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Search Results for " mesylate "

20

Compounds

Cat No. Product Name Synonyms Targets
T15675 Tirbanibulin Mesylate KX2-391 Mesylate,KX01 Mesylate Microtubule Associated , Src
Tirbanibulin Mesylate (KX01 Mesylate) is an inhibitor of Src that targets the peptide substrate site of Src (GI50: 9-60 nM in cancer cell lines).
T11578L Encequidar mesylate HM30181 mesylate,HM30181A mesylate P-gp
Encequidar mesylate (HM30181A mesylate) is a competitive P-glycoprotein inhibitor.
T7212 Delavirdine mesylate U 90152 (mesylate),BHAP-U 90152 (mesylate),Delavirdine (mesylate) HIV Protease , Reverse Transcriptase
Delavirdine mesylate (BHAP-U 90152 (mesylate)) is a non-nucleoside reverse transcriptase inhibitor (NNRTI).
T2346L Enasidenib mesylate AG221 mesylate,AG 221 mesylate,AG-221 mesylate Dehydrogenase
Enasidenib mesylate (AG-221 mesylate) is a potent and selective IDH2 mutase inhibitor that promotes differentiation of leukemia myeloid cells for the treatment of acute myeloid leukemia.
T4342 PF-04929113 Mesylate PF-04929113 (Mesylate),SNX-5422 Mesylate HSP , HER
PF-04929113 Mesylate (SNX-5422 Mesylate), a prodrug of SNX-2112, is an orally available Hsp90 inhibitor (Kd: 41 nM) and also induces Her-2 degradation (IC50: 37 nM).
T13687 Eribulin mesylate B1939 mesylate,ER-086526 mesylate,E7389 mesylate Apoptosis , Others , Microtubule Associated
Eribulin mesylate (E7389 mesylate) (E7389 mesylate) inhibits the proliferation of cancer cells by binding microtubule proteins and microtubules. Eribulin mesylate (E7389 mesylate) is a microtubule targeting agent that is...
T7547 Ralfinamide mesylate FCE-26742A (mesylate) Sodium Channel
Ralfinamide mesylate (FCE-26742A (mesylate)) is an orally available Na+ channel blocker.
T11949 Masupirdine mesylate SUVN-502 mesylate,SVN-502 mesylate 5-HT Receptor
Masupirdine mesylate (SUVN-502 mesylate) is a selective 5-HT6 receptor antagonist that crosses the blood-brain barrier.Masupirdine mesylate is used in the study of neurological disorders such as Alzheimer's disease and d...
T10960L Darbufelone mesylate CI-1004 mesylate Prostaglandin Receptor , LTR
Darbufelone mesylate (CI-1004 mesylate) inhibited PGF2α and LTB4 in cells. Darbufelone mesylate inhibited PGHS-2 with IC50 value of 0.19 μM and PGHS-1 with IC50 value of 20 μM.
T12059L Mitoquinone mesylate MitoQ mesylate,MitoQ10 mesylate Reactive Oxygen Species
Mitoquinone mesylate (MitoQ10 mesylate) is a TPP-based, mitochondrially targeted antioxidant to protect against oxidative damage.
T0425 Pefloxacin Mesylate Pefloxacinium mesylate Topoisomerase , Antibacterial , Antibiotic
Pefloxacin Mesylate (Pefloxacinium mesylate) is a synthetic broad-spectrum fluoroquinolone antibacterial agent active against most gram-negative and gram-positive bacteria.
T2545 Lomitapide Mesylate BMS-201038 mesylate,AEGR-733 mesylate CETP
Lomitapide Mesylate (BMS-201038 mesylate) is a methanesulfonic acid form of lomitapide, a small molecule inhibitor of microsomal triglyceride transfer protein.
T28978 Tirilazad mesylate U-74006 mesylate,U74006 mesylate,U 74006 mesylate,U 74006F mesylate,U-74006F mesylate,U74006F mesylate Antiviral
Tirilazad mesylate (U 74006F) is a non-glucocorticoid, lipid peroxidation inhibitor with antiviral activity and neuroprotective activity.Tirilazad mesylate confines intracellular intramembranous foci, attenuates spinal c...
T3634 Osimertinib mesylate Mereletinib mesylate,AZD-9291 mesylate EGFR
Osimertinib mesylate (Mereletinib mesylate) is an irreversible and mutant selective EGFR inhibitor (IC50s: 12/1 nM for EGFR(L858R) and EGFR(L858R/T790M)).
T2190 Methiothepin mesylate Ro 8-6837 mesylate,Metitepine mesylate Dopamine Receptor , 5-HT Receptor
Methiothepin mesylate (Metitepine mesylate) is a potent and non-selective 5-HT2 receptor antagonist, used as an antipsychotic.
T71699 Lanopepden mesylate GSK 1322322 mesylate,GSK-1322322J mesylate Antibacterial
Lanopepden mesylate is a peptide deformylase inhibitor against Staphylococcus aureus.
T6835 Fenoldopam mesylate Fenoldopam methanesulfonate,SKF-82526 mesylate,Corlopam mesylate,mesylate,SKF 82526 Dopamine Receptor
Fenoldopam mesylate (Corlopam mesylate) is a selective dopamine-1 receptor (DA1) agonist with natriuretic/diuretic properties. It lowers blood pressure through arteriolar vasodilation.
T3533 Apilimod mesylate STA 5326 mesylate IL Receptor , PI3K , Interleukin
Apilimod mesylate (STA 5326 mesylate) is a potent IL-12/IL-23 inhibitor.
T11043 Dihydroergocristine mesylate DHEC (mesylate) Beta Amyloid
Dihydroergocristine mesylate (DHEC (mesylate))(DHEC mesylate) is the methanesulfonic acid salt of dihydroergocristine. It has been used as the for the symptomatic treatment of mental deterioration associated with cerebro...
T1336 Benztropine mesylate Benzotropine mesylate,Benzatropine mesylate,Benztropine methanesulfonate Dopamine Receptor , AChR , Histamine Receptor
Benztropine mesylate (Benztropine methanesulfonate) is a centrally active muscarinic antagonist that has been used in the symptomatic treatment of PARKINSON DISEASE. Benztropine also inhibits the uptake of dopamine.

Compounds

Tirbanibulin Mesylate
T15675
Synonym: KX2-391 Mesylate,KX01 Mesylate
Target: Microtubule Associated, Src
Encequidar mesylate
T11578L
Synonym: HM30181 mesylate,HM30181A mesylate
Target: P-gp
Delavirdine mesylate
T7212
Synonym: U 90152 (mesylate),BHAP-U 90152 (mesylate),Delavirdine (mesylate)
Target: HIV Protease, Reverse Transcriptase
Enasidenib mesylate
T2346L
Synonym: AG221 mesylate,AG 221 mesylate,AG-221 mesylate
Target: Dehydrogenase
PF-04929113 Mesylate
T4342
Synonym: PF-04929113 (Mesylate),SNX-5422 Mesylate
Target: HSP, HER
Eribulin mesylate
T13687
Synonym: B1939 mesylate,ER-086526 mesylate,E7389 mesylate
Target: Apoptosis, Others, Microtubule Associated
Ralfinamide mesylate
T7547
Synonym: FCE-26742A (mesylate)
Target: Sodium Channel
Masupirdine mesylate
T11949
Synonym: SUVN-502 mesylate,SVN-502 mesylate
Target: 5-HT Receptor
Darbufelone mesylate
T10960L
Synonym: CI-1004 mesylate
Target: Prostaglandin Receptor, LTR
Mitoquinone mesylate
T12059L
Synonym: MitoQ mesylate,MitoQ10 mesylate
Target: Reactive Oxygen Species
Pefloxacin Mesylate
T0425
Synonym: Pefloxacinium mesylate
Target: Topoisomerase, Antibacterial, Antibiotic
Lomitapide Mesylate
T2545
Synonym: BMS-201038 mesylate,AEGR-733 mesylate
Target: CETP
Tirilazad mesylate
T28978
Synonym: U-74006 mesylate,U74006 mesylate,U 74006 mesylate,U 74006F mesylate,U-74006F mesylate,U74006F mesylate
Target: Antiviral
Osimertinib mesylate
T3634
Synonym: Mereletinib mesylate,AZD-9291 mesylate
Target: EGFR
Methiothepin mesylate
T2190
Synonym: Ro 8-6837 mesylate,Metitepine mesylate
Target: Dopamine Receptor, 5-HT Receptor
Lanopepden mesylate
T71699
Synonym: GSK 1322322 mesylate,GSK-1322322J mesylate
Target: Antibacterial
Fenoldopam mesylate
T6835
Synonym: Fenoldopam methanesulfonate,SKF-82526 mesylate,Corlopam mesylate,mesylate,SKF 82526
Target: Dopamine Receptor
Apilimod mesylate
T3533
Synonym: STA 5326 mesylate
Target: IL Receptor, PI3K, Interleukin
Dihydroergocristine mesylate
T11043
Synonym: DHEC (mesylate)
Target: Beta Amyloid
Benztropine mesylate
T1336
Synonym: Benzotropine mesylate,Benzatropine mesylate,Benztropine methanesulfonate
Target: Dopamine Receptor, AChR, Histamine Receptor
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TargetMol