Powder: -20°C for 3 years | In solvent: -80°C for 1 year
CYP17-IN-1 is an effective oral inhibitor of CYP17 that can inhibit CYP17 in rats and humans with IC50 of 15.8 and 20.1 nM.
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
1 mg | In stock | $ 195.00 | |
2 mg | In stock | $ 293.00 | |
5 mg | In stock | $ 448.00 | |
10 mg | In stock | $ 658.00 | |
25 mg | In stock | $ 987.00 | |
50 mg | In stock | $ 1,380.00 | |
100 mg | In stock | $ 1,890.00 | |
1 mL * 10 mM (in DMSO) | In stock | $ 437.00 |
Description | CYP17-IN-1 is an effective oral inhibitor of CYP17 that can inhibit CYP17 in rats and humans with IC50 of 15.8 and 20.1 nM. |
Targets&IC50 | Rat CYP17:15.8 nM , Human CYP17:20.1 nM |
In vitro | The IC50 value of CYP17-IN-1 for CYP3A4 is 8.5 µM[1]. |
In vivo | CYP17-IN-1 dose-dependently reduced plasma testosterone levels in Sprague-Dawley rats[1]. |
Molecular Weight | 312.4 |
Formula | C18H17FN2S |
CAS No. | 2093317-51-0 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 3.12 mg/mL (10 mM), Sonification is recommended
You can also refer to dose conversion for different animals. More
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CYP17-IN-1 2093317-51-0 Metabolism P450 CYP17IN1 CYP17 IN 1 CYP-17-IN-1 inhibitor inhibit