Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Masupirdine mesylate (SUVN-502 mesylate) shows high selectivity over 5-HT2A receptor and other 100 target sites, and has potential for treatment of Alzheimer's disease. Masupirdine mesylate (SUVN-502 mesylate) is a potent, selective, orally bioavailable, and brain penetrant 5-HT6 receptor antagonist (Ki of 2.04 nM for human 5-HT6 receptor).
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
25 mg | In stock | $ 920.00 | |
50 mg | In stock | $ 1,180.00 | |
100 mg | In stock | $ 1,790.00 |
Description | Masupirdine mesylate (SUVN-502 mesylate) shows high selectivity over 5-HT2A receptor and other 100 target sites, and has potential for treatment of Alzheimer's disease. Masupirdine mesylate (SUVN-502 mesylate) is a potent, selective, orally bioavailable, and brain penetrant 5-HT6 receptor antagonist (Ki of 2.04 nM for human 5-HT6 receptor). |
Targets&IC50 | 5-HT6 receptor:2.04 nM (ki) |
Synonyms | SUVN-502 mesylate |
Molecular Weight | 670.61 |
Formula | C23H32BrN3O9S3 |
CAS No. | 1791396-46-7 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
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Masupirdine mesylate 1791396-46-7 GPCR/G Protein Neuroscience 5-HT Receptor SUVN-502 Mesylate Masupirdine Mesylate SUVN-502 mesylate SUVN 502 Mesylate SUVN502 Mesylate inhibitor inhibit