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20

Compounds

Cat No. Product Name Synonyms Targets
T26834 BL-1020 Mesylate CYP-1020 Mesylate Dopamine Receptor , GABA Receptor
BL-1020 Mesylate (CYP-1020 Mesylate) is an orally available GABA A receptor agonist and D2 antagonist that decreases dopamine activity and enhances GABAA activity.BL-1020 Mesylate has been used in the study of schizophre...
T10922 CYP11B2-IN-1 P450
CYP11B2-IN-1 is an effective and selective inhibitor of CYP11B2 with IC50s of 2.3 nM and 142 nM for CYP11B2 and CYP11B1.
T10923 CYP17-IN-1 P450
CYP17-IN-1 is an effective oral inhibitor of CYP17 that can inhibit CYP17 in rats and humans with IC50 of 15.8 and 20.1 nM.
T5786 TETRAHYDROPIPERINE Cosmoperine P450 , TRP/TRPV Channel
Tetrahydropiperine (Cosmoperine) is a natural product derived from piperine, can be used to treat convulsion, epilepsy, relieve pain, and control insects.
T1011 Itraconazole R51211 P450 , Hedgehog/Smoothened , Antibiotic , Autophagy , Antifungal
Itraconazole (R51211) is a triazole antifungal agent that inhibits cytochrome P-450-dependent enzymes required for ERGOSTEROL synthesis.
T27109 CYP1A1 inhibitor 8a
CYP1A1 inhibitor 8a is a potent and selective CYP1A1 inhibitor. It antagonizes B[a]P mediated activation of aromatic hydrocarbon receptor (AhR) in yeast cells, thereby protects human cells from CYP1A1-mediated B[a]P toxi...
T6S0923 Hypericin Hypericine,Cyclosan Apoptosis , Antiviral , Influenza Virus , Tyrosine Kinases , Antibacterial , PKC
1. Hypericin (Cyclosan) has antineoplastic activity. 2. Hypericin has antibiotic and antiviral activities. 3. Hypericin has antidepressive activity through inhibiting monoamine oxidase enzyme. 4. Hypericin inhibits RANKL...
T6420 BMS-707035 HIV Protease
BMS-707035 is a specific HIV-I integrase (IN) inhibitor with IC50 of 15 nM. Phase 2.
T72501 CYP4A11/CYP4F2-IN-1 P450
CYP4A11/CYP4F2-IN-1 is a cytochrome P450 (CYP) 4A11 and CYP4F2 inhibitor. CYP4A11/CYP4F2-IN-1 can be used to study kidney diseases and cardiovascular and cerebrovascular diseases.
T67916 CYP4A11/CYP4F2-IN-2 P450
CYP4A11/CYP4F2-IN-2 is a potent and orally active dual inhibitor of cytochrome P450 (CYP) 4A11 and CYP4F2, with IC50 values of 140 nM and 40 nM, respectively. CYP4A11/CYP4F2-IN-2 can be extracted from liver and kidney an...
T77698 HCYP3A4 Fluorogenic substrate 1 Others
hCYP3A4 Fluorogenic substrate 1 is a phthalimide derivative and shows low activity against COX.
T73040 CYP1B1-IN-4 P450
CYP1B1-IN-4, a 2,4-diarylthiazole compound, exhibits selective inhibition of CYP1B1 (IC50=0.2 nM), demonstrating minimal cytotoxicity and high stability in human and rat liver microsomes [1].
T6814 Cyproheptadine hydrochloride Periactin hydrochloride,Anarexol,Cyproheptadine HCl,Nuran 5-HT Receptor
Cyproheptadine hydrochloride (Periactin hydrochloride) is a hydrochloride salt form of cyproheptadine which is a histamine receptor antagonist.
T5709 Cyperotundone Others
Cyperotundone is a natural product from Cyperus rotundus
T0168 Estradiol (cypionate) Depofemin,Estradiol cypionate Estrogen Receptor/ERR , Estrogen/progestogen Receptor
Estradiol cypionate (Depofemin), the 17 β-cyclopentylpropinate ester of estradiol, inhibits ET-1 synthesis via estrogen receptor.
T1025 Tranylcypromine (2-PCPA) hydrochloride Tranylcypromine (2-PCPA) HCl,SKF-385 HCl Histone Demethylase , MAO
Tranylcypromine (2-PCPA) hydrochloride (SKF-385 HCl), a Monoamine Oxidase inhibitor, is effective in the treatment of major depression, dysthymic disorder, and atypical depression.
T73042 CYP1B1-IN-5 P450
CYP1B1-IN-5 is a selective and potent cytochrome P450 1B1 (CYP1B1) inhibitor with an IC50 of 4.7 nM.CYP1B1-IN-5 can be used for the study of metabolism-related diseases.
T0174 Cyproheptadine hydrochloride sesquihydrate Peritol,Periactin hydrochloride,Cyproheptadine hydrochloride 5-HT Receptor , Histone Methyltransferase , Histamine Receptor
Cyproheptadine hydrochloride sesquihydrate (Peritol), an antihistamine, is an antagonist of serotonin and histamine2.
T19213 Boldenone Cypionate Others , Androgen Receptor
Boldenone Cypionate is an androgenic anabolic steroid used by recreational bodybuilders and regular gym members.
T20968 CyPPA Potassium Channel , Dopamine Receptor
CyPPA, a subtype-selective positive modulator of SK channels, decreased spontaneous firing rate, increased the duration of the apamin-sensitive afterhyperpolarization.

Compounds

BL-1020 Mesylate
T26834
Synonym: CYP-1020 Mesylate
Target: Dopamine Receptor, GABA Receptor
CYP11B2-IN-1
T10922
Synonym:
Target: P450
CYP17-IN-1
T10923
Synonym:
Target: P450
TETRAHYDROPIPERINE
T5786
Synonym: Cosmoperine
Target: P450, TRP/TRPV Channel
Itraconazole
T1011
Synonym: R51211
Target: P450, Hedgehog/Smoothened, Antibiotic, Autophagy, Antifungal
CYP1A1 inhibitor 8a
T27109
Synonym:
Target:
Hypericin
T6S0923
Synonym: Hypericine,Cyclosan
Target: Apoptosis, Antiviral, Influenza Virus, Tyrosine Kinases, Antibacterial, PKC
BMS-707035
T6420
Synonym:
Target: HIV Protease
CYP4A11/CYP4F2-IN-1
T72501
Synonym:
Target: P450
CYP4A11/CYP4F2-IN-2
T67916
Synonym:
Target: P450
hCYP3A4 Fluorogenic substrate 1
T77698
Synonym:
Target: Others
CYP1B1-IN-4
T73040
Synonym:
Target: P450
Cyproheptadine hydrochloride
T6814
Synonym: Periactin hydrochloride,Anarexol,Cyproheptadine HCl,Nuran
Target: 5-HT Receptor
Cyperotundone
T5709
Synonym:
Target: Others
Estradiol (cypionate)
T0168
Synonym: Depofemin,Estradiol cypionate
Target: Estrogen Receptor/ERR, Estrogen/progestogen Receptor
Tranylcypromine (2-PCPA) hydrochloride
T1025
Synonym: Tranylcypromine (2-PCPA) HCl,SKF-385 HCl
Target: Histone Demethylase, MAO
CYP1B1-IN-5
T73042
Synonym:
Target: P450
Cyproheptadine hydrochloride sesquihydrate
T0174
Synonym: Peritol,Periactin hydrochloride,Cyproheptadine hydrochloride
Target: 5-HT Receptor, Histone Methyltransferase, Histamine Receptor
Boldenone Cypionate
T19213
Synonym:
Target: Others, Androgen Receptor
CyPPA
T20968
Synonym:
Target: Potassium Channel, Dopamine Receptor
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TargetMol