate) is a potent and non-selective 5-HT2 receptor antagonist, used as an antipsychotic. | |||
T71699 | Lanopepden mesylate | GSK 1322322 mesylate,GSK-1322322J mesylate | Antibacterial |
Lanopepden mesylate is a peptide deformylase inhibitor against Staphylococcus aureus. | |||
T6835 | Fenoldopam mesylate | Fenoldopam methanesulfonate,SKF-82526 mesylate,Corlopam mesylate,mesylate,SKF 82526 | Dopamine Receptor |
Fenoldopam mesylate (Corlopam mesylate) is a selective dopamine-1 receptor (DA1) agonist with natriuretic/diuretic properties. It lowers blood pressure through arteriolar vasodilation. | |||
T3533 | Apilimod mesylate | STA 5326 mesylate | IL Receptor , PI3K , Interleukin |
Apilimod mesylate (STA 5326 mesylate) is a potent IL-12/IL-23 inhibitor. | |||
T11043 | Dihydroergocristine mesylate | DHEC (mesylate) | Beta Amyloid |
Dihydroergocristine mesylate (DHEC (mesylate))(DHEC mesylate) is the methanesulfonic acid salt of dihydroergocristine. It has been used as the for the symptomatic treatment of mental deterioration associated with cerebro... | |||
T1336 | Benztropine mesylate | Benzotropine mesylate,Benzatropine mesylate,Benztropine methanesulfonate | Dopamine Receptor , AChR , Histamine Receptor |
Benztropine mesylate (Benztropine methanesulfonate) is a centrally active muscarinic antagonist that has been used in the symptomatic treatment of PARKINSON DISEASE. Benztropine also inhibits the uptake of dopamine. |