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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T26834 | BL-1020 Mesylate | CYP-1020 Mesylate | Dopamine Receptor , GABA Receptor |
BL-1020 Mesylate (CYP-1020 Mesylate) is an orally available GABA A receptor agonist and D2 antagonist that decreases dopamine activity and enhances GABAA activity.BL-1020 Mesylate has been used in the study of schizophre... | |||
T10922 | CYP11B2-IN-1 | P450 | |
CYP11B2-IN-1 is an effective and selective inhibitor of CYP11B2 with IC50s of 2.3 nM and 142 nM for CYP11B2 and CYP11B1. | |||
T10923 | CYP17-IN-1 | P450 | |
CYP17-IN-1 is an effective oral inhibitor of CYP17 that can inhibit CYP17 in rats and humans with IC50 of 15.8 and 20.1 nM. | |||
T5786 | TETRAHYDROPIPERINE | Cosmoperine | P450 , TRP/TRPV Channel |
Tetrahydropiperine (Cosmoperine) is a natural product derived from piperine, can be used to treat convulsion, epilepsy, relieve pain, and control insects. | |||
T1011 | Itraconazole | R51211 | P450 , Hedgehog/Smoothened , Antibiotic , Autophagy , Antifungal |
Itraconazole (R51211) is a triazole antifungal agent that inhibits cytochrome P-450-dependent enzymes required for ERGOSTEROL synthesis. | |||
T27109 | CYP1A1 inhibitor 8a | ||
CYP1A1 inhibitor 8a is a potent and selective CYP1A1 inhibitor. It antagonizes B[a]P mediated activation of aromatic hydrocarbon receptor (AhR) in yeast cells, thereby protects human cells from CYP1A1-mediated B[a]P toxi... | |||
T6S0923 | Hypericin | Hypericine,Cyclosan | Apoptosis , Antiviral , Influenza Virus , Tyrosine Kinases , Antibacterial , PKC |
1. Hypericin (Cyclosan) has antineoplastic activity. 2. Hypericin has antibiotic and antiviral activities. 3. Hypericin has antidepressive activity through inhibiting monoamine oxidase enzyme. 4. Hypericin inhibits RANKL... | |||
T6420 | BMS-707035 | HIV Protease | |
BMS-707035 is a specific HIV-I integrase (IN) inhibitor with IC50 of 15 nM. Phase 2. | |||
T72501 | CYP4A11/CYP4F2-IN-1 | P450 | |
CYP4A11/CYP4F2-IN-1 is a cytochrome P450 (CYP) 4A11 and CYP4F2 inhibitor. CYP4A11/CYP4F2-IN-1 can be used to study kidney diseases and cardiovascular and cerebrovascular diseases. | |||
T67916 | CYP4A11/CYP4F2-IN-2 | P450 | |
CYP4A11/CYP4F2-IN-2 is a potent and orally active dual inhibitor of cytochrome P450 (CYP) 4A11 and CYP4F2, with IC50 values of 140 nM and 40 nM, respectively. CYP4A11/CYP4F2-IN-2 can be extracted from liver and kidney an... | |||
T77698 | HCYP3A4 Fluorogenic substrate 1 | Others | |
hCYP3A4 Fluorogenic substrate 1 is a phthalimide derivative and shows low activity against COX. | |||
T73040 | CYP1B1-IN-4 | P450 | |
CYP1B1-IN-4, a 2,4-diarylthiazole compound, exhibits selective inhibition of CYP1B1 (IC50=0.2 nM), demonstrating minimal cytotoxicity and high stability in human and rat liver microsomes [1]. | |||
T6814 | Cyproheptadine hydrochloride | Periactin hydrochloride,Anarexol,Cyproheptadine HCl,Nuran | 5-HT Receptor |
Cyproheptadine hydrochloride (Periactin hydrochloride) is a hydrochloride salt form of cyproheptadine which is a histamine receptor antagonist. | |||
T5709 | Cyperotundone | Others | |
Cyperotundone is a natural product from Cyperus rotundus | |||
T0168 | Estradiol (cypionate) | Depofemin,Estradiol cypionate | Estrogen Receptor/ERR , Estrogen/progestogen Receptor |
Estradiol cypionate (Depofemin), the 17 β-cyclopentylpropinate ester of estradiol, inhibits ET-1 synthesis via estrogen receptor. | |||
T1025 | Tranylcypromine (2-PCPA) hydrochloride | Tranylcypromine (2-PCPA) HCl,SKF-385 HCl | Histone Demethylase , MAO |
Tranylcypromine (2-PCPA) hydrochloride (SKF-385 HCl), a Monoamine Oxidase inhibitor, is effective in the treatment of major depression, dysthymic disorder, and atypical depression. | |||
T73042 | CYP1B1-IN-5 | P450 | |
CYP1B1-IN-5 is a selective and potent cytochrome P450 1B1 (CYP1B1) inhibitor with an IC50 of 4.7 nM.CYP1B1-IN-5 can be used for the study of metabolism-related diseases. | |||
T0174 | Cyproheptadine hydrochloride sesquihydrate | Peritol,Periactin hydrochloride,Cyproheptadine hydrochloride | 5-HT Receptor , Histone Methyltransferase , Histamine Receptor |
Cyproheptadine hydrochloride sesquihydrate (Peritol), an antihistamine, is an antagonist of serotonin and histamine2. | |||
T19213 | Boldenone Cypionate | Others , Androgen Receptor | |
Boldenone Cypionate is an androgenic anabolic steroid used by recreational bodybuilders and regular gym members. | |||
T20968 | CyPPA | Potassium Channel , Dopamine Receptor | |
CyPPA, a subtype-selective positive modulator of SK channels, decreased spontaneous firing rate, increased the duration of the apamin-sensitive afterhyperpolarization. |